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Romeo Romagnoli

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Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cara Carlota Lopez; Cruz-Lopez Olga; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonietta; Pipitone Maria Rosaria; Balzarini Jan; Zonta Nicola; Brancale Andrea; Hamel Ernest
Design, synthesis and structure-activity relationship of 2-(3',4',5'-trimethoxybenzoyl)-benzo[b]furan derivatives as a novel class of inhibitors of tubulin polymerization.
Romagnoli Romeo; Baraldi Pier Giovanni; Cruz-Lopez Olga; Preti Delia; Bermejo Jaime; Estévez Francisco
alpha-Bromoacrylamido N-substituted isatin derivatives as potent inducers of apoptosis in human myeloid leukemia cells.
Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cruz-Lopez Olga; Cara Carlota Lopez; Basso Giuseppe; Viola Giampietro; Khedr Mohammed; Balzarini Jan; Mahboobi Siavosh; Sellmer Andreas; Brancale Andrea; Hamel Ernest
2-Arylamino-4-amino-5-aroylthiazoles. "One-pot" synthesis and biological evaluation of a new class of inhibitors of tubulin polymerization.

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All Publications

2009: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cara Carlota Lopez; Cruz-Lopez Olga; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonietta; Pipitone Maria Rosaria; Balzarini Jan; Zonta Nicola; Brancale Andrea; Hamel Ernest
Design, synthesis and structure-activity relationship of 2-(3',4',5'-trimethoxybenzoyl)-benzo[b]furan derivatives as a novel class of inhibitors of tubulin polymerization.
Bioorganic & medicinal chemistry 2009;17(19):6862-71.
2009: Romagnoli Romeo; Baraldi Pier Giovanni; Cruz-Lopez Olga; Preti Delia; Bermejo Jaime; Estévez Francisco
alpha-Bromoacrylamido N-substituted isatin derivatives as potent inducers of apoptosis in human myeloid leukemia cells.
ChemMedChem 2009;4(10):1668-76.
2009: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cruz-Lopez Olga; Cara Carlota Lopez; Basso Giuseppe; Viola Giampietro; Khedr Mohammed; Balzarini Jan; Mahboobi Siavosh; Sellmer Andreas; Brancale Andrea; Hamel Ernest
2-Arylamino-4-amino-5-aroylthiazoles. "One-pot" synthesis and biological evaluation of a new class of inhibitors of tubulin polymerization.
Journal of medicinal chemistry 2009;52(17):5551-5.
2009: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cruz-Lopez Olga; Cara Carlota Lopez; Balzarini Jan; Hamel Ernest; Canella Alessandro; Fabbri Enrica; Gambari Roberto; Basso Giuseppe; Viola Giampietro
Hybrid alpha-bromoacryloylamido chalcones. Design, synthesis and biological evaluation.
Bioorganic & medicinal chemistry letters 2009;19(7):2022-8.
2009: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Fruttarolo Francesca; Romagnoli Romeo; Preti Delia
Recent improvements in the development of A(2B) adenosine receptor agonists.
Purinergic signalling 2009;5(1):3-19.
2009: Romagnoli Romeo; Baraldi Pier Giovanni; Cruz-Lopez Olga; Lopez-Cara Carlota; Preti Delia
alpha-halogenoacrylic derivatives of antitumor agents.
Mini reviews in medicinal chemistry 2009;9(1):81-94.
2008: Baraldi Pier Giovanni; Preti Delia; Tabrizi Mojgan Aghazadeh; Romagnoli Romeo; Saponaro Giulia; Baraldi Stefania; Botta Maurizio; Bernardini Cesare; Tafi Andrea; Tuccinardi Tiziano; Martinelli Adriano; Varani Katia; Borea Pier Andrea
Structure-activity relationship studies of a new series of imidazo[2,1-f]purinones as potent and selective A(3) adenosine receptor antagonists.
Bioorganic & medicinal chemistry 2008;16(24):10281-94.
2008: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Fruttarolo Francesca; Romagnoli Romeo; Preti Delia
Recent improvements in the development of A(2B) adenosine receptor agonists.
Purinergic signalling 2008;4(4):287-303.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Sarkar Taradas; Cara Carlota Lopez; Lopez Olga Cruz; Carrion Maria Dora; Preti Delia; Tolomeo Manlio; Balzarini Jan; Hamel Ernest
Synthesis and biological evaluation of 2-aroyl-4-phenyl-5-hydroxybenzofurans as a new class of antitubulin agents.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2008;4(6):558-64.
2008: Simoni Daniele; Romagnoli Romeo; Baruchello Riccardo; Rondanin Riccardo; Grisolia Giuseppina; Eleopra Marco; Rizzi Michele; Tolomeo Manlio; Giannini Giuseppe; Alloatti Domenico; Castorina Massimo; Marcellini Marcella; Pisano Claudio
Novel A-ring and B-ring modified combretastatin A-4 (CA-4) analogues endowed with interesting cytotoxic activity.
