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Giuseppe Ronsisvalle

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Chemicals & Drugs

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Carmela Parenti; Giuseppina Aricò; Agostino Marrazzo; Orazio Prezzavento; Giuseppe Ronsisvalle; Simone Ronsisvalle; Giovanna M. Scoto; Rita Turnaturi; L Pasquinucci
Antinociceptive profile of LP1, a non-peptide multitarget opioid ligand.
Carmela Parenti; Giuseppe Ronsisvalle; Giuseppina Aricò; Giovanna M. Scoto
Supraspinal injection of Substance P attenuates allodynia and hyperalgesia in a rat model of inflammatory pain.
Agostino Marrazzo; giuseppina marrazzo; Carmela Parenti; L Pasquinucci; Orazio Prezzavento; Giuseppina Aricò; Enrique J Cobos; Nicola A Colabufo; Marialessandra Contino; Luis G González; Simone Ronsisvalle; Giovanna M. Scoto; Giuseppe Ronsisvalle
Novel potent and selective σ ligands: evaluation of their agonist and antagonist properties.

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All Publications

2012: Carmela Parenti; Giuseppina Aricò; Agostino Marrazzo; Orazio Prezzavento; Giuseppe Ronsisvalle; Simone Ronsisvalle; Giovanna M. Scoto; Rita Turnaturi; L Pasquinucci
Antinociceptive profile of LP1, a non-peptide multitarget opioid ligand.
Life sciences 2012;90(25-26):957-61.
2012: Carmela Parenti; Giuseppe Ronsisvalle; Giuseppina Aricò; Giovanna M. Scoto
Supraspinal injection of Substance P attenuates allodynia and hyperalgesia in a rat model of inflammatory pain.
Peptides 2012;34(2):412-8.
2011: Agostino Marrazzo; giuseppina marrazzo; Carmela Parenti; L Pasquinucci; Orazio Prezzavento; Giuseppina Aricò; Enrique J Cobos; Nicola A Colabufo; Marialessandra Contino; Luis G González; Simone Ronsisvalle; Giovanna M. Scoto; Giuseppe Ronsisvalle
Novel potent and selective σ ligands: evaluation of their agonist and antagonist properties.
Journal of medicinal chemistry 2011;54(10):3669-73.
2011: Vuokko Antonini; Marino Coradazzi; Giulio Kleiner; Agostino Marrazzo; Orazio Prezzavento; Giuseppe Ronsisvalle; Simone Ronsisvalle; G Leanza
Anti-amnesic and neuroprotective actions of the sigma-1 receptor agonist (-)-MR22 in rats with selective cholinergic lesion and amyloid infusion.
Journal of Alzheimer's disease : JAD 2011;24(3):569-86.
2011: Agostino Marrazzo; Jole Fiorito; Laura Zappalà; Orazio Prezzavento; Simone Ronsisvalle; L Pasquinucci; Giovanna M. Scoto; Renato Bernardini; Giuseppe Ronsisvalle
Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells.
European journal of medicinal chemistry 2011;46(1):433-8.
2010: Orazio Prezzavento; Agata Campisi; Carmela Parenti; Simone Ronsisvalle; Giuseppina Aricò; Emanuela Arena; Marco Pistolozzi; Giovanna M. Scoto; Carlo Bertucci; Angelo Vanella; Giuseppe Ronsisvalle
Synthesis and resolution of cis-(+/-)-methyl (1R,2S/1S,2R)-2-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-1-(4-methylphenyl)cyclopropanecarboxylate [(+/-)-PPCC)]: new sigma receptor ligands with neuroprotective effect.
Journal of medicinal chemistry 2010;53(15):5881-5.
2010: L Pasquinucci; Orazio Prezzavento; Agostino Marrazzo; Emanuele Amata; Simone Ronsisvalle; Zafiroula Georgoussi; Danai-Dionysia Fourla; Giovanna M. Scoto; Carmela Parenti; Giuseppina Aricò; Giuseppe Ronsisvalle
Evaluation of N-substitution in 6,7-benzomorphan compounds.
