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William Roush

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TOP 3
Ming Chen; William R Roush
Enantioselective synthesis of (+)-crocacin C. An example of a highly challenging mismatched double asymmetric δ-stannylcrotylboration reaction.
Yanchen Zhou; Juliet Agudelo; Sean M Amberg; Yen Ting Chen; Charles S Craik; David H Goetz; Elizabeth Hansell; Kai Lu; James McKerrow; William R Roush; Graham Simmons
Inhibitors of SARS-CoV entry--identification using an internally-controlled dual envelope pseudovirion assay.
Huikai Sun; Jason R Abbott; William R Roush
Stereoselective synthesis of a model C(18)-C(35) spiroketal fragment of integramycin.

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All Publications

2012: Ming Chen; William R Roush
Enantioselective synthesis of (+)-crocacin C. An example of a highly challenging mismatched double asymmetric δ-stannylcrotylboration reaction.
Organic letters 2012;14(7):1880-3.
2011: Yanchen Zhou; Juliet Agudelo; Sean M Amberg; Yen Ting Chen; Charles S Craik; David H Goetz; Elizabeth Hansell; Kai Lu; James McKerrow; William R Roush; Graham Simmons
Inhibitors of SARS-CoV entry--identification using an internally-controlled dual envelope pseudovirion assay.
Antiviral research 2011;92(2):187-94.
2011: Huikai Sun; Jason R Abbott; William R Roush
Stereoselective synthesis of a model C(18)-C(35) spiroketal fragment of integramycin.
Organic letters 2011;13(10):2734-7.
2010: Franck Madoux; Scott Simanski; Peter Chase; Jitendra K Mishra; William R Roush; Nagi Ayad; Peter Hodder
An ultra-high throughput cell-based screen for wee1 degradation inhibitors.
Journal of biomolecular screening 2010;15(8):907-17.
2010: Ming Chen; William R Roush
Highly (E)-selective BF(3).Et(2)O-promoted allylboration of chiral nonracemic alpha-substituted allylboronates and analysis of the origin of stereocontrol.
Organic letters 2010;12(12):2706-9.
2010: Ming Chen; Daniel H Ess; William R Roush
Enantioselective synthesis of (E)-delta-stannyl homoallylic alcohols via aldehyde allylboration using alpha-stannylallylboranes generated by allene hydroboration followed by a highly diastereoselective 1,3-boratropic shift.
Journal of the American Chemical Society 2010;132(23):7881-3.
2010: Chen He; George P Nora; Eric L Schneider; Iain D Kerr; Elizabeth Hansell; Ken Hirata; David Gonzalez; Mohammed Sajid; Sarah E Boyd; Petr Hruz; Eduardo R Cobo; Christine Le; Wei-Ting Liu; Lars Eckmann; Pieter dorrestein; Eric R Houpt; Linda S Brinen; Charles S Craik; William R Roush; James McKerrow; Sharon L Reed
A novel Entamoeba histolytica cysteine proteinase, EhCP4, is key for invasive amebiasis and a therapeutic target.
The Journal of biological chemistry 2010;285(24):18516-27.
2009: Jeremy Kister; Amy C DeBaillie; Ricardo Lira; William R Roush
Stereoselective synthesis of gamma-substituted (Z)-allylic boranes via kinetically controlled hydroboration of allenes with 10-TMS-9-borabicyclo[3.3.2]decane.
Journal of the American Chemical Society 2009;131(40):14174-5.
2009: Fangzheng Li; William R Roush
Stereoselective synthesis of syn,syn- and syn,anti-1,3,5-triols via intramolecular hydrosilylation of substituted pent-3-en-1,5-diols.
Organic letters 2009;11(13):2932-5.
2008: Mariola Tortosa; Neal A Yakelis; William R Roush
Total synthesis of (+)-superstolide A.
The Journal of organic chemistry 2008;73(24):9657-67.
2008: Joshua R Dunetz; Lisa D Julian; Jason S Newcom; William R Roush
Total syntheses of (+)-tedanolide and (+)-13-deoxytedanolide.
Journal of the American Chemical Society 2008;130(48):16407-16.
2008: Robert H Bates; J Brad Shotwell; William R Roush
Stereoselective syntheses of the C(1)-C(9) fragment of amphidinolide C.
Organic letters 2008;10(19):4343-6.