Journal of medicinal chemistry 2008;51(19):6211-5.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Sarkar Taradas; Carrion Maria Dora; Cruz-Lopez Olga; Lopez Cara Carlota; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonietta; Pipitone Maria Rosaria; Balzarini Jan; Gambari Roberto; Ilaria Lampronti; Saletti Roberto; Brancale Andrea; Hamel Ernest
Synthesis and biological evaluation of 2-(3',4',5'-trimethoxybenzoyl)-3-N,N-dimethylamino benzo[b]furan derivatives as inhibitors of tubulin polymerization.
Bioorganic & medicinal chemistry 2008;16(18):8419-26.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cara Carlota Lopez; Cruz-Lopez Olga; Iaconinoto Maria Antonietta; Preti Delia; Shryock John C; Moorman Allan R; Vincenzi Fabrizio; Varani Katia; Andrea Borea Pier
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N-(substituted) piperazin-1-yl]thiophenes as potent allosteric enhancers of the A1 adenosine receptor.
Journal of medicinal chemistry 2008;51(18):5875-9.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cruz-Lopez Olga; Cara Carlota Lopez; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonietta; Pipitone Maria Rosa; Balzarini Jan; Kandil Sahar; Brancale Andrea; Sarkar Taradas; Hamel Ernest
Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxybenzoyl)-6-substituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine derivatives as antimitotic agents and inhibitors of tubulin polymerization.
Bioorganic & medicinal chemistry letters 2008;18(18):5041-5.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cara Carlota Lopez; Cruz-Lopez Olga; Preti Delia; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonella; Zonta Nicola; Balzarini Jan; Brancale Andrea; Sarkar Taradas; Hamel Ernest
Design, synthesis, and biological evaluation of thiophene analogues of chalcones.
Bioorganic & medicinal chemistry 2008;16(10):5367-76.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Cruz-Lopez Olga; Lopez-Cara Carlota; Preti Delia; Borea Pier Andrea; Gessi Stefania
The P2X7 receptor as a therapeutic target.
Expert opinion on therapeutic targets 2008;12(5):647-61.
2008: Romagnoli Romeo; Baraldi Pier Giovanni; Sarkar Taradas; Carrion Maria Dora; Cara Carlota Lopez; Cruz-Lopez Olga; Preti Delia; Tabrizi Mojgan Aghazadeh; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonella; Zonta Nicola; Balzarini Jan; Brancale Andrea; Hsieh Hsing-Pang; Hamel Ernest
Synthesis and biological evaluation of 1-methyl-2-(3',4',5'-trimethoxybenzoyl)-3-aminoindoles as a new class of antimitotic agents and tubulin inhibitors.
Journal of medicinal chemistry 2008;51(5):1464-8.
2008: Tabrizi Mojgan Aghazadeh; Baraldi Pier Giovanni; Preti Delia; Romagnoli Romeo; Saponaro Giulia; Baraldi Stefania; Moorman Allan R; Zaid Abdel Naser; Varani Katia; Borea Pier Andrea
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists.
Bioorganic & medicinal chemistry 2008;16(5):2419-30.
2007: Romagnoli Romeo; Baraldi Pier Giovanni; Remusat Vincent; Carrion Maria Dora; Cara Carlota Lopez; Cruz-Lopez Olga; Preti Delia; Fruttarolo Francesca; Tabrizi Mojgan Aghazadeh; Balzarini Jan; Hamel Ernest
Synthesis and biological evaluation of 2-amino-3-(3', 4', 5'-trimethoxy-phenylsulfonyl)-5-aryl thiophenes as a new class of antitubulin agents.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2007;3(6):507-12.
2007: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cara Carlota Lopez; Preti Delia; Cruz-Lopez Olga; Tabrizi Mojgan Aghazadeh; Moorman Allan R; Gessi Stefania; Fogli Eleonora; Sacchetto Valeria; Borea Pier Andrea
From tyrosine to glycine: synthesis and biological activity of potent antagonists of the purinergic P2X7 receptor.
Journal of medicinal chemistry 2007;50(15):3706-15.
2007: Baraldi Pier Giovanni; Iaconinoto Maria Antonietta; Moorman Allan R; Carrion Maria Dora; Cara Carlota Lopez; Preti Delia; López Olga Cruz; Fruttarolo Francesca; Tabrizi Mojgan Aghazade; Romagnoli Romeo
Allosteric enhancers for A1 adenosine receptor.
Mini reviews in medicinal chemistry 2007;7(6):559-69.
2007: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Lopez Cara Carlota; Preti Delia; Fruttarolo Francesca; Pavani Maria Giovanna; Tabrizi Mojgan Aghazadeh; Tolomeo Manlio; Grimaudo Stefania; Di Cristina Antonella; Balzarini Jan; Hadfield John A; Brancale Andrea; Hamel Ernest
Synthesis and biological evaluation of 2- and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization.
