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Joseph Duffy

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Scott B Hoyt; Nina Jochnowitz; Gregory J Kaczorowski; Bindhu V Karanam; Xiaohua Li; Clare London; Kathryn A Lyons; Erin McGowan; Birgit T Priest; McHardy M Smith; Brande S Thomas-Fowlkes; Vivien A Warren; Catherine Abbadie; John P Felix; Maria L Garcia; Joseph L Duffy
A novel benzazepinone sodium channel blocker with oral efficacy in a rat model of neuropathic pain.
Pengcheng P Shao; McHardy M Smith; Shu-Yu Sun; Andrew M Swensen; Deepu J Varughese; Vivien A Warren; Feng Ye; Catherine Abbadie; Randal M Bugianesi; Prasun K Chakravarty; Ge Dai; Maria L Garcia; Mitchell Green; Rodolfo J Haedo; James B Herrington; Nina Jochnowitz; Gregory J Kaczorowski; Xiaohua Li; Kathryn A Lyons; Erin McGowan; Owen B McManus; Shruti Mistry; Joseph L Duffy
Aminopiperidine sulfonamide Cav2.2 channel inhibitors for the treatment of chronic pain.
Andrew M Swensen; Vivien A Warren; David Parker; Kevin S Ratliff; McHardy Smith; Terrance P Snutch; Stephen P Arneric; Randal M Bugianesi; Ge Dai; Joseph L Duffy; Cyrus Eduljee; Rodolfo J Haedo; James Herrington; Scott B Hoyt; Gregory J Kaczorowski; Clare London; Owen B McManus
Characterization of the substituted N-triazole oxindole TROX-1, a small-molecule, state-dependent inhibitor of Ca(V)2 calcium channels.

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All Publications

2013: Scott B Hoyt; Nina Jochnowitz; Gregory J Kaczorowski; Bindhu V Karanam; Xiaohua Li; Clare London; Kathryn A Lyons; Erin McGowan; Birgit T Priest; McHardy M Smith; Brande S Thomas-Fowlkes; Vivien A Warren; Catherine Abbadie; John P Felix; Maria L Garcia; Joseph L Duffy
A novel benzazepinone sodium channel blocker with oral efficacy in a rat model of neuropathic pain.
Bioorganic & medicinal chemistry letters 2013;23(12):3640-5.
2012: Pengcheng P Shao; McHardy M Smith; Shu-Yu Sun; Andrew M Swensen; Deepu J Varughese; Vivien A Warren; Feng Ye; Catherine Abbadie; Randal M Bugianesi; Prasun K Chakravarty; Ge Dai; Maria L Garcia; Mitchell Green; Rodolfo J Haedo; James B Herrington; Nina Jochnowitz; Gregory J Kaczorowski; Xiaohua Li; Kathryn A Lyons; Erin McGowan; Owen B McManus; Shruti Mistry; Joseph L Duffy
Aminopiperidine sulfonamide Cav2.2 channel inhibitors for the treatment of chronic pain.
Journal of medicinal chemistry 2012;55(22):9847-55.
2012: Andrew M Swensen; Vivien A Warren; David Parker; Kevin S Ratliff; McHardy Smith; Terrance P Snutch; Stephen P Arneric; Randal M Bugianesi; Ge Dai; Joseph L Duffy; Cyrus Eduljee; Rodolfo J Haedo; James Herrington; Scott B Hoyt; Gregory J Kaczorowski; Clare London; Owen B McManus
Characterization of the substituted N-triazole oxindole TROX-1, a small-molecule, state-dependent inhibitor of Ca(V)2 calcium channels.
Molecular pharmacology 2012;81(3):488-97.
2011: S Tyagarajan; Prasun K Chakravarty; Min Park; Bishan Zhou; James B Herrington; Kevin Ratliff; Randal M Bugianesi; Brande Williams; Rodolfo J Haedo; Andrew M Swensen; Vivien A Warren; McHardy Smith; Maria Garcia; Gregory J Kaczorowski; Owen B McManus; Kathryn A Lyons; Xiaohua Li; Maria Madeira; Bindhu V Karanam; Mitchell Green; Michael J Forrest; Catherine Abbadie; Erin McGowan; Shruti Mistry; Nina Jochnowitz; Joseph L Duffy
A potent and selective indole N-type calcium channel (Ca(v)2.2) blocker for the treatment of pain.
Bioorganic & medicinal chemistry letters 2011;21(2):869-73.
