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William Padgett

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Dan Shi; William L Padgett; John W Daly
Caffeine analogs: effects on ryanodine-sensitive calcium-release channels and GABAA receptors.
Christa E Müller; Mark Thorand; Ramatullah Qurishi; Martina Diekmann; Kenneth Alan Jacobson; William L Padgett; John W Daly
Imidazo[2,1-i]purin-5-ones and related tricyclic water-soluble purine derivatives: potent A(2A)- and A(3)-adenosine receptor antagonists.
John W Daly; Tara Gupta; William L Padgett; Xue-Feng Pei
6beta-Acyloxy(nor)tropanes: affinities for antagonist/agonist binding sites on transfected and native muscarinic receptors.

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All Publications

2003: Dan Shi; William L Padgett; John W Daly
Caffeine analogs: effects on ryanodine-sensitive calcium-release channels and GABAA receptors.
Cellular and molecular neurobiology 2003;23(3):331-47.
2002: Christa E Müller; Mark Thorand; Ramatullah Qurishi; Martina Diekmann; Kenneth Alan Jacobson; William L Padgett; John W Daly
Imidazo[2,1-i]purin-5-ones and related tricyclic water-soluble purine derivatives: potent A(2A)- and A(3)-adenosine receptor antagonists.
Journal of medicinal chemistry 2002;45(16):3440-50.
2000: John W Daly; Tara Gupta; William L Padgett; Xue-Feng Pei
6beta-Acyloxy(nor)tropanes: affinities for antagonist/agonist binding sites on transfected and native muscarinic receptors.
Journal of medicinal chemistry 2000;43(13):2514-22.
2000: S F Lu; Brian Herbert; Günter Haufe; K W Laue; William L Padgett; O Oshunleti; John W Daly; Kenneth L Kirk
Syntheses of (R)- and (S)-2- and 6-fluoronorepinephrine and (R)- and (S)-2- and 6-fluoroepinephrine: effect of stereochemistry on fluorine-induced adrenergic selectivities.
Journal of medicinal chemistry 2000;43(8):1611-9.
1998: Xue-Feng Pei; Tara Gupta; B Badio; William L Padgett; John W Daly
6beta-Acetoxynortropane: a potent muscarinic agonist with apparent selectivity toward M2-receptors.
Journal of medicinal chemistry 1998;41(12):2047-55.
1997: John W Daly; William L Padgett; R L Saunders; John F Cover
Absence of tetrodotoxins in a captive-raised riparian frog, Atelopus varius.
Toxicon : official journal of the International Society on Toxinology 1997;35(5):705-9.
1997: B Badio; H Martin Garraffo; William L Padgett; N H Greig; John W Daly
Pseudophrynaminol: a potent noncompetitive blocker of nicotinic receptor-channels.
Biochemical pharmacology 1997;53(5):671-6.
1997: B Badio; H Martin Garraffo; C V Plummer; William L Padgett; John W Daly
Synthesis and nicotinic activity of epiboxidine: an isoxazole analogue of epibatidine.
European journal of pharmacology 1997;321(2):189-94.
1997: B Badio; William L Padgett; John W Daly
Ibogaine: a potent noncompetitive blocker of ganglionic/neuronal nicotinic receptors.
Molecular pharmacology 1997;51(1):1-5.
1996: B Badio; D Shi; Y Shin; K D Hutchinson; William L Padgett; John W Daly
Spiropyrrolizidines: a new class of blockers of nicotinic receptors.
Biochemical pharmacology 1996;52(6):933-9.
1996: AM van Rhee; S M Siddiqi; Neli Melman; D Shi; William L Padgett; John W Daly; Kenneth Alan Jacobson
Tetrahydrobenzothiophenone derivatives as a novel class of adenosine receptor antagonists.
Journal of medicinal chemistry 1996;39(2):398-406.
1995: John W Daly; J Lueders; William L Padgett; Y Shin; F Gusovsky
Maitotoxin-elicited calcium influx in cultured cells. Effect of calcium-channel blockers.
