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Maurizio Anzini

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Claudia Sticozzi; Maurizio Anzini; Giuseppe Belmonte; Mariangela Biava; Andrea Cappelli; Franco Cervellati; Angela Di Capua; Antonio Giordani; Emanuela Maioli; Giuseppe Valacchi
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes.
Maurizio Anzini; Veronica Benetti; Paola Anzellotti; Simone Brogi; Vincenzo Calderone; Andrea Cappelli; Luisa Chiasserini; Angela Di Capua; Lorenzo Di Cesare Mannelli; Melania Dovizio; Carla Ghelardini; Antonio Giordani; Gianluca Giorgi; Germano Giuliani; Alma Martelli; Simona Pace; Paola Patrignani; Giovanna Poce; Antonietta Rossi; Michele Rovini; Lidia Sautebin; Alessandro Sega; Lara Testai; Salvatore Valenti; Salvatore Vomero; Mariangela Biava
Novel analgesic/anti-inflammatory agents: 1,5-diarylpyrrole nitrooxyalkyl ethers and related compounds as cyclooxygenase-2 inhibiting nitric oxide donors.
Mariangela Biava; Vincenzo Calderone; Sara Consalvi; Lorenzo Di Cesare Mannelli; Carla Ghelardini; Antonio Giordani; Alma Martelli; Paola Patrignani; Giovanna Poce; Giulio Cesare Porretta; Antonietta Rossi; Lidia Sautebin; Silvia Schenone; Lara Testai; Salvatore Alfonso; Claudio Battilocchio; Maurizio Anzini
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme.

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All Publications

2013: Claudia Sticozzi; Maurizio Anzini; Giuseppe Belmonte; Mariangela Biava; Andrea Cappelli; Franco Cervellati; Angela Di Capua; Antonio Giordani; Emanuela Maioli; Giuseppe Valacchi
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 2013;49(2):133-41.
2013: Maurizio Anzini; Veronica Benetti; Paola Anzellotti; Simone Brogi; Vincenzo Calderone; Andrea Cappelli; Luisa Chiasserini; Angela Di Capua; Lorenzo Di Cesare Mannelli; Melania Dovizio; Carla Ghelardini; Antonio Giordani; Gianluca Giorgi; Germano Giuliani; Alma Martelli; Simona Pace; Paola Patrignani; Giovanna Poce; Antonietta Rossi; Michele Rovini; Lidia Sautebin; Alessandro Sega; Lara Testai; Salvatore Valenti; Salvatore Vomero; Mariangela Biava
Novel analgesic/anti-inflammatory agents: 1,5-diarylpyrrole nitrooxyalkyl ethers and related compounds as cyclooxygenase-2 inhibiting nitric oxide donors.
Journal of medicinal chemistry 2013;56(8):3191-206.
2012: Mariangela Biava; Vincenzo Calderone; Sara Consalvi; Lorenzo Di Cesare Mannelli; Carla Ghelardini; Antonio Giordani; Alma Martelli; Paola Patrignani; Giovanna Poce; Giulio Cesare Porretta; Antonietta Rossi; Lidia Sautebin; Silvia Schenone; Lara Testai; Salvatore Alfonso; Claudio Battilocchio; Maurizio Anzini
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme.
European journal of medicinal chemistry 2012;58():287-98.
2012: Antonella Fioravanti; Mauro Galeazzi; Antonio Giordani; Antonello Lamboglia; Silvia Niccolini; Nicola Antonio Pascarelli; Laura Tinti; Angela Di Capua; Mariangela Biava; Andrea Cappelli; Maurizio Anzini
In vitro effects of VA441, a new selective cyclooxygenase-2 inhibitor, on human osteoarthritic chondrocytes exposed to IL-1β.
Journal of pharmacological sciences 2012;120(1):6-14.