2008: Joshua R Dunetz; William R Roush
Concerning the synthesis of the tedanolide C(13)-C(23) fragment via anti-aldol reaction.
Organic letters 2008;10(10):2059-62.
2008: SusAnn M Winbush; Dustin J Mergott; William R Roush
Total synthesis of (-)-spinosyn A: examination of structural features that govern the stereoselectivity of the key transannular Diels-Alder reaction.
The Journal of organic chemistry 2008;73(5):1818-29.
2008: Mariola Tortosa; Neal A Yakelis; William R Roush
Total synthesis of +-superstolide A.
Journal of the American Chemical Society 2008;130(9):2722-3.
2008: Jacqueline D Hicks; William R Roush
Synthesis of the C(26)-C(42) and C(43)-C(67) pyran-containing fragments of amphidinol 3 via a common pyran intermediate.
Organic letters 2008;10(4):681-4.
2008: Masaki Handa; William J Smith; William R Roush
Studies on the synthesis of apoptolidin A. 2. Synthesis of the disaccharide unit.
The Journal of organic chemistry 2008;73(3):1036-9.
2008: Masaki Handa; Karl A Scheidt; Martin Bossart; Nan Zheng; William R Roush
Studies on the synthesis of apoptolidin A. 1. Synthesis of the C(1)-C(11) fragment.
The Journal of organic chemistry 2008;73(3):1031-5.
2007: Jacqueline D Hicks; Chan Woo Huh; Ashley D Legg; William R Roush
Concerning the selective protection of (Z)-1,5-syn-ene-diols and (E)-1,5-anti-ene-diols as allylic triethylsilyl ethers.
Organic letters 2007;9(26):5621-4.
2007: Ricardo Lira; William R Roush
Enantio- and diastereoselective synthesis of syn-beta-hydroxyallylsilanes via a chiral (Z)-gamma-silylallylboronate.
Organic letters 2007;9(21):4315-8.
2007: D H Goetz; Youngchool Choe; Elizabeth Hansell; Y T Chen; M McDowell; C B Jonsson; William R Roush; James H McKerrow; Charles S Craik
Substrate specificity profiling and identification of a new class of inhibitor for the major protease of the SARS coronavirus.
Biochemistry 2007;46(30):8744-52.
2007: Samuel G Meléndez-López; Scott Herdman; Ken Hirata; Min-Ho Choi; Youngchool Choe; Charles Craik; Conor R Caffrey; Elizabeth Hansell; Bibiana Chávez-Munguía; Yen Ting Chen; William R Roush; James H McKerrow; Lars Eckmann; Jianhua Guo; Samuel L Stanley; Sharon L Reed
Use of recombinant Entamoeba histolytica cysteine proteinase 1 to identify a potent inhibitor of amebic invasion in a human colonic model.
Eukaryotic cell 2007;6(7):1130-6.
2007: Ricardo Lira; William R Roush
Stereoselective synthesis of the C(1)-C(19) fragment of tetrafibricin.
Organic letters 2007;9(3):533-6.
2007: Porino Va; William R Roush
Synthesis of 2-epi-amphidinolide E: an unexpected and highly selective C(2)inversion during an esterification reaction.
Organic letters 2007;9(2):307-10.
2006: Porino Va; William R Roush
Total synthesis of amphidinolide E.
Journal of the American Chemical Society 2006;128(50):15960-1.
2006: Tony K Trullinger; Jun Qi; William R Roush
Studies on the synthesis of quartromicins a(3) and d(3): synthesis of the vertical and horizontal bis-spirotetronate fragments.
The Journal of organic chemistry 2006;71(18):6915-22.
2006: Jun Qi; William R Roush
Synthesis of precursors of the agalacto (exo) fragment of the quartromicins via an auxiliary-controlled exo-selective Diels-Alder reaction.
Organic letters 2006;8(13):2795-8.
2005: Reema K Thalji; William R Roush
Remarkable phosphine-effect on the intramolecular aldol reactions of unsaturated 1,5-diketones: highly regioselective synthesis of cross-conjugated dienones.
Journal of the American Chemical Society 2005;127(48):16778-9.
2005: Jacqueline D Hicks; Eric M Flamme; William R Roush
Synthesis of the C(43)-C(67) fragment of amphidinol 3.
Organic letters 2005;7(24):5509-12.
2005: William T Lambert; William R Roush
Synthesis of the A-B subunit of angelmicin B.
