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Thi M-D Nguyen

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Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Peter W Schiller
Potent opioid peptide agonists containing 4'-[N-((4'-phenyl)-phenethyl)carboxamido]phenylalanine (Bcp) in place of Tyr.
Stefica Horvat; Maja Roscić; Carole Lemieux; Thi M-D Nguyen; Peter W Schiller
Formation pathways and opioid activity data for 3-hydroxypyridinium compounds derived from glucuronic acid and opioid peptides by Maillard processes.
Yixin Lu; Tze Keong Lum; Yoon Wui Leow Augustine; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Peter W Schiller
Replacement of the N-terminal tyrosine residue in opioid peptides with 3-(2,6-dimethyl-4-carbamoylphenyl)propanoic acid (Dcp) results in novel opioid antagonists.

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2008: Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Peter W Schiller
Potent opioid peptide agonists containing 4'-[N-((4'-phenyl)-phenethyl)carboxamido]phenylalanine (Bcp) in place of Tyr.
Chemical biology & drug design 2008;72(5):337-40.
2007: Stefica Horvat; Maja Roscić; Carole Lemieux; Thi M-D Nguyen; Peter W Schiller
Formation pathways and opioid activity data for 3-hydroxypyridinium compounds derived from glucuronic acid and opioid peptides by Maillard processes.
Chemical biology & drug design 2007;70(1):30-9.
2006: Yixin Lu; Tze Keong Lum; Yoon Wui Leow Augustine; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Peter W Schiller
Replacement of the N-terminal tyrosine residue in opioid peptides with 3-(2,6-dimethyl-4-carbamoylphenyl)propanoic acid (Dcp) results in novel opioid antagonists.
Journal of medicinal chemistry 2006;49(17):5382-5.
2003: Claire L Neilan; Adam J Janvey; Elizabeth A Bolan; Irena Berezowska; Thi M-D Nguyen; Peter W Schiller; Gavril W Pasternak
Characterization of the binding of [3H][Dmt1]H-Dmt-D-Arg-Phe-Lys-NH2, a highly potent opioid peptide.
The Journal of pharmacology and experimental therapeutics 2003;306(2):430-6.
2003: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Yixin Lu
Conversion of delta-, kappa- and mu-receptor selective opioid peptide agonists into delta-, kappa- and mu-selective antagonists.
Life sciences 2003;73(6):691-8.
2002: Pal Riba; Yong Ben; Thi M-D Nguyen; Susanna Furst; Peter W Schiller; Nancy M Lee
[Dmt(1)]DALDA is highly selective and potent at mu opioid receptors, but is not cross-tolerant with systemic morphine.
Current medicinal chemistry 2002;9(1):31-9.
2001: Yixin Lu; Thi M-D Nguyen; Grazyna Weltrowska; Irena Berezowska; Carole Lemieux; Nga N Chung; Peter W Schiller
[2',6'-Dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: potent and selective kappa opioid antagonists.
Journal of medicinal chemistry 2001;44(19):3048-53.
2001: Claire L Neilan; Thi M-D Nguyen; Peter W Schiller; Gavril W Pasternak
Pharmacological characterization of the dermorphin analog [Dmt(1)]DALDA, a highly potent and selective mu-opioid peptide.
European journal of pharmacology 2001;419(1):15-23.
2000: Peter W Schiller; Thi M-D Nguyen; Irena Berezowska; S Dupuis; Grazyna Weltrowska; Nga N Chung; Carole Lemieux
Synthesis and in vitro opioid activity profiles of DALDA analogues.
European journal of medicinal chemistry 2000;35(10):895-901.
2000: Peter W Schiller; Irena Berezowska; Thi M-D Nguyen; Ralf Schmidt; Carole Lemieux; Nga N Chung; M L Falcone-Hindley; W Yao; J Liu; S Iwama; A B Smith; Ralph Hirschmann
Novel ligands lacking a positive charge for the delta- and mu-opioid receptors.
Journal of medicinal chemistry 2000;43(4):551-9.
1999: Peter W Schiller; Marian E Fundytus; L Merovitz; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Terence J Coderre
The opioid mu agonist/delta antagonist DIPP-NH(2)[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats.
Journal of medicinal chemistry 1999;42(18):3520-6.
1999: Peter W Schiller; Grazyna Weltrowska; Irena Berezowska; Thi M-D Nguyen; Brian C Wilkes; Carole Lemieux; Nga N Chung
The TIPP opioid peptide family: development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists.
Biopolymers 1999;51(6):411-25.