Bioorganic & medicinal chemistry 2010;18(14):4975-82.
2010: Giovanna M. Scoto; Giuseppina Aricò; Attilio Iemolo; Giuseppe Ronsisvalle; Carmela Parenti
Selective inhibition of the NOP receptor in the ventrolateral periaqueductal gray attenuates the development and the expression of tolerance to morphine-induced antinociception in rats.
Peptides 2010;31(4):696-700.
2008: Gloria Cristalli; Péter Mátyus; Peter Mohr; Giuseppe Ronsisvalle; Noël de Souza; Anna Tsantili-Kakoulidou
European medicinal chemistry education: the transformational accomplishments and challenges.
ChemMedChem 2008;3(4):561-3.
2008: Orazio Prezzavento; Carmela Parenti; Agostino Marrazzo; Simone Ronsisvalle; Franco Vittorio; Giuseppina Aricò; Giovanna M. Scoto; Giuseppe Ronsisvalle
A new sigma ligand, (+/-)-PPCC, antagonizes kappa opioid receptor-mediated antinociceptive effect.
Life sciences 2008;82(11-12):549-53.
2008: Natale Alfredo Santagati; Loredana Salerno; Giuseppina Attaguile; Francesca Savoca; Giuseppe Ronsisvalle
Simultaneous determination of catechins, rutin, and gallic acid in Cistus species extracts by HPLC with diode array detection.
Journal of chromatographic science 2008;46(2):150-6.
2007: L Pasquinucci; Manuela Iadanza; Agostino Marrazzo; Orazio Prezzavento; Simone Ronsisvalle; Giovanna M. Scoto; Carmela Parenti; L De Luca; Giuseppe Ronsisvalle
New benzomorphan derivatives of MPCB as MOP and KOP receptor ligands.
Die Pharmazie 2007;62(11):813-24.
2007: Orazio Prezzavento; Agata Campisi; Simone Ronsisvalle; Giovanni Li Volti; Agostino Marrazzo; Vincenzo Bramanti; Giuseppe Cannavò; Luca Vanella; Alfredo Cagnotto; Tiziana Mennini; Riccardo Ientile; Giuseppe Ronsisvalle
Novel sigma receptor ligands: synthesis and biological profile.
Journal of medicinal chemistry 2007;50(5):951-61.
2007: Simona Collina; Guya Loddo; Mariangela Urbano; Laura Linati; Aliria Callegari; Francesco Ortuso; Stefano Alcaro; Christian Laggner; Thierry Langer; Orazio Prezzavento; Giuseppe Ronsisvalle; Ornella Azzolina
Design, synthesis, and SAR analysis of novel selective sigma1 ligands.
Bioorganic & medicinal chemistry 2007;15(2):771-83.
2006: Annamaria Panico; Venera Cardile; S Avondo; Floriana Garufi; Barbara Gentile; carmelo puglia; Francesco Bonina; Natale Alfredo Santagati; Giuseppe Ronsisvalle
The in vitro effect of a lyophilized extract of wine obtained from Jacquez grapes on human chondrocytes.
Phytomedicine : international journal of phytotherapy and phytopharmacology 2006;13(7):522-6.
2006: Claudio Bucolo; Agostino Marrazzo; Simone Ronsisvalle; Giuseppe Ronsisvalle; Salvatore Cuzzocrea; Emanuela Mazzon; Achille Caputi; Filippo Drago
A novel adamantane derivative attenuates retinal ischemia-reperfusion damage in the rat retina through sigma1 receptors.
European journal of pharmacology 2006;536(1-2):200-3.
2006: Agostino Marrazzo; Carmela Parenti; Valentina Scavo; Simone Ronsisvalle; Giovanna M. Scoto; Giuseppe Ronsisvalle
In vivo evaluation of (+)-MR200 as a new selective sigma ligand modulating MOP, DOP and KOP supraspinal analgesia.
Life sciences 2006;78(21):2449-53.
