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Peter Schiller

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Irena Berezowska; Nga N Chung; Jinguo Ding; Carole Lemieux; Peter W Schiller
Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists.
Hazel H Szeto; Peter W Schiller
Novel therapies targeting inner mitochondrial membrane--from discovery to clinical development.
Peter W Schiller
Bi- or multifunctional opioid peptide drugs.

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All Publications

2012: Irena Berezowska; Nga N Chung; Jinguo Ding; Carole Lemieux; Peter W Schiller
Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists.
Bioorganic & medicinal chemistry letters 2012;22(5):1899-902.
2011: Hazel H Szeto; Peter W Schiller
Novel therapies targeting inner mitochondrial membrane--from discovery to clinical development.
Pharmaceutical research 2011;28(11):2669-79.
2010: Peter W Schiller
Bi- or multifunctional opioid peptide drugs.
Life sciences 2010;86(15-16):598-603.
2010: Grazyna Weltrowska; Nga N Chung; Carole Lemieux; Jianxin Guo; Yixin Lu; Brian C Wilkes; Peter W Schiller
"Carba"-analogues of fentanyl are opioid receptor agonists.
Journal of medicinal chemistry 2010;53(7):2875-81.
2010: Grazyna Weltrowska; Irena Berezowska; Carole Lemieux; Nga N Chung; Brian C Wilkes; Peter W Schiller
N-methylated cyclic enkephalin analogues retain high opioid receptor binding affinity.
Chemical biology & drug design 2010;75(2):182-8.
2009: Irena Berezowska; Nga N Chung; Carole Lemieux; Brian C Wilkes; Peter W Schiller
Agonist vs antagonist behavior of delta opioid peptides containing novel phenylalanine analogues in place of Tyr(1).
Journal of medicinal chemistry 2009;52(21):6941-5.
2009: Irena Berezowska; Carole Lemieux; Nga N Chung; Brian C Wilkes; Peter W Schiller
Cyclic opioid peptide agonists and antagonists obtained via ring-closing metathesis.
Chemical biology & drug design 2009;74(4):329-34.
2009: Jerzy Ciarkowski; A Zieleniak; S Rodziewicz-Motowidło; Ł Rusak; Nga N Chung; Cezary Czaplewski; E Witkowska; Peter W Schiller; Jan Izdebski
Deltorphin analogs restricted via a urea bridge: structure and opioid activity.
Advances in experimental medicine and biology 2009;611():491-2.
2009: Jerzy Ciarkowski; Cezary Czaplewski; Sylwia Łuczak; Sylwia Rodziewicz-Motowidło; Irena Berezowska; Peter W Schiller
Conformation-activity relationships of cyclo-constrained mu/delta opioid agonists derived from the N-terminal tetrapeptide segment of dermorphin/deltorphin.
Advances in experimental medicine and biology 2009;611():489-90.
2009: Grazyna Weltrowska; Carole Lemieux; Nga N Chung; Brian C Wilkes; Peter W Schiller
Stereoselective synthesis of (3S)- and (3R)-3-hydroxy-3-(2,6-dimethyl-4-hydroxyphenyl)propanoic acid and its incorporation into a cyclic enkephalin analogue.
Advances in experimental medicine and biology 2009;611():207-8.
2008: Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Peter W Schiller
Potent opioid peptide agonists containing 4'-[N-((4'-phenyl)-phenethyl)carboxamido]phenylalanine (Bcp) in place of Tyr.
Chemical biology & drug design 2008;72(5):337-40.
2008: Animesh Ghosh; Jie Luo; Chen Liu; Grazyna Weltrowska; Carole Lemieux; Nga N Chung; Yixin Lu; Peter W Schiller
Novel opioid peptide derived antagonists containing (2S)-2-methyl-3-(2,6-dimethyl-4-carbamoylphenyl)propanoic acid [(2S)-Mdcp].
Journal of medicinal chemistry 2008;51(18):5866-70.
2007: Irena Berezowska; Nga N Chung; Carole Lemieux; Brian C Wilkes; Peter W Schiller
Dicarba analogues of the cyclic enkephalin peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) retain high opioid activity.
Journal of medicinal chemistry 2007;50(6):1414-7.