Journal of medicinal chemistry 2007;50(9):2273-7.
2007: Romagnoli Romeo; Baraldi Pier Giovanni; Carrion Maria Dora; Cruz-Lopez Olga; Preti Delia; Tabrizi Mojgan Aghazadeh; Fruttarolo Francesca; Heilmann Jörg; Bermejo Jaime; Estévez Francisco
Hybrid molecules containing benzo[4,5]imidazo[1,2-d][1,2,4]thiadiazole and alpha-bromoacryloyl moieties as potent apoptosis inducers on human myeloid leukaemia cells.
Bioorganic & medicinal chemistry letters 2007;17(10):2844-8.
2007: Baraldi Pier Giovanni; Preti Delia; Tabrizi Mojgan Aghazadeh; Fruttarolo Francesca; Saponaro Giulia; Baraldi Stefania; Romagnoli Romeo; Moorman Allan R; Gessi Stefania; Varani Katia; Borea Pier Andrea
N(6)-[(hetero)aryl/(cyclo)alkyl-carbamoyl-methoxy-phenyl]-(2-chloro)-5'-N-ethylcarboxamido-adenosines: the first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor.
Bioorganic & medicinal chemistry 2007;15(7):2514-27.
2007: Baraldi Pier Giovanni; Preti Delia; Tabrizi Mojgan Aghazadeh; Fruttarolo Francesca; Romagnoli Romeo; Carrion Maria Dora; Cara Luisa Carlota Lopez; Moorman Allan R; Varani Katia; Borea Pier Andrea
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]- 9H-purin-9-yl]-N-ethyl-beta-D-ribofuranuronamide derivatives as useful templates for the development of A2B adenosine receptor agonists.
Journal of medicinal chemistry 2007;50(2):374-80.
2007: Cortesi R; Esposito E; Cuccu I; Romagnoli R; Menegatti E; Zaid A N; Nastruzzi C
Liposomes and micellar dispersions for delivery of benzoheterocyclic derivatives of distamycin A.
Drug delivery 2007;14(1):1-8.
2007: Baraldi Pier Giovanni; Preti Delia; Fruttarolo Francesca; Tabrizi Mojgan Aghazadeh; Romagnoli Romeo
Hybrid molecules between distamycin A and active moieties of antitumor agents.
Bioorganic & medicinal chemistry 2007;15(1):17-35.
2006: Romagnoli Romeo; Baraldi Pier Giovanni; Moorman Allan R; Iaconinoto Maria Antonietta; Carrion Maria Dora; Cara Carlota Lopez; Tabrizi Mojgan Aghazadeh; Preti Delia; Fruttarolo Francesca; Baker Stephen P; Varani Katia; Borea Pier Andrea
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A(1) receptor.
Bioorganic & medicinal chemistry letters 2006;16(21):5530-3.
2006: Romagnoli Romeo; Baraldi Pier Giovanni; Remusat Vincent; Carrion Maria Dora; Cara Carlota Lopez; Preti Delia; Fruttarolo Francesca; Pavani Maria Giovanna; Tabrizi Mojgan Aghazadeh; Tolomeo Manlio; Grimaudo Stefania; Balzarini Jan; Jordan Mary Ann; Hamel Ernest
Synthesis and biological evaluation of 2-(3',4',5'-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors.
Journal of medicinal chemistry 2006;49(21):6425-8.
2006: Romagnoli Romeo; Baraldi Pier Giovanni; Pavani Maria Giovanna; Tabrizi Mojgan Aghazadeh; Preti Delia; Fruttarolo Francesca; Piccagli Laura; Jung M Katherine; Hamel Ernest; Borgatti Monica; Gambari Roberto
Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxybenzoyl)-5-aryl thiophenes as a new class of potent antitubulin agents.
Journal of medicinal chemistry 2006;49(13):3906-15.
2006: Simoni Daniele; Romagnoli Romeo; Baruchello Riccardo; Rondanin Riccardo; Rizzi Michele; Pavani Maria Giovanna; Alloatti Domenico; Giannini Giuseppe; Marcellini Marcella; Riccioni Teresa; Castorina Massimo; Guglielmi Mario B; Bucci Federica; Carminati Paolo; Pisano Claudio
Novel combretastatin analogues endowed with antitumor activity.
Journal of medicinal chemistry 2006;49(11):3143-52.
2006: Baraldi Pier Giovanni; Pavani Maria Giovanna; Leung Edward; Moorman Allan R; Varani Katia; Vincenzi Fabrizio; Borea Pier Andrea; Romagnoli Romeo
Synthesis and biological characterization of [3H] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A1 allosteric enhancer.
Bioorganic & medicinal chemistry letters 2006;16(5):1402-4.