2011: Mariangela Biava; Annalisa Bruno; Vincenzo Calderone; Lorenzo Di Cesare Mannelli; Carla Ghelardini; Antonio Giordani; Gianluca Giorgi; Alma Martelli; Giuseppina Papa; Paola Patrignani; Giovanna Poce; Giulio Cesare Porretta; Antonietta Rossi; Michele Rovini; Lidia Sautebin; Lara Testai; Salvatore Valenti; Salvatore Alfonso; Paola Anzellotti; Claudio Battilocchio; Maurizio Anzini
Novel analgesic/anti-inflammatory agents: diarylpyrrole acetic esters endowed with nitric oxide releasing properties.
Journal of medicinal chemistry 2011;54(22):7759-71.
2011: Andrea Cappelli; Alessandra Concas; Lorenzo Di Cesare Mannelli; Carla Ghelardini; Antonio Giordani; Gianluca Giorgi; Germano Giuliani; Francesco Makovec; Marco Paolino; Patrizia Porcu; Luigi Piero Stasi; Salvatore Valenti; Salvatore Vomero; Maurizio Anzini; Giulia Bini; Giovanni Biggio
Synthesis and structure-activity relationship studies in translocator protein ligands based on a pyrazolo[3,4-b]quinoline scaffold.
Journal of medicinal chemistry 2011;54(20):7165-75.
2011: Maurizio Anzini; Laura Betti; Stefano Alcaro; Carlo Braile; Andrea Cappelli; Simona Daniele; Carla Ghelardini; Gino Giannaccini; Gianluca Giorgi; Vittorio Limongelli; Antonio Lucacchini; Luciana Marinelli; Claudia Martini; Maria Paola Mascia; Ettore Novellino; Francesco Ortuso; Salvatore Valenti; Salvatore Vomero; Lorenzo Di Cesare Mannelli; Giovanni Biggio
New insight into the central benzodiazepine receptor-ligand interactions: design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds.
Journal of medicinal chemistry 2011;54(16):5694-711.
2011: Germano Giuliani; Andrea Cappelli; Mario Matarrese; Valeria Masiello; Elia Anna Turolla; Cristina Monterisi; Ferruccio Fazio; Maurizio Anzini; Gal la Pericot Mohr; Daniela Riitano; Federica Finetti; Lucia Morbidelli; Marina Ziche; Gianluca Giorgi; Salvatore Vomero
Non-peptide NK1 receptor ligands based on the 4-phenylpyridine moiety.
Bioorganic & medicinal chemistry 2011;19(7):2242-51.
2011: Mariangela Biava; Giulio Cesare Porretta; Giovanna Poce; Claudio Battilocchio; Maurizio Botta; Fabrizio Manetti; M Rovini; Andrea Cappelli; Lidia Sautebin; Antonietta Rossi; Carlo Pergola; Carla Ghelardini; N Galeotti; Francesco Makovec; A Giordani; P Anzellotti; S Tacconelli; Paola Patrignani; Maurizio Anzini
Enlarging the NSAIDs family: ether, ester and acid derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents.
Current medicinal chemistry 2011;18(10):1540-54.
2010: Andrea Cappelli; Salvatore Valenti; Alessandra Mancini; Germano Giuliani; Maurizio Anzini; Saverio Altieri; Silva Bortolussi; Cinzia Ferrari; Anna Maria Clerici; Cecilia Zonta; Fabio Carraro; Irene Filippi; Gianluca Giorgi; Alessandro Donati; Sandra Ristori; Salvatore Vomero; Alessandra Concas; Giovanni Biggio
Carborane-conjugated 2-quinolinecarboxamide ligands of the translocator protein for boron neutron capture therapy.
Bioconjugate chemistry 2010;21(12):2213-21.
2010: Andrea Cappelli; Chiara Nannicini; Salvatore Valenti; Germano Giuliani; Maurizio Anzini; Laura Mennuni; Antonio Giordani; Gianfranco Caselli; Luigi Piero Stasi; Francesco Makovec; Gianluca Giorgi; Salvatore Vomero
Design, synthesis, and preliminary biological evaluation of pyrrolo[3,4-c]quinolin-1-one and oxoisoindoline derivatives as aggrecanase inhibitors.
ChemMedChem 2010;5(5):739-48.