2010: S Tyagarajan; Prasun K Chakravarty; Bishan Zhou; Brett Taylor; Ronsar Eid; Michael H Fisher; William H Parsons; Matthew J Wyvratt; Kathryn A Lyons; Tracy Klatt; Xiaohua Li; Sanjeev Kumar; Brande Williams; John Felix; Birgit T Priest; Richard Brochu; Vivien A Warren; McHardy Smith; Maria Garcia; Gregory J Kaczorowski; William J Martin; Catherine Abbadie; Erin McGowan; Nina Jochnowitz; Ann Weber; Joseph L Duffy
Discovery of a novel class of biphenyl pyrazole sodium channel blockers for treatment of neuropathic pain.
Bioorganic & medicinal chemistry letters 2010;20(24):7479-82.
2010: Catherine Abbadie; Owen B McManus; Shu-Yu Sun; Randal M Bugianesi; Ge Dai; Rodolfo J Haedo; James B Herrington; Gregory J Kaczorowski; McHardy Smith; Andrew M Swensen; Vivien A Warren; Brande Williams; Stephen P Arneric; Cyrus Eduljee; Terrance P Snutch; Elizabeth W Tringham; Nina Jochnowitz; Annie Liang; D Euan MacIntyre; Erin McGowan; Shruti Mistry; Valerie V White; Scott B Hoyt; Clare London; Kathryn A Lyons; Patricia B Bunting; Sylvia Volksdorf; Joseph L Duffy
Analgesic effects of a substituted N-triazole oxindole (TROX-1), a state-dependent, voltage-gated calcium channel 2 blocker.
The Journal of pharmacology and experimental therapeutics 2010;334(2):545-55.
2008: Cheng Zhu; Alexa R Hansen; Thomas Bateman; Zhesheng Chen; Tom Holt; James A Hubert; Bindhu V Karanam; Susan J Lee; Jie Pan; Su Qian; Vijay B G Reddy; Marc L Reitman; Alison M Strack; Vincent Tong; Drew T Weingarth; Michael S Wolff; Douglas J MacNeil; Ann E Weber; Joseph L Duffy; Scott D Edmondson
Discovery of imidazole carboxamides as potent and selective CCK1R agonists.
Bioorganic & medicinal chemistry letters 2008;18(15):4393-6.
2008: Clare London; Scott B Hoyt; William H Parsons; Brande S Williams; Vivien A Warren; Richard A Tschirret-Guth; McHardy Smith; Birgit T Priest; Erin McGowan; William J Martin; Kathryn A Lyons; Xiaohua Li; Bindhu V Karanam; Nina Jochnowitz; Maria L Garcia; John P Felix; Brian Dean; Catherine Abbadie; Gregory J Kaczorowski; Joseph L Duffy
Imidazopyridines: a novel class of hNav1.7 channel blockers.
Bioorganic & medicinal chemistry letters 2008;18(5):1696-701.
2007: Brande S Williams; John P Felix; Birgit T Priest; Richard Brochu; Kefei Dai; Scott B Hoyt; Clare London; Yui S Tang; Joseph L Duffy; William H Parsons; Gregory J Kaczorowski; Maria L Garcia
Characterization of a new class of potent inhibitors of the voltage-gated sodium channel Nav1.7.
Biochemistry 2007;46(50):14693-703.
2007: Scott B Hoyt; Clare London; Hyun O Ok; Edward Gonzalez; Joseph L Duffy; Catherine Abbadie; Brian Dean; John P Felix; Maria L Garcia; Nina Jochnowitz; Bindhu V Karanam; Xiaohua Li; Kathryn A Lyons; Erin McGowan; D Euan MacIntyre; William J Martin; Birgit T Priest; McHardy Smith; Richard A Tschirret-Guth; Vivien A Warren; Brande S Williams; Gregory J Kaczorowski; William H Parsons
Benzazepinone Nav1.7 blockers: potential treatments for neuropathic pain.
Bioorganic & medicinal chemistry letters 2007;17(22):6172-7.
2007: David E Kaelin; Abigail L Smenton; George J Eiermann; Huaibing He; Barbara Leiting; Kathryn A Lyons; Reshma A Patel; Sangita B Patel; Aleksandr Petrov; Giovanna Scapin; Joseph K Wu; Nancy A Thornberry; Ann E Weber; Joseph L Duffy
4-arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV.
Bioorganic & medicinal chemistry letters 2007;17(21):5806-11.