2006: Baraldi Pier Giovanni; Romagnoli Romeo; Preti Delia; Fruttarolo Francesca; Carrion Maria Dora; Tabrizi Mojgan Aghazadeh
Ligands for A2B adenosine receptor subtype.
Current medicinal chemistry 2006;13(28):3467-82.
2005: Romagnoli Romeo; Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Bermejo Jaime; Estévez Francisco; Borgatti Monica; Gambari Roberto
Design, synthesis, and biological evaluation of hybrid molecules containing alpha-methylene-gamma-butyrolactones and alpha-bromoacryloyl moieties.
Journal of medicinal chemistry 2005;48(24):7906-10.
2005: Penolazzi Letizia; Bianchini Ercolina; Lambertini Elisabetta; Baraldi Pier Giovanni; Romagnoli Romeo; Piva Roberta; Gambari Roberto
N-Arylpiperazine modified analogues of the P2X7 receptor KN-62 antagonist are potent inducers of apoptosis of human primary osteoclasts.
Journal of biomedical science 2005;12(6):1013-20.
2005: Romagnoli Romeo; Baraldi Pier Giovanni; Iaconinoto Maria Antonietta; Carrion Maria Dora; Tabrizi Mojgan Aghazadeh; Gambari Roberto; Borgatti Monica; Heilmann Jörg
Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates.
European journal of medicinal chemistry 2005;40(11):1123-8.
2005: Romagnoli Romeo; Baraldi Pier Giovanni; Jung M Katherine; Iaconinoto Maria Antonietta; Carrion Maria Dora; Remusat Vincent; Preti Delia; Tabrizi Mojgan Aghazadeh; Francesca Fruttarolo; De Clercq Erik; Balzarini Jan; Hamel Ernest
Synthesis and preliminary biological evaluation of new anti-tubulin agents containing different benzoheterocycles.
Bioorganic & medicinal chemistry letters 2005;15(18):4048-52.
2005: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Preti Delia; Bovero Andrea; Fruttarolo Francesca; Romagnoli Romeo; Zaid Naser Abdel; Moorman Allan R; Varani Katia; Borea Pier Andrea
New 2-arylpyrazolo[4,3-c]quinoline derivatives as potent and selective human A3 adenosine receptor antagonists.
Journal of medicinal chemistry 2005;48(15):5001-8.
2005: Baraldi Pier Giovanni; Preti Delia; Tabrizi Mojgan Aghazadeh; Fruttarolo Francesca; Romagnoli Romeo; Zaid Naser Abdel; Moorman Allan R; Merighi Stefania; Varani Katia; Borea Pier Andrea
New pyrrolo[2,1-f]purine-2,4-dione and imidazo[2,1-f]purine-2,4-dione derivatives as potent and selective human A3 adenosine receptor antagonists.
Journal of medicinal chemistry 2005;48(14):4697-701.
2005: Baraldi Pier Giovanni; Romagnoli Romeo; Tabrizi Mojgan Aghazadeh; Bovero Andrea; Preti Delia; Fruttarolo Francesca; Moorman Allan R; Borea Pier Andrea
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2.
Farmaco (Società chimica italiana : 1989) 2005;60(3):185-202.
2005: Di Virgilio Francesco; Baricordi O Roberto; Romagnoli Romeo; Baraldi Pier Giovanni
Leukocyte P2 receptors: a novel target for anti-inflammatory and anti-tumor therapy.
Current drug targets. Cardiovascular & haematological disorders 2005;5(1):85-99.
2005: Simoni Daniele; Grisolia Giuseppina; Giannini Giuseppe; Roberti Marinella; Rondanin Riccardo; Piccagli Laura; Baruchello Riccardo; Rossi Marcello; Romagnoli Romeo; Invidiata Francesco Paolo; Grimaudo Stefania; Jung M Katherine; Hamel Ernest; Gebbia Nicola; Crosta Lucia; Abbadessa Vincenzo; Di Cristina Antonietta; Dusonchet Luisa; Meli Maria; Tolomeo Manlio
Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines.
Journal of medicinal chemistry 2005;48(3):723-36.
2005: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Romagnoli Romeo; Fruttarolo Francesca; Merighi Stefania; Varani Katia; Gessi Stefania; Borea Pier Andrea
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine ligands, new tools to characterize A3 adenosine receptors in human tumor cell lines.
Current medicinal chemistry 2005;12(11):1319-29.
2004: Romagnoli Romeo; Baraldi Pier Giovanni; Pavani Maria Giovanna; Tabrizi Mojgan Aghazadeh; Moorman Allan R; Di Virgilio Francesco; Cattabriga Elena; Pancaldi Cecilia; Gessi Stefania; Borea Pier Andrea
Synthesis, radiolabeling, and preliminary biological evaluation of [3H]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl)-piperazine, a potent antagonist radioligand for the P2X7 receptor.
