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Vincenza Andrisano
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49
Cavrini, Vanni
35
Bartolini, Manuela
26
Gotti, Roberto
23
Cavalli, Andrea
22
Melchiorre, Carlo
22
Recanatini, Maurizio
16
Rosini, Michela
16
Bolognesi, Maria Laura
14
Bertucci, Carlo
12
Tumiatti, Vincenzo
11
Rampa, Angela
11
Minarini, Anna
10
Fiori, Jessica
10
Mancini, Francesca
9
Bisi, Alessandra
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All Publications
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2009: Camps Pelayo; Formosa Xavier; Galdeano Carles; Muñoz-Torrero Diego; Ramírez Lorena; Gómez Elena; Isambert Nicolás; Lavilla Rodolfo; Badia Albert; Clos M Victòria; Bartolini Manuela; Mancini Francesca; Andrisano Vincenza; Arce Mariana P; Rodríguez-Franco M Isabel; Huertas Oscar; Dafni Thomai; Luque F Javier
Pyrano[3,2-c]quinoline-6-chlorotacrine hybrids as a novel family of acetylcholinesterase- and beta-amyloid-directed anti-Alzheimer compounds.
Journal of medicinal chemistry 2009;52(17):5365-79.
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2009: Mancini Francesca; Bolognesi Maria Laura; Melchiorre Carlo; Andrisano Vincenza
Investigation of the photostability properties of memoquin, a quinone derivative for the treatment of Alzheimer's disease.
Journal of pharmaceutical and biomedical analysis 2009;50(2):164-70.
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2009: Bolognesi Maria Laura; Bartolini Manuela; Rosini Michela; Andrisano Vincenza; Melchiorre Carlo
Structure-activity relationships of memoquin: Influence of the chain chirality in the multi-target mechanism of action.
Bioorganic & medicinal chemistry letters 2009;19(15):4312-5.
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2009: Rizzo Stefano; Cavalli Andrea; Ceccarini Luisa; Bartolini Manuela; Belluti Federica; Bisi Alessandra; Andrisano Vincenza; Recanatini Maurizio; Rampa Angela
Structure-activity relationships and binding mode in the human acetylcholinesterase active site of pseudo-irreversible inhibitors related to xanthostigmine.
ChemMedChem 2009;4(4):670-9.
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2009: Bartolini Manuela; Greig Nigel H; Yu Qian-Sheng; Andrisano Vincenza
Immobilized butyrylcholinesterase in the characterization of new inhibitors that could ease Alzheimer's disease.
Journal of chromatography. A 2009;1216(13):2730-8.
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2009: Bolognesi M L; Rosini M; Andrisano V; Bartolini M; Minarini A; Tumiatti V; Melchiorre C
MTDL design strategy in the context of Alzheimer's disease: from lipocrine to memoquin and beyond.
Current pharmaceutical design 2009;15(6):601-13.
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2008: Tumiatti Vincenzo; Milelli Andrea; Minarini Anna; Rosini Michela; Bolognesi Maria Laura; Micco Marialuisa; Andrisano Vincenza; Bartolini Manuela; Mancini Francesca; Recanatini Maurizio; Cavalli Andrea; Melchiorre Carlo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 4. Further investigation on the inner spacer.
Journal of medicinal chemistry 2008;51(22):7308-12.
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2008: Rosini Michela; Simoni Elena; Bartolini Manuela; Cavalli Andrea; Ceccarini Luisa; Pascu Nicoleta; McClymont David W; Tarozzi Andrea; Bolognesi Maria L; Minarini Anna; Tumiatti Vincenzo; Andrisano Vincenza; Mellor Ian R; Melchiorre Carlo
Inhibition of acetylcholinesterase, beta-amyloid aggregation, and NMDA receptors in Alzheimer's disease: a promising direction for the multi-target-directed ligands gold rush.
Journal of medicinal chemistry 2008;51(15):4381-4.
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2008: Camps Pelayo; Formosa Xavier; Galdeano Carles; Gómez Tània; Muñoz-Torrero Diego; Scarpellini Michele; Viayna Elisabet; Badia Albert; Clos M Victòria; Camins Antoni; Pallàs Mercè; Bartolini Manuela; Mancini Francesca; Andrisano Vincenza; Estelrich Joan; Lizondo Mònica; Bidon-Chanal Axel; Luque F Javier
Novel donepezil-based inhibitors of acetyl- and butyrylcholinesterase and acetylcholinesterase-induced beta-amyloid aggregation.
