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Fabrizio Bordi

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Caterina Carmi; Andrea Cavazzoni; Gabriele Costantino; Elena Galvani; Alessio Lodola; Stefania Aiello; Roberta R Alfieri; Andrea Ardizzoni; Fabrizio Bordi; Pier Giorgio Petronini; Silvia Rivara; Simonetta Russo; Federica Vacondio; Marco Mor
Irreversible inhibition of epidermal growth factor receptor activity by 3-aminopropanamides.
Fabrizio Bordi; Caterina Carmi; Elisa Dallaturca; Lisa Flammini; Alessio Lodola; Vigilio Ballabeni; Elisabetta Barocelli; Simona Bertoni; Daniele Pala; Silvia Rivara; Federica Vacondio; sha mor
Dibasic biphenyl H3 receptor antagonists: Steric tolerance for a lipophilic side chain.
Federica Vacondio; Giovanni Morini; Claudia Silva; Elisabetta Barocelli; Fabrizio Bordi; Lisa Flammini; sha mor
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H3-receptor antagonist UPR1056 in rat plasma.

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All Publications

2012: Caterina Carmi; Andrea Cavazzoni; Gabriele Costantino; Elena Galvani; Alessio Lodola; Stefania Aiello; Roberta R Alfieri; Andrea Ardizzoni; Fabrizio Bordi; Pier Giorgio Petronini; Silvia Rivara; Simonetta Russo; Federica Vacondio; Marco Mor
Irreversible inhibition of epidermal growth factor receptor activity by 3-aminopropanamides.
Journal of medicinal chemistry 2012;55(5):2251-64.
2012: Fabrizio Bordi; Caterina Carmi; Elisa Dallaturca; Lisa Flammini; Alessio Lodola; Vigilio Ballabeni; Elisabetta Barocelli; Simona Bertoni; Daniele Pala; Silvia Rivara; Federica Vacondio; sha mor
Dibasic biphenyl H3 receptor antagonists: Steric tolerance for a lipophilic side chain.
European journal of medicinal chemistry 2012;48():214-30.
2011: Federica Vacondio; Giovanni Morini; Claudia Silva; Elisabetta Barocelli; Fabrizio Bordi; Lisa Flammini; sha mor
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H3-receptor antagonist UPR1056 in rat plasma.
Journal of separation science 2011;34(14):1656-63.
2010: Caterina Carmi; Andrea Cavazzoni; Stefano Vezzosi; Fabrizio Bordi; Federica Vacondio; Claudia Silva; Silvia Rivara; Alessio Lodola; Roberta R Alfieri; Silvia La Monica; Maricla Galetti; Andrea Ardizzoni; Pier Giorgio Petronini; sha mor
Novel irreversible epidermal growth factor receptor inhibitors by chemical modulation of the cysteine-trap portion.
Journal of medicinal chemistry 2010;53(5):2038-50.
2009: Valentina Zuliani; Caterina Carmi; Mirko Rivara; Marco Fantini; Alessio Lodola; Federica Vacondio; Fabrizio Bordi; Pier Vincenzo Plazzi; Andrea Cavazzoni; Maricla Galetti; Roberta R Alfieri; Pier Giorgio Petronini; sha mor
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line.
European journal of medicinal chemistry 2009;44(9):3471-9.
2008: Giovanni Morini; Mara Comini; Mirko Rivara; Silvia Rivara; Fabrizio Bordi; Pier Vincenzo Plazzi; Lisa Flammini; Francesca Saccani; Simona Bertoni; Vigilio Ballabeni; Elisabetta Barocelli; sha mor
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity.
Bioorganic & medicinal chemistry 2008;16(23):9911-24.
2008: Andrea Cavazzoni; Roberta R Alfieri; Caterina Carmi; Valentina Zuliani; Maricla Galetti; Claudia Fumarola; Raffaele Frazzi; Mara A Bonelli; Fabrizio Bordi; Alessio Lodola; sha mor; Pier Giorgio Petronini
Dual mechanisms of action of the 5-benzylidene-hydantoin UPR1024 on lung cancer cell lines.
Molecular cancer therapeutics 2008;7(2):361-70.
2008: Federica Vacondio; Claudia Silva; Alessandro Fioni; sha mor; Mirko Rivara; Fabrizio Bordi; Lisa Flammini; Vigilio Ballabeni; Elisabetta Barocelli
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H3 antagonist ROS203 in rat plasma.
Journal of pharmaceutical and biomedical analysis 2008;46(1):200-5.