2007: Joseph L Duffy; Brian A Kirk; Liping Wang; George J Eiermann; Huaibing He; Barbara Leiting; Kathryn A Lyons; Reshma A Patel; Sangita B Patel; Aleksandr Petrov; Giovanna Scapin; Joseph K Wu; Nancy A Thornberry; Ann E Weber
4-aminophenylalanine and 4-aminocyclohexylalanine derivatives as potent, selective, and orally bioavailable inhibitors of dipeptidyl peptidase IV.
Bioorganic & medicinal chemistry letters 2007;17(10):2879-85.
2006: Sheila M Cohen; Joseph L Duffy; Corin Miller; Brian A Kirk; Mari Rios Candelore; Victor D H Ding; Gregory Kaczorowski; Laurie M Tota; Jeffrey G Werrmann; Michael Wright; Emma R Parmee; James R Tata; Bei B Zhang
Direct observation (NMR) of the efficacy of glucagon receptor antagonists in murine liver expressing the human glucagon receptor.
Bioorganic & medicinal chemistry 2006;14(5):1506-17.
2005: Scott D Edmondson; Anthony Mastracchio; Joseph L Duffy; George J Eiermann; Huaibing He; Ida Ita; Barbara Leiting; Joseph F Leone; Kathryn A Lyons; Amanda M Makarewicz; Reshma A Patel; Aleksandr Petrov; Joseph K Wu; Nancy A Thornberry; Ann E Weber
Discovery of potent and selective orally bioavailable beta-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors.
Bioorganic & medicinal chemistry letters 2005;15(12):3048-52.
2005: Joseph L Duffy; Brian A Kirk; Zenon Konteatis; Elizabeth L Campbell; Rui Liang; Edward J Brady; Mari Rios Candelore; Victor D H Ding; Guoqiang Jiang; Frank Liu; Sajjad A Qureshi; Richard Saperstein; Deborah Szalkowski; Sharon Tong; Laurie M Tota; Dan Xie; Xiaodong Yang; Peter Zafian; Song Zheng; Kevin Chapman; Bei B Zhang; James R Tata
Discovery and investigation of a novel class of thiophene-derived antagonists of the human glucagon receptor.
Bioorganic & medicinal chemistry letters 2005;15(5):1401-5.
2004: Sajjad A Qureshi; Mari Rios Candelore; Dan Xie; Xiaodong Yang; Laurie M Tota; Victor D H Ding; Zhihua Li; Alka Bansal; Corin Miller; Sheila M Cohen; Guoqiang Jiang; Edward J Brady; Richard Saperstein; Joseph L Duffy; James R Tata; Kevin Chapman; David E Moller; Bei B Zhang
A novel glucagon receptor antagonist inhibits glucagon-mediated biological effects.
Diabetes 2004;53(12):3267-73.
2003: Nancy J Kevin; Joseph L Duffy; Brian A Kirk; Kevin Chapman; William A Schleif; David B Olsen; Mark Stahlhut; Carrie A Rutkowski; Lawrence C Kuo; Lixia Jin; Jiunn H Lin; Emilio A Emini; James R Tata
Novel HIV-1 protease inhibitors active against multiple PI-resistant viral strains: coadministration with indinavir.
Bioorganic & medicinal chemistry letters 2003;13(22):4027-30.
2003: Joseph L Duffy; Brian A Kirk; Nancy J Kevin; Kevin Chapman; William A Schleif; David B Olsen; Mark Stahlhut; Carrie A Rutkowski; Lawrence C Kuo; Lixia Jin; Jiunn H Lin; Emilio A Emini; James R Tata
HIV-1 protease inhibitors with picomolar potency against PI-resistant HIV-1 by modification of the P1' substituent.
Bioorganic & medicinal chemistry letters 2003;13(19):3323-6.
2003: Joseph L Duffy; Thomas A Rano; Nancy J Kevin; Kevin Chapman; William A Schleif; David B Olsen; Mark Stahlhut; Carrie A Rutkowski; Lawrence C Kuo; Lixia Jin; Jiunn H Lin; Emilio A Emini; James R Tata
HIV protease inhibitors with picomolar potency against PI-Resistant HIV-1 by extension of the P3 substituent.
Bioorganic & medicinal chemistry letters 2003;13(15):2569-72.
2002: Joseph L Duffy; Nancy J Kevin; Brian A Kirk; Kevin Chapman; William A Schleif; David B Olsen; Mark Stahlhut; Carrie A Rutkowski; Lawrence C Kuo; Lixia Jin; Jiunn H Lin; Emilio A Emini; James R Tata
Synthesis and activity of novel HIV protease inhibitors with improved potency against multiple PI-resistant viral strains.
Bioorganic & medicinal chemistry letters 2002;12(17):2423-6.