2006: Yixin Lu; Tze Keong Lum; Yoon Wui Leow Augustine; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Peter W Schiller
Replacement of the N-terminal tyrosine residue in opioid peptides with 3-(2,6-dimethyl-4-carbamoylphenyl)propanoic acid (Dcp) results in novel opioid antagonists.
Journal of medicinal chemistry 2006;49(17):5382-5.
2006: Irena Berezowska; Nga N Chung; Carole Lemieux; Brian C Wilkes; Peter W Schiller
Cyclic dermorphin tetrapeptide analogues obtained via ring-closing metathesis.
Acta biochimica Polonica 2006;53(1):73-6.
2005: Peter W Schiller; Irena Berezowska; Grazyna Weltrowska; H Chen; Carole Lemieux; Nga N Chung
Type and location of fluorescent probes incorporated into the potent mu-opioid peptide [Dmt]DALDA affect potency, receptor selectivity and intrinsic efficacy.
The journal of peptide research : official journal of the American Peptide Society 2005;65(6):556-63.
2005: Peter W Schiller
Opioid peptide-derived analgesics.
The AAPS journal 2005;7(3):E560-5.
2005: Grazyna Weltrowska; Carole Lemieux; Nga N Chung; Peter W Schiller
Cyclic enkephalin analogs containing various para-substituted phenylalanine derivatives in place of Tyr1 are potent opioid agonists.
The journal of peptide research : official journal of the American Peptide Society 2005;65(1):36-41.
2005: Heru Chen; Nga N Chung; Carole Lemieux; Bogumil Zelent; Jane M Vanderkooi; Ignacy Gryczynski; Brian C Wilkes; Peter W Schiller
[Aladan3]TIPP: a fluorescent delta-opioid antagonist with high delta-receptor binding affinity and delta selectivity.
Biopolymers 2005;80(2-3):325-31.
2005: Hazel H Szeto; Peter W Schiller; Kesheng Zhao; Guoxiong Luo
Fluorescent dyes alter intracellular targeting and function of cell-penetrating tetrapeptides.
FASEB journal : official publication of the Federation of American Societies for Experimental Biology 2005;19(1):118-20.
2004: Grazyna Weltrowska; Yixin Lu; Carole Lemieux; Nga N Chung; Peter W Schiller
A novel cyclic enkephalin analogue with potent opioid antagonist activity.
Bioorganic & medicinal chemistry letters 2004;14(18):4731-3.
2004: Kesheng Zhao; Guo-Min Zhao; Dunli Wu; Yi Soong; Alex V Birk; Peter W Schiller; Hazel H Szeto
Cell-permeable peptide antioxidants targeted to inner mitochondrial membrane inhibit mitochondrial swelling, oxidative cell death, and reperfusion injury.
The Journal of biological chemistry 2004;279(33):34682-90.
2004: Haibao Wan; Edward S Umstot; Hazel H Szeto; Peter W Schiller; Dominic M Desiderio
Quantitative analysis of [Dmt(1)]DALDA in ovine plasma by capillary liquid chromatography-nanospray ion-trap mass spectrometry.
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 2004;803(1):83-90.
2004: Grazyna Weltrowska; Carole Lemieux; Nga N Chung; Peter W Schiller
A chimeric opioid peptide with mixed mu agonist/delta antagonist properties.
The journal of peptide research : official journal of the American Peptide Society 2004;63(2):63-8.
2004: Irena Berezowska; Carole Lemieux; Nga N Chung; Bogumil Zelent; Peter W Schiller
Dansylated analogues of the opioid peptide [Dmt1]DALDA: in vitro activity profiles and fluorescence parameters.
Acta biochimica Polonica 2004;51(1):107-13.
2003: Guo-Min Zhao; Xuanxuan Qian; Peter W Schiller; Hazel H Szeto
Comparison of [Dmt1]DALDA and DAMGO in binding and G protein activation at mu, delta, and kappa opioid receptors.
The Journal of pharmacology and experimental therapeutics 2003;307(3):947-54.
2003: Irena Berezowska; Nga N Chung; Carole Lemieux; Bogumil Zelent; Hazel H Szeto; Peter W Schiller
Highly potent fluorescent analogues of the opioid peptide [Dmt1] DALDA.
