FIND

researchers

DISCOVER

relevant articles

PROMOTE

your research

now for free

Violetta Cecchetti

Research Profile

Concepts & Ideas

Chemicals & Drugs

Procedures

Microbial Sensitivity Tests

Physiology

Living Beings

Anatomy

Cell Line

Genes & Molecular Sequences

Molecular Structure

Co-author Network

Publications

TOP 3
Maria Letizia Barreca; Amartya Basu; U Helena Danielson; Nunzio Iraci; Neerja Kaushik-Basu; Ramalingam Krishnan; Pieter Leyssen; Giuseppe Manfroni; Johan Neyts; Jan Paeshuyse; Stefano Sabatini; Oriana Tabarrini; Johan Winquist; Violetta Cecchetti
Structure-based discovery of pyrazolobenzothiazine derivatives as inhibitors of hepatitis C virus replication.
Oriana Tabarrini; Scott G Franzblau; Serena Massari; Marco Pieroni; Stefano Sabatini; Violetta Cecchetti
6-hydrogen-8-methylquinolones active against replicating and non-replicating Mycobacterium tuberculosis.
Stefano Sabatini; Serena Serritella; Oriana Tabarrini; Milena Villarini; Francesca Gosetto; Nunzio Iraci; Glenn W Kaatz; Giuseppe Manfroni; Jean Pierre Brincat; Emanuele Carosati; Violetta Cecchetti
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-dioxide: a promising new class of Staphylococcus aureus NorA efflux pump inhibitors.

Register for free to view:

Visualized networks:

See your personal network in
sophisticated graphical views

GeoTargeted Searches:

Locate experts around the world
and connect with global collaborators

Research Profiles:

See the research activity
of experts around the globe

Geonetwork of Violetta Cecchetti (preview)

Cities where this author has publications
Cities where co-authors of this author have publications