Bioorganic & medicinal chemistry letters 2004;14(22):5709-12.
2004: Baraldi Pier Giovanni; Fruttarolo Francesca; Tabrizi Mojgan Aghazadeh; Romagnoli Romeo; Preti Delia; Bovero Andrea; Pineda de Las Infantas Maria Josè; Moorman Allan; Varani Katia; Borea Pier Andrea
Synthesis and biological evaluation of novel N6-[4-(substituted)sulfonamidophenylcarbamoyl]adenosine-5'-uronamides as A3 adenosine receptor agonists.
Journal of medicinal chemistry 2004;47(22):5535-40.
2004: Baraldi Pier Giovanni; Pavani Maria Giovanna; Shryock John C; Moorman Allan R; Iannotta Valeria; Borea Pier Andrea; Romagnoli Romeo
Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A1 receptor.
European journal of medicinal chemistry 2004;39(10):855-65.
2004: Baraldi Pier Giovanni; Beria Italo; Cozzi Paolo; Geroni Cristina; Espinosa Antonio; Gallo Miguel A; Entrena Antonio; Bingham John P; Hartley John A; Romagnoli Romeo
Cinnamoyl nitrogen mustard derivatives of pyrazole analogues of tallimustine modified at the amidino moiety: design, synthesis, molecular modeling and antitumor activity studies.
Bioorganic & medicinal chemistry 2004;12(14):3911-21.
2004: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Preti Delia; Bovero Andrea; Fruttarolo Francesca; Romagnoli Romeo; Moorman Allan R; Gessi Stefania; Merighi Stefania; Varani Katia; Borea Pier Andrea
[3H]-MRE 2029-F20, a selective antagonist radioligand for the human A2B adenosine receptors.
Bioorganic & medicinal chemistry letters 2004;14(13):3607-10.
2004: Baraldi Pier Giovanni; Bovero Andrea; Fruttarolo Francesca; Preti Delia; Tabrizi Mojgan Aghazadeh; Pavani Maria Giovanna; Romagnoli Romeo
DNA minor groove binders as potential antitumor and antimicrobial agents.
Medicinal research reviews 2004;24(4):475-528.
2004: Baraldi Pier Giovanni; Del Carmen Nunez Maria; Tabrizi Mojgan Aghazadeh; De Clercq Erik; Balzarini Jan; Bermejo Jaime; Estévez Francisco; Romagnoli Romeo
Design, synthesis, and biological evaluation of hybrid molecules containing alpha-methylene-gamma-butyrolactones and polypyrrole minor groove binders.
Journal of medicinal chemistry 2004;47(11):2877-86.
2004: Beria Italo; Baraldi Pier Giovanni; Cozzi Paolo; Caldarelli Marina; Geroni Cristina; Marchini Sergio; Mongelli Nicola; Romagnoli Romeo
Cytotoxic alpha-halogenoacrylic derivatives of distamycin A and congeners.
Journal of medicinal chemistry 2004;47(10):2611-23.
2004: Cortesi R; Romagnoli R; Menegatti E; Esposito E; Cervellati F; Nastruzzi C
Liposomes containing distamycins: preparation, characterization and antiproliferative activity.
Drug delivery 2004;11(2):83-8.
2004: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Preti Delia; Bovero Andrea; Romagnoli Romeo; Fruttarolo Francesca; Zaid Naser Abdel; Moorman Allan R; Varani Katia; Gessi Stefania; Merighi Stefania; Borea Pier Andrea
Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists.
Journal of medicinal chemistry 2004;47(6):1434-47.
2004: Mischiati Carlo; Finotti Alessia; Sereni Alessia; Boschetti Sindi; Baraldi Pier Giovanni; Romagnoli Romeo; Feriotto Giordana; Jeang Kuan-Teh; Bianchi Nicoletta; Borgatti Monica; Gambari Roberto
Binding of hybrid molecules containing pyrrolo [2,1-c][1,4]benzodiazepine (PBD) and oligopyrrole carriers to the human immunodeficiency type 1 virus TAR-RNA.
Biochemical pharmacology 2004;67(3):401-10.
2004: Baraldi Pier Giovanni; Romagnoli Romeo; Del Carmen Nuñez Maria; Perretti Mauro; Paul-Clark Mark J; Ferrario Massimiliano; Govoni Mirco; Benedini Francesca; Ongini Ennio
Synthesis of nitro esters of prednisolone, new compounds combining pharmacological properties of both glucocorticoids and nitric oxide.
Journal of medicinal chemistry 2004;47(3):711-9.
2004: Baraldi Pier Giovanni; Di Virgilio Francesco; Romagnoli Romeo
Agonists and antagonists acting at P2X7 receptor.
Current topics in medicinal chemistry 2004;4(16):1707-17.
2004: Baraldi Pier Giovanni; Nûnez Maria del Carmen; Espinosa Antonio; Romagnoli Romeo
Distamycin A as stem of DNA minor groove alkylating agents.
