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Eric Dawson

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Jon Jacobs; Craig W Lindsley; Andrew D Mesecar; Anna M Mielech; S Adrian Saldanha; Yahira M Baez-Santos; Susan C Baker; Peter Chase; Eric S Dawson; Aimee Eggler; Valerie Grum-Tokars; Peter Hodder; Sakshi Tomar; Mark Turlington; Ya Zhou; Shaun R Stauffer
Discovery, synthesis, and structure-based optimization of a series of N-(tert-butyl)-2-(N-arylamido)-2-(pyridin-3-yl) acetamides (ML188) as potent noncovalent small molecule inhibitors of the severe acute respiratory syndrome coronavirus (SARS-CoV) 3CL protease.
Alice L Rodriguez; J Scott Daniels; Thomas Steckler; Paige N Vinson; Richard Williams; Ya Zhou; José M Bartolomé; C David Weaver; Eric S Dawson; P Jeffrey Conn; Carrie K Jones; Hilde Lavreysen; Craig W Lindsley; Gregor J Macdonald; Claire Mackie; Colleen M Niswender; Shaun R Stauffer
Discovery and SAR of a novel series of non-MPEP site mGlu₅ PAMs based on an aryl glycine sulfonamide scaffold.
Ralf Mueller; Colleen M Niswender; C David Weaver; Mariusz Butkiewicz; P Jeffrey Conn; Eric S Dawson; Corey R Hopkins; Craig W Lindsley; Jens Meiler
Iterative experimental and virtual high-throughput screening identifies metabotropic glutamate receptor subtype 4 positive allosteric modulators.

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All Publications

2013: Jon Jacobs; Craig W Lindsley; Andrew D Mesecar; Anna M Mielech; S Adrian Saldanha; Yahira M Baez-Santos; Susan C Baker; Peter Chase; Eric S Dawson; Aimee Eggler; Valerie Grum-Tokars; Peter Hodder; Sakshi Tomar; Mark Turlington; Ya Zhou; Shaun R Stauffer
Discovery, synthesis, and structure-based optimization of a series of N-(tert-butyl)-2-(N-arylamido)-2-(pyridin-3-yl) acetamides (ML188) as potent noncovalent small molecule inhibitors of the severe acute respiratory syndrome coronavirus (SARS-CoV) 3CL protease.
Journal of medicinal chemistry 2013;56(2):534-46.
2012: Alice L Rodriguez; J Scott Daniels; Thomas Steckler; Paige N Vinson; Richard Williams; Ya Zhou; José M Bartolomé; C David Weaver; Eric S Dawson; P Jeffrey Conn; Carrie K Jones; Hilde Lavreysen; Craig W Lindsley; Gregor J Macdonald; Claire Mackie; Colleen M Niswender; Shaun R Stauffer
Discovery and SAR of a novel series of non-MPEP site mGlu₅ PAMs based on an aryl glycine sulfonamide scaffold.
Bioorganic & medicinal chemistry letters 2012;22(24):7388-92.
2012: Ralf Mueller; Colleen M Niswender; C David Weaver; Mariusz Butkiewicz; P Jeffrey Conn; Eric S Dawson; Corey R Hopkins; Craig W Lindsley; Jens Meiler
Iterative experimental and virtual high-throughput screening identifies metabotropic glutamate receptor subtype 4 positive allosteric modulators.
Journal of molecular modeling 2012;18(9):4437-46.
2012: Ralf Mueller; Colleen M Niswender; Christopher M Olsen; Alice L Rodriguez; Danny G Winder; Jens Meiler; Usha N Menon; Brittney S Bates; Brian A Chauder; P Jeffrey Conn; Eric S Dawson; Kyle A Emmitte; Andrew S Felts; Karen J Gregory; Sataywan B Jadhav; Carrie K Jones; Alexander S Kane; Jeffrey P Lamb; Craig W Lindsley
Discovery of 2-(2-benzoxazoyl amino)-4-aryl-5-cyanopyrimidine as negative allosteric modulators (NAMs) of metabotropic glutamate receptor 5 (mGlu₅): from an artificial neural network virtual screen to an in vivo tool compound.
ChemMedChem 2012;7(3):406-14.
2011: Keith Henry; Hideki Iwamoto; Miriam T Jacobs; Kristian Kaufmann; Jens Meiler; Sergei Y Noskov; Gary Rudnick; Ernesto Solis; Igor Zdravkovic; Steven Combs; Eric S Dawson; Louis J DeFelice; Bruce Felts; Julie R Field; Chelsea Adams; Vanessa Armstrong; Randy D Blakely
A conserved asparagine residue in transmembrane segment 1 (TM1) of serotonin transporter dictates chloride-coupled neurotransmitter transport.
The Journal of biological chemistry 2011;286(35):30823-36.
2009: Kristian W Kaufmann; Eric S Dawson; Keith Henry; Julie R Field; Randy D Blakely; Jens Meiler
Structural determinants of species-selective substrate recognition in human and Drosophila serotonin transporters revealed through computational docking studies.
Proteins 2009;74(3):630-42.
2008: Susan M Hanson; Eric S Dawson; Derek J Francis; Ned Van Eps; Candice S Klug; Wayne L Hubbell; Jens Meiler; Vsevolod V Gurevich
A model for the solution structure of the rod arrestin tetramer.
Structure (London, England : 1993) 2008;16(6):924-34.
2006: Simona G Codreanu; Deanna G Adams; Eric S Dawson; Brian E Wadzinski; Daniel C Liebler
Inhibition of protein phosphatase 2A activity by selective electrophile alkylation damage.
Biochemistry 2006;45(33):10020-9.
2006: Elizabeth M Hadac; Eric S Dawson; James W Darrow; Elizabeth E Sugg; Terry P Lybrand; Laurence J Miller
Novel benzodiazepine photoaffinity probe stereoselectively labels a site deep within the membrane-spanning domain of the cholecystokinin receptor.
Journal of medicinal chemistry 2006;49(3):850-63.
2004: Kaleeckal harikumar; Delia I Pinon; William Wessels; Eric S Dawson; Terry P Lybrand; Franklyn G Prendergast; Laurence J Miller
Measurement of intermolecular distances for the natural agonist Peptide docked at the cholecystokinin receptor expressed in situ using fluorescence resonance energy transfer.
Molecular pharmacology 2004;65(1):28-35.
2002: Eric S Dawson; Randel M Henne; Laurence J Miller; Terry P Lybrand
Moleular models for cholecystokinin-A receptor.
Pharmacology & toxicology 2002;91(6):290-6.
2001: Eric S Dawson; JN Wells
Determination of amino acid residues that are accessible from the ligand binding crevice in the seventh transmembrane-spanning region of the human A(1) adenosine receptor.
Molecular pharmacology 2001;59(5):1187-95.