Flash Player Required

All Publications

2013: Maria Letizia Barreca; Amartya Basu; U Helena Danielson; Nunzio Iraci; Neerja Kaushik-Basu; Ramalingam Krishnan; Pieter Leyssen; Giuseppe Manfroni; Johan Neyts; Jan Paeshuyse; Stefano Sabatini; Oriana Tabarrini; Johan Winquist; Violetta Cecchetti
Structure-based discovery of pyrazolobenzothiazine derivatives as inhibitors of hepatitis C virus replication.
Journal of medicinal chemistry 2013;56(6):2270-82.
2012: Oriana Tabarrini; Scott G Franzblau; Serena Massari; Marco Pieroni; Stefano Sabatini; Violetta Cecchetti
6-hydrogen-8-methylquinolones active against replicating and non-replicating Mycobacterium tuberculosis.
Chemical biology & drug design 2012;80(5):781-6.
2012: Stefano Sabatini; Serena Serritella; Oriana Tabarrini; Milena Villarini; Francesca Gosetto; Nunzio Iraci; Glenn W Kaatz; Giuseppe Manfroni; Jean Pierre Brincat; Emanuele Carosati; Violetta Cecchetti
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-dioxide: a promising new class of Staphylococcus aureus NorA efflux pump inhibitors.
Journal of medicinal chemistry 2012;55(7):3568-72.
2012: Giuseppe Manfroni; Serena Massari; Francesco Meschini; Johan Neyts; Stefano Sabatini; Alberta Samuele; Maria Letizia Barreca; Nunzio Iraci; Pieter Leyssen; Giovanni Maga; Violetta Cecchetti
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase.
Bioorganic & medicinal chemistry 2012;20(2):866-76.
2011: Stefano Sabatini; Oriana Tabarrini; Francesca Gosetto; Glenn W Kaatz; Giuseppe Manfroni; Diixa Patel; Violetta Cecchetti
Evolution from a natural flavones nucleus to obtain 2-(4-Propoxyphenyl)quinoline derivatives as potent inhibitors of the S. aureus NorA efflux pump.
Journal of medicinal chemistry 2011;54(16):5722-36.
2011: Oriana Tabarrini; Stefano Sabatini; Luca Sancineto; Violetta Cecchetti; Dirk Daelemans; Giuseppe Manfroni; Serena Massari; Christophe Pannecouque
Structural investigation of the naphthyridone scaffold: identification of a 1,6-naphthyridone derivative with potent and selective anti-HIV activity.
ChemMedChem 2011;6(7):1249-57.
2011: Maria Letizia Barreca; Nunzio Iraci; Giuseppe Manfroni; Violetta Cecchetti
Allosteric inhibition of the hepatitis C virus NS5B polymerase: in silico strategies for drug discovery and development.
Future medicinal chemistry 2011;3(8):1027-55.
2010: Oriana Tabarrini; Serena Massari; Dirk Daelemans; Francesco Meschini; Giuseppe Manfroni; Laura Bottega; Barbara Gatto; Manlio Palumbo; Christophe Pannecouque; Violetta Cecchetti
Studies of anti-HIV transcription inhibitor quinolones: identification of potent N1-vinyl derivatives.
ChemMedChem 2010;5(11):1880-92.
2010: Oriana Tabarrini; Serena Massari; Violetta Cecchetti
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
Future medicinal chemistry 2010;2(7):1161-80.
2010: Arianna Loregian; Beatrice Mercorelli; Giulia Muratore; Elisa Sinigalia; Silvana Pagni; Serena Massari; Giorgio Gribaudo; Barbara Gatto; Manlio Palumbo; Oriana Tabarrini; Violetta Cecchetti; Giorgio Palù
The 6-aminoquinolone WC5 inhibits human cytomegalovirus replication at an early stage by interfering with the transactivating activity of viral immediate-early 2 protein.
Antimicrobial agents and chemotherapy 2010;54(5):1930-40.
2010: Serena Massari; Dirk Daelemans; Maria Letizia Barreca; Anna Knezevich; Stefano Sabatini; Violetta Cecchetti; Alessandro Marcello; Christophe Pannecouque; Oriana Tabarrini
A 1,8-naphthyridone derivative targets the HIV-1 Tat-mediated transcription and potently inhibits the HIV-1 replication.
Journal of medicinal chemistry 2010;53(2):641-8.
2009: Barbara Gatto; Oriana Tabarrini; Serena Massari; Giulia Giaretta; Stefano Sabatini; Claudia Del Vecchio; Cristina Parolin; Arnaldo Fravolini; Manlio Palumbo; Violetta Cecchetti
2-Phenylquinolones as inhibitors of the HIV-1 Tat-TAR interaction.
ChemMedChem 2009;4(6):935-8.
2009: Giuseppe Manfroni; Jan Paeshuyse; Serena Massari; Samantha Zanoli; Barbara Gatto; Giovanni Maga; Oriana Tabarrini; Violetta Cecchetti; Arnaldo Fravolini; Johan Neyts