Current topics in medicinal chemistry 2004;4(2):231-9.
2003: Boschi Alessandra; Uccelli Licia; Duatti Adriano; Bolzati Cristina; Refosco Fiorenzo; Tisato Francesco; Romagnoli Romeo; Baraldi Pier Giovanni; Varani Katia; Borea Pier Andrea
Asymmetrical nitrido tc-99m heterocomplexes as potential imaging agents for benzodiazepine receptors.
Bioconjugate chemistry 2003;14(6):1279-88.
2003: Baraldi Pier Giovanni; Bovero Andrea; Fruttarolo Francesca; Romagnoli Romeo; Tabrizi Mojgan Aghazadeh; Preti Delia; Varani Katia; Borea Pier Andrea; Moorman Allan R
New strategies for the synthesis of A3 adenosine receptor antagonists.
Bioorganic & medicinal chemistry 2003;11(19):4161-9.
2003: Baraldi Pier Giovanni; Romagnoli Romeo; Bianchi Nicoletta; Gambari Roberto
Benzoyl nitrogen mustard derivatives of benzoheterocyclic analogues of netropsin: synthesis and biological activity.
Bioorganic & medicinal chemistry 2003;11(11):2381-8.
2003: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Bovero Andrea; Avitabile Barbara; Preti Delia; Fruttarolo Francesca; Romagnoli Romeo; Varani Katia; Borea Pier Andrea
Recent developments in the field of A2A and A3 adenosine receptor antagonists.
European journal of medicinal chemistry 2003;38(4):367-82.
2003: Baraldi Pier Giovanni; Fruttarolo Francesca; Tabrizi Mojgan Aghazadeh; Preti Delia; Romagnoli Romeo; El-Kashef Hussein; Moorman Allan; Varani Katia; Gessi Stefania; Merighi Stefania; Borea Pier Andrea
Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists.
Journal of medicinal chemistry 2003;46(7):1229-41.
2003: Baraldi Pier Giovanni; Beria Italo; Cozzi Paolo; Bianchi Nicoletta; Gambari Roberto; Romagnoli Romeo
Synthesis and growth inhibition activity of alpha-bromoacrylic heterocyclic and benzoheterocyclic derivatives of distamycin A modified on the amidino moiety.
Bioorganic & medicinal chemistry 2003;11(6):965-75.
2003: Baraldi Pier Giovanni; Romagnoli Romeo; Pavani Maria Giovanna; Nuñez Maria del Carmen; Tabrizi Mojgan Aghazadeh; Shryock John C; Leung Edward; Moorman Allan R; Uluoglu Canan; Iannotta Valeria; Merighi Stefania; Borea Pier Andrea
Synthesis and biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptor.
Journal of medicinal chemistry 2003;46(5):794-809.
2003: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Pavani Maria Giovanna; Nuñez Maria del Carmen; Makaeva Rimma; Gambari Roberto; La Colla Paolo; Romagnoli Romeo
Design, synthesis and in vitro cytotoxicity of a cis-dichloroplatinum (II) complex linked to the minor groove binder stallimycin.
Arzneimittel-Forschung 2003;53(2):107-13.
2002: Baraldi Pier Giovanni; Romagnoli Romeo; Guadix Antonio Entrena; Pineda de las Infantas Maria Josè; Gallo Miguel Angel; Espinosa Antonio; Martinez Alberto; Bingham John P; Hartley John A
Design, synthesis, and biological activity of hybrid compounds between uramustine and DNA minor groove binder distamycin A.
Journal of medicinal chemistry 2002;45(17):3630-8.
2002: Baraldi Pier Giovanni; Romagnoli Romeo; Giovanna Pavani Maria; del Carmen Nunez Maria; Bingham John P; Hartley John A
Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: synthesis and antitumour activity.
Bioorganic & medicinal chemistry 2002;10(5):1611-8.
2002: Baraldi Pier Giovanni; Pavani Maria Giovanna; Nuñez Maria del Carmen; Brigidi Patrizia; Vitali Beatrice; Gambari Roberto; Romagnoli Romeo
Antimicrobial and antitumor activity of N-heteroimmine-1,2,3-dithiazoles and their transformation in triazolo-, imidazo-, and pyrazolopirimidines.
Bioorganic & medicinal chemistry 2002;10(2):449-56.
2002: Baraldi Pier Giovanni; Cacciari Barbara; Romagnoli Romeo; Spalluto Giampiero; Monopoli Angela; Ongini Ennio; Varani Katia; Borea Pier Andrea
7-Substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: a study on the importance of modifications at the side chain on the activity and solubility.
Journal of medicinal chemistry 2002;45(1):115-26.