2010: Mariangela Biava; Giulio Cesare Porretta; Giovanna Poce; Claudio Battilocchio; Fabrizio Manetti; Maurizio Botta; Stefano Forli; Lidia Sautebin; Antonietta Rossi; Carlo Pergola; Carla Ghelardini; Nicoletta Galeotti; Francesco Makovec; Antonio Giordani; Paola Anzellotti; Paola Patrignani; Maurizio Anzini
Novel ester and acid derivatives of the 1,5-diarylpyrrole scaffold as anti-inflammatory and analgesic agents. Synthesis and in vitro and in vivo biological evaluation.
Journal of medicinal chemistry 2010;53(2):723-33.
2010: Maurizio Anzini; Alessia Chelini; Alessandra Mancini; Andrea Cappelli; Maria Frosini; Lorenzo Ricci; massimo valoti; Jacopo Magistretti; Loretta Castelli; Antonio Giordani; Francesco Makovec; Salvatore Vomero
Synthesis and biological evaluation of amidine, guanidine, and thiourea derivatives of 2-amino(6-trifluoromethoxy)benzothiazole as neuroprotective agents potentially useful in brain diseases.
Journal of medicinal chemistry 2010;53(2):734-44.
2010: Simone Galeazzi; Thomas M Hermans; Marco Paolino; Maurizio Anzini; Laura Mennuni; Antonio Giordani; Gianfranco Caselli; Francesco Makovec; E W Meijer; Salvatore Vomero; Andrea Cappelli
Multivalent supramolecular dendrimer-based drugs.
Biomacromolecules 2010;11(1):182-6.
2010: Anna Maria Aloisi; Ilaria Ceccarelli; Paolo Fiorenzani; Melinda Maddalena; Alessandra Rossi; Valentina Tomei; Giuseppina Sorda; Barbara Danielli; Michele Rovini; Andrea Cappelli; Maurizio Anzini; Antonio Giordano
Aromatase and 5-alpha reductase gene expression: modulation by pain and morphine treatment in male rats.
Molecular pain 2010;6():69.
2010: Andrea Cappelli; Stefania Butini; Antonella Brizzi; Sandra Gemma; Salvatore Valenti; Germano Giuliani; Maurizio Anzini; Laura Mennuni; Giuseppe Campiani; Vittorio Brizzi; Salvatore Vomero
The interactions of the 5-HT3 receptor with quipazine-like arylpiperazine ligands: the journey track at the end of the first decade of the third millennium.
Current topics in medicinal chemistry 2010;10(5):504-26.
2008: Mariangela Biava; Giulio C Porretta; Giovanna Poce; Sibilla Supino; Fabrizio Manetti; Stefano Forli; Maurizio Botta; Lidia Sautebin; Antonietta Rossi; Carlo Pergola; Carla Ghelardini; Monica Norcini; Francesco Makovec; Antonio Giordani; Paola Anzellotti; Roberto Cirilli; Rosella Ferretti; Bruno Gallinella; Francesco La Torre; Maurizio Anzini; Paola Patrignani
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents.
Bioorganic & medicinal chemistry 2008;16(17):8072-81.
2008: Maurizio Anzini; Carlo Braile; Salvatore Valenti; Andrea Cappelli; Salvatore Vomero; Luciana Marinelli; Vittorio Limongelli; Ettore Novellino; Laura Betti; Gino Giannaccini; Antonio Lucacchini; Carla Ghelardini; Monica Norcini; Francesco Makovec; Gianluca Giorgi; R Ian Fryer
Ethyl 8-fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as novel, highly potent, and safe antianxiety agent.
Journal of medicinal chemistry 2008;51(15):4730-43.
2008: Maurizio Anzini; Michele Rovini; Andrea Cappelli; Salvatore Vomero; Fabrizio Manetti; Maurizio Botta; Lidia Sautebin; Antonietta Rossi; Carlo Pergola; Carla Ghelardini; Monica Norcini; Antonio Giordani; Francesco Makovec; Paola Anzellotti; Paola Patrignani; Mariangela Biava
Synthesis, biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity.
Journal of medicinal chemistry 2008;51(15):4476-81.