Inhibition of subgenomic hepatitis C virus RNA replication by acridone derivatives: identification of an NS3 helicase inhibitor.
Journal of medicinal chemistry 2009;52(10):3354-65.
2009: Giuseppe Manfroni; Barbara Gatto; Oriana Tabarrini; Stefano Sabatini; Violetta Cecchetti; Giulia Giaretta; Cristina Parolin; Claudia Del Vecchio; Arianna Calistri; Manlio Palumbo; Arnaldo Fravolini
Synthesis and biological evaluation of 2-phenylquinolones targeted at Tat/TAR recognition.
Bioorganic & medicinal chemistry letters 2009;19(3):714-7.
2009: Serena Massari; Dirk Daelemans; Giuseppe Manfroni; Stefano Sabatini; Oriana Tabarrini; Christophe Pannecouque; Violetta Cecchetti
Studies on anti-HIV quinolones: new insights on the C-6 position.
Bioorganic & medicinal chemistry 2009;17(2):667-74.
2009: Beatrice Mercorelli; Giulia Muratore; Elisa Sinigalia; Oriana Tabarrini; Maria Angela Biasolo; Violetta Cecchetti; Giorgio Palù; Arianna Loregian
A 6-aminoquinolone compound, WC5, with potent and selective anti-human cytomegalovirus activity.
Antimicrobial agents and chemotherapy 2009;53(1):312-5.
2008: Jan Paeshuyse; Inge Vliegen; Lotte Coelmont; Pieter Leyssen; Oriana Tabarrini; Piet Herdewijn; Harald Mittendorfer; Johnny Easmon; Violetta Cecchetti; Ralf Bartenschlager; Gerhard Puerstinger; Johan Neyts
Comparative in vitro anti-hepatitis C virus activities of a selected series of polymerase, protease, and helicase inhibitors.
Antimicrobial agents and chemotherapy 2008;52(9):3433-7.
2007: Miguel Stevens; Michela Pollicita; Christophe Pannecouque; Erik Verbeken; Oriana Tabarrini; Violetta Cecchetti; Stefano Aquaro; Carlo Federico Perno; Arnaldo Fravolini; Erik De Clercq; Dominique Schols; Jan Balzarini
Novel in vivo model for the study of human immunodeficiency virus type 1 transcription inhibitors: evaluation of new 6-desfluoroquinolone derivatives.
Antimicrobial agents and chemotherapy 2007;51(4):1407-13.
2006: Oriana Tabarrini; Giuseppe Manfroni; Arnaldo Fravolini; Violetta Cecchetti; Stefano Sabatini; Erik De Clercq; Jef Rozenski; Bruno Canard; Hélène Dutartre; Jan Paeshuyse; Johan Neyts
Synthesis and anti-BVDV activity of acridones as new potential antiviral agents.
Journal of medicinal chemistry 2006;49(8):2621-7.
2006: Violetta Cecchetti; Oriana Tabarrini; Stefano Sabatini
From cromakalim to different structural classes of K(ATP) channel openers.
Current topics in medicinal chemistry 2006;6(10):1049-68.
2005: Miguel Stevens; Jan Balzarini; Oriana Tabarrini; Graciela Andrei; Robert Snoeck; Violetta Cecchetti; Arnaldo Fravolini; Erik De Clercq; Christophe Pannecouque
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation.
The Journal of antimicrobial chemotherapy 2005;56(5):847-55.
2005: Emanuele Carosati; Horst Lemoine; Roberto Spogli; Dagmar Grittner; Raimund Mannhold; Oriana Tabarrini; Stefano Sabatini; Violetta Cecchetti
Binding studies and GRIND/ALMOND-based 3D QSAR analysis of benzothiazine type K(ATP)-channel openers.
Bioorganic & medicinal chemistry 2005;13(19):5581-91.
2005: Alba Minelli; Ilaria Bellezza; Emanuela Siciliano; Lavinia Liguori; Oriana Tabarrini; Violetta Cecchetti; Arnaldo Fravolini
Inhibition of cell growth and induction of apoptosis in human prostate cancer cell lines by 6-aminoquinolone WM13.
Oncology reports 2005;13(6):1113-20.
2004: Oriana Tabarrini; Miguel Stevens; Violetta Cecchetti; Stefano Sabatini; Micaela Dell'Uomo; Giuseppe Manfroni; Manlio Palumbo; Christophe Pannecouque; Erik De Clercq; Arnaldo Fravolini
Structure modifications of 6-aminoquinolones with potent anti-HIV activity.
Journal of medicinal chemistry 2004;47(22):5567-78.
2004: Giampietro Viola; Laura Facciolo; Stefano Dall'Acqua; Fabio Di Lisa; Marcella Canton; Daniela Vedaldi; Arnaldo Fravolini; Oriana Tabarrini; Violetta Cecchetti
6-Aminoquinolones: photostability, cellular distribution and phototoxicity.
Toxicology in vitro : an international journal published in association with BIBRA 2004;18(5):581-92.
