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Antonio Di Stefano

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TOP 3
Piera Sozio; Anna Abbadessa; Laura Serafina Cerasa; Antonio Di Stefano
Designing prodrugs for the treatment of Parkinson's disease.
S Zara; Antonio Di Stefano; Cinzia Nasuti; Monica Rapino; Piera Sozio; A Cataldi
Ibuprofen and lipoic acid codrug 1 control Alzheimer's disease progression by down-regulating protein kinase C ε-mediated metalloproteinase 2 and 9 levels in β-amyloid infused Alzheimer's disease rat model.
Antonio Di Stefano; Antonio Iannitelli; Sara Laserra; Piera Sozio
Drug delivery strategies for Alzheimer's disease treatment.

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All Publications

2012: Piera Sozio; Anna Abbadessa; Laura Serafina Cerasa; Antonio Di Stefano
Designing prodrugs for the treatment of Parkinson's disease.
Expert opinion on drug discovery 2012;7(5):385-406.
2011: S Zara; Antonio Di Stefano; Cinzia Nasuti; Monica Rapino; Piera Sozio; A Cataldi
Ibuprofen and lipoic acid codrug 1 control Alzheimer's disease progression by down-regulating protein kinase C ε-mediated metalloproteinase 2 and 9 levels in β-amyloid infused Alzheimer's disease rat model.
Brain research 2011;1412():79-87.
2011: Antonio Di Stefano; Antonio Iannitelli; Sara Laserra; Piera Sozio
Drug delivery strategies for Alzheimer's disease treatment.
Expert opinion on drug delivery 2011;8(5):581-603.
2011: Susi Zara; Antonio Di Stefano; Cinzia Nasuti; Monica Rapino; Antonia Patruno; Mirko Pesce; Piera Sozio; Laura S Cerasa; Amelia Cataldi
NOS-mediated morphological and molecular modifications in rats infused with Aβ (1-40), as a model of Alzheimer's disease, in response to a new lipophilic molecular combination codrug-1.
Experimental gerontology 2011;46(4):273-81.
2011: Francesco Pinnen; Piera Sozio; Ivana Cacciatore; Catia Cornacchia; Adriano Mollica; Antonio Iannitelli; Eleonora D'Aurizio; Amelia Cataldi; Susi Zara; Cinzia Nasuti; Antonio Di Stefano
Ibuprofen and glutathione conjugate as a potential therapeutic agent for treating Alzheimer's disease.
Archiv der Pharmazie 2011;344(3):139-48.
2011: Antonio Iannitelli; Sara Laserra; Cecilia Paolini; Feliciano Protasi; Piera Sozio; Lucinda Janete Bessa; Mara Di Giulio; Antonio Di Stefano; Rossella Grande; Luigina Cellini
Potential Antibacterial Activity of Carvacrol-Loaded Poly(DL-lactide-co-glycolide) (PLGA) Nanoparticles against Microbial Biofilm.
International journal of molecular sciences 2011;12(8):5039-51.
2010: Antonio Di Stefano; Piera Sozio; L S Cerasa; Antonio Iannitelli; A Cataldi; S Zara; Gianfabio Giorgioni; Cinzia Nasuti
Ibuprofen and lipoic acid diamide as co-drug with neuroprotective activity: pharmacological properties and effects in beta-amyloid (1-40) infused Alzheimer's disease rat model.
International journal of immunopathology and pharmacology 2010;23(2):589-99.
2010: Ivana Cacciatore; Catia Cornacchia; Francesco Pinnen; Adriano Mollica; Antonio Di Stefano
Prodrug approach for increasing cellular glutathione levels.
Molecules (Basel, Switzerland) 2010;15(3):1242-64.
2010: Piera Sozio; Eleonora D'Aurizio; Antonio Iannitelli; Amelia Cataldi; Susi Zara; Franco Cantalamessa; Cinzia Nasuti; Antonio Di Stefano
Ibuprofen and lipoic acid diamides as potential codrugs with neuroprotective activity.
Archiv der Pharmazie 2010;343(3):133-42.