Organic letters 2005;7(24):5501-4.
2005: Eric Mertz; Jennifer M Tinsley; William R Roush
[3 + 2]-annulation reactions of chiral allylsilanes and chiral aldehydes. studies on the synthesis of bis-tetrahydrofuran substructures of annonaceous acetogenins.
The Journal of organic chemistry 2005;70(20):8035-46.
2005: Jennifer M Tinsley; Eric Mertz; Pek Y Chong; Robert-André F Rarig; William R Roush
Synthesis of (+)-bullatacin via the highly diastereoselective [3+2] annulation reaction of a racemic aldehyde and a nonracemic allylsilane.
Organic letters 2005;7(19):4245-8.
2005: Robert M. Owen; William R Roush
Stereoselective synthesis of the C(1)-C(11) fragment of peloruside A.
Organic letters 2005;7(18):3941-4.
2005: Jennifer M Tinsley; William R Roush
Total synthesis of asimicin via highly stereoselective [3 + 2] annulation reactions of substituted allylsilanes.
Journal of the American Chemical Society 2005;127(31):10818-9.
2005: Cheryl L Heitzman; William T Lambert; Eric Mertz; J Brad Shotwell; Jennifer M Tinsley; Porino Va; William R Roush
Efficient protiodesilylation of unactivated C(sp3)-SiMe2Ph bonds using tetrabutylammonium fluoride.
Organic letters 2005;7(12):2405-8.
2005: Lisa D Julian; Jason S Newcom; William R Roush
Total synthesis of (+)-13-deoxytedanolide.
Journal of the American Chemical Society 2005;127(17):6186-7.
2005: Christopher M Liu; William J Smith; Darin J Gustin; William R Roush
Experimental evidence for chair-like transition states in aldol reactions of methyl ketone lithium enolates: stereoselective synthesis and utilization of a deuterium-labeled enolate as a probe of reaction stereochemistry.
Journal of the American Chemical Society 2005;127(16):5770-1.
2005: Eric M Flamme; William R Roush
Synthesis of the C(1)-C(25) fragment of amphidinol 3: application of the double-allylboration reaction for synthesis of 1,5-diols.
Organic letters 2005;7(7):1411-4.
2005: Thomas A Dineen; William R Roush
Stereoselective synthesis of the octahydronaphthalene unit of integramycin via an intramolecular Diels-Alder reaction.
Organic letters 2005;7(7):1355-8.
2005: Eric M Flamme; William R Roush
Synthesis of 2,6-trans-disubstituted 5,6-dihydropyrans from (Z)-1,5-syn-endiols.
Beilstein journal of organic chemistry 2005;1(1):7.
2004: J Brad Shotwell; William R Roush
Synthesis of the C11-C29 fragment of amphidinolide F.
Organic letters 2004;6(21):3865-8.
2004: Sridhar Narayan; William R Roush
Studies toward the total synthesis of angelmicin B (hibarimicin B): synthesis of a model CD-D' arylnaphthoquinone.
Organic letters 2004;6(21):3789-92.
2004: Dustin J Mergott; Scott A Frank; William R Roush
Total synthesis of (-)-spinosyn A.
Proceedings of the National Academy of Sciences of the United States of America 2004;101(33):11955-9.
2004: Timothy B Durham; Nicolas Blanchard; Brad M Savall; Noel A Powell; William R Roush
Total synthesis of formamicin.
Journal of the American Chemical Society 2004;126(30):9307-17.
2004: William R Roush; R Jeffrey Neitz
Studies on the synthesis of landomycin A. Synthesis of the originally assigned structure of the aglycone, landomycinone, and revision of structure.
The Journal of organic chemistry 2004;69(15):4906-12.
2004: Thomas A Dineen; William R Roush
Total synthesis of cochleamycin A.
Organic letters 2004;6(12):2043-6.
2003: Thomas A Dineen; William R Roush
Probing the Lewis acid-catalyzed intramolecular Diels-Alder cyclizations of allylic alkoxy-substituted (Z)-1,3-dienes.
Organic letters 2003;5(24):4725-8.
2003: Joey L Methot; William R Roush
Synthetic studies toward FR182877. Remarkable solvent effect in the vinylogous morita-baylis-hillman cyclization.
Organic letters 2003;5(22):4223-6.