2008: Mirko Rivara; Federica Vacondio; Claudia Silva; Valentina Zuliani; Marco Fantini; Fabrizio Bordi; Pier Vincenzo Plazzi; Simona Bertoni; Vigilio Ballabeni; Lisa Flammini; Elisabetta Barocelli; sha mor
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
Chemistry & biodiversity 2008;5(1):140-52.
2006: Caterina Carmi; Andrea Cavazzoni; Valentina Zuliani; Alessio Lodola; Fabrizio Bordi; Pier Vincenzo Plazzi; Roberta R Alfieri; Pier Giorgio Petronini; sha mor
5-benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity.
Bioorganic & medicinal chemistry letters 2006;16(15):4021-5.
2006: Giovanni Morini; Mara Comini; Mirko Rivara; Silvia Rivara; Simone Lorenzi; Fabrizio Bordi; sha mor; Lisa Flammini; Simona Bertoni; Vigilio Ballabeni; Elisabetta Barocelli; Pier Vincenzo Plazzi
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid biphenyl scaffold.
Bioorganic & medicinal chemistry letters 2006;16(15):4063-7.
2006: Mirko Rivara; Valentina Zuliani; Giuseppe Cocconcelli; Giovanni Morini; Mara Comini; Silvia Rivara; sha mor; Fabrizio Bordi; Elisabetta Barocelli; Vigilio Ballabeni; Simona Bertoni; Pier Vincenzo Plazzi
Synthesis and biological evaluation of new non-imidazole H3-receptor antagonists of the 2-aminobenzimidazole series.
Bioorganic & medicinal chemistry 2006;14(5):1413-24.
2005: sha mor; Silvia Rivara; Alessio Lodola; Simone Lorenzi; Fabrizio Bordi; Pier Vincenzo Plazzi; Gilberto Spadoni; Annalida Bedini; Andrea Duranti; Andrea Tontini; Giorgio Tarzia
Application of 3D-QSAR in the rational design of receptor ligands and enzyme inhibitors.
Chemistry & biodiversity 2005;2(11):1438-51.
2005: Simone Lorenzi; sha mor; Fabrizio Bordi; Silvia Rivara; Mirko Rivara; Giovanni Morini; Simona Bertoni; Vigilio Ballabeni; Elisabetta Barocelli; Pier Vincenzo Plazzi
Validation of a histamine H3 receptor model through structure-activity relationships for classical H3 antagonists.
Bioorganic & medicinal chemistry 2005;13(19):5647-57.
2004: Federica Vacondio; sha mor; Claudia Silva; Valentina Zuliani; Mirko Rivara; Silvia Rivara; Fabrizio Bordi; Pier Vincenzo Plazzi; Francesca Magnanini; Simona Bertoni; Vigilio Ballabeni; Elisabetta Barocelli; Pierre-Alain Carrupt; Bernard Testa
Imidazole H3-antagonists: relationship between structure and ex vivo binding to rat brain H3-receptors.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 2004;23(1):89-98.
2004: Valeria Lucini; Marilou Pannacci; Francesco Scaglione; Franco Fraschini; Silvia Rivara; sha mor; Fabrizio Bordi; Pier Vincenzo Plazzi; Gilberto Spadoni; Annalida Bedini; Giovanni Piersanti; Giuseppe Diamantini; Giorgio Tarzia
Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity.
Journal of medicinal chemistry 2004;47(17):4202-12.
2004: sha mor; Fabrizio Bordi; Claudia Silva; Silvia Rivara; Valentina Zuliani; Federica Vacondio; Mirko Rivara; Elisabetta Barocelli; Simona Bertoni; Vigilio Ballabeni; Francesca Magnanini; Mariannina Impicciatore; Pier Vincenzo Plazzi
Synthesis, biological activity, QSAR and QSPR study of 2-aminobenzimidazole derivatives as potent H3-antagonists.
Bioorganic & medicinal chemistry 2004;12(4):663-74.
2003: Valentina Zuliani; Fabrizio Bordi; Mirko Rivara; Claudia Silva; Federica Vacondio; Giovanni Morini; Silvia Rivara; Elisabetta Barocelli; Vigilio Ballabeni; Simona Bertoni; Francesca Magnanini; Pier Vincenzo Plazzi
The role of HB-donor groups in the heterocyclic polar fragment of H3-antagonists. I. Synthesis and biological assays.
Farmaco (Società chimica italiana : 1989) 2003;58(9):891-9.