2002: Baraldi Pier Giovanni; Makaeva Rimma; Pavani Maria Giovanna; Nuñez Maria del Carmen; Spalluto Giampiero; Moro Stefano; Falzoni Simonetta; Di Virgilio Francesco; Romagnoli Romeo
Synthesis, biological activity and molecular modeling studies of 1,2,3,4-tetrahydroisoquinoline derivatives as conformationally constrained analogues of KN62, a potent antagonist of the P2X7-receptor containing a tyrosine moiety.
Arzneimittel-Forschung 2002;52(4):273-85.
2001: Baraldi P G; Cacciari B; Moro S; Romagnoli R; Ji Xd; Jacobson K A; Gessi S; Borea P A; Spalluto G
Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalized pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: irreversible antagonists at the human A3 adenosine receptor and molecular modeling studies.
Journal of medicinal chemistry 2001;44(17):2735-42.
2001: Baraldi P G; Balboni G; Pavani M G; Spalluto G; Tabrizi M A; Clercq E D; Balzarini J; Bando T; Sugiyama H; Romagnoli R
Design, synthesis, DNA binding, and biological evaluation of water-soluble hybrid molecules containing two pyrazole analogues of the alkylating cyclopropylpyrroloindole (CPI) subunit of the antitumor agent CC-1065 and polypyrrole minor groove binders.
Journal of medicinal chemistry 2001;44(16):2536-43.
2000: Baraldi P G; Zaid A N; Lampronti I; Fruttarolo F; Pavani M G; Tabrizi M A; Shryock J C; Leung E; Romagnoli R
Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor.
Bioorganic & medicinal chemistry letters 2000;10(17):1953-7.
2000: Baraldi P G; Cacciari B; Guiotto A; Romagnoli R; Spalluto G; Leoni A; Bianchi N; Feriotto G; Rutigliano C; Mischiati C; Gambari R
[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding to transcription factor Sp1.
Nucleosides, nucleotides & nucleic acids 2000;19(8):1219-29.
2000: Baraldi P G; Romagnoli R; Beria I; Cozzi P; Geroni C; Mongelli N; Bianchi N; Mischiati C; Gambari R
Synthesis and antitumor activity of new benzoheterocyclic derivatives of distamycin A.
Journal of medicinal chemistry 2000;43(14):2675-84.
2000: Baraldi P G; Romagnoli R; Duatti A; Bolzati C; Piffanelli A; Bianchi N; Mischiati C; Gambari R
Synthesis of hybrid distamycin-cysteine labeled with 99mTc: a model for a novel class of cancer imaging agents.
Bioorganic & medicinal chemistry letters 2000;10(12):1397-400.
2000: Varani K; Merighi S; Gessi S; Klotz K N; Leung E; Baraldi P G; Cacciari B; Romagnoli R; Spalluto G; Borea P A
[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.
Molecular pharmacology 2000;57(5):968-75.
2000: Baraldi P G; Romagnoli R; Tabrizi M A; Falzoni S; di Virgilio F
Synthesis of conformationally constrained analogues of KN62, a potent antagonist of the P2X7-receptor.
Bioorganic & medicinal chemistry letters 2000;10(7):681-4.
2000: Baraldi P G; Romagnoli R; Spalluto G; Cozzi P; Mongelli N; Bianchi N; Gambari R
DNA sequence-recognizing properties of minor groove alkylating agents. Effects of the replacement of N-methylpyrrole by an N-methylimidazole on tallimustine and its own homologue.
Arzneimittel-Forschung 2000;50(3):309-15.
2000: Baraldi P G; Cacciari B; Romagnoli R; Merighi S; Varani K; Borea P A; Spalluto G
A(3) adenosine receptor ligands: history and perspectives.
Medicinal research reviews 2000;20(2):103-28.
2000: Baraldi P G; Cacciari B; Romagnoli R; Varani K; Merighi S; Gessi S; Borea P A; Leung E; Hickey S L; Spalluto G
Synthesis and preliminary biological evaluation of [3H]-MRE 3008-F20: the first high affinity radioligand antagonist for the human A3 adenosine receptors.
Bioorganic & medicinal chemistry letters 2000;10(3):209-11.
1999: Baraldi P G; Cacciari B; Romagnoli R; Spalluto G
1H-pyrazolo[2,3-d][1,2,4]triazine-3,7-diones as a new class of human leukocyte elastase inhibitors.
Arzneimittel-Forschung 1999;49(12):997-1000.
1999: Baraldi P G; Balboni G; Cacciari B; Guiotto A; Manfredini S; Romagnoli R; Spalluto G; Thurston D E; Howard P W; Bianchi N; Rutigliano C; Mischiati C; Gambari R
Synthesis, in vitro antiproliferative activity, and DNA-binding properties of hybrid molecules containing pyrrolo[2,1-c][1, 4]benzodiazepine and minor-groove-binding oligopyrrole carriers.
Journal of medicinal chemistry 1999;42(25):5131-41.
