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Simone Carradori

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TOP 3
Y Ragazzoni; Daniela Secci; Antonio Candiloro; Simone Carradori; Maria Condello; T De Luca; Donatella Del Bufalo; Marianna Desideri; Chiara Gabellini; Stefania Meschini; R Nescatelli; Daniela Trisciuoglio
The thiazole derivative CPTH6 impairs autophagy.
Simone Carradori
Selective carbonic anhydrase IX inhibitors based on coumarin scaffold as promising antimetastatic agents: WO2012070024.
Simone Carradori; Melissa D'Ascenzio; Celeste De Monte; Daniela Secci; Matilde Yáñez
Synthesis and selective human monoamine oxidase B inhibition of heterocyclic hybrids based on hydrazine and thiazole scaffolds.

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All Publications

2013: Y Ragazzoni; Daniela Secci; Antonio Candiloro; Simone Carradori; Maria Condello; T De Luca; Donatella Del Bufalo; Marianna Desideri; Chiara Gabellini; Stefania Meschini; R Nescatelli; Daniela Trisciuoglio
The thiazole derivative CPTH6 impairs autophagy.
Cell death & disease 2013;4():e524.
2013: Simone Carradori
Selective carbonic anhydrase IX inhibitors based on coumarin scaffold as promising antimetastatic agents: WO2012070024.
Expert opinion on therapeutic patents 2013;23(6):751-6.
2013: Simone Carradori; Melissa D'Ascenzio; Celeste De Monte; Daniela Secci; Matilde Yáñez
Synthesis and selective human monoamine oxidase B inhibition of heterocyclic hybrids based on hydrazine and thiazole scaffolds.
Archiv der Pharmazie 2013;346(1):17-22.
2012: Simone Carradori; Roberto Cirilli; Simona Dei Cicchi; Rosella Ferretti; Sergio Menta; Marco Pierini; Daniela Secci
3-methylcyclohexanone thiosemicarbazone: determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes.
Journal of chromatography. A 2012;1269():168-77.
2012: Daniela Secci; Adriana Bolasco; Simone Carradori; Melissa D'Ascenzio; Riccardo Nescatelli; Matilde Yáñez
Recent advances in the development of selective human MAO-B inhibitors: (hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines.
European journal of medicinal chemistry 2012;58():405-17.
2012: Simone Carradori; Celeste De Monte; Daniela Secci; Adriana Bolasco; Matilde Yáñez
Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives.
Archiv der Pharmazie 2012;345(12):973-9.
2012: Simone Carradori; Paola Chimenti; Adriana Bolasco; Daniela Secci; Melissa D'Ascenzio
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential.
Expert opinion on therapeutic patents 2012;22(7):759-801.
2012: Daniela Secci; Bruna Bizzarri; Adriana Bolasco; Simone Carradori; Melissa D'Ascenzio; Emanuela Mari; Lucia Polletta; Daniela Rivanera; Alessandra Zicari
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives.
European journal of medicinal chemistry 2012;53():246-53.
2012: Simone Carradori; Cristiano Cristini; Vincenzo Gentile; Caterina Gulia; Daniela Secci; Giovanni Battista Di Pierro
Current and emerging strategies in bladder cancer.
Anti-cancer agents in medicinal chemistry 2012;12(6):589-603.
2012: Daniela Trisciuoglio; Bruna Bizzarri; Adriana Bolasco; Simone Carradori; Chiara Cavaliere; Igea D'Agnano; Marianna Desideri; patrizia filetici; Chiara Gabellini; Giovanna Maresca; Riccardo Nescatelli; Andrea Pelosi; Ylenia Ragazzoni; Lucia Ricci-Vitiani; Maria Giulia Rizzo; Daniela Secci; Donatella Del Bufalo
CPTH6, a thiazole derivative, induces histone hypoacetylation and apoptosis in human leukemia cells.
Clinical cancer research : an official journal of the American Association for Cancer Research 2012;18(2):475-86.
2012: Daniela Secci; Bruna Bizzarri; Adriana Bolasco; Simone Carradori; Melissa D'Ascenzio; Elias Maccioni
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors.
Current topics in medicinal chemistry 2012;12(20):2240-57.
2011: Daniela Secci; Matilde Yáñez; Adriana Bolasco; Simone Carradori; Paola Chimenti; Francesco Ortuso; Stefano Alcaro
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives.
European journal of medicinal chemistry 2011;46(10):4846-52.
2011: Simone Carradori; Daniela Secci; Antonello Mai
Epigenetic modulation of PGC-1α activity by GCN5 inhibitors: WO2010007085.
Expert opinion on therapeutic patents 2011;21(10):1651-6.
2011: Franco Chimenti; Bruna Bizzarri; Adriana Bolasco; Daniela Secci; Paola Chimenti; Arianna Granese; Simone Carradori; Melissa D'Ascenzio; Daniela Lilli; Daniela Rivanera
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents.
European journal of medicinal chemistry 2011;46(1):378-82.
2010: Franco Chimenti; Daniela Secci; Adriana Bolasco; Paola Chimenti; Arianna Granese; Simone Carradori; Matilde Yáñez; Matilde Yañez; M Luisa Sanna; Bruno Gallinella; Roberto Cirilli
Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines.
Journal of medicinal chemistry 2010;53(17):6516-20.
2010: Franco Chimenti; Bruna Bizzarri; Adriana Bolasco; Daniela Secci; Paola Chimenti; Arianna Granese; Simone Carradori; Daniela Rivanera; Alessandra Zicari; M Maddalena Scaltrito; Francesca Sisto
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides.
Bioorganic & medicinal chemistry letters 2010;20(16):4922-6.
2010: Franco Chimenti; Adriana Bolasco; Daniela Secci; Paola Chimenti; Arianna Granese; Simone Carradori; Matilde Yáñez; Matilde Yañez; Francesco Ortuso; Stefano Alcaro
Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors.
Bioorganic & medicinal chemistry 2010;18(15):5715-23.
2010: Franco Chimenti; Daniela Secci; Adriana Bolasco; Paola Chimenti; Arianna Granese; Simone Carradori; Elias Maccioni; M Cristina Cardia; Matilde Yáñez; Matilde Yañez; Stefano Alcaro; Francesco Ortuso; Roberto Cirilli; Rosella Ferretti; Simona Distinto; Johannes Kirchmair; Thierry Langer
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors.
Bioorganic & medicinal chemistry 2010;18(14):5063-70.
2010: Adriana Bolasco; Simone Carradori; Rossella Fioravanti
Focusing on new monoamine oxidase inhibitors.
Expert opinion on therapeutic patents 2010;20(7):909-39.
2010: Franco Chimenti; Simone Carradori; Daniela Secci; Adriana Bolasco; Bruna Bizzarri; Paola Chimenti; Arianna Granese; Matilde Yáñez; Matilde Yañez
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives.
European journal of medicinal chemistry 2010;45(2):800-4.
2009: Franco Chimenti; Bruna Bizzarri; Adriana Bolasco; Daniela Secci; Paola Chimenti; Simone Carradori; Arianna Granese; Daniela Rivanera; Nathan Frishberg; Claudia Bordón; LORRAINE BRANDO
Synthesis and evaluation of 4-acyl-2-thiazolylhydrazone derivatives for anti-Toxoplasma efficacy in vitro.
Journal of medicinal chemistry 2009;52(15):4574-7.
2009: Franco Chimenti; Daniela Secci; Adriana Bolasco; Paola Chimenti; Bruna Bizzarri; Arianna Granese; Simone Carradori; Matilde Yáñez; Matilde Yañez; Francesco Ortuso; Stefano Alcaro
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins.
Journal of medicinal chemistry 2009;52(7):1935-42.
2009: Franco Chimenti; Bruna Bizzarri; Elias Maccioni; Daniela Secci; Adriana Bolasco; Paola Chimenti; Rossella Fioravanti; Arianna Granese; Simone Carradori; Federica Tosi; Paola Ballario; Stefano Vernarecci; patrizia filetici
A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone.
Journal of medicinal chemistry 2009;52(2):530-6.
2008: Franco Chimenti; Elias Maccioni; Daniela Secci; Adriana Bolasco; Paola Chimenti; Arianna Granese; Simone Carradori; Stefano Alcaro; Francesco Ortuso; Matilde Yáñez; Matilde Yañez; Roberto Cirilli; Rosella Ferretti; Francesco La Torre
Synthesis, stereochemical identification, and selective inhibitory activity against human monoamine oxidase-B of 2-methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones.
Journal of medicinal chemistry 2008;51(16):4874-80.
2007: Roberto Cirilli; Rosella Ferretti; Francesco La Torre; Daniela Secci; Adriana Bolasco; Simone Carradori; M Pierini
High-performance liquid chromatographic separation of enantiomers and diastereomers of 2-methylcyclohexanone thiosemicarbazone, and determination of absolute configuration and configurational stability.
Journal of chromatography. A 2007;1172(2):160-9.
2007: Franco Chimenti; Bruna Bizzarri; Elias Maccioni; Daniela Secci; Adriana Bolasco; Rossella Fioravanti; Paola Chimenti; Arianna Granese; Simone Carradori; Daniela Rivanera; Daniela Lilli; Alessandra Zicari; Simona Distinto
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
Bioorganic & medicinal chemistry letters 2007;17(16):4635-40.
2007: Franco Chimenti; Bruna Bizzarri; Adriana Bolasco; Daniela Secci; Paola Chimenti; Simone Carradori; Arianna Granese; Daniela Rivanera; Daniela Lilli; Alessandra Zicari; M Maddalena Scaltrito; Francesca Sisto
A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives.
Bioorganic & medicinal chemistry letters 2007;17(11):3065-71.
2006: Franco Chimenti; Daniela Secci; Adriana Bolasco; Paola Chimenti; Arianna Granese; Simone Carradori; Olivia Befani; Paola Turini; Stefano Alcaro; Francesco Ortuso
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides.
Bioorganic & medicinal chemistry letters 2006;16(15):4135-40.
2006: Franco Chimenti; Bruna Bizzarri; Adriana Bolasco; Daniela Secci; Paola Chimenti; Simone Carradori; Arianna Granese; Daniela Rivanera; Daniela Lilli; M Maddalena Scaltrito; Maria Immacolata Brenciaglia
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides.
European journal of medicinal chemistry 2006;41(2):208-12.