2008: Andrea Cappelli; Germano Giuliani; Maurizio Anzini; Daniela Riitano; Gianluca Giorgi; Salvatore Vomero
Design, synthesis, and structure-affinity relationship studies in NK1 receptor ligands based on azole-fused quinolinecarboxamide moieties.
Bioorganic & medicinal chemistry 2008;16(14):6850-9.
2008: Andrea Cappelli; Alessandra Mancini; Francesco Sudati; Salvatore Valenti; Maurizio Anzini; Sara Belloli; Rosa Maria Moresco; Mario Matarrese; Mauro Vaghi; Andrea Fabro; Ferruccio Fazio; Salvatore Vomero
Synthesis and biological characterization of novel 2-quinolinecarboxamide ligands of the peripheral benzodiazepine receptors bearing technetium-99m or rhenium.
Bioconjugate chemistry 2008;19(6):1143-53.
2008: Andrea Cappelli; Chiara Nannicini; Andrea Gallelli; Germano Giuliani; Salvatore Valenti; Gal la Pericot Mohr; Maurizio Anzini; Laura Mennuni; Flora Ferrari; Gianfranco Caselli; Antonio Giordani; Walter Peris; Francesco Makovec; Gianluca Giorgi; Salvatore Vomero
Design, synthesis, and biological evaluation of AT1 angiotensin II receptor antagonists based on the pyrazolo[3,4-b]pyridine and related heteroaromatic bicyclic systems.
Journal of medicinal chemistry 2008;51(7):2137-46.
2008: Andrea Cappelli; Germano Giuliani; Salvatore Valenti; Maurizio Anzini; Salvatore Vomero; Gianluca Giorgi; Cristiana Sogliano; Elisabetta Maciocco; Giovanni Biggio; Alessandra Concas
Synthesis and structure-activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidem.
Bioorganic & medicinal chemistry 2008;16(6):3428-37.
2007: Filippo Carlucci; Maurizio Anzini; Michele Rovini; Dario Cattaneo; Simona Merlini; Antonella Tabucchi
Development of a CE method for the determination of mycophenolic acid in human plasma: a comparison with HPLC.
Electrophoresis 2007;28(21):3908-14.
2007: Mariangela Biava; Giulio Cesare Porretta; Giovanna Poce; Sibilla Supino; Stefano Forli; Michele Rovini; Andrea Cappelli; Fabrizio Manetti; Maurizio Botta; Lidia Sautebin; Antonietta Rossi; Carlo Pergola; Carla Ghelardini; Elisa Vivoli; Francesco Makovec; Paola Anzellotti; Paola Patrignani; Maurizio Anzini
Cyclooxygenase-2 inhibitors. 1,5-diarylpyrrol-3-acetic esters with enhanced inhibitory activity toward cyclooxygenase-2 and improved cyclooxygenase-2/cyclooxygenase-1 selectivity.
Journal of medicinal chemistry 2007;50(22):5403-11.
2006: Andrea Cappelli; Valter Travagli; Iacopo Zanardi; Maurizio Anzini; Gianluca Giorgi; Alessandro Donati; Marianna Aggravi; Mario Casolaro; Massimo Fresta; Eugenio Paccagnini; Francesco Makovec; Salvatore Vomero
Physicochemical and biopharmaceutical characterization of endo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1H-benz[e]isoindol-1-one (CR3124) a novel potent 5-HT3 receptor antagonist.
Journal of pharmaceutical sciences 2006;95(12):2706-21.
2006: Andrea Cappelli; Gal la Pericot Mohr; Germano Giuliani; Simone Galeazzi; Maurizio Anzini; Laura Mennuni; Flora Ferrari; Francesco Makovec; Eva M Kleinrath; Thierry Langer; massimo valoti; Gianluca Giorgi; Salvatore Vomero
Further studies on imidazo[4,5-b]pyridine AT1 angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4-phenylisoquinolinone or 1-phenylindene scaffolds.
Journal of medicinal chemistry 2006;49(22):6451-64.
