FIND

researchers

DISCOVER

relevant articles

PROMOTE

your research

now for free

Amaury Farce

Research Profile

Concepts & Ideas

Anatomy

Tumor Cell Line

Genes & Molecular Sequences

Occupations

Drug Design

Chemicals & Drugs

Co-author Network

Publications

TOP 3
Alina Ghinet; Marie Leman; Benoît Rigo; Vivien Stocker; Aurélien Tourteau; Joëlle Dubois; Amaury Farce; Philippe Gautret
Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin.
Nicolas Renault; Pierre Desreumaux; Jamal El Bakali; Amaury Farce; Christophe Furman; Philippe Gervois; Xavier Laurent; Roxane Mansouri; Régis Millet; Philippe CHAVATTE
Virtual screening of CB(2) receptor agonists from bayesian network and high-throughput docking: structural insights into agonist-modulated GPCR features.
Cristina-Maria Abuhaie; Dalila Belei; Joëlle Dubois; Amaury Farce; Philippe Gautret; Alina Ghinet; Benoît Rigo; Elena Bîcu
Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors.

Register for free to view:

Visualized networks:

See your personal network in
sophisticated graphical views

GeoTargeted Searches:

Locate experts around the world
and connect with global collaborators

Research Profiles:

See the research activity
of experts around the globe

Geonetwork of Amaury Farce (preview)

Cities where this author has publications
Cities where co-authors of this author have publications