2005: Annamaria Panico; Venera Cardile; Floriana Garufi; carmelo puglia; Francesco Bonina; Giuseppe Ronsisvalle
Protective effect of Capparis spinosa on chondrocytes.
Life sciences 2005;77(20):2479-88.
2005: Agostino Marrazzo; Filippo Caraci; Elisa Trovato Salinaro; Tsung-Ping Su; Agata Copani; Giuseppe Ronsisvalle
Neuroprotective effects of sigma-1 receptor agonists against beta-amyloid-induced toxicity.
Neuroreport 2005;16(11):1223-6.
2005: Natale Alfredo Santagati; Salvatore Tropea; Giuseppe Ronsisvalle
Analysis of ecdysteroids by micellar electrokinetic chromatography with on-line preconcentration.
Journal of chromatography. A 2005;1081(1):77-86.
2005: Natale Alfredo Santagati; Roberto Gotti; Giuseppe Ronsisvalle
Simultaneous determination of phenytoin and dextromethorphan in urine by solid-phase extraction and HPLC-DAD.
Journal of separation science 2005;28(11):1157-62.
2005: Emanuela Sperlinga; Piotr Kosson; Zofia Urbanczyk-Lipkowska; Giuseppe Ronsisvalle; Daniel B Carr; Andrzej W Lipkowski
6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid mimics active conformation of tyrosine in opioid peptides.
Bioorganic & medicinal chemistry letters 2005;15(10):2467-9.
2005: Luca Costantino; Francesca Gandolfi; Claudia Sorbi; Silvia Franchini; Orazio Prezzavento; Franco Vittorio; Giuseppe Ronsisvalle; Amedeo Leonardi; Elena Poggesi; Livio Brasili
Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.
Journal of medicinal chemistry 2005;48(1):266-73.
2004: Annamaria Panico; Paola Vicini; G Massimo; Venera Cardile; Barbara Gentile; S Avondo; Franco Vittorio; Giuseppe Ronsisvalle
Protective effects of benzisothiazolylamidines on IL-1 beta induced alterations in human articular chondrocyte metabolism.
Inflammation 2004;28(4):231-5.
2003: Annamaria Panico; Venera Cardile; Franco Vittorio; Giuseppe Ronsisvalle; Giovanna M. Scoto; Carmela Parenti; Barbara Gentile; R Morrone; G Nicolosi
Different in vitro activity of flurbiprofen and its enantiomers on human articular cartilage.
Farmaco (Società chimica italiana : 1989) 2003;58(12):1339-44.
2003: Natale Alfredo Santagati; Ennio Bousquet; A Garozzo; Orazio Prezzavento; Spadaro Angelo; Giuseppe Ronsisvalle
Synthesis and anti-measles virus activity of new isoquinolin-4-one derivatives.
Farmaco (Società chimica italiana : 1989) 2003;58(12):1217-25.
2003: Delphine Moison; Philippe De Deurwaerdère; Alfredo Cagnotto; Agostino Marrazzo; Orazio Prezzavento; Giuseppe Ronsisvalle; Tiziana Mennini; Umberto Spampinato
Intrastriatal administration of sigma ligands inhibits basal dopamine release in vivo.
Neuropharmacology 2003;45(7):945-53.
2003: Annamaria Panico; Venera Cardile; Barbara Gentile; Floriana Garufi; Paolo Fama'; Giuseppe Bonfiglio; Giuseppe Ronsisvalle
Effects of leflunomide on human cartilage.
Farmaco (Società chimica italiana : 1989) 2003;58(9):983-7.
2003: Maria S Pappalardo; Ennio Bousquet; Agata Annino; Gabriella Lombardo; Renato Bernardini; Giuseppe Ronsisvalle
Synthesis of new P3CS derivatives and their mitogenic activity on in vitro mice splenocytes.
Farmaco (Società chimica italiana : 1989) 2003;58(4):329-36.