2006: Andrea Cappelli; Mario Matarrese; Rosa Maria Moresco; Salvatore Valenti; Maurizio Anzini; Salvatore Vomero; Elia Anna Turolla; Sara Belloli; Pasquale Simonelli; Maria Azzurra Filannino; Michela Lecchi; Ferruccio Fazio
Synthesis, labeling, and biological evaluation of halogenated 2-quinolinecarboxamides as potential radioligands for the visualization of peripheral benzodiazepine receptors.
Bioorganic & medicinal chemistry 2006;14(12):4055-66.
2005: Andrea Cappelli; Andrea Gallelli; Monica Manini; Maurizio Anzini; Laura Mennuni; Francesco Makovec; M Cristina Menziani; Stefano Alcaro; Francesco Ortuso; Salvatore Vomero
Further studies on the interaction of the 5-hydroxytryptamine3 (5-HT3) receptor with arylpiperazine ligands. development of a new 5-HT3 receptor ligand showing potent acetylcholinesterase inhibitory properties.
Journal of medicinal chemistry 2005;48(10):3564-75.
2005: Andrea Cappelli; Germano Giuliani; Andrea Gallelli; Salvatore Valenti; Maurizio Anzini; Laura Mennuni; Francesco Makovec; Aroldo Cupello; Salvatore Vomero
Structure-affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5HT3 receptor.
Bioorganic & medicinal chemistry 2005;13(10):3455-60.
2005: Mariangela Biava; Giulio Cesare Porretta; Andrea Cappelli; Salvatore Vomero; Fabrizio Manetti; Maurizio Botta; Lidia Sautebin; Antonietta Rossi; Francesco Makovec; Maurizio Anzini
1,5-Diarylpyrrole-3-acetic acids and esters as novel classes of potent and highly selective cyclooxygenase-2 inhibitors.
Journal of medicinal chemistry 2005;48(9):3428-32.
2004: Andrea Cappelli; Gianluca Giorgi; Maurizio Anzini; Salvatore Vomero; Sandra Ristori; Claudio Rossi; Alessandro Donati
Characterization of persistent intramolecular C-H...X(N,O) bonds in solid state and solution.
Chemistry (Weinheim an der Bergstrasse, Germany) 2004;10(13):3177-83.
2004: Andrea Cappelli; Gal la Pericot Mohr Gl; Andrea Gallelli; Milena Rizzo; Maurizio Anzini; Salvatore Vomero; Laura Mennuni; Flora Ferrari; Francesco Makovec; M Cristina Menziani; Pier G De Benedetti; Gianluca Giorgi
Design, synthesis, structural studies, biological evaluation, and computational simulations of novel potent AT(1) angiotensin II receptor antagonists based on the 4-phenylquinoline structure.
Journal of medicinal chemistry 2004;47(10):2574-86.
2004: M Rizzo; D Ventrice; F Monforte; S Procopio; G De Sarro; Maurizio Anzini; Andrea Cappelli; Francesco Makovec
Sensitive SPE-HPLC method to determine a novel angiotensin-AT1 antagonist in biological samples.
Journal of pharmaceutical and biomedical analysis 2004;35(2):321-9.
2004: Andrea Cappelli; Germano Giuliani; Gal la Pericot Mohr Gl; Andrea Gallelli; Maurizio Anzini; Salvatore Vomero; Aroldo Cupello; Simona Scarrone; Mario Matarrese; Rosa Maria Moresco; Ferruccio Fazio; Federica Finetti; Lucia Morbidelli; Marina Ziche
A non-peptide NK1 receptor agonist showing subpicomolar affinity.
Journal of medicinal chemistry 2004;47(6):1315-8.
2003: Andrea Cappelli; Gal la Pericot Mohr; Maurizio Anzini; Salvatore Vomero; Alessandro Donati; Mario Casolaro; Raniero Mendichi; Gianluca Giorgi; Francesco Makovec
Synthesis and characterization of a new benzofulvene polymer showing a thermoreversible polymerization behavior.
The Journal of organic chemistry 2003;68(24):9473-6.
2003: M Rizzo; Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; D Ventrice; G De Sarro; S Procopio; N Costa; Francesco Makovec
Determination of a novel angiotensin-AT1 antagonist CR 3210 in biological samples by HPLC.
