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Harshad Rami

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Susan M Westaway; Mervyn Thompson; Harshad K Rami; Geoffrey Stemp; Leontine S Trouw; Darren J Mitchell; Jon T Seal; Stephen J Medhurst; Sarah C Lappin; James Biggs; James Wright; Sandra Arpino; Jeffrey C Jerman; Jennifer E Cryan; Vicky Holland; Kim Y Winborn; Tanya Coleman; Alexander J Stevens; John B Davis; Martin J Gunthorpe
Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1.
Martin Gunthorpe; Sara Luis Hannan; Darren Smart; Jeffrey C Jerman; Sandra Arpino; Graham D Smith; Stephen J Brough; Jim Wright; Julie Egerton; Sarah C Lappin; Vicky Holland; Kim Y Winborn; Mervyn Thompson; Harshad K Rami; Andrew Randall; John B Davis
Characterization of SB-705498, a potent and selective vanilloid receptor-1 (VR1/TRPV1) antagonist that inhibits the capsaicin-, acid-, and heat-mediated activation of the receptor.
Susan M Westaway; Ying-Kit Chung; John B Davis; Vicky Holland; Jeffrey C Jerman; Stephen J Medhurst; Harshad K Rami; Geoffrey Stemp; Alexander J Stevens; Mervyn Thompson; Kim Y Winborn; James Wright
N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1.

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2008: Susan M Westaway; Mervyn Thompson; Harshad K Rami; Geoffrey Stemp; Leontine S Trouw; Darren J Mitchell; Jon T Seal; Stephen J Medhurst; Sarah C Lappin; James Biggs; James Wright; Sandra Arpino; Jeffrey C Jerman; Jennifer E Cryan; Vicky Holland; Kim Y Winborn; Tanya Coleman; Alexander J Stevens; John B Davis; Martin J Gunthorpe
Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1.
Bioorganic & medicinal chemistry letters 2008;18(20):5609-13.
2007: Martin Gunthorpe; Sara Luis Hannan; Darren Smart; Jeffrey C Jerman; Sandra Arpino; Graham D Smith; Stephen J Brough; Jim Wright; Julie Egerton; Sarah C Lappin; Vicky Holland; Kim Y Winborn; Mervyn Thompson; Harshad K Rami; Andrew Randall; John B Davis
Characterization of SB-705498, a potent and selective vanilloid receptor-1 (VR1/TRPV1) antagonist that inhibits the capsaicin-, acid-, and heat-mediated activation of the receptor.
The Journal of pharmacology and experimental therapeutics 2007;321(3):1183-92.
2006: Susan M Westaway; Ying-Kit Chung; John B Davis; Vicky Holland; Jeffrey C Jerman; Stephen J Medhurst; Harshad K Rami; Geoffrey Stemp; Alexander J Stevens; Mervyn Thompson; Kim Y Winborn; James Wright
N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1.
Bioorganic & medicinal chemistry letters 2006;16(17):4533-6.
2006: Harshad K Rami; Mervyn Thompson; Geoffrey Stemp; Steve Fell; Jeffrey C Jerman; Alexander J Stevens; Darren Smart; Becky Sargent; Dominic Sanderson; Andrew D Randall; Martin Gunthorpe; John B Davis
Discovery of SB-705498: a potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development.
Bioorganic & medicinal chemistry letters 2006;16(12):3287-91.
2005: Peter J Atkinson; Steven M Bromidge; Mark S Duxon; Laramie M Gaster; Michael S Hadley; Beverley Hammond; Christopher N Johnson; Derek N Middlemiss; Stephanie E North; Gary W Price; Harshad K Rami; Graham J Riley; Claire M Scott; Tracey E Shaw; Kathryn R Starr; Geoffrey Stemp; Kevin M Thewlis; David R Thomas; Mervyn Thompson; Antonio K K Vong; Jeannette M Watson
3,4-Dihydro-2H-benzoxazinones are 5-HT(1A) receptor antagonists with potent 5-HT reuptake inhibitory activity.
Bioorganic & medicinal chemistry letters 2005;15(3):737-41.
2004: Karen A Augustine-Rauch; Qin J Zhang; Jennifer L Leonard; Antony Chadderton; Michael J Welsh; Harshad K Rami; Mervyn Thompson; Laramie M Gaster; Patrick J Wier
Evidence for a molecular mechanism of teratogenicity of SB-236057, a 5-HT1B receptor inverse agonist that alters axial formation.
Birth defects research. Part A, Clinical and molecular teratology 2004;70(10):789-807.
2004: Harshad K Rami; Mervyn Thompson; Paul A Wyman; Jeffrey C Jerman; Julie Egerton; Stephen J Brough; Alexander J Stevens; Andrew D Randall; Darren Smart; Martin Gunthorpe; John B Davis
Discovery of small molecule antagonists of TRPV1.
Bioorganic & medicinal chemistry letters 2004;14(14):3631-4.
2004: Martin Gunthorpe; Harshad K Rami; Jeffrey C Jerman; Darren Smart; Catherine H Gill; Ellen M Soffin; S Luis Hannan; Sarah C Lappin; Julie Egerton; Graham D Smith; Angela Worby; L Howett; D Owen; S Nasir; Ceri H Davies; Mervyn Thompson; Paul A Wyman; Andrew D Randall; John B Davis
Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist.
Neuropharmacology 2004;46(1):133-49.