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Susanna Nencetti

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Elisa Nuti; Elisabetta Orlandini; Silvia Salerno; Salvatore Santamaria; Sabrina Taliani; Kazuhiro Yamamoto; Francesca Casalini; Federico Da Settimo; Valeria La Pietra; Luciana Marinelli; Anna Maria Marini; Hideaki Nagase; Susanna Nencetti; Ettore Novellino; Armando Rossello
Arylsulfonamide inhibitors of aggrecanases as potential therapeutic agents for osteoarthritis: synthesis and biological evaluation.
Anna M Marini; Robert McKenna; Susanna Nencetti; Elisa Nuti; Elisabetta Orlandini; Armando Rossello; Silvia Salerno; Andrea Scozzafava; Francesca Simorini; Mayank Aggarwal; Federico Da Settimo; Concettina La Motta; Alfonso Maresca; Sabrina Taliani; Claudiu T Supuran
Tricyclic sulfonamides incorporating benzothiopyrano[4,3-c]pyrazole and pyridothiopyrano[4,3-c]pyrazole effectively inhibit α- and β-carbonic anhydrase: X-ray crystallography and solution investigations on 15 isoforms.
Maria Letizia Trincavelli; Gemma Navarro; Susanna Nencetti; Elisa Nuti; Elisabetta Orlandini; Armando Rossello; Vicent Casadó; Simona Daniele; Chiara Giacomelli; Peter Gmeiner; Harald Huebner; Carme Lluís; Marco Macchia; Claudia Martini
A new D₂ dopamine receptor agonist allosterically modulates A(2A) adenosine receptor signalling by interacting with the A(2A)/D₂ receptor heteromer.

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All Publications

2013: Elisa Nuti; Elisabetta Orlandini; Silvia Salerno; Salvatore Santamaria; Sabrina Taliani; Kazuhiro Yamamoto; Francesca Casalini; Federico Da Settimo; Valeria La Pietra; Luciana Marinelli; Anna Maria Marini; Hideaki Nagase; Susanna Nencetti; Ettore Novellino; Armando Rossello
Arylsulfonamide inhibitors of aggrecanases as potential therapeutic agents for osteoarthritis: synthesis and biological evaluation.
European journal of medicinal chemistry 2013;62():379-94.
2012: Anna M Marini; Robert McKenna; Susanna Nencetti; Elisa Nuti; Elisabetta Orlandini; Armando Rossello; Silvia Salerno; Andrea Scozzafava; Francesca Simorini; Mayank Aggarwal; Federico Da Settimo; Concettina La Motta; Alfonso Maresca; Sabrina Taliani; Claudiu T Supuran
Tricyclic sulfonamides incorporating benzothiopyrano[4,3-c]pyrazole and pyridothiopyrano[4,3-c]pyrazole effectively inhibit α- and β-carbonic anhydrase: X-ray crystallography and solution investigations on 15 isoforms.
Journal of medicinal chemistry 2012;55(22):9619-29.
2012: Maria Letizia Trincavelli; Gemma Navarro; Susanna Nencetti; Elisa Nuti; Elisabetta Orlandini; Armando Rossello; Vicent Casadó; Simona Daniele; Chiara Giacomelli; Peter Gmeiner; Harald Huebner; Carme Lluís; Marco Macchia; Claudia Martini
A new D₂ dopamine receptor agonist allosterically modulates A(2A) adenosine receptor signalling by interacting with the A(2A)/D₂ receptor heteromer.
Cellular signalling 2012;24(4):951-60.
2012: Susanna Nencetti; E Orlandini
TTR fibril formation inhibitors: is there a SAR?
Current medicinal chemistry 2012;19(15):2356-79.
2011: Susanna Nencetti; Maria R Mazzoni; Gabriella Ortore; Annalina Lapucci; Janette Giuntini; Elisabetta Orlandini; Irene Banti; Elisa Nuti; Antonio Lucacchini; Gino Giannaccini; Armando Rossello
Synthesis, molecular docking and binding studies of selective serotonin transporter inhibitors.
European journal of medicinal chemistry 2011;46(3):825-34.