2010: Gianfabio Giorgioni; F Claudi; Sabrina Ruggieri; Massimo Ricciutelli; Giovanni F Palmieri; Antonio Di Stefano; Piera Sozio; Laura S Cerasa; Annalisa Chiavaroli; Claudio Ferrante; Giustino Orlando; Richard A Glennon
Design, synthesis, and preliminary pharmacological evaluation of new imidazolinones as L-DOPA prodrugs.
Bioorganic & medicinal chemistry 2010;18(5):1834-43.
2009: S Heuking; Antonio Iannitelli; Antonio Di Stefano; G Borchard
Toll-like receptor-2 agonist functionalized biopolymer for mucosal vaccination.
International journal of pharmaceutics 2009;381(2):97-105.
2009: Antonio Di Stefano; Eleonora D'Aurizio; Oriana Trubiani; Rossella Grande; Emanuela Di Campli; Mara Di Giulio; Sabrina Di Bartolomeo; Piera Sozio; Antonio Iannitelli; Antonia Nostro; Luigina Cellini
Viscoelastic properties of Staphylococcus aureus and Staphylococcus epidermidis mono-microbial biofilms.
Microbial biotechnology 2009;2(6):634-41.
2009: Antonio Di Stefano; Piera Sozio; Antonio Iannitelli; Laura Serafina Cerasa
New drug delivery strategies for improved Parkinson's disease therapy.
Expert opinion on drug delivery 2009;6(4):389-404.
2009: Francesco Pinnen; Ivana Cacciatore; Catia Cornacchia; Piera Sozio; Laura Serafina Cerasa; Antonio Iannitelli; Cinzia Nasuti; Franco Cantalamessa; Durairaj Sekar; Rosita Gabbianelli; Maria Letizia Falcioni; Antonio Di Stefano
Codrugs linking L-dopa and sulfur-containing antioxidants: new pharmacological tools against Parkinson's disease.
Journal of medicinal chemistry 2009;52(2):559-63.
2008: Antonio Di Stefano; Piera Sozio; Antonio Iannitelli; Laura Serafina Cerasa; Antonella Fontana; Giuseppe Di Biase; Guglielmo D'Amico; Mara Di Giulio; Carmen Carpentiero; Lucia Grumetto; Francesco Barbato
Characterization of alkanoyl-10-O-minocyclines in micellar dispersions as potential agents for treatment of human neurodegenerative disorders.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 2008;34(2-3):118-28.
2008: Piera Sozio; Antonio Iannitelli; Laura Serafina Cerasa; Ivana Cacciatore; Catia Cornacchia; Gianfabio Giorgioni; Massimo Ricciutelli; Cinzia Nasuti; Franco Cantalamessa; Antonio Di Stefano
New L-dopa codrugs as potential antiparkinson agents.
Archiv der Pharmazie 2008;341(7):412-7.
2008: Gianfabio Giorgioni; S Ruggieri; Antonio Di Stefano; P Sozio; B Cinque; L Di Marzio; Giorgio Santoni; F Claudi
Glycosyl and polyalcoholic prodrugs of lonidamine.
Bioorganic & medicinal chemistry letters 2008;18(7):2445-50.
2008: Antonio Di Stefano; Piera Sozio; Laura Serafina Cerasa
Antiparkinson prodrugs.
Molecules (Basel, Switzerland) 2008;13(1):46-68.
2008: Gianfabio Giorgioni; S Ruggieri; F Claudi; Antonio Di Stefano; E Ljung; T Carlsson
Synthesis and pharmacological evaluation of 4-phenoxy-1,2,3,4-tetrahydroisoquinolines and 4,5,6,6a-tetrahydrochromeno[2,3,4-de]isoquinolines.
Medicinal chemistry (Shāriqah (United Arab Emirates)) 2008;4(1):1-10.
2007: Francesco Pinnen; Ivana Cacciatore; Catia Cornacchia; Piera Sozio; Antonio Iannitelli; Mara Costa; Laura Pecci; Cinzia Nasuti; Franco Cantalamessa; Antonio Di Stefano
Synthesis and study of L-dopa-glutathione codrugs as new anti-Parkinson agents with free radical scavenging properties.
Journal of medicinal chemistry 2007;50(10):2506-15.
2007: Cinzia Nasuti; Rosita Gabbianelli; Maria Letizia Falcioni; Antonio Di Stefano; Piera Sozio; Franco Cantalamessa
Dopaminergic system modulation, behavioral changes, and oxidative stress after neonatal administration of pyrethroids.