Farmaco (Società chimica italiana : 1989) 2003;58(9):837-44.
2003: Maurizio Anzini; Laura Canullo; Carlo Braile; Andrea Cappelli; Andrea Gallelli; Salvatore Vomero; M Cristina Menziani; Pier G De Benedetti; Milena Rizzo; Simona Collina; Ornella Azzolina; Massimo Sbacchi; Carla Ghelardini; Nicoletta Galeotti
Synthesis, biological evaluation, and receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as kappa-opioid receptor agonists endowed with antinociceptive and antiamnesic activity.
Journal of medicinal chemistry 2003;46(18):3853-64.
2003: Andrea Cappelli; Gal la Pericot Mohr; Andrea Gallelli; Germano Giuliani; Maurizio Anzini; Salvatore Vomero; Massimo Fresta; Patrizia Porcu; Elisabetta Maciocco; Alessandra Concas; Giovanni Biggio; Alessandro Donati
Structure-activity relationships in carboxamide derivatives based on the targeted delivery of radionuclides and boron atoms by means of peripheral benzodiazepine receptor ligands.
Journal of medicinal chemistry 2003;46(17):3568-71.
2002: Andrea Cappelli; Andrea Gallelli; Carlo Braile; Maurizio Anzini; Salvatore Vomero; Laura Mennuni; Francesco Makovec; M Cristina Menziani; Pier G De Benedetti; Alessandro Donati; Gianluca Giorgi
Novel potent 5-HT(3) receptor ligands based on the pyrrolidone structure. Effects of the quaternization of the basic nitrogen on the interaction with 5-HT(3) receptor.
Bioorganic & medicinal chemistry 2002;10(8):2681-91.
2002: Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; Laura Mennuni; Francesco Makovec; Michel Hamon; Pier G De Benedetti; M Cristina Menziani
The Interactions of the 5-HT(3) receptor with arylpiperazine, tropane, and quinuclidine ligands.
Current topics in medicinal chemistry 2002;2(6):599-624.
2002: Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; Laura Mennuni; Francesco Makovec; Edith Doucet; Michel Hamon; M Cristina Menziani; Pier G De Benedetti; Gianluca Giorgi; Carla Ghelardini; Simona Collina
Novel potent 5-HT(3) receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities.
Bioorganic & medicinal chemistry 2002;10(3):779-801.
2001: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; M Seeber; M Cristina Menziani; Thierry Langer; B Hagen; C Manzoni; J J Bourguignon
Mapping and fitting the peripheral benzodiazepine receptor binding site by carboxamide derivatives. Comparison of different approaches to quantitative ligand-receptor interaction modeling.
Journal of medicinal chemistry 2001;44(8):1134-50.
2001: Mario Matarrese; Rosa Maria Moresco; Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; Pasquale Simonelli; E Verza; Fulvio Magni; Francesco Sudati; Dmitri Soloviev; Sergio Todde; Assunta Carpinelli; Marzia Galli Kienle; Ferruccio Fazio
Labeling and evaluation of N-[11C]methylated quinoline-2-carboxamides as potential radioligands for visualization of peripheral benzodiazepine receptors.
Journal of medicinal chemistry 2001;44(4):579-85.
2001: Ornella Azzolina; Simona Collina; Laura Linati; Maurizio Anzini; Andrea Cappelli; Mark A Scheideler; Massimo Sbacchi
Enantiomers of 2-[(Acylamino)ethyl]-1,4-benzodiazepines, potent ligands of kappa-opioid receptor: chiral chromatographic resolution, configurational assignment and biological activity.
Chirality 2001;13(9):606-12.
1999: Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; L Canullo; Laura Mennuni; Francesco Makovec; Edith Doucet; Michel Hamon; M Cristina Menziani; Pier G De Benedetti; Giancarlo Bruni; M R Romeo; Gianluca Giorgi; Alessandro Donati
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 2. Molecular basis of the intrinsic efficacy of arylpiperazine derivatives at the central 5-HT3 receptors.