2003: Anthony E Boitano; Cory D Emal; Francesco Leonetti; Neal Blatt; Thomas A Dineen; Jonathan A Ellman; William R Roush; Anthony William Opipari Jr; Gary D Glick
Structure activity studies of a novel cytotoxic benzodiazepine.
Bioorganic & medicinal chemistry letters 2003;13(19):3327-30.
2003: Jason J Reddick; Jianming Cheng; William R Roush
Relative rates of Michael reactions of 2'-(phenethyl)thiol with vinyl sulfones, vinyl sulfonate esters, and vinyl sulfonamides relevant to vinyl sulfonyl cysteine protease inhibitors.
Organic letters 2003;5(11):1967-70.
2003: Timothy B Durham; William R Roush
Stereoselective synthesis of functionalized precursors of the CDEF and CDE 2,6-dideoxy-tetra- and trisaccharide units of durhamycins A and B.
Organic letters 2003;5(11):1875-8.
2003: Timothy B Durham; William R Roush
Stereoselective synthesis of 2-deoxy-beta-galactosides via 2-deoxy-2-bromo- and 2-deoxy-2-iodo-galactopyranosyl donors.
Organic letters 2003;5(11):1871-4.
2003: Neal A Yakelis; William R Roush
Synthesis of the C(21)-C(26) fragment of superstolide A: concerning the stereochemistry of (E)-crotylboration reactions of alaninal derivatives.
The Journal of organic chemistry 2003;68(10):3838-43.
2003: Jung-Nyoung Heo; Edward B Holson; William R Roush
Common-intermediate strategy for synthesis of conduritols and inositols via beta-hydroxy cyclohexenylsilanes.
Organic letters 2003;5(10):1697-700.
2003: Jung-Nyoung Heo; Glenn C. Micalizio; William R Roush
Enantio- and diastereoselective synthesis of cyclic beta-hydroxy allylsilanes via sequential aldehyde gamma-silylallylboration and ring-closing metathesis reactions.
Organic letters 2003;5(10):1693-6.
2003: Sherry R Chemler; William R Roush
Stereochemistry of the allylation and crotylation reactions of alpha-methyl-beta-hydroxy aldehydes with allyl- and crotyltrifluorosilanes. Synthesis of anti,anti-dipropionate stereotriads and stereodivergent pathways for the reactions with 2,3-anti- and 2,3-syn-alpha-methyl-beta-hydroxy aldehydes.
The Journal of organic chemistry 2003;68(4):1319-33.
2003: Brad M Savall; Nicolas Blanchard; William R Roush
Total synthesis of the formamicin aglycon, formamicinone.
Organic letters 2003;5(3):377-9.
2003: Nicolas Blanchard; William R Roush
2-Deoxy-2-iodo-beta-glucopyranosyl fluorides: mild and highly stereoselective glycosyl donors for the synthesis of 2-deoxy-beta-glycosides from beta-hydroxy ketones.
Organic letters 2003;5(1):81-4.
2003: Bhaskar R Shenai; Belinda J Lee; Alejandro Alvarez-Hernandez; Pek Y Chong; Cory D Emal; R Jeffrey Neitz; William R Roush; Philip J Rosenthal
Structure-activity relationships for inhibition of cysteine protease activity and development of Plasmodium falciparum by peptidyl vinyl sulfones.
Antimicrobial agents and chemotherapy 2003;47(1):154-60.
2002: William R Roush; Jason S Newcom
Studies on the synthesis of tedanolide. 2. Stereoselective synthesis of a protected C(1)-C(12) fragment.
Organic letters 2002;4(26):4739-42.
2002: Pek Y Chong; William R Roush
Concerning the origin of the high beta-selectivity of glycosidation reactions of 2-deoxy-2-iodo-glucopyranosyl trichloroacetimidates.
Organic letters 2002;4(25):4523-6.
2002: Eric M Flamme; William R Roush
Enantioselective synthesis of 1,5-anti- and 1,5-syn-diols using a highly diastereoselective one-pot double allylboration reaction sequence.
Journal of the American Chemical Society 2002;124(46):13644-5.
2002: Edward B Holson; William R Roush
Synthesis of the C(2)-C(13) fragment (the A-B spiroketal unit) of spongistatin 1 (altohyrtin A): use of a common intermediate for the synthesis of both spongistatin spiroketals.
Organic letters 2002;4(21):3723-5.