Peptides 2003;24(8):1195-200.
2003: Claire L Neilan; Adam J Janvey; Elizabeth A Bolan; Irena Berezowska; Thi M-D Nguyen; Peter W Schiller; Gavril W Pasternak
Characterization of the binding of [3H][Dmt1]H-Dmt-D-Arg-Phe-Lys-NH2, a highly potent opioid peptide.
The Journal of pharmacology and experimental therapeutics 2003;306(2):430-6.
2003: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Yixin Lu
Conversion of delta-, kappa- and mu-receptor selective opioid peptide agonists into delta-, kappa- and mu-selective antagonists.
Life sciences 2003;73(6):691-8.
2003: Claire L Neilan; Michael A King; Grace Rossi; Micheal Ansonoff; John E Pintar; Peter W Schiller; Gavril W Pasternak
Differential sensitivities of mouse strains to morphine and [Dmt1]DALDA analgesia.
Brain research 2003;974(1-2):254-7.
2003: Kesheng Zhao; Guoxiong Luo; Guo-Min Zhao; Peter W Schiller; Hazel H Szeto
Transcellular transport of a highly polar 3+ net charge opioid tetrapeptide.
The Journal of pharmacology and experimental therapeutics 2003;304(1):425-32.
2002: Brian C Wilkes; Laurent Masaro; Peter W Schiller; Katharine A Carpenter
Angiotensin II vs its type I antagonists: conformational requirements for receptor binding assessed from NMR spectroscopic and receptor docking experiments.
Journal of medicinal chemistry 2002;45(20):4410-8.
2002: Guo-Min Zhao; Dunli Wu; Yi Soong; Megumi Shimoyama; Irena Berezowska; Peter W Schiller; Hazel H Szeto
Profound spinal tolerance after repeated exposure to a highly selective mu-opioid peptide agonist: role of delta-opioid receptors.
The Journal of pharmacology and experimental therapeutics 2002;302(1):188-96.
2001: Yixin Lu; Thi M-D Nguyen; Grazyna Weltrowska; Irena Berezowska; Carole Lemieux; Nga N Chung; Peter W Schiller
[2',6'-Dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: potent and selective kappa opioid antagonists.
Journal of medicinal chemistry 2001;44(19):3048-53.
2001: Hazel H Szeto; J L Lovelace; G Fridland; Y Soong; J Fasolo; D Wu; Dominic M Desiderio; Peter W Schiller
In vivo pharmacokinetics of selective mu-opioid peptide agonists.
The Journal of pharmacology and experimental therapeutics 2001;298(1):57-61.
2001: Claire L Neilan; Thi M-D Nguyen; Peter W Schiller; Gavril W Pasternak
Pharmacological characterization of the dermorphin analog [Dmt(1)]DALDA, a highly potent and selective mu-opioid peptide.
European journal of pharmacology 2001;419(1):15-23.
2001: Yixin Lu; Grazyna Weltrowska; Carole Lemieux; Nga N Chung; Peter W Schiller
Stereospecific synthesis of (2S)-2-methyl-3-(2',6'-dimethyl-4'-hydroxyphenyl)-propionic acid (Mdp) and its incorporation into an opioid peptide.
Bioorganic & medicinal chemistry letters 2001;11(3):323-5.
2000: Peter W Schiller; Thi M-D Nguyen; Irena Berezowska; S Dupuis; Grazyna Weltrowska; Nga N Chung; Carole Lemieux
Synthesis and in vitro opioid activity profiles of DALDA analogues.
European journal of medicinal chemistry 2000;35(10):895-901.
2000: Dominic M Desiderio; U Wirth; J L Lovelace; G Fridland; Edward S Umstot; T M Nguyen; Peter W Schiller; H S Szeto; J F Clapp
Matrix-assisted laser desorption/ionization mass spectrometric quantification of the mu opioid receptor agonist DAMGO in ovine plasma.
Journal of mass spectrometry : JMS 2000;35(6):725-33.
2000: Hiroshi Ueda; M Inoue; Grazyna Weltrowska; Peter W Schiller
An enzymatically stable kyotorphin analog induces pain in subattomol doses.
Peptides 2000;21(5):717-22.