Journal of medicinal chemistry 2008;51(12):3588-98.
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2008: Rizzo Stefano; Rivière Céline; Piazzi Lorna; Bisi Alessandra; Gobbi Silvia; Bartolini Manuela; Andrisano Vincenza; Morroni Fabiana; Tarozzi Andrea; Monti Jean-Pierre; Rampa Angela
Benzofuran-based hybrid compounds for the inhibition of cholinesterase activity, beta amyloid aggregation, and abeta neurotoxicity.
Journal of medicinal chemistry 2008;51(10):2883-6.
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2008: Olmo Stefano; Gotti Roberto; Naldi Marina; Andrisano Vincenza; Calonghi Natalia; Parolin Carola; Masotti Lanfranco; Cavrini Vanni
Analysis of human histone H4 by capillary electrophoresis in a pullulan-coated capillary, LC-ESI-MS and MALDI-TOF-MS.
Analytical and bioanalytical chemistry 2008;390(7):1881-8.
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2008: Petraglio Gabriele; Bartolini Manuela; Branduardi Davide; Andrisano Vincenza; Recanatini Maurizio; Gervasio Francesco Luigi; Cavalli Andrea; Parrinello Michele
The role of Li+, Na+, and K+ in the ligand binding inside the human acetylcholinesterase gorge.
Proteins 2008;70(3):779-85.
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2008: Piazzi Lorna; Cavalli Andrea; Colizzi Francesco; Belluti Federica; Bartolini Manuela; Mancini Francesca; Recanatini Maurizio; Andrisano Vincenza; Rampa Angela
Multi-target-directed coumarin derivatives: hAChE and BACE1 inhibitors as potential anti-Alzheimer compounds.
Bioorganic & medicinal chemistry letters 2008;18(1):423-6.
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2007: Bolognesi Maria Laura; Cavalli Andrea; Valgimigli Luca; Bartolini Manuela; Rosini Michela; Andrisano Vincenza; Recanatini Maurizio; Melchiorre Carlo
Multi-target-directed drug design strategy: from a dual binding site acetylcholinesterase inhibitor to a trifunctional compound against Alzheimer's disease.
Journal of medicinal chemistry 2007;50(26):6446-9.
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2007: Mancini Francesca; Naldi Marina; Cavrini Vanni; Andrisano Vincenza
Development and characterization of beta-secretase monolithic micro-immobilized enzyme reactor for on-line high-performance liquid chromatography studies.
Journal of chromatography. A 2007;1175(2):217-26.
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2007: Mancini Francesca; Bolognesi Maria L; Melchiorre Carlo; Cavalli Andrea; Andrisano Vincenza
Monolithic stationary phase coupled with coulometric detection: development of an ion-pair HPLC method for the analysis of quinone-bearing compounds.
Journal of separation science 2007;30(17):2935-42.
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2007: Bartolini Manuela; Bertucci Carlo; Bolognesi Maria Laura; Cavalli Andrea; Melchiorre Carlo; Andrisano Vincenza
Insight into the kinetic of amyloid beta (1-42) peptide self-aggregation: elucidation of inhibitors' mechanism of action.
Chembiochem : a European journal of chemical biology 2007;8(17):2152-61.
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2007: Bolognesi Maria Laura; Banzi Rita; Bartolini Manuela; Cavalli Andrea; Tarozzi Andrea; Andrisano Vincenza; Minarini Anna; Rosini Michela; Tumiatti Vincenzo; Bergamini Christian; Fato Romana; Lenaz Giorgio; Hrelia Patrizia; Cattaneo Antonino; Recanatini Maurizio; Melchiorre Carlo
Novel class of quinone-bearing polyamines as multi-target-directed ligands to combat Alzheimer's disease.
Journal of medicinal chemistry 2007;50(20):4882-97.
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2007: Piazzi Lorna; Cavalli Andrea; Belluti Federica; Bisi Alessandra; Gobbi Silvia; Rizzo Stefano