2002: Edward B Holson; William R Roush
Diastereoselective synthesis of the C(17)-C(28) fragment (the C-D spiroketal unit) of spongistatin 1 (altohyrtin A) via a kinetically controlled iodo-spiroketalization reaction.
Organic letters 2002;4(21):3719-22.
2002: Benjamin W Gung; Xiaowen Xue; William R Roush
The origin of diastereofacial control in allylboration reactions using tartrate ester derived allylboronates: attractive interactions between the Lewis acid coordinated aldehyde carbonyl group and an ester carbonyl oxygen.
Journal of the American Chemical Society 2002;124(36):10692-7.
2002: Dustin J Mergott; Scott A Frank; William R Roush
Application of the intramolecular vinylogous Morita-Baylis-Hillman reaction toward the synthesis of the spinosyn A tricyclic nucleus.
Organic letters 2002;4(18):3157-60.
2002: Alejandro Alvarez Hernandez; William R Roush
Recent advances in the synthesis, design and selection of cysteine protease inhibitors.
Current opinion in chemical biology 2002;6(4):459-65.
2002: Karl A Scheidt; Thomas D Bannister; Akihiro Tasaka; Michael D Wendt; Brad M Savall; Glenn J Fegley; William R Roush
Total synthesis of (-)-bafilomycin A(1).
Journal of the American Chemical Society 2002;124(24):6981-90.
2002: Scott A Frank; William R Roush
Studies on the synthesis of (-)-spinosyn a: application of the steric directing group strategy to transannular Diels-Alder reactions.
The Journal of organic chemistry 2002;67(12):4316-24.
2002: William R Roush; Thomas D Bannister; Michael D Wendt; Michael S VanNieuwenhze; Darin J Gustin; Garrett J Dilley; Gregory C Lane; Karl A Scheidt; William J Smith
An NMR method for assigning relative stereochemistry to beta-hydroxy ketones deriving from aldol reactions of methyl ketones.
The Journal of organic chemistry 2002;67(12):4284-9.
2002: William R Roush; Thomas D Bannister; Michael D Wendt; JIll Jablonowski; Karl A Scheidt
Studies on the synthesis of bafilomycin A(1): stereochemical aspects of the fragment assembly aldol reaction for construction of the C(13)-C25) segment.
The Journal of organic chemistry 2002;67(12):4275-83.
2002: William R Roush; Chris Limberakis; Roxanne K Kunz; David A Barda
Diastereoselective synthesis of the endo- and exo-spirotetronate subunits of the quartromicins. The first enantioselective Diels-Alder reaction of an acyclic (Z)-1,3-diene.
Organic letters 2002;4(9):1543-6.
2002: William R Roush; David A Barda
Partial stereochemical assignment of quartromicins A3 and D3.
Organic letters 2002;4(9):1539-42.
2002: Scott A Frank; Dustin J Mergott; William R Roush
The vinylogous intramolecular Morita-Baylis-Hillman reaction: synthesis of functionalized cyclopentenes and cyclohexenes with trialkylphosphines as nucleophilic catalysts.
Journal of the American Chemical Society 2002;124(11):2404-5.
2001: Conor R Caffrey; Elizabeth Hansell; Kimberley D Lucas; Linda S Brinen; Alejandro Alvarez-Hernandez; J Cheng; S L Gwaltney; William R Roush; Y D Stierhof; Matthew Bogyo; Dietmar Steverding; James H McKerrow
Active site mapping, biochemical properties and subcellular localization of rhodesain, the major cysteine protease of Trypanosoma brucei rhodesiense.
Molecular and biochemical parasitology 2001;118(1):61-73.
2001: William R Roush; J Cheng; B Knapp-Reed; Alejandro Alvarez-Hernandez; James H McKerrow; Elizabeth Hansell; Juan C Engel
Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain.
Bioorganic & medicinal chemistry letters 2001;11(20):2759-62.
2001: William R Roush; CE Bennett; S E Roberts
Studies on the synthesis of landomycin A: synthesis and glycosidation reactions of L-rhodinosyl acetate derivatives.
The Journal of organic chemistry 2001;66(19):6389-93.
2001: Brad M Savall; Noel A Powell; William R Roush
Highly diastereoselective synthesis of propargylic 1,2-anti-diol derivatives using alpha-alkoxypropargylstannanes.
Organic letters 2001;3(19):3057-60.