2010: Elisa Nuti; Francesca Casalini; Stanislava I Avramova; Salvatore Santamaria; Marina Fabbi; Silvano Ferrini; Luciana Marinelli; Valeria La Pietra; Vittorio Limongelli; Ettore Novellino; Giovanni Cercignani; Elisabetta Orlandini; Susanna Nencetti; Armando Rossello
Potent arylsulfonamide inhibitors of tumor necrosis factor-alpha converting enzyme able to reduce activated leukocyte cell adhesion molecule shedding in cancer cell models.
Journal of medicinal chemistry 2010;53(6):2622-35.
2009: Elisa Nuti; Laura Panelli; Francesca Casalini; Stanislava I Avramova; Elisabetta Orlandini; Salvatore Santamaria; Susanna Nencetti; Tiziano Tuccinardi; Adriano Martinelli; Giovanni Cercignani; Nicola D'Amelio; Alessandro Maiocchi; Fulvio Uggeri; Armando Rossello
Design, synthesis, biological evaluation, and NMR studies of a new series of arylsulfones as selective and potent matrix metalloproteinase-12 inhibitors.
Journal of medicinal chemistry 2009;52(20):6347-61.
2009: Elisa Nuti; Francesca Casalini; Stanislava I Avramova; Salvatore Santamaria; Giovanni Cercignani; Luciana Marinelli; Valeria La Pietra; Ettore Novellino; Elisabetta Orlandini; Susanna Nencetti; Tiziano Tuccinardi; Adriano Martinelli; Ngee-Han Lim; Robert Visse; Hideaki Nagase; Armando Rossello
N-O-isopropyl sulfonamido-based hydroxamates: design, synthesis and biological evaluation of selective matrix metalloproteinase-13 inhibitors as potential therapeutic agents for osteoarthritis.
Journal of medicinal chemistry 2009;52(15):4757-73.
2009: Irene Banti; Susanna Nencetti; Elisabetta Orlandini; Annalina Lapucci; Maria Cristina Breschi; Stefano Fogli
Synthesis and in-vitro antitumour activity of new naphthyridine derivatives on human pancreatic cancer cells.
The Journal of pharmacy and pharmacology 2009;61(8):1057-66.
2009: Satheesh K Palaninathan; Nilofar N Mohamedmohaideen; Elisabetta Orlandini; Gabriella Ortore; Susanna Nencetti; Annalina Lapucci; Armando Rossello; Joel S Freundlich; James C Sacchettini
Novel transthyretin amyloid fibril formation inhibitors: synthesis, biological evaluation, and X-ray structural analysis.
PloS one 2009;4(7):e6290.
2008: Musa Ahmed; Susanna Nencetti; Maria R Mazzoni; Francesca Porchia; Federica Antonelli; Annalina Lapucci
Allosteric inhibition of [(125I)] ET-1 binding to ET(A) receptors by aldoxime and hydroxamic acid derivatives.
Medicinal chemistry (Shāriqah (United Arab Emirates)) 2008;4(4):298-308.
2007: Susanna Nencetti; Gian Carlo Demontis; Maria R Mazzoni; Laura Betti; Irene Banti; Armando Rossello; Annalina Lapucci
3-[(Aryl)(4-fluorobenzyloxy)methyl]piperidine derivatives: high-affinity ligands for the serotonin transporter.
The Journal of pharmacy and pharmacology 2007;59(10):1439-45.
2007: Elisa Nuti; Elisabetta Orlandini; Susanna Nencetti; Armando Rossello; Alessio Innocenti; Andrea Scozzafava; Claudiu T Supuran
Carbonic anhydrase and matrix metalloproteinase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozyme I and II with sulfonylated hydroxamates.
Bioorganic & medicinal chemistry 2007;15(6):2298-311.
2007: Elisabetta Orlandini; Simona Rapposelli; Susanna Nencetti; Gino Giannaccini; Laura Betti; Aldo Balsamo
Synthesis and 5-HT2A, 5-HT1A and alpha1-binding affinities of 2-[2-Hydroxy-3-(pyridin-3-yl-methyl)amino]-, 2-[2-hydroxy-3-(2-pyridin-2-yl-ethyl)amino]- and 2-[2-hydroxy-3-(4-N-methyl-piperazin-1-yl)-amino]propoxybenzaldehyde-O-(substituted) benzyl oximes.