Flash Player Required

All Publications

2013: Alina Ghinet; Marie Leman; Benoît Rigo; Vivien Stocker; Aurélien Tourteau; Joëlle Dubois; Amaury Farce; Philippe Gautret
Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin.
Bioorganic & medicinal chemistry 2013;21(11):2932-40.
2013: Nicolas Renault; Pierre Desreumaux; Jamal El Bakali; Amaury Farce; Christophe Furman; Philippe Gervois; Xavier Laurent; Roxane Mansouri; Régis Millet; Philippe CHAVATTE
Virtual screening of CB(2) receptor agonists from bayesian network and high-throughput docking: structural insights into agonist-modulated GPCR features.
Chemical biology & drug design 2013;81(4):442-54.
2013: Cristina-Maria Abuhaie; Dalila Belei; Joëlle Dubois; Amaury Farce; Philippe Gautret; Alina Ghinet; Benoît Rigo; Elena Bîcu
Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors.
European journal of medicinal chemistry 2013;59():101-10.
2013: Valérie Verones; Nicole Wattez; Marie Lecoeur; Amelie Lemoine; Christine Mahieu; Brigitte Baldeyrou; Pascal Berthelot; Amaury Farce; Nathalie Flouquet; Jean-François Goossens; Amélie Lansiaux; Nicolas Lebegue
Synthesis, antiproliferative activity and tubulin targeting effect of acridinone and dioxophenothiazine derivatives.
European journal of medicinal chemistry 2013;59():39-47.
2013: Cristina-Maria Abuhaie; Dalila Belei; Elena Bîcu; Joëlle Dubois; Amaury Farce; Philippe Gautret; Benoît Rigo; Alina Ghinet
Synthesis and anticancer activity of analogues of phenstatin, with a phenothiazine A-ring, as a new class of microtubule-targeting agents.
Bioorganic & medicinal chemistry letters 2013;23(1):147-52.
2012: Morgan Le Naour; Véronique Leclerc; Michel Lonchampt; Bart Staels; Valérie Audinot-Bouchez; Pascal Berthelot; Jean-Albert Boutin; Daniel-Henri Caignard; Catherine Dacquet; Amaury Farce; Nathalie Hennuyer; Alain Ktorza; Nicolas Lebegue
Effect of oxime ether incorporation in acyl indole derivatives on PPAR subtype selectivity.
ChemMedChem 2012;7(12):2179-93.
2012: Lavinia Baciu-Atudosie; Dalila Belei; Joëlle Dubois; Amaury Farce; Alina Ghinet; Elena Bîcu
Synthesis and biological evaluation of new phenothiazine derivatives bearing a pyrazole unit as protein farnesyltransferase inhibitors.
Bioorganic & medicinal chemistry letters 2012;22(22):6896-902.
2012: Alina Ghinet; Jean-Pierre Henichart; Souhila Oudir; Jean Pommery; Benoît Rigo; Joseph Vamecq; Amaury Farce; Philippe Gautret
Antioxidant activity of new benzo[de]quinolines and lactams: 2D-quantitative structure-activity relationships.
Medicinal chemistry (Shāriqah (United Arab Emirates)) 2012;8(5):942-6.
2012: Dalila Belei; Elena Bîcu; Joëlle Dubois; Carmen Dumea; Amaury Farce; Alexandrina Samson; Alina Ghinet
New farnesyltransferase inhibitors in the phenothiazine series.
Bioorganic & medicinal chemistry letters 2012;22(14):4517-22.
2012: Céline Pirat; Nicolas Renault; Silvia Speca; Saïd Yous; Pierre Desreumaux; Amaury Farce; Christophe Furman; Nicolas Lebègue; Régis Millet; Pascal Berthelot; Philippe CHAVATTE
Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.
Journal of medicinal chemistry 2012;55(9):4027-61.
2012: Antonio Garofalo; Laurence Goossens; Amélie Lemoine; Séverine Ravez; Perrine Six; Philippe CHAVATTE; Amaury Farce; Patrick Depreux
Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitors.
Journal of medicinal chemistry 2012;55(3):1189-204.
2011: christian lacks lino cardenas; Jean-Marc Lo-Guidice; Nicolas Renault; Amaury Farce; Michel Lhermitte; Delphine Allorge; Franck Broly; Christelle Cauffiez; Philippe CHAVATTE; Dany Chevalier
Genetic polymorphism of CYP4A11 and CYP4A22 genes and in silico insights from comparative 3D modelling in a French population.
Gene 2011;487(1):10-20.
2011: Delphine Le Broc-Ryckewaert; Jean Pommery; Nicole Pommery; Benoît Rigo; Jean-François Wiart; Amaury Farce; Philippe Gautret; Alina Ghinet; Jean-Pierre Hénichart
In vitro metabolism of phenstatin: potential pharmacological consequences.
Drug metabolism letters 2011;5(3):209-15.
2011: Véronique Leclerc; Mohamed Ettaoussi; Marouan Rami; Amaury Farce; Jean A Boutin; Philippe Delagrange; Daniel-Henri Caignard; Pierre Renard; Pascal Berthelot; Saïd Yous
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3.
European journal of medicinal chemistry 2011;46(5):1622-9.
2011: Antonio Garofalo; Laurence Goossens; Perrine Six; Amélie Lemoine; Séverine Ravez; Amaury Farce; Patrick Depreux
Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors.
Bioorganic & medicinal chemistry letters 2011;21(7):2106-12.
2011: Nicolas Wlodarczyk; Delphine Le Broc-Ryckewaert; Pauline Gilleron; Amélie Lemoine; Amaury Farce; Philippe CHAVATTE; Joëlle Dubois; Nicole Pommery; Jean-Pierre Hénichart; Christophe Furman; Régis Millet
Potent farnesyltransferase inhibitors with 1,4-diazepane scaffolds as novel destabilizing microtubule agents in hormone-resistant prostate cancer.
Journal of medicinal chemistry 2011;54(5):1178-90.
2010: Valerie Verones; Nathalie Flouquet; Amaury Farce; Pascal Carato; stephane leonce; Bruno Pfeiffer; Pascal Berthelot; Nicolas Lebegue
Synthesis, biological evaluation and docking studies of 4-amino-tetrahydroquinazolino[3,2-e]purine derivatives.
European journal of medicinal chemistry 2010;45(12):5678-84.
2010: Nicolas Renault; Arnaud Gohier; Philippe CHAVATTE; Amaury Farce
Novel structural insights for drug design of selective 5-HT(2C) inverse agonists from a ligand-biased receptor model.
European journal of medicinal chemistry 2010;45(11):5086-99.
2010: Antonio Garofalo; Laurence Goossens; Amelie Lemoine; Amaury Farce; Yannick Arlot; Patrick Depreux
Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancer.