2003: Silvia Rivara; sha mor; Fabrizio Bordi; Claudia Silva; Valentina Zuliani; Federica Vacondio; Giovanni Morini; Pier Vincenzo Plazzi; Pierre-Alain Carrupt; Bernard Testa
Synthesis and three-dimensional quantitative structure-activity relationship analysis of H3 receptor antagonists containing a neutral heterocyclic polar group.
Drug design and discovery 2003;18(2-3):65-79.
2000: Claudia Silva; Pier Vincenzo Plazzi; Fabrizio Bordi; Silvia Rivara; Federica Vacondio; Valentina Zuliani; A Caretta; sha mor
Structure-property relationships on histamine H3-antagonists: binding of phenyl-substituted alkylthioimidazole derivatives to rat plasma proteins.
Farmaco (Società chimica italiana : 1989) 2000;55(4):239-45.
2000: Elisabetta Barocelli; Vigilio Ballabeni; M Chiavarini; Simona Bertoni; sha mor; Pier Vincenzo Plazzi; Fabrizio Bordi; Mariannina Impicciatore
Pharmacological characterization of H3 receptor antagonists with imidazole, thioimidazole and thioimidazoline polar groups in the side chain.
Inflammation research : official journal of the European Histamine Research Society ... [et al.] 2000;49 Suppl 1():S62-3.
2000: sha mor; Fabrizio Bordi; Claudia Silva; Silvia Rivara; Valentina Zuliani; Federica Vacondio; Giovanni Morini; Elisabetta Barocelli; Vigilio Ballabeni; Mariannina Impicciatore; Pier Vincenzo Plazzi
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups.
Farmaco (Società chimica italiana : 1989) 2000;55(1):27-34.
1998: sha mor; Silvia Rivara; Claudia Silva; Fabrizio Bordi; Pier Vincenzo Plazzi; Gilberto Spadoni; Giuseppe Diamantini; C Balsamini; Giorgio Tarzia; Franco Fraschini; Valeria Lucini; R Nonno; BM Stankov
Melatonin receptor ligands: synthesis of new melatonin derivatives and comprehensive comparative molecular field analysis (CoMFA) study.
Journal of medicinal chemistry 1998;41(20):3831-44.
1997: sha mor; Fabrizio Bordi; Claudia Silva; Silvia Rivara; P Crivori; Pier Vincenzo Plazzi; Vigilio Ballabeni; A Caretta; Elisabetta Barocelli; Mariannina Impicciatore; Pierre-Alain Carrupt; Bernard Testa
H3-receptor antagonists: synthesis and structure-activity relationships of para- and meta-substituted 4(5)-phenyl-2-[[2-[4(5)-imidazolyl]ethyl]thio]imidazoles.
Journal of medicinal chemistry 1997;40(16):2571-8.
1997: Pier Vincenzo Plazzi; Fabrizio Bordi; sha mor; P Cozzini; P Domiano
H3-receptor antagonists: conformational analysis of thioperamide and x-ray crystal structure of the analog N-cyclohexyl-4-methylpiperidine-1-carbothioamide.
Farmaco (Società chimica italiana : 1989) 1997;52(6-7):399-404.
1997: Elisabetta Barocelli; Vigilio Ballabeni; A Caretta; Simona Bertoni; Fabrizio Bordi; Silvia Rivara; Claudia Silva; sha mor; Mariannina Impicciatore
In vitro characterization of potency, affinity and selectivity of H3-antagonists: from thioperamide to thioperamide unrelated imidazole derivatives.
Farmaco (Società chimica italiana : 1989) 1997;52(6-7):463-9.
1997: Claudia Silva; sha mor; Fabrizio Bordi; Silvia Rivara; A Caretta; Vigilio Ballabeni; Elisabetta Barocelli; Pier Vincenzo Plazzi
Plasma concentration and brain penetration of the H3-receptor antagonist thioperamide in rats.
Farmaco (Società chimica italiana : 1989) 1997;52(6-7):457-62.
1997: Pier Vincenzo Plazzi; sha mor; Fabrizio Bordi; Claudia Silva; Silvia Rivara; A Caretta; Vigilio Ballabeni; Mariannina Impicciatore; T Vitali
Ligands of the histamine H3-receptor: new potent antagonists of the 2-thioimidazole type.
Farmaco (Società chimica italiana : 1989) 1997;52(5):295-302.
1996: Pier Vincenzo Plazzi; sha mor; Claudia Silva; Fabrizio Bordi; Giovanni Morini; M Crivori; A Caretta
Rat protein binding and cerebral phospholipid affinity of the H3-receptor antagonist thioperamide.