Archiv der Pharmazie 2007;340(3):135-9.
2005: Armando Rossello; Elisa Nuti; Paolo Carelli; Elisabetta Orlandini; Marco Macchia; Susanna Nencetti; Maurizio Zandomeneghi; Federica Balzano; Gloria Uccello-Barretta; Adriana Albini; Roberto Benelli; Giovanni Cercignani; Gillian Murphy; Aldo Balsamo
N-i-Propoxy-N-biphenylsulfonylaminobutylhydroxamic acids as potent and selective inhibitors of MMP-2 and MT1-MMP.
Bioorganic & medicinal chemistry letters 2005;15(5):1321-6.
2003: Annalina Lapucci; Susanna Nencetti; Gian Carlo Demontis
Synthesis and affinity for serotonin and dopamine transporters of some benzophenone oxime ether derivatives.
Farmaco (Società chimica italiana : 1989) 2003;58(9):977-81.
2003: Aldo Balsamo; Isabella Coletta; Angelo Guglielmotti; Carla Landolfi; Francesca Mancini; Adriano Martinelli; Claudio Milanese; Filippo Minutolo; Susanna Nencetti; Elisabetta Orlandini; Mario Pinza; Simona Rapposelli; Armando Rossello
Synthesis of heteroaromatic analogues of (2-aryl-1-cyclopentenyl-1-alkylidene)-(arylmethyloxy)amine COX-2 inhibitors: effects on the inhibitory activity of the replacement of the cyclopentene central core with pyrazole, thiophene or isoxazole ring.
European journal of medicinal chemistry 2003;38(2):157-68.
2002: Bruno Macchia; Clementina Manera; Adriano Martinelli; Susanna Nencetti; Elisabetta Orlandini; Maria Cristina Breschi; Claudia Martini; Enrica Martinotti
Spirotetrahydronaphthalene analogues of sympathomimetic catecholamines. Synthesis and adrenergic activity of 5,6- and 6,7-dihydroxy-3,4-dihydrospiro[naphthalen-1 (2H)-3'-piperidines].
The Journal of pharmacy and pharmacology 2002;54(5):649-60.
2002: Aldo Balsamo; Annalina Lapucci; Clementina Manera; Adriano Martinelli; Susanna Nencetti; Elisabetta Orlandini; Vincenzo Calderone; Gino Giannaccini; Paola Nieri
Conformationally restrained analogues of sympathomimetic catecholamines. Synthesis and adrenergic activity of 5,6- and 6,7-dihydroxy-3,4-dihydrospiro[naphthalen-1(2H)-2',5'-morpholines].
European journal of medicinal chemistry 2002;37(1):11-22.
2001: Marco Macchia; teresina laragione; Simone Bertini; Valeria Di Bussolo; L Gattuso; Marco Gesi; Mahmoud Hamdan; Karl-Norbert Klotz; T Laragione; Antonio Lucacchini; Filippo Minutolo; Susanna Nencetti; Chiara Papi; Daniela Tuscano; Claudia Martini
7-Nitrobenzofurazan (NBD) derivatives of 5'-N-ethylcarboxamidoadenosine (NECA) as new fluorescent probes for human A(3) adenosine receptors.
Bioorganic & medicinal chemistry letters 2001;11(23):3023-6.
2001: Aldo Balsamo; Simone Bertini; Gianbattista Gervasi; Annalina Lapucci; Susanna Nencetti; Elisabetta Orlandini; Simona Rapposelli; Armando Rossello; Giulio Soldani
Enantiopure 3-(arylmethylidene)aminoxy-2-methylpropionic acids: synthesis and antiinflammatory properties.
European journal of medicinal chemistry 2001;36(10):799-807.
1999: D Gentili; Marco Macchia; E Menchini; Susanna Nencetti; Elisabetta Orlandini; Armando Rossello; G Broccali; D Limonta
Synthesis and antimicrobial properties of cephalosporin derivatives substituted on the C(7) nitrogen with arylmethyloxyimino or arylmethyloxyamino alkanoyl groups.