Journal of enzyme inhibition and medicinal chemistry 2010;25(2):158-71.
2009: Jamal El Bakali; Frédérique Klupsch; Aurore Guédin; Bertrand BRASSART; Gaëlle Fontaine; Amaury Farce; Pascal Roussel; Raymond Houssin; Jean-Luc Bernier; Philippe CHAVATTE; Jean-Louis Mergny; Jean-François Riou; Jean-Pierre Hénichart
2,6-Diphenylthiazolo[3,2-b][1,2,4]triazoles as telomeric G-quadruplex stabilizers.
Bioorganic & medicinal chemistry letters 2009;19(13):3434-8.
2009: Amaury Farce; N Renault; P Chavatte
Structural insight into PPARgamma ligands binding.
Current medicinal chemistry 2009;16(14):1768-89.
2008: Nicolas Kambia; Nicolas Renault; Sebastien Dilly; Amaury Farce; Thierry Dine; Bernard Gressier; Michel Luyckx; Claude Brunet; Philippe CHAVATTE
Molecular modelling of phthalates - PPARs interactions.
Journal of enzyme inhibition and medicinal chemistry 2008;23(5):611-6.
2008: Amaury Farce; Anton O Chugunov; Cédric Logé; Ahmed Sabaouni; Saïd Yous; Sebastien Dilly; Nicolas Renault; Gérard Vergoten; Roman G Efremov; Daniel Lesieur; Philippe CHAVATTE
Homology modeling of MT1 and MT2 receptors.
European journal of medicinal chemistry 2008;43(9):1926-44.
2007: Amaury Graulich; Sebastien Dilly; Amaury Farce; Jacqueline Scuvée-Moreau; Olivier Waroux; Cédric Lamy; Philippe CHAVATTE; Vincent Seutin; Jean-François Liégeois
Synthesis and radioligand binding studies of bis-isoquinolinium derivatives as small conductance Ca(2+)-activated K(+) channel blockers.
Journal of medicinal chemistry 2007;50(21):5070-5.
2007: Anne-Catherine Durand; Amaury Farce; Pascal Carato; Sebastien Dilly; Saïd Yous; Pascal Berthelot; Philippe CHAVATTE
Quantitative structure-activity relationships studies of antioxidant hexahydropyridoindoles and flavonoid derivatives.
Journal of enzyme inhibition and medicinal chemistry 2007;22(5):556-62.
2007: Pauline Gilleron; Nicolas Wlodarczyk; Raymond Houssin; Amaury Farce; Guillaume Laconde; Jean-François Goossens; Amélie Lemoine; Nicole Pommery; Jean-Pierre Hénichart; Régis Millet
Design, synthesis and biological evaluation of substituted dioxodibenzothiazepines and dibenzocycloheptanes as farnesyltransferase inhibitors.
Bioorganic & medicinal chemistry letters 2007;17(19):5465-71.
2007: Aurélie Telliez; Matthieu Desroses; Nicole Pommery; Olivier Briand; Amaury Farce; Guillaume Laconde; Amélie Lemoine; Patrick Depreux; Jean-Pierre Hénichart
Derivatives of Iressa, a specific epidermal growth factor receptor inhibitor, are powerful apoptosis inducers in PC3 prostatic cancer cells.
ChemMedChem 2007;2(3):318-32.
2006: Elodie Blanc-Delmas; Nicolas Lebegue; Valérie Wallez; Véronique Leclerc; Saïd Yous; Pascal Carato; Amaury Farce; Caroline Bennejean; Pierre Renard; Daniel-Henri Caignard; Valérie Audinot-Bouchez; Pascale Chomarat; Jean Boutin; Nathalie Hennuyer; Katie Louche; MARI CARMEN CARMONA; Bart Staels; Luc Pénicaud; Louis Casteilla; Michel Lonchampt; Catherine Dacquet; Philippe CHAVATTE; Pascal Berthelot; Daniel Lesieur
Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARgamma agonists.
Bioorganic & medicinal chemistry 2006;14(22):7377-91.
2006: Anton O Chugunov; Amaury Farce; Philippe CHAVATTE; Roman G Efremov
Differences in binding sites of two melatonin receptors help to explain their selectivity to some melatonin analogs: a molecular modeling study.
Journal of biomolecular structure & dynamics 2006;24(2):91-107.
2006: Amaury Farce; Sebastien Dilly; Saïd Yous; Pascal Berthelot; Philippe CHAVATTE
Homology modelling of the serotoninergic 5-HT2c receptor.
Journal of enzyme inhibition and medicinal chemistry 2006;21(3):285-92.
2006: Pauline Gilleron; Régis Millet; Raymond Houssin; Nicolas Wlodarczyk; Amaury Farce; Amélie Lemoine; Jean-François Goossens; Philippe CHAVATTE; Nicole Pommery; Jean-Pierre Hénichart
Solid-phase synthesis and pharmacological evaluation of a library of peptidomimetics as potential farnesyltransferase inhibitors: an approach to new lead compounds.
European journal of medicinal chemistry 2006;41(6):745-55.
2006: Philippe CHAVATTE; Amaury Farce
A computational view of COX-2 inhibition.
Anti-cancer agents in medicinal chemistry 2006;6(3):239-49.
2006: Pauline Gilleron; Régis Millet; Juozas Domarkas; Amaury Farce; Raymond Houssin; Jean-Pierre Hénichart
Synthesis of a novel conformationally restricted Val-Phe dipeptidomimetic.
Journal of peptide science : an official publication of the European Peptide Society 2006;12(2):140-6.
2006: Eric Stern; Giulio G Muccioli; Régis Millet; Jean-François Goossens; Amaury Farce; Philippe CHAVATTE; Jacques H Poupaert; Didier M Lambert; Patrick Depreux; Jean-Pierre Hénichart
Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling.
Journal of medicinal chemistry 2006;49(1):70-9.
2005: Sebastien Dilly; Amaury Graulich; Amaury Farce; Vincent Seutin; Jean-Francois Liegeois; Philippe CHAVATTE
Identification of a pharmacophore of SKCa channel blockers.
Journal of enzyme inhibition and medicinal chemistry 2005;20(6):517-23.
2005: Christel Rousseaux; Bruno Lefebvre; Laurent Dubuquoy; Philippe Lefebvre; Olivier Romano; Johan Auwerx; Daniel Metzger; Walter Wahli; Béatrice Desvergne; Gian Carlo Naccari; Philippe CHAVATTE; Amaury Farce; Philippe Bulois; Antoine Cortot; Jean-Frédéric Colombel; Pierre Desreumaux
Intestinal antiinflammatory effect of 5-aminosalicylic acid is dependent on peroxisome proliferator-activated receptor-gamma.
The Journal of experimental medicine 2005;201(8):1205-15.
2004: Amaury Farce; Cedric Loge; Sebastien Gallet; Nicolas Lebegue; Pascal Carato; Philippe CHAVATTE; Pascal Berthelot; Daniel Lesieur
Docking study of ligands into the colchicine binding site of tubulin.
Journal of enzyme inhibition and medicinal chemistry 2004;19(6):541-7.