2002: Venera Cardile; Annamaria Panico; Athina Geronikaki; Barbara Gentile; Giuseppe Ronsisvalle
In vitro evaluation of thiazolyl and benzothiazolyl Schiff bases on pig cartilage.
Farmaco (Società chimica italiana : 1989) 2002;57(12):1009-13.
2002: Ennio Bousquet; Spadaro Angelo; Natale Alfredo Santagati; Santo Scalia; Giuseppe Ronsisvalle
Determination of undecylenic and sorbic acids in cosmetic preparations by high performance liquid chromatography with electrochemical detection.
Journal of pharmaceutical and biomedical analysis 2002;30(4):947-54.
2002: Manuela Iadanza; Monika Höltje; Giuseppe Ronsisvalle; Hans-Dieter Höltje
Kappa-opioid receptor model in a phospholipid bilayer: molecular dynamics simulation.
Journal of medicinal chemistry 2002;45(22):4838-46.
2002: Natale Alfredo Santagati; Giuseppina Ferrara; Agostino Marrazzo; Giuseppe Ronsisvalle
Simultaneous determination of amphetamine and one of its metabolites by HPLC with electrochemical detection.
Journal of pharmaceutical and biomedical analysis 2002;30(2):247-55.
2002: Annamaria Panico; Paola Vicini; Matteo Incerti; Venera Cardile; Barbara Gentile; Giuseppe Ronsisvalle
Amidinobenzisothiazole derivatives with antidegenerative activity on cartilage.
Farmaco (Società chimica italiana : 1989) 2002;57(8):671-5.
2002: Natale Alfredo Santagati; Ennio Bousquet; Spadaro Angelo; Giuseppe Ronsisvalle
Analysis of aliphatic amines in air samples by HPLC with electrochemical detection.
Journal of pharmaceutical and biomedical analysis 2002;29(6):1105-11.
2002: Giuseppe Ronsisvalle; Orazio Prezzavento; Agostino Marrazzo; Franco Vittorio; Michele Massimino; Giovanna Murari; santi spampinato
Synthesis of (+)-cis-N-(4-isothiocyanatobenzyl)-N-normetazocine, an isothiocyanate derivative of N-benzylnormetazocine as acylant agent for the sigma(1) receptor.
Journal of medicinal chemistry 2002;45(12):2662-5.
2002: Natale Alfredo Santagati; Orazio Prezzavento; Ennio Bousquet; Giuseppe Ronsisvalle; santi spampinato
Synthesis and spasmolytic action of 2-substituted thienopyrimidin-4-one derivatives.
The Journal of pharmacy and pharmacology 2002;54(5):717-28.
2002: Orazio Prezzavento; Fulvio Gualtieri; Agostino Marrazzo; Maria Novella Romanelli; Giuseppe Ronsisvalle; Elisabetta Teodori
Sigma receptor binding profile of a series of analgesic tropane derivatives.
Archiv der Pharmazie 2002;335(1):39-43.
2002: Agostino Marrazzo; Orazio Prezzavento; Maria S Pappalardo; Ennio Bousquet; Manuela Iadanza; Victor W Pike; Giuseppe Ronsisvalle
Synthesis of (+)- and (-)-cis-2-[(1-adamantylamino)-methyl]-1-phenylcyclopropane derivatives as high affinity probes for sigma1 and sigma2 binding sites.
Farmaco (Società chimica italiana : 1989) 2002;57(1):45-53.
2001: Agostino Marrazzo; Orazio Prezzavento; L Pasquinucci; Franco Vittorio; Giuseppe Ronsisvalle
Synthesis and pharmacological evaluation of potent and enantioselective sigma 1, and sigma 2 ligands.
Farmaco (Società chimica italiana : 1989) 2001;56(3):181-9.
2001: Giuseppe Ronsisvalle; Agostino Marrazzo; L Pasquinucci; Orazio Prezzavento; Maria S Pappalardo; Franco Vittorio
Specific kappa opioid receptor agonists.
Farmaco (Società chimica italiana : 1989) 2001;56(1-2):121-5.