The Journal of pharmacy and pharmacology 1996;48(7):712-7.
1996: sha mor; F Zani; P Mazza; Claudia Silva; Fabrizio Bordi; Giovanni Morini; Pier Vincenzo Plazzi
Biological studies on 1,2-benzisothiazole derivatives V. Antimicrobial properties of N-alkanoic, N-arylalkanoic and N-aryloxyalkanoic derivatives of 1,2-benzisothiazolin-3-one: QSAR study and genotoxicity evaluation.
Farmaco (Società chimica italiana : 1989) 1996;51(7):493-501.
1994: Fabrizio Bordi; sha mor; Giovanni Morini; Pier Vincenzo Plazzi; Claudia Silva; T Vitali; A Caretta
QSAR study on H3-receptor affinity of benzothiazole derivatives of thioperamide.
Farmaco (Società chimica italiana : 1989) 1994;49(3):153-66.
1993: Elisabetta Barocelli; Vigilio Ballabeni; A Caretta; Fabrizio Bordi; Claudia Silva; Giovanni Morini; Mariannina Impicciatore
Pharmacological profile of new thioperamide derivatives at histamine peripheral H1-, H2-, H3-receptors in guinea-pig.
Agents and actions 1993;38(3-4):158-64.
1993: Elisabetta Barocelli; M Chiavarini; Vigilio Ballabeni; Fabrizio Bordi; Mariannina Impicciatore
Interaction of selective compounds with muscarinic receptors at dispersed intestinal smooth muscle cells.
British journal of pharmacology 1993;108(2):393-7.
1992: Fabrizio Bordi; sha mor; Pier Vincenzo Plazzi; Claudia Silva; Giovanni Morini; A Caretta; Elisabetta Barocelli; Mariannina Impicciatore
Synthesis and binding assays of H3-receptor ligands.
Farmaco (Società chimica italiana : 1989) 1992;47(11):1343-65.
1992: Fabrizio Bordi; sha mor; Pier Vincenzo Plazzi; Claudia Silva; A Caretta; Giovanni Morini
HPLC detection of thioperamide from biological samples and its determination in rat blood and brain after systemic administration.
Farmaco (Società chimica italiana : 1989) 1992;47(7-8):1095-103.
1992: Vigilio Ballabeni; Elisabetta Barocelli; M Chiavarini; Fabrizio Bordi; Mariannina Impicciatore
Neuronal and myogenic muscarinic effects of McN-A-343 on guinea pig longitudinal smooth muscle-myenteric plexus.
Bollettino della Società italiana di biologia sperimentale 1992;68(7):437-44.
1992: Fabrizio Bordi; sha mor; Pier Vincenzo Plazzi; Claudia Silva; Giovanni Morini; Mariannina Impicciatore; Elisabetta Barocelli; M Chiavarini
4-(1,2-Benzisothiazol-3-yl)alkanoic and phenylalkanoic acids: synthesis and anti-inflammatory, analgesic and antipyretic activities.
Farmaco (Società chimica italiana : 1989) 1992;47(5):551-65.
1989: Pier Vincenzo Plazzi; Fabrizio Bordi; Claudia Silva; Giovanni Morini; P L Catellani; G Vaona; Mariannina Impicciatore
H2-antagonists: synthesis and activity of 2-amino-5-thiazolyl derivatives.
Farmaco (Società chimica italiana : 1989) 1989;44(11):1011-30.
1989: Fabrizio Bordi; P L Catellani; Giovanni Morini; Pier Vincenzo Plazzi; Claudia Silva; Elisabetta Barocelli; M Chiavarini
[4-(3-Oxo-1,2-benzisothiazolin-2-yl)alkanoic, phenyl and phenoxyalkanoic acids: synthesis and anti-inflammatory, analgesic, and antipyretic properties].
Farmaco (Società chimica italiana : 1989) 1989;44(9):795-807.
1989: M Chiavarini; Giovanni Morini; Elisabetta Barocelli; Fabrizio Bordi; Pier Vincenzo Plazzi; T Vitali; Mariannina Impicciatore
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H2-receptor antagonist activity in gastric fistula cat.
Agents and actions 1989;27(1-2):192-4.
1988: M Chiavarini; Giovanni Morini; Elisabetta Barocelli; Mariannina Impicciatore; Fabrizio Bordi
Effects of antimuscarinic agents, H2-blockers and omeprazole on rat chronic gastric ulcer after long- and short-term administration.
Il Farmaco; edizione scientifica 1988;43(5):479-87.