2004: Giovanni Cianchetta; Raimund Mannhold; Gabriele Cruciani; Massimo Baroni; Violetta Cecchetti
Chemometric studies on the bactericidal activity of quinolones via an extended VolSurf approach.
Journal of medicinal chemistry 2004;47(12):3193-201.
2003: Violetta Cecchetti; Vincenzo Calderone; Oriana Tabarrini; Stefano Sabatini; Enrica Filipponi; Lara Testai; Roberto Spogli; Enrica Martinotti; Arnaldo Fravolini
Highly potent 1,4-benzothiazine derivatives as K(ATP)-channel openers.
Journal of medicinal chemistry 2003;46(17):3670-9.
2003: Cristina Parolin; Barbara Gatto; Claudia Del Vecchio; Teresa Pecere; Enzo Tramontano; Violetta Cecchetti; Arnaldo Fravolini; Sara Masiero; Manlio Palumbo; Giorgio Palù
New anti-human immunodeficiency virus type 1 6-aminoquinolones: mechanism of action.
Antimicrobial agents and chemotherapy 2003;47(3):889-96.
2002: Giorgia Miolo; Giampietro Viola; Daniela Vedaldi; Francesco Dall'Acqua; Arnaldo Fravolini; Oriana Tabarrini; Violetta Cecchetti
In vitro phototoxic properties of new 6-desfluoro and 6-fluoro-8-methylquinolones.
Toxicology in vitro : an international journal published in association with BIBRA 2002;16(6):683-93.
2001: Oriana Tabarrini; Violetta Cecchetti; Andrea Temperini; Enrica Filipponi; M G Lamperti; Arnaldo Fravolini
Velnacrine thiaanalogues as potential agents for treating Alzheimer's disease.
Bioorganic & medicinal chemistry 2001;9(11):2921-8.
2001: Enrica Filipponi; Gabriele Cruciani; Oriana Tabarrini; Violetta Cecchetti; Arnaldo Fravolini
QSAR study and VolSurf characterization of anti-HIV quinolone library.
Journal of computer-aided molecular design 2001;15(3):203-17.
2000: Violetta Cecchetti; Cristina Parolin; Stefano Moro; Teresa Pecere; Enrica Filipponi; Arianna Calistri; Oriana Tabarrini; Barbara Gatto; Manlio Palumbo; Arnaldo Fravolini; G Palu'
6-Aminoquinolones as new potential anti-HIV agents.
Journal of medicinal chemistry 2000;43(20):3799-802.
2000: Violetta Cecchetti; Fausto Schiaffella; Oriana Tabarrini; Arnaldo Fravolini
(1,4-Benzothiazinyloxy)alkylpiperazine derivatives as potential antihypertensive agents.
Bioorganic & medicinal chemistry letters 2000;10(5):465-8.
2000: Enrica Filipponi; Violetta Cecchetti; Oriana Tabarrini; D Bonelli; Arnaldo Fravolini
Chemometric rationalization of the structural and physicochemical basis for selective cyclooxygenase-2 inhibition: toward more specific ligands.
Journal of computer-aided molecular design 2000;14(3):277-91.
1999: Violetta Cecchetti; Oriana Tabarrini; Stefano Sabatini; H Miao; Enrica Filipponi; Arnaldo Fravolini
Studies on 6-aminoquinolones: synthesis and antibacterial evaluation of 6-amino-8-ethyl- and 6-amino-8-methoxyquinolones.
Bioorganic & medicinal chemistry 1999;7(11):2465-71.
1999: Angela De Sarro; Violetta Cecchetti; V Fravolini; Francesco Naccari; Oriana Tabarrini; Giovambattista De Sarro
Effects of novel 6-desfluoroquinolones and classic quinolones on pentylenetetrazole-induced seizures in mice.
Antimicrobial agents and chemotherapy 1999;43(7):1729-36.
1999: Oriana Tabarrini; Violetta Cecchetti; Arnaldo Fravolini; Giuseppe Nocentini; A Barzi; Stefano Sabatini; H Miao; Claudia Sissi
Design and synthesis of modified quinolones as antitumoral acridones.
Journal of medicinal chemistry 1999;42(12):2136-44.
1998: Claudia Sissi; M Andreolli; Violetta Cecchetti; Arnaldo Fravolini; Barbara Gatto; Manlio Palumbo
Mg(2+)-mediated binding of 6-substituted quinolones to DNA: relevance to biological activity.
Bioorganic & medicinal chemistry 1998;6(9):1555-61.
1997: Maria Carbone; Maria Teresa Fera; Violetta Cecchetti; Oriana Tabarrini; Elena Losi; Valentina Valeria Cusumano; Giuseppe Teti
In vitro activities of new quinolones against Helicobacter pylori.
Antimicrobial agents and chemotherapy 1997;41(12):2790-2.
1997: Violetta Cecchetti; Gabriele Cruciani; Enrica Filipponi; Arnaldo Fravolini; Oriana Tabarrini; T Xin