2000: Peter W Schiller; Irena Berezowska; Thi M-D Nguyen; Ralf Schmidt; Carole Lemieux; Nga N Chung; M L Falcone-Hindley; W Yao; J Liu; S Iwama; A B Smith; Ralph Hirschmann
Novel ligands lacking a positive charge for the delta- and mu-opioid receptors.
Journal of medicinal chemistry 2000;43(4):551-9.
1999: Peter W Schiller; Marian E Fundytus; L Merovitz; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Terence J Coderre
The opioid mu agonist/delta antagonist DIPP-NH(2)[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats.
Journal of medicinal chemistry 1999;42(18):3520-6.
1999: Peter W Schiller; Grazyna Weltrowska; Irena Berezowska; Thi M-D Nguyen; Brian C Wilkes; Carole Lemieux; Nga N Chung
The TIPP opioid peptide family: development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists.
Biopolymers 1999;51(6):411-25.
1999: Peter W Schiller; Grazyna Weltrowska; Ralf Schmidt; Irena Berezowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; Katharine A Carpenter; Brian C Wilkes
Subtleties of structure-agonist versus antagonist relationships of opioid peptides and peptidomimetics.
Journal of receptor and signal transduction research 1999;19(1-4):573-88.
1998: Katharine A Carpenter; Peter W Schiller
Aggregation behaviour and Zn2+ binding properties of secretin.
Biochemistry 1998;37(48):16967-74.
1998: Brian C Wilkes; Thi M-D Nguyen; Grazyna Weltrowska; Katharine A Carpenter; Carole Lemieux; Nga N Chung; Peter W Schiller
The receptor-bound conformation of H-Tyr-Tic-(Phe-Phe)-OH-related delta-opioid antagonists contains all trans peptide bonds.
The journal of peptide research : official journal of the American Peptide Society 1998;51(5):386-94.
1998: Katharine A Carpenter; Brian C Wilkes; Peter W Schiller
The octapeptide angiotensin II adopts a well-defined structure in a phospholipid environment.
European journal of biochemistry / FEBS 1998;251(1-2):448-53.
1998: Hazel H Szeto; James F Clapp; Dominic M Desiderio; Peter W Schiller; O O Grigoriants; YI Soong; D Wu; N Olariu; JL Tseng; RR Becklin
In vivo disposition of dermorphin analog (DALDA) in nonpregnant and pregnant sheep.
The Journal of pharmacology and experimental therapeutics 1998;284(1):61-5.
1997: Ralf Schmidt; D Menard; C Mrestani-Klaus; Nga N Chung; Carole Lemieux; Peter W Schiller
Structural modifications of the N-terminal tetrapeptide segment of [D-Ala2]deltorphin I: effects on opioid receptor affinities and activities in vitro and on antinociceptive potency.
Peptides 1997;18(10):1615-21.
1997: Katharine A Carpenter; Brian C Wilkes; André De Léan; Alain Fournier; Peter W Schiller
Hydrophobic forces are responsible for the folding of a highly potent natriuretic peptide analogue at a membrane mimetic surface: an NMR study.
Biopolymers 1997;42(1):37-48.
1996: R Schmidt; Brian C Wilkes; Nga N Chung; Carole Lemieux; Peter W Schiller
Effect of aromatic amino acid substitutions in the 3-position of cyclic beta-casomorphin analogues on mu-opioid agonist/delta-opioid antagonist properties.
International journal of peptide and protein research 1996;48(5):411-9.
1996: Katharine A Carpenter; Brian C Wilkes; Grazyna Weltrowska; Peter W Schiller
Role of hydrophobic substituents in the interaction of opioid Tyr-Tic dipeptide analogs with dodecylphosphocholine micelles. Molecular partitioning in model membrane systems.
European journal of biochemistry / FEBS 1996;241(3):756-64.
1996: Katharine A Carpenter; Peter W Schiller; R Schmidt; Brian C Wilkes
Distinct conformational preferences of three cyclic beta-casomorphin-5 analogs determined using NMR spectroscopy and theoretical analysis.
International journal of peptide and protein research 1996;48(1):102-11.
1996: Carmen Mrestani-Klaus; Wolfgang Brandt; R Schmidt; Klaus Neubert; Peter W Schiller
Proton NMR conformational analysis of cyclic beta-casomorphin analogues of the type Tyr-cyclo[N omega-D-Orn-Xaa-Yaa-Gly-].