Farmaco (Società chimica italiana : 1989) 1999;54(4):224-31.
1998: Aldo Balsamo; Maria Cristina Breschi; Grazia Chiellini; Annalina Lapucci; N Lazzeri; Marco Macchia; Adriano Martinelli; E Micali; Susanna Nencetti; Armando Rossello
Synthesis and beta-adrenergic properties of (Z)-N-[3-(alkylamino)-2-hydroxypropylidene](aryl-methyloxy)amines: effects of the configuration around the methyloxyiminomethyl (MOIM) double bond on the biopharmacological properties of MOIM-type beta-blocking agents.
Bioorganic & medicinal chemistry 1998;6(11):2151-60.
1998: Marco Macchia; Silvia Barontini; Adriano Martinelli; E Menchini; Susanna Nencetti; Elisabetta Orlandini; F Romagnoli
Synthesis and aldose reductase inhibitory activity of new N-(benzyloxy) glycine derivatives.
Farmaco (Società chimica italiana : 1989) 1998;53(5):369-73.
1996: Marco Macchia; Clementina Manera; Susanna Nencetti; Armando Rossello; G Broccali; D Limonta
Synthesis and antimicrobial activity of benzo[a]dihydrocarbazole and benzotetrahydrocyclohept[1,2-b]indole derivatives.
Farmaco (Società chimica italiana : 1989) 1996;51(1):75-8.
1995: D Gentili; A Lapucci; B Macchia; Marco Macchia; Adriano Martinelli; Susanna Nencetti; Elisabetta Orlandini; G Ferni; M Pinza
Synthesis and beta-adrenergic activity of a series of 3-(substituted-benzylideneaminoxy)propanolamine derivatives.
Farmaco (Società chimica italiana : 1989) 1995;50(7-8):519-26.
1994: B Macchia; Aldo Balsamo; Maria Cristina Breschi; G Chiellini; Marco Macchia; Adriano Martinelli; Claudia Martini; C Nardini; Susanna Nencetti; Armando Rossello
The [(methyloxy)imino]methyl moiety as a bioisoster of aryl. A novel class of completely aliphatic beta-adrenergic receptor antagonists.
Journal of medicinal chemistry 1994;37(10):1518-25.
1994: Aldo Balsamo; A Lapucci; Marco Macchia; Adriano Martinelli; Susanna Nencetti; Armando Rossello; T Cristina
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity.
Farmaco (Società chimica italiana : 1989) 1994;49(2):77-82.
1990: B Macchia; Aldo Balsamo; A Lapucci; F Macchia; Adriano Martinelli; Susanna Nencetti; Elisabetta Orlandini; M Baldacci; Grazia Mengozzi; Giulio Soldani
Molecular design, synthesis, and antiinflammatory activity of a series of beta-aminoxypropionic acids.
Journal of medicinal chemistry 1990;33(5):1423-30.
1989: Aldo Balsamo; Maria Cristina Breschi; A Lapucci; B Macchia; F Macchia; Enrica Martinotti; Susanna Nencetti; Paola Nieri; Elisabetta Orlandini
Synthesis and evaluation of the pharmacological activity of rigid analogues of sympathomimetic catecholamines derived from bicyclo[2.2.1]heptane.
Journal of medicinal chemistry 1989;32(4):856-9.
1988: B Macchia; Aldo Balsamo; A Lapucci; F Macchia; Clementina Manera; Susanna Nencetti; Maria Cristina Breschi; Antonio Lucacchini; Claudia Martini; Enrica Martinotti
An anomalous effect of N-isopropyl substitution in determining beta-adrenergic activity.
Drug design and delivery 1988;2(4):257-62.
1986: B Macchia; Aldo Balsamo; E Epifani; A Lapucci; Susanna Nencetti; F Macchia; Maria Cristina Breschi; Enrica Martinotti; R Ceserani
Conformational effects on the activity of drugs. 11. Stereostructural models for the direct activation of the alpha- and beta-adrenergic receptor.
Journal of medicinal chemistry 1986;29(5):740-7.