Biochemical pharmacology 1995;50(8):1187-97.
1993: Kenneth Alan Jacobson; O Nikodijević; William L Padgett; C Gallo-Rodriguez; M Maillard; John W Daly
8-(3-Chlorostyryl)caffeine (CSC) is a selective A2-adenosine antagonist in vitro and in vivo.
FEBS letters 1993;323(1-2):141-4.
1993: John W Daly; William L Padgett; S I Secunda; R D Thompson; R A Olsson
Structure-activity relationships for 2-substituted adenosines at A1 and A2 adenosine receptors.
Pharmacology 1993;46(2):91-100.
1992: F Gusovsky; William L Padgett; C R Creveling; John W Daly
Interaction of pumiliotoxin B with an "alkaloid-binding domain" on the voltage-dependent sodium channel.
Molecular pharmacology 1992;42(6):1104-8.
1992: John W Daly; William L Padgett
Agonist activity of 2- and 5'-substituted adenosine analogs and their N6-cycloalkyl derivatives at A1- and A2-adenosine receptors coupled to adenylate cyclase.
Biochemical pharmacology 1992;43(5):1089-93.
1992: I Hide; William L Padgett; Kenneth Alan Jacobson; John W Daly
A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase.
Molecular pharmacology 1992;41(2):352-9.
1992: C R Creveling; William L Padgett; E T McNeal; L A Cohen; K L Kirk
Incorporation of 2-fluorohistidine in murine protein in vivo.
Life sciences 1992;51(15):1197-204.
1992: OKSOON CHOI; William L Padgett; John W Daly
Effects of the amphiphilic peptides melittin and mastoparan on calcium influx, phosphoinositide breakdown and arachidonic acid release in rat pheochromocytoma PC12 cells.
The Journal of pharmacology and experimental therapeutics 1992;260(1):369-75.
1991: John W Daly; Y Nishizawa; William L Padgett; T Tokuyama; A L Smith; A B Holmes; C Kibayashi; R S Aronstam
5,8-disubstituted indolizidines: a new class of noncompetitive blockers for nicotinic receptor-channels.
Neurochemical research 1991;16(11):1213-8.
1991: John W Daly; Y Nishizawa; William L Padgett; T Tokuyama; P J McCloskey; L Waykole; A G Schultz; R S Aronstam
Decahydroquinoline alkaloids: noncompetitive blockers for nicotinic acetylcholine receptor-channels in pheochromocytoma cells and Torpedo electroplax.
Neurochemical research 1991;16(11):1207-12.
1991: A Adejare; J Y Nie; D Hebel; L E Brackett; OKSOON CHOI; F Gusovsky; William L Padgett; John W Daly; C R Creveling; K L Kirk
Effect of fluorine substitution on the adrenergic properties of 3-(tert-butylamino)-1-(3,4-dihydroxyphenoxy)-2-propanol.
Journal of medicinal chemistry 1991;34(3):1063-8.
1990: F Gusovsky; Y Nishizawa; William L Padgett; E T McNeal; K Rice; C H Kim; C R Creveling; John W Daly
Voltage-dependent sodium channels in synaptoneurosomes: studies with 22Na+ influx and [3H]saxitoxin and [3H]batrachotoxinin-A 20-alpha-benzoate binding. Effects of proparacaine isothiocyanate.
Brain research 1990;518(1-2):101-6.
1990: OKSOON CHOI; William L Padgett; Y Nishizawa; F Gusovsky; T Yasumoto; John W Daly
Maitotoxin: effects on calcium channels, phosphoinositide breakdown, and arachidonate release in pheochromocytoma PC12 cells.
Molecular pharmacology 1990;37(2):222-30.
1989: M T Shamim; D Ukena; William L Padgett; John W Daly
Effects of 8-phenyl and 8-cycloalkyl substituents on the activity of mono-, di-, and trisubstituted alkylxanthines with substitution at the 1-, 3-, and 7-positions.
Journal of medicinal chemistry 1989;32(6):1231-7.