Archiv der Pharmazie 1996;329(3):133-42.
1995: Katharine A Carpenter; Brian C Wilkes; Peter W Schiller
Influence of sample pH on the conformational backbone dynamics of a pseudotripeptide (H-Tyr-Tic psi [CH2-NH]Phe-OH) incorporating a reduced peptide bond: an NMR investigation.
Biopolymers 1995;36(6):735-49.
1995: Marian E Fundytus; Peter W Schiller; M Shapiro; Grazyna Weltrowska; Terence J Coderre
Attenuation of morphine tolerance and dependence with the highly selective delta-opioid receptor antagonist TIPP[psi].
European journal of pharmacology 1995;286(1):105-8.
1995: R Schmidt; A Kálmán; Nga N Chung; Carole Lemieux; C Horváth; Peter W Schiller
Structure-activity relationships of dermorphin analogues containing N-substituted amino acids in the 2-position of the peptide sequence.
International journal of peptide and protein research 1995;46(1):47-55.
1995: Colette T Dooley; R A Kaplan; Nga N Chung; Peter W Schiller; Jean M Bidlack; Richard A Houghten
Six highly active mu-selective opioid peptides identified from two synthetic combinatorial libraries.
Peptide research 1995;8(3):124-37.
1995: Brian C Wilkes; Peter W Schiller
Comparative analysis of various proposed models of the receptor-bound conformation of H-Tyr-Tic-Phe-OH related delta-opioid antagonists.
Biopolymers 1995;37(6):391-400.
1994: Colette T Dooley; Nga N Chung; Brian C Wilkes; Peter W Schiller; Jean M Bidlack; Gavril W Pasternak; Richard A Houghten
An all D-amino acid opioid peptide with central analgesic activity from a combinatorial library.
Science (New York, N.Y.) 1994;266(5193):2019-22.
1994: Brian C Wilkes; Peter W Schiller
Theoretical conformational analysis of the opioid delta antagonist H-Tyr-Tic-Phe-OH and the mu agonist H-Tyr-D-Tic-Phe-NH2.
Biopolymers 1994;34(9):1213-9.
1994: R Schmidt; D Vogel; Carmen Mrestani-Klaus; Wolfgang Brandt; Klaus Neubert; Nga N Chung; Carole Lemieux; Peter W Schiller
Cyclic beta-casomorphin analogues with mixed mu agonist/delta antagonist properties: synthesis, pharmacological characterization, and conformational aspects.
Journal of medicinal chemistry 1994;37(8):1136-44.
1993: Colette T Dooley; Nga N Chung; Peter W Schiller; Richard A Houghten
Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries.
Proceedings of the National Academy of Sciences of the United States of America 1993;90(22):10811-5.
1993: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Brian C Wilkes; Nga N Chung; Carole Lemieux
TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity.
Journal of medicinal chemistry 1993;36(21):3182-7.
1993: B J Marsden; Thi M-D Nguyen; Peter W Schiller
Spontaneous degradation via diketopiperazine formation of peptides containing a tetrahydroisoquinoline-3-carboxylic acid residue in the 2-position of the peptide sequence.
International journal of peptide and protein research 1993;41(3):313-6.
1993: Peter W Schiller; Thi M-D Nguyen; Grazyna Weltrowska; Nga N Chung; Carole Lemieux; B J Marsden; Brian C Wilkes
The use of conformational restriction and molecular modeling techniques in the development of receptor-specific opioid peptide agonists and antagonists.
NIDA research monograph 1993;134():238-52.
1992: Peter W Schiller; Thi M-D Nguyen; Grazyna Weltrowska; Brian C Wilkes; B J Marsden; Carole Lemieux; Nga N Chung
Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists.
Proceedings of the National Academy of Sciences of the United States of America 1992;89(24):11871-5.
1992: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Brian C Wilkes; Nga N Chung; Carole Lemieux
Conformationally restricted deltorphin analogues.
Journal of medicinal chemistry 1992;35(21):3956-61.
1992: Brian C Wilkes; Peter W Schiller
Molecular dynamics simulations of opioid peptide analogs containing multiple conformational restrictions.