1999: Baraldi P G; Cacciari B; Romagnoli R; Spalluto G; Klotz K N; Leung E; Varani K; Gessi S; Merighi S; Borea P A
Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists.
Journal of medicinal chemistry 1999;42(22):4473-8.
1999: Baraldi P G; Cacciari B; Romagnoli R; Spalluto G; Boyce C W; Boger D L
Resolution of a CPzI precursor, synthesis and biological evaluation of (+) and (-)-N-Boc-CPzI: a further validation of the relationship between chemical solvolytic stability and cytotoxicity.
Bioorganic & medicinal chemistry letters 1999;9(21):3087-92.
1999: Baraldi P G; Balboni G; Romagnoli R; Spalluto G; Cozzi P; Geroni C; Mongelli N; Rutigliano C; Bianchi N; Gambari R
PNU 157977: a new potent antitumour agent exhibiting low in vivo toxicity in mice injected with L1210 leukaemia cells.
Anti-cancer drug design 1999;14(1):71-6.
1999: Baraldi P G; Cozzi P; Geroni C; Mongelli N; Romagnoli R; Spalluto G
Novel benzoyl nitrogen mustard derivatives of pyrazole analogues of distamycin A: synthesis and antileukemic activity.
Bioorganic & medicinal chemistry 1999;7(2):251-62.
1999: Baraldi P G; Cacciari B; Guiotto A; Romagnoli R; Zaid A N; Spalluto G
DNA minor-groove binders: results and design of new antitumor agents.
Farmaco (Società chimica italiana : 1989) 1999;54(1-2):15-25.
1998: Baraldi P G; Cacciari B; Guiotto A; Leoni A; Romagnoli R; Spalluto G; Mongelli N; Howard P W; Thurston D E; Bianchi N; Gambari R
Design, synthesis and biological activity of a pyrrolo [2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid.
Bioorganic & medicinal chemistry letters 1998;8(21):3019-24.
1998: Baraldi P G; Cacciari B; Pineda de Las Infantas M J; Romagnoli R; Spalluto G; Volpini R; Costanzi S; Vittori S; Cristalli G; Melman N; Park K S; Ji X D; Jacobson K A
Synthesis and biological activity of a new series of N6-arylcarbamoyl, 2-(Ar)alkynyl-N6-arylcarbamoyl, and N6-carboxamido derivatives of adenosine-5'-N-ethyluronamide as A1 and A3 adenosine receptor agonists.
Journal of medicinal chemistry 1998;41(17):3174-85.
1998: Baraldi P G; Cacciari B; Guiotto A; Romagnoli R; Zaid A N; Spalluto G
Heterocyclic analogs of DNA minor groove alkylating agents.
Current pharmaceutical design 1998;4(3):249-76.
1997: Baraldi P G; Cacciari B; Guiotto A; Romagnoli R; Spalluto G; Zaid A N; Capolongo L; Cozzi P; Geroni C; Mongelli N
Synthesis, solvolytic stability and cytotoxicity of a modified derivative of CPzI, a pyrazole analog of the alkylation subunit of the antitumor agent CC-1065: effect of the nitrogen substitution on the functional reactivity.
Farmaco (Società chimica italiana : 1989) 1997;52(12):717-23.
1997: Baraldi P G; Cacciari B; Guiotto A; Romagnoli R; Spalluto G; Zaid A N; Cozzi P; Geroni C; Mongelli N
Synthesis, cytotoxicity and antitumor activity of some new simplified pyrazole analogs of the antitumor agent CC-1065. Effect of an hydrophobic group on antitumor activity.
Farmaco (Società chimica italiana : 1989) 1997;52(12):711-6.
1997: Baraldi P G; Cacciari B; Romagnoli R; Spalluto G; Gambari R; Bianchi N; Passadore M; Ambrosino P; Mongelli N; Cozzi P; Geroni C
Synthesis, cytotoxicity, antitumor activity and sequence selective binding of two pyrazole analogs structurally related to the antitumor agents U-71,184 and adozelesin.
Anti-cancer drug design 1997;12(7):555-76.
1997: Baraldi P G; Cacciari B; Pineda de las Infantas M J; Romagnoli R; Spalluto G; Cozzi P; Mongelli N
Synthesis, chemical solvolytic stability and preliminary biological evaluation of (+/-)-N-Boc-CPzI: a pyrazole analog of the left-hand segment of the antitumor agent CC-1065.
Anti-cancer drug design 1997;12(1):67-74.
1996: Baraldi P G; Cacciari B; Romagnoli R; Spalluto G; Garuti L; Roberti M; Pani A; Perra G; Scintu F; Pinna N; Musiu C; La Colla P
Synthesis, antiviral and antiproliferative activity of a new class of 5-(alkyl or arylthio)-6-vinyl uracils.
Anti-cancer drug design 1996;11(8):597-609.

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