1987: Mariannina Impicciatore; Giovanni Morini; M Chiavarini; Elisabetta Barocelli; Fabrizio Bordi; Pier Vincenzo Plazzi; F Vitali
Are histamine receptors involved in the stimulant activities of thiazolylethylamines supposed as cyclic models of dimaprit?
Agents and actions 1987;20(3-4):262-4.
1986: T Vitali; Mariannina Impicciatore; Pier Vincenzo Plazzi; Fabrizio Bordi; Giovanni Morini
[Thiazolylalkylamines: synthesis of analogs of imidazolylethylamines and their effect on gastric secretion].
Il Farmaco; edizione scientifica 1986;41(6):483-98.
1986: Mariannina Impicciatore; Giovanni Morini; M Chiavarini; Pier Vincenzo Plazzi; Fabrizio Bordi; F Vitali
Pharmacological activities of two new histamine analogs.
Agents and actions 1986;18(1-2):134-6.
1986: Elisabetta Barocelli; Giovanni Morini; Claudia Silva; Fabrizio Bordi; Pier Vincenzo Plazzi; Mariannina Impicciatore
Antipyretic activity of new compounds 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenylalkanoic acids, their esters, amides and 1,1-dioxide derivatives.
Pharmacological research communications 1986;18(2):171-85.
1985: Pier Vincenzo Plazzi; Fabrizio Bordi; Mariannina Impicciatore
[The preparation and histaminergic properties of 2-(2-oxo-4-imidazolin-4-yl)ethylamine].
Il Farmaco; edizione scientifica 1985;40(3):218-20.
1984: Pier Vincenzo Plazzi; Fabrizio Bordi; F Vitali; Claudia Silva; M Chiavarini; Giovanni Morini; Mariannina Impicciatore
[Synthesis and analgesic activity of 4-(3-oxo-1,2-benzoisothiazoline-2-yl)phenylalkanoic derivatives].
Il Farmaco; edizione scientifica 1984;39(9):788-96.
1984: Pier Vincenzo Plazzi; Fabrizio Bordi; Claudia Silva; F Vitali; Mariannina Impicciatore; Giovanni Morini
[3-Benzyl-1,2-benzoisothiazoles: spasmolytic properties of the aminoalkyl derivatives].
Il Farmaco; edizione scientifica 1984;39(8):649-59.
1984: M Chiavarini; Giovanni Morini; Elisabetta Barocelli; Fabrizio Bordi; Pier Vincenzo Plazzi; Mariannina Impicciatore
[Pharmacological actions of alkylaminoalkyl-phenylbenzisothazole compounds on the gastrointestinal tract].
Bollettino della Società italiana di biologia sperimentale 1984;60(4):797-803.
1984: Giovanni Morini; M Chiavarini; Fabrizio Bordi; Pier Vincenzo Plazzi; F Vitali; Mariannina Impicciatore
[Imidazolic H2-agonists: importance of 2-amino substitution for pharmacological activity].
Bollettino della Società italiana di biologia sperimentale 1984;60(4):789-95.
1984: T Vitali; Mariannina Impicciatore; Pier Vincenzo Plazzi; Fabrizio Bordi; M Vitto
[Imidazole H-2 agonists. Synthesis and activity of 2-(2-amino-4-imidazolyl)ethylamine (2-aminohistamine) dihydrochloride].
Il Farmaco; edizione scientifica 1984;39(1):70-80.
1983: Giovanni Morini; Mariannina Impicciatore; Fabrizio Bordi; Pier Vincenzo Plazzi; M Vitto
[Synthesis of new derivatives of 3-benzyl-1,2-benzisothiazole and a study of analgesic activity in mice].
Il Farmaco; edizione scientifica 1983;38(10):794-800.
1983: Mariannina Impicciatore; Giovanni Morini; M Chiavarini; Fabrizio Bordi
A possible physiological role of histamine H2-receptors in rat mesenteric circulation.
European journal of pharmacology 1983;90(2-3):231-5.
1981: Pier Vincenzo Plazzi; Fabrizio Bordi; M Vitto; Mariannina Impicciatore
[Synthesis and biological activity of substituted 2-(4-imidazolyl)ethylamines].
Il Farmaco; edizione scientifica 1981;36(11):931-31.
1980: Giovanni Morini; Pier Vincenzo Plazzi; Fabrizio Bordi; Mariannina Impicciatore
[Study of substances analagous to dimaprit affecting gastric secretion in vitro].
Bollettino della Società italiana di biologia sperimentale 1980;56(1):88-94.