2001: Giuseppe Ronsisvalle; Orazio Prezzavento; Agostino Marrazzo; Franco Vittorio; Ennio Bousquet; Rosanna Di Toro; santi spampinato
Synthesis and binding affinity of cis-(-)- and cis-(+)-N-ethyleneamino-N-nordeoxymetazocine and cis-(-)-N-normetazocine analogues at sigma1, sigma2 and kappa opioid receptors.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 2001;12(3):277-84.
2000: Giuseppe Ronsisvalle; L Pasquinucci; V Pittalà; Agostino Marrazzo; Orazio Prezzavento; Rosanna Di Toro; B Falcucci; santi spampinato
Nonpeptide analogues of dynorphin A(1-8): design, synthesis, and pharmacological evaluation of kappa-selective agonists.
Journal of medicinal chemistry 2000;43(16):2992-3004.
2000: Giuseppe Ronsisvalle; Agostino Marrazzo; Orazio Prezzavento; L Pasquinucci; B Falcucci; Rosanna Di Toro; santi spampinato
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites.
Bioorganic & medicinal chemistry 2000;8(6):1503-13.
2000: Antonio Lavecchia; Giovanni Greco; Ettore Novellino; Franco Vittorio; Giuseppe Ronsisvalle
Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations.
Journal of medicinal chemistry 2000;43(11):2124-34.
1999: Natale Alfredo Santagati; Ennio Bousquet; Spadaro Angelo; Giuseppe Ronsisvalle
4-quinazolinones: synthesis and reduction of prostaglandin E2 production.
Farmaco (Società chimica italiana : 1989) 1999;54(11-12):780-4.
1998: Giuseppe Ronsisvalle; Agostino Marrazzo; Orazio Prezzavento; L Pasquinucci; Franco Vittorio; V Pittalà; Maria S Pappalardo; S Cacciaguerra; santi spampinato
(+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties.
Journal of medicinal chemistry 1998;41(10):1574-80.
1997: Giuseppe Ronsisvalle; Orazio Prezzavento; L Pasquinucci; Maria S Pappalardo; Agostino Marrazzo; Franco Vittorio; L Carboni; santi spampinato
Synthesis of (+)-(1'R,2'S) and (1'S,2'R)-6,11-dimethyl-1,2,3,4,5,6 -hexahydro-3-[[2'-(alkoxycarbonyl)-2'-phenylcyclopropyl]methyl]-2 ,6 -methano-3-benzazocin-8-ol. Comparison of the affinities for sigma 1 and opioid receptors with in the diastereoisomeric MPCB and CCB.
Farmaco (Società chimica italiana : 1989) 1997;52(6-7):471-6.
1997: L Carboni; Gabriele Campana; S Cacciaguerra; Giovanna Murari; Ester Speroni; Maria S Pappalardo; Giuseppe Ronsisvalle; santi spampinato
Agonist binding properties for recombinant kappa opioid receptors expressed in CHO-K1 cells.
Annals of the New York Academy of Sciences 1997;812():203-4.
1995: Franco Vittorio; Giuseppe Ronsisvalle; Agostino Marrazzo; G Blandino
Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hydrazones.
Farmaco (Società chimica italiana : 1989) 1995;50(4):265-72.
1995: Giuseppe Ronsisvalle; Orazio Prezzavento; L Pasquinucci; Agostino Marrazzo; Franco Vittorio; J A Gomez-Vidal; L Carboni; santi spampinato
CCB, a novel specific kappa opioid agonist, which discriminates between opioid and sigma 1 recognition sites.
Life sciences 1995;57(16):1487-95.
1994: Franco Vittorio; Maria S Pappalardo; Giuseppe Ronsisvalle; A Caruso; Vincenza Maria Cutuli; Matilde Amico-Roxas
Synthesis and pharmacological evaluation of 3H-pyridazino[4,5-b][1,4]benzothiazin-4(10H)-one derivatives.
Farmaco (Società chimica italiana : 1989) 1994;49(4):237-44.