Synthesis and antibacterial evaluation of [1,3]benzothiazino[3,2-a]quinoline- and [3,1]benzothiazino[1,2-a]quinoline-6-carboxylic acid derivatives.
Bioorganic & medicinal chemistry 1997;5(7):1339-44.
1997: Violetta Cecchetti; Enrica Filipponi; Arnaldo Fravolini; Oriana Tabarrini; D Bonelli; M Clementi; Gabriele Cruciani; S Clementi
Chemometric methodologies in a quantitative structure-activity relationship study: the antibacterial activity of 6-aminoquinolones.
Journal of medicinal chemistry 1997;40(11):1698-706.
1996: Violetta Cecchetti; Arnaldo Fravolini; Manlio Palumbo; Claudia Sissi; Oriana Tabarrini; P Terni; T Xin
Potent 6-desfluoro-8-methylquinolones as new lead compounds in antibacterial chemotherapy.
Journal of medicinal chemistry 1996;39(25):4952-7.
1996: Violetta Cecchetti; Arnaldo Fravolini; M C Lorenzini; Oriana Tabarrini; P Terni; T Xin
Studies on 6-aminoquinolones: synthesis and antibacterial evaluation of 6-amino-8-methylquinolones.
Journal of medicinal chemistry 1996;39(2):436-45.
1995: Violetta Cecchetti; S Clementi; Gabriele Cruciani; Arnaldo Fravolini; P G Pagella; A Savino; Oriana Tabarrini
6-Aminoquinolones: a new class of quinolone antibacterials?
Journal of medicinal chemistry 1995;38(6):973-82.
1995: Richard Wise; P G Pagella; Violetta Cecchetti; Arnaldo Fravolini; Oriana Tabarrini
In vitro activity of MF 5137, a new potent 6-aminoquinolone.
Drugs 1995;49 Suppl 2():272-3.
1994: Violetta Cecchetti; Arnaldo Fravolini; P G Pagella; Oriana Tabarrini; Andrea Temperini
7-(Disubstituted thiazolyl)-3,5-dihydroxy-6-heptenoic/heptanoic acid derivatives as HMG-CoA reductase inhibitors.
Bioorganic & medicinal chemistry 1994;2(8):799-806.
1993: Violetta Cecchetti; Arnaldo Fravolini; P G Pagella; A Savino; Oriana Tabarrini
Quinolinecarboxylic acids. 3. Synthesis and antibacterial evaluation of 2-substituted-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de] [1,4]benzothiazine-6-carboxylic acids related to rufloxacin.
Journal of medicinal chemistry 1993;36(22):3449-54.
1993: Violetta Cecchetti; Arnaldo Fravolini; Fausto Schiaffella; Oriana Tabarrini; Giancarlo Bruni; G Segre
o-Chlorobenzenesulfonamidic derivatives of (aryloxy)propanolamines as beta-blocking/diuretic agents.
Journal of medicinal chemistry 1993;36(1):157-61.
1990: Fausto Schiaffella; Renata Fringuelli; Violetta Cecchetti; Arnaldo Fravolini; P Angeli; G Marucci
Enantiomers of 8-(3-tert-butylamino-2-hydroxypropoxy)-3,4-dihydro-3-oxo-2H- (1,4)benzothiazine: racemic resolution, chiral synthesis and biological activity.
Farmaco (Società chimica italiana : 1989) 1990;45(12):1299-307.
1989: Fausto Schiaffella; Renata Fringuelli; Violetta Cecchetti; Arnaldo Fravolini; Giancarlo Bruni; F M Runci
Synthesis and antiinflammatory/analgesic activities of N-heterocyclic carboxamides of thiopyrano-1,2-benzothiazine.
Farmaco (Società chimica italiana : 1989) 1989;44(11):1031-44.
1987: Violetta Cecchetti; Arnaldo Fravolini; Renata Fringuelli; G Mascellani; P Pagella; M Palmioli; G Segre; P Terni
Quinolonecarboxylic acids. 2. Synthesis and antibacterial evaluation of 7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzothiazine-6-carboxylic acids.
Journal of medicinal chemistry 1987;30(3):465-73.
1987: Violetta Cecchetti; Arnaldo Fravolini; Renata Fringuelli; Fausto Schiaffella; G Mascellani; P G Pagella; P L Rugarli
Synthesis and beta-adrenergic blocking activity of oxipropanolamines of 3,4-dihydro-3-oxo-2H(1,4)benzothiazine.
Il Farmaco; edizione scientifica 1987;42(1):61-75.
1984: E Bousquet; Violetta Cecchetti; M De Regis; E Mannucci; G Orzalesi; I Volpato
[Quaternary salts of aminoethyl-p-aminobenzoates and aminoethyl-p-aminobenzamides. Synthesis and pharmacologic activity].
Il Farmaco; edizione scientifica 1984;39(1):3-15.
1983: Violetta Cecchetti; Arnaldo Fravolini; Fausto Schiaffella; M De Regis; G Orzalesi; I Volpato
[Synthesis and pharmacologic activity of the carboxamides of pyrazolo-1,2-benzothiazine and isoxazolo-1,2-benzothiazine (I)].
Il Farmaco; edizione scientifica 1983;38(1):35-44.