1988: John W Daly; William L Padgett; Kurt Eger
7-Deaza-9-phenyladenines. A new class of adenosine receptor antagonists.
Biochemical pharmacology 1988;37(19):3749-53.
1988: Kenneth Alan Jacobson; R de la Cruz; R Schulick; L Kiriasis; William L Padgett; Wolfgang Pfleiderer; K L Kirk; J L Neumeyer; John W Daly
8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.
Biochemical pharmacology 1988;37(19):3653-61.
1988: A Adejare; F Gusovsky; William L Padgett; C R Creveling; John W Daly; K L Kirk
Syntheses and adrenergic activities of ring-fluorinated epinephrines.
Journal of medicinal chemistry 1988;31(10):1972-7.
1988: M T Shamim; D Ukena; William L Padgett; OKSOON CHOI; John W Daly
8-Aryl-and 8-cycloalkyl-1,3-dipropylxanthines: further potent and selective antagonists for A1-adenosine receptors.
Journal of medicinal chemistry 1988;31(3):613-7.
1988: John W Daly; OKSOON CHOI; William L Padgett; M T Shamim; Kenneth Alan Jacobson; D Ukena
Non-xanthine heterocycles: activity as antagonists of A1- and A2-adenosine receptors.
Biochemical pharmacology 1988;37(4):655-64.
1988: OKSOON CHOI; M T Shamim; William L Padgett; John W Daly
Caffeine and theophylline analogues: correlation of behavioral effects with activity as adenosine receptor antagonists and as phosphodiesterase inhibitors.
Life sciences 1988;43(5):387-98.
1987: D Ukena; William L Padgett; OKSOON CHOI; John W Daly; D T Daly; R A Olsson
N6-substituted 9-methyladenines: a new class of adenosine receptor antagonists.
FEBS letters 1987;215(2):203-8.
1986: D Ukena; Kenneth Alan Jacobson; William L Padgett; C Ayala; M T Shamim; K L Kirk; R O Olsson; John W Daly
Species differences in structure-activity relationships of adenosine agonists and xanthine antagonists at brain A1 adenosine receptors.
FEBS letters 1986;209(1):122-8.
1986: D Ukena; M T Shamim; William L Padgett; John W Daly
Analogs of caffeine: antagonists with selectivity for A2 adenosine receptors.
Life sciences 1986;39(8):743-50.
1986: John W Daly; William L Padgett; M T Shamim
Analogues of 1,3-dipropyl-8-phenylxanthine: enhancement of selectivity at A1-adenosine receptors by aryl substituents.
Journal of medicinal chemistry 1986;29(8):1520-4.
1986: John W Daly; William L Padgett; M T Shamim
Analogues of caffeine and theophylline: effect of structural alterations on affinity at adenosine receptors.
Journal of medicinal chemistry 1986;29(7):1305-8.
1985: John W Daly; William L Padgett; M T Shamim; P Butts-Lamb; J Waters
1,3-Dialkyl-8-(p-sulfophenyl)xanthines: potent water-soluble antagonists for A1- and A2-adenosine receptors.
Journal of medicinal chemistry 1985;28(4):487-92.
1983: J W Daly; P Butts-Lamb; William L Padgett
Subclasses of adenosine receptors in the central nervous system: interaction with caffeine and related methylxanthines.
Cellular and molecular neurobiology 1983;3(1):69-80.
1981: J W Daly; William L Padgett; C R Creveling; D Cantacuzene; K L Kirk
Cyclic AMP-generating systems: regional differences in activation by adrenergic receptors in rat brain.
The Journal of neuroscience : the official journal of the Society for Neuroscience 1981;1(1):49-59.
1980: J W Daly; William L Padgett; Y Nimitkitpaisan; C R Creveling; D Cantacuzene; K L Kirk
Fluoronorepinephrines: specific agonists for the activation of alpha and beta adrenergic-sensitive cyclic AMP-generating systems in brain slices.
The Journal of pharmacology and experimental therapeutics 1980;212(3):382-9.