Toxicology 2007;229(3):194-205.
2006: m carafa; Carlotta Marianecci; V Annibaldi; Antonio Di Stefano; Piera Sozio; Eleonora Santucci
Novel O-palmitoylscleroglucan-coated liposomes as drug carriers: development, characterization and interaction with leuprolide.
International journal of pharmaceutics 2006;325(1-2):155-62.
2006: Antonio Di Stefano; Piera Sozio; Antonio Iannitelli; Carlotta Marianecci; Eleonora Santucci; m carafa
Maleic- and fumaric-diamides of (O,O-diacetyl)-L-Dopa-methylester as anti-Parkinson prodrugs in liposomal formulation.
Journal of drug targeting 2006;14(9):652-61.
2006: Antonio Di Stefano; Piera Sozio; Alessandra Cocco; Antonio Iannitelli; Eleonora Santucci; Mara Costa; Laura Pecci; Cinzia Nasuti; Franco Cantalamessa; Francesco Pinnen
L-dopa- and dopamine-(R)-alpha-lipoic acid conjugates as multifunctional codrugs with antioxidant properties.
Journal of medicinal chemistry 2006;49(4):1486-93.
2005: Ivana Cacciatore; Anna Maria Caccuri; Alessandra Cocco; Francesca De Maria; Antonio Di Stefano; Grazia Luisi; Francesco Pinnen; Giorgio Ricci; Piera Sozio; Paola Turella
Potent isozyme-selective inhibition of human glutathione S-transferase A1-1 by a novel glutathione S-conjugate.
Amino acids 2005;29(3):255-61.
2005: Antonio Di Stefano; Piera Sozio; Ivana Cacciatore; Alessandra Cocco; Gianfabio Giorgioni; Barbara Costa; Marina Montali; Antonio Lucacchini; Claudia Martini; Giuseppe Spoto; Francesco Di Pietrantonio; Elisabetta Di Matteo; Francesco Pinnen
Preparation and pharmacological characterization of trans-2-amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes as D2-like dopamine receptor agonists.
Journal of medicinal chemistry 2005;48(7):2646-54.
2004: Antonio Di Stefano; m carafa; Piera Sozio; Francesco Pinnen; Daniela Braghiroli; Giustino Orlando; Giuseppe Cannazza; Massimo Ricciutelli; Carlotta Marianecci; Eleonora Santucci
Evaluation of rat striatal L-dopa and DA concentration after intraperitoneal administration of L-dopa prodrugs in liposomal formulations.
Journal of controlled release : official journal of the Controlled Release Society 2004;99(2):293-300.
2004: Vincenzo Rispoli; Domenicantonio Rotiroti; Vincenzo Carelli; Felice Liberatore; Luigi Scipione; Rosario Marra; Gianfabio Giorgioni; Antonio Di Stefano
Choline pivaloyl esters improve in rats cognitive and memory performances impaired by scopolamine treatment or lesions of the nucleus basalis of Meynert.
Neuroscience letters 2004;356(3):199-202.
2004: Ivana Cacciatore; Antonio Di Stefano; Grazia Luisi; Francesco Pinnen; Piera Sozio
Transition state isosteres of the gamma-glutamyl peptide bond hydrolysis: synthesis and characterization of the psi (CH2NH) pseudopeptide analogue of glutathione.
Journal of peptide science : an official publication of the European Peptide Society 2004;10(2):109-14.
2003: Vincenzo Carelli; Felice Liberatore; Luigi Scipione; Gianfabio Giorgioni; Antonio Di Stefano; Mariannina Impicciatore; Vigilio Ballabeni; Francesco Calcina; Francesca Magnanini; Elisabetta Barocelli
Synthesis and biological evaluation of GABA derivatives able to cross the blood-brain barrier in rats.
Bioorganic & medicinal chemistry letters 2003;13(21):3765-9.
2003: Ivana Cacciatore; Anna Maria Caccuri; Antonio Di Stefano; Grazia Luisi; Marianna Nalli; Francesco Pinnen; Giorgio Ricci; Piera Sozio
Synthesis and activity of novel glutathione analogues containing an urethane backbone linkage.