International journal of peptide and protein research 1992;40(3-4):249-54.
1991: Peter W Schiller; Grazyna Weltrowska; Thi M-D Nguyen; Carole Lemieux; Nga N Chung; B J Marsden; Brian C Wilkes
Conformational restriction of the phenylalanine residue in a cyclic opioid peptide analogue: effects on receptor selectivity and stereospecificity.
Journal of medicinal chemistry 1991;34(10):3125-32.
1991: Brian C Wilkes; Peter W Schiller
Comparative conformational analysis of [D-Pen2,D-Pen5]enkephalin (DPDPE): a molecular mechanics study.
Journal of computer-aided molecular design 1991;5(4):293-302.
1991: Peter W Schiller
Development of receptor-specific opioid peptide analogues.
Progress in medicinal chemistry 1991;28():301-40.
1991: Peter W Schiller
Development of opioid peptide analogs as pharmacologic tools and as potential drugs: current status and future directions.
NIDA research monograph 1991;112():180-97.
1990: Brian C Wilkes; Peter W Schiller
Conformation-activity relationships of cyclic dermorphin analogues.
Biopolymers 1990;29(1):89-95.
1990: Peter W Schiller; Thi M-D Nguyen; Nga N Chung; G Dionne; R Martel
Peripheral antinociceptive effect of an extremely mu-selective polar dermorphin analog (DALDA).
Progress in clinical and biological research 1990;328():53-6.
1989: Peter W Schiller; Thi M-D Nguyen; Nga N Chung; Carole Lemieux
Dermorphin analogues carrying an increased positive net charge in their "message" domain display extremely high mu opioid receptor selectivity.
Journal of medicinal chemistry 1989;32(3):698-703.
1988: Peter W Schiller
Role of the conformational element in peptide-receptor interactions. Studies with cyclic opioid peptide analogs.
Biophysical chemistry 1988;31(1-2):63-9.
1988: Peter W Schiller; Brian C Wilkes
Conformational analysis of cyclic opioid peptide analogs.
NIDA research monograph 1988;87():60-73.
1987: Peter W Schiller; Thi M-D Nguyen; L A Maziak; Brian C Wilkes; Carole Lemieux
Structure-activity relationships of cyclic opioid peptide analogues containing a phenylalanine residue in the 3-position.
Journal of medicinal chemistry 1987;30(11):2094-9.
1987: Peter W Schiller; L A Maziak; Thi M-D Nguyen; J Godin; R Garcia; A DeLéan; M Cantin
Superactive analogs of the atrial natriuretic peptide (ANP).
Biochemical and biophysical research communications 1987;143(2):499-505.
1986: Peter W Schiller; L A Maziak; Carole Lemieux; Thi M-D Nguyen
Side chain to side chain cyclization of an enkephalin analog results in loss of opioid receptor selectivity.
International journal of peptide and protein research 1986;28(5):493-7.
1986: Peter W Schiller; F Bellini; G Dionne; L A Maziak; R Garcia; A DeLéan; M Cantin
Synthesis and activity profiles of atrial natriuretic peptide (ANP) analogs with reduced ring size.
Biochemical and biophysical research communications 1986;138(2):880-6.
1985: Peter W Schiller; Thi M-D Nguyen; Carole Lemieux; L A Maziak
Synthesis and activity profiles of novel cyclic opioid peptide monomers and dimers.
Journal of medicinal chemistry 1985;28(12):1766-71.
1985: Peter W Schiller; Thi M-D Nguyen; Carole Lemieux; L A Maziak
A novel side-chain-linked antiparallel cyclic dimer of enkephalin.
FEBS letters 1985;191(2):231-4.
1985: Peter W Schiller; L Maziak; Thi M-D Nguyen; J Godin; R Garcia; A De Léan; M Cantin
Synthesis and biological activity of a linear fragment of the atrial natriuretic factor (ANF).
Biochemical and biophysical research communications 1985;131(3):1056-62.
1985: Peter W Schiller; Thi M-D Nguyen; L Maziak; Carole Lemieux
A novel cyclic opioid peptide analog showing high preference for mu-receptors.
Biochemical and biophysical research communications 1985;127(2):558-64.