2001: Glenn C. Micalizio; William R Roush
Studies on the synthesis of pectenotoxin II: synthesis of a C(11)-C(26) fragment precursor via [3 + 2]-annulation reactions of chiral allylsilanes.
Organic letters 2001;3(12):1949-52.
2001: Robert Ménard; C Therrien; Paule Lachance; Traian Sulea; H Qo; Alejandro Alvarez-Hernandez; William R Roush
Cathepsins X and B display distinct activity profiles that can be exploited for inhibitor design.
Biological chemistry 2001;382(5):839-45.
2001: N A Yakelis; William R Roush
Lewis acid catalyzed intramolecular Diels-Alder reactions of acyclic (Z)-substituted 1,3-dienes.
Organic letters 2001;3(6):957-60.
2001: C Therrien; Paule Lachance; Traian Sulea; Enrico O Purisima; Hongtao Qi; Edmund Ziomek; Alejandro Alvarez-Hernandez; William R Roush; Robert Ménard
Cathepsins X and B can be differentiated through their respective mono- and dipeptidyl carboxypeptidase activities.
Biochemistry 2001;40(9):2702-11.
2001: Noel A Powell; William R Roush
Studies on the total synthesis of formamicin: synthesis of the C(1)-C(11) fragment.
Organic letters 2001;3(3):453-6.
2000: Glenn C. Micalizio; A N Pinchuk; William R Roush
Synthesis of the C(29)-C(45) bis-pyran subunit (E-F) of spongistatin 1 (Altohyrtin A).
The Journal of organic chemistry 2000;65(25):8730-6.
2000: Scott A Frank; H Chen; R K Kunz; M J Schnaderbeck; William R Roush
Use of thallium(I) ethoxide in Suzuki cross coupling reactions.
Organic letters 2000;2(17):2691-4.
2000: Linda S Brinen; Elizabeth Hansell; J Cheng; William R Roush; James H McKerrow; Robert J Fletterick
A target within the target: probing cruzain's P1' site to define structural determinants for the Chagas' disease protease.
Structure (London, England : 1993) 2000;8(8):831-40.
2000: William R Roush; L A Pfeifer
Total synthesis of mycalamide A and 7-epi-mycalamide A.
Organic letters 2000;2(6):859-62.
2000: Glenn C. Micalizio; William R Roush
A three-component coupling strategy for tetrahydrofuran synthesis: application of the diisopropyl tartrate modified (E)-gamma-(dimethylphenylsilyl)allylboronate as an alpha,gamma-allyl dianion equivalent.
Organic letters 2000;2(4):461-4.
1999: William R Roush; Sridhar Narayan
2-Deoxy-2-iodo-alpha-mannopyranosyl and -talopyranosyl acetates: highly stereoselective glycosyl donors for the synthesis of 2-deoxy-alpha-glycosides.
Organic letters 1999;1(6):899-902.
1999: William R Roush; Sridhar Narayan; CE Bennett; K Briner
Iodoacetoxylation of glycals using cerium(IV) ammonium nitrate, sodium iodide, and acetic acid: stereoselective synthesis of 2-deoxy-2-iodo-alpha-mannopyranosyl acetates.
Organic letters 1999;1(6):895-7.
1999: William R Roush; Benjamin W Gung; CE Bennett
2-Deoxy-2-iodo- and 2-deoxy-2-bromo-alpha-glucopyranosyl trichloroacetimidates: highly reactive and stereoselective donors for the synthesis of 2-deoxy-beta-glycosides.
Organic letters 1999;1(6):891-3.
1999: William R Roush; G C Lane
Studies on the synthesis of tedanolide: synthesis of the C(5)-C(21) segment via a highly stereoselective fragment assembly aldol reaction of a chiral beta,gamma-unsaturated methyl ketone.
Organic letters 1999;1(1):95-8.
1998: Karl A Scheidt; William R Roush; James H McKerrow; P M Selzer; Elizabeth Hansell; P J Rosenthal
Structure-based design, synthesis and evaluation of conformationally constrained cysteine protease inhibitors.
Bioorganic & medicinal chemistry 1998;6(12):2477-94.
1998: William R Roush; Florenci V González; James H McKerrow; Elizabeth Hansell
Design and synthesis of dipeptidyl alpha',beta'-epoxy ketones, potent irreversible inhibitors of the cysteine protease cruzain.
Bioorganic & medicinal chemistry letters 1998;8(19):2809-12.