Farmaco (Società chimica italiana : 1989) 2003;58(9):787-93.
2003: Mario Paglialunga Paradisi; Adriano Mollica; Ivana Cacciatore; Antonio Di Stefano; Francesco Pinnen; Anna Maria Caccuri; Giorgio Ricci; Silvestro Duprè; Alessandra Spirito; Gino Lucente
Proline-glutamate chimeras in isopeptides. Synthesis and biological evaluation of conformationally restricted glutathione analogues.
Bioorganic & medicinal chemistry 2003;11(8):1677-83.
2003: Ivana Cacciatore; Antonio Di Stefano; Silvestro Duprè; Enrico Morera; Francesco Pinnen; Alessandra Spirito
Synthesis and biological evaluation of the disulfide form of the glutathione analogue gamma-(L-glutamyl)-L-cysteinyl-L-aspartyl-L-cysteine.
Bioorganic chemistry 2003;31(2):109-21.
2002: Luigi Brunetti; Ivana Cacciatore; Antonio Di Stefano; Silvestro Duprè; Alessandra Giorgi; Grazia Luisi; Barbara Michelotto; Giustino Orlando; Francesco Pinnen; Lucia Recinella; Piera Sozio; Alessandra Spirito
Synthesis and biological evaluation of a novel pyroglutamyl-modified TRH analogue.
Farmaco (Società chimica italiana : 1989) 2002;57(6):479-86.
2002: Antonio Di Stefano; Piera Sozio; Grazia Luisi; Ivana Cacciatore; Barbara Mosciatti; Barbara Costa; Antonio Lucacchini; Claudia Martini; Francesco Pinnen
Synthesis and preliminary pharmacological evaluation of trans-2-amino-5(6)-chloro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes as dopamine receptor ligands.
Farmaco (Società chimica italiana : 1989) 2002;57(4):303-13.
2001: GM Cingolani; Antonio Di Stefano; F Napolitani; Barbara Mosciatti; Gianfabio Giorgioni; N Cinone; Luigi Brunetti; Grazia Luisi; Barbara Michelotto; Giustino Orlando; Barbara Costa; Antonio Lucacchini; Claudia Martini; F Claudi
Synthesis and preliminary pharmacological evaluation of 5-hydroxy- and 5,6-dihydroxy-1,2,3,7,12,12a-hexahydrobenzo[5,6]cyclohepta[1,2,3-ij]isoquinoline derivatives as dopamine receptor ligands.
Bioorganic & medicinal chemistry 2001;9(6):1447-58.
2001: Antonio Di Stefano; Barbara Mosciatti; GM Cingolani; Gianfabio Giorgioni; Massimo Ricciutelli; Ivana Cacciatore; Piera Sozio; F Claudi
Dimeric L-dopa derivatives as potential prodrugs.
Bioorganic & medicinal chemistry letters 2001;11(8):1085-8.
2000: GM Cingolani; Antonio Di Stefano; Barbara Mosciatti; F Napolitani; Gianfabio Giorgioni; Massimo Ricciutelli; F Claudi
Synthesis of L-(+)-3-(3-hydroxy-4-pivaloyloxybenzyl)-2,5-diketomorpholine as potential prodrug of L-dopa.
Bioorganic & medicinal chemistry letters 2000;10(12):1385-8.
2000: F Claudi; Antonio Di Stefano; F Napolitani; GM Cingolani; Gianfabio Giorgioni; Jose A Fontenla; GY Montenegro; ME Rivas; E Rosa; Barbara Michelotto; Giustino Orlando; Luigi Brunetti
Binding and preliminary evaluation of 5-hydroxy- and 10-hydroxy-2,3, 12,12a-tetrahydro-1H-[1]benzoxepino[2,3,4-ij]isoquinolines as dopamine receptor ligands.
Journal of medicinal chemistry 2000;43(4):599-608.
1999: A Calcagni; P G Ciattini; Antonio Di Stefano; Silvestro Duprè; Grazia Luisi; Francesco Pinnen; D Rossi; Alessandra Spirito
psi(SO2NH) transition state isosteres of peptides. Synthesis and bioactivity of sulfonamido pseudopeptides related to carnosine.
Farmaco (Società chimica italiana : 1989) 1999;54(10):673-7.