1993: Giuseppe Ronsisvalle; L Pasquinucci; Maria S Pappalardo; Franco Vittorio; G Fronza; C Romagnoli; E Pistacchio; santi spampinato; S Ferri
Non-peptide ligands for opioid receptors. Design of kappa-specific agonists.
Journal of medicinal chemistry 1993;36(13):1860-5.
1991: Giuseppe Ronsisvalle; Maria S Pappalardo; santi spampinato; A Mele
Opioid receptors: development of selective peptidomimetics with agonist or antagonist activity.
Farmaco (Società chimica italiana : 1989) 1991;46(1 Suppl):171-5.
1990: Francesco Guerrera; L Salerno; Maria Angela Siracusa; Giuseppe Ronsisvalle; A Caruso; M G Leone; Alex Felice
Synthesis and pharmacological properties of 2-nitro-3-substituted-amino benzo[b]thiophenes and 1-substituted benzothieno[2,3-d]imidazoles.
Farmaco (Società chimica italiana : 1989) 1990;45(1):29-38.
1989: Franco Vittorio; Maria S Pappalardo; Giuseppe Ronsisvalle; A Caruso; M G Leone; Matilde Amico-Roxas
Chemical and pharmacological investigations on 2H-pyridazino[4,5-b] [1,4]benzothiazin-1(10H)-one derivatives.
Farmaco (Società chimica italiana : 1989) 1989;44(10):911-32.
1989: L Vio; Maria Grazia Mamolo; Giuseppe Ronsisvalle; S Oliveri; A M Grego
Synthesis and antifungal activity of some amidrazone derivatives.
Farmaco (Società chimica italiana : 1989) 1989;44(9):819-29.
1989: Giuseppe Ronsisvalle; Maria S Pappalardo; Franco Vittorio; L Pasquinucci; E Bousquet; S Oliveri; E Cammarata
Synthesis of substituted pyrimidines, pyrazole[3,4-d]pyrimidines and imidazo[4,5-d]pyrimidines and evaluation of their antifungal activity.
Farmaco (Società chimica italiana : 1989) 1989;44(4):383-90.
1988: Francesco Guerrera; M C Sarvà; Maria Angela Siracusa; Giuseppe Ronsisvalle; G Conforto; S Dibennardo; G Failla; M Matera
[Synthesis and anti-ulcer activity of 3-arylprop-2-enthionoethyl esters].
Il Farmaco; edizione scientifica 1988;43(6):551-8.
1988: Giuseppe Romeo; E Bousquet; Maria S Pappalardo; Giuseppe Ronsisvalle; S Oliveri; E Cammarata
[Synthesis and antifungal activity of new derivatives of 5-(4-halobenzoyl)-4-amino-3-(2-dialkylaminoethylthio)thieno [2,3-c] and [3,2-d] isothiazole].
Il Farmaco; edizione scientifica 1988;43(5):457-67.
1988: Franco Vittorio; Maria S Pappalardo; Giuseppe Ronsisvalle; G Blandino
Studies on isoquinoline derivatives. IV. Synthesis and evaluation of the antimicrobial and antifungal activities of N2-arylidene-substituted 3-carbazoyl-isoquinolines.
Il Farmaco; edizione scientifica 1988;43(3):239-50.
1985: Franco Vittorio; Giuseppe Ronsisvalle; Maria S Pappalardo; G Blandino
Synthesis and antibacterial activity of 3-(2-arylvinylen)-2-isoxazolines.
Il Farmaco; edizione scientifica 1985;40(5):359-68.
1983: Giuseppe Ronsisvalle; Franco Vittorio; Maria S Pappalardo
Synthesis and biological activity of some di(nitrothienyl)- and di(acetylaminothienyl)sulfones.
Il Farmaco; edizione scientifica 1983;38(11):877-83.
1981: Giuseppe Ronsisvalle; G Blandino
Synthesis, spectral behaviour and microbiological properties of some di(nitrothienyl)sulfides.
Il Farmaco; edizione scientifica 1981;36(9):785-93.