Journal of medicinal chemistry 1999;42(9):1556-75.
1998: Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; Laura Mennuni; Francesco Makovec; Edith Doucet; Michel Hamon; Giancarlo Bruni; M R Romeo; M Cristina Menziani; Pier G De Benedetti; Thierry Langer
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 1. Mapping the central 5-HT3 receptor binding site by arylpiperazine derivatives.
Journal of medicinal chemistry 1998;41(5):728-41.
1997: Giuseppe Campiani; Andrea Cappelli; Vito Nacci; Maurizio Anzini; Salvatore Vomero; Michel Hamon; Alfredo Cagnotto; Claudia Fracasso; C Uboldi; S Caccia; S Consolo; Tiziana Mennini
Novel and highly potent 5-HT3 receptor agonists based on a pyrroloquinoxaline structure.
Journal of medicinal chemistry 1997;40(22):3670-8.
1997: Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; Pier G De Benedetti; M Cristina Menziani; Gianluca Giorgi; C Manzoni
Mapping the peripheral benzodiazepine receptor binding site by conformationally restrained derivatives of 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3- isoquinolinecarboxamide (PK11195).
Journal of medicinal chemistry 1997;40(18):2910-21.
1996: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; Gianluca Giorgi; T Langer; Giancarlo Bruni; M R Romeo; Anthony Basile
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem.
Journal of medicinal chemistry 1996;39(21):4275-84.
1996: Andrea Cappelli; A Donati; Maurizio Anzini; Salvatore Vomero; Pier G De Benedetti; M Cristina Menziani; T Langer
Molecular structure and dynamics of some potent 5-HT3 receptor antagonists. Insight into the interaction with the receptor.
Bioorganic & medicinal chemistry 1996;4(8):1255-69.
1996: Andrea Cappelli; Maurizio Anzini; Salvatore Vomero; M Cristina Menziani; Pier G De Benedetti; M Sbacchi; G D Clarke; Laura Mennuni
Synthesis, biological evaluation, and quantitative receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as novel tifluadom-like ligands with high affinity and selectivity for kappa-opioid receptors.
Journal of medicinal chemistry 1996;39(4):860-72.
1995: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; Gianluca Giorgi; T Langer; Michel Hamon; N Merahi; B M Emerit; Alfredo Cagnotto; M Skorupska
Novel, potent, and selective 5-HT3 receptor antagonists based on the arylpiperazine skeleton: synthesis, structure, biological activity, and comparative molecular field analysis studies.
Journal of medicinal chemistry 1995;38(14):2692-704.
1993: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; Alfredo Cagnotto; M Skorupska
Synthesis and receptor binding studies of 2-functionalized 1,4-benzodiazepine derivatives as potential metaclazepam-like antianxiety agents.
Farmaco (Società chimica italiana : 1989) 1993;48(7):897-905.
1992: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; Alfredo Cagnotto; M Skorupska
Synthesis and benzodiazepine receptors affinity of 2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinolin-1-one and 3-carbethoxy-4-phenylquinoline derivatives.
Farmaco (Società chimica italiana : 1989) 1992;47(2):191-202.
1991: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; Giuseppe Campiani; Alfredo Cagnotto; M Skorupska
Synthesis and 5-HT receptors binding studies of some 3-substituted-2-(4-methyl-1-piperazinyl)-4-phenylquinolines.
Farmaco (Società chimica italiana : 1989) 1991;46(12):1435-47.
1990: Maurizio Anzini; Andrea Cappelli; Salvatore Vomero; Maurizio Botta; Alfredo Cagnotto
5-HT and benzodiazepine receptor ligands. III. Synthesis and receptor affinities of 1,2,4-triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one derivatives.
Farmaco (Società chimica italiana : 1989) 1990;45(11):1169-79.
1989: Maurizio Anzini; Salvatore Vomero; Antonio Garofalo; Andrea Cappelli; Alfredo Cagnotto
Synthesis and 5HT-receptors affinity of some 4-phenylquinoline derivatives.
Farmaco (Società chimica italiana : 1989) 1989;44(6):555-63.