1999: Peter W Schiller; Grazyna Weltrowska; Ralf Schmidt; Irena Berezowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Katharine A Carpenter; Brian C Wilkes
Subtleties of structure-agonist versus antagonist relationships of opioid peptides and peptidomimetics.
Journal of receptor and signal transduction research 1999;19(1-4):573-88.
1998: Brian C Wilkes; Thi M-D Nguyen; Grazyna Weltrowska; Katharine A Carpenter; Carole Lemieux; Nga N Chung; Peter W Schiller
The receptor-bound conformation of H-Tyr-Tic-(Phe-Phe)-OH-related delta-opioid antagonists contains all trans peptide bonds.
The journal of peptide research : official journal of the American Peptide Society 1998;51(5):386-94.
1993: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Brian C Wilkes; Nga N Chung; Carole Lemieux
TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity.
Journal of medicinal chemistry 1993;36(21):3182-7.
1993: B J Marsden; Thi M-D Nguyen; Peter W Schiller
Spontaneous degradation via diketopiperazine formation of peptides containing a tetrahydroisoquinoline-3-carboxylic acid residue in the 2-position of the peptide sequence.
International journal of peptide and protein research 1993;41(3):313-6.
1993: Peter W Schiller; Thi M-D Nguyen; Grazyna Weltrowska; Nga N Chung; Carole Lemieux; B J Marsden; Brian C Wilkes
The use of conformational restriction and molecular modeling techniques in the development of receptor-specific opioid peptide agonists and antagonists.
NIDA research monograph 1993;134():238-52.
1992: Peter W Schiller; Thi M-D Nguyen; Grazyna Weltrowska; Brian C Wilkes; B J Marsden; Carole Lemieux; Nga N Chung
Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists.
Proceedings of the National Academy of Sciences of the United States of America 1992;89(24):11871-5.
1992: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Brian C Wilkes; Nga N Chung; Carole Lemieux
Conformationally restricted deltorphin analogues.
Journal of medicinal chemistry 1992;35(21):3956-61.
1991: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; B J Marsden; Brian C Wilkes
Conformational restriction of the phenylalanine residue in a cyclic opioid peptide analogue: effects on receptor selectivity and stereospecificity.
Journal of medicinal chemistry 1991;34(10):3125-32.
1990: Peter W Schiller; Thi M-D Nguyen; Nga N Chung; G Dionne; R Martel
Peripheral antinociceptive effect of an extremely mu-selective polar dermorphin analog (DALDA).
Progress in clinical and biological research 1990;328():53-6.
1989: Peter W Schiller; Thi M-D Nguyen; Nga N Chung; Carole Lemieux
Dermorphin analogues carrying an increased positive net charge in their "message" domain display extremely high mu opioid receptor selectivity.
Journal of medicinal chemistry 1989;32(3):698-703.
1987: Peter W Schiller; Thi M-D Nguyen; L A Maziak; Brian C Wilkes; Carole Lemieux
Structure-activity relationships of cyclic opioid peptide analogues containing a phenylalanine residue in the 3-position.
Journal of medicinal chemistry 1987;30(11):2094-9.
1987: Peter W Schiller; L A Maziak; Thi M-D Nguyen; J Godin; R Garcia; A DeLéan; M Cantin
Superactive analogs of the atrial natriuretic peptide (ANP).
Biochemical and biophysical research communications 1987;143(2):499-505.
1986: Peter W Schiller; L A Maziak; Carole Lemieux; Thi M-D Nguyen
Side chain to side chain cyclization of an enkephalin analog results in loss of opioid receptor selectivity.
International journal of peptide and protein research 1986;28(5):493-7.
1985: Peter W Schiller; Thi M-D Nguyen; Carole Lemieux; L A Maziak
Synthesis and activity profiles of novel cyclic opioid peptide monomers and dimers.
Journal of medicinal chemistry 1985;28(12):1766-71.
1985: Peter W Schiller; Thi M-D Nguyen; Carole Lemieux; L A Maziak
A novel side-chain-linked antiparallel cyclic dimer of enkephalin.
FEBS letters 1985;191(2):231-4.
1985: Peter W Schiller; L Maziak; Thi M-D Nguyen; J Godin; R Garcia; A De Léan; M Cantin
Synthesis and biological activity of a linear fragment of the atrial natriuretic factor (ANF).
Biochemical and biophysical research communications 1985;131(3):1056-62.
1985: Peter W Schiller; Thi M-D Nguyen; L Maziak; Carole Lemieux
A novel cyclic opioid peptide analog showing high preference for mu-receptors.
Biochemical and biophysical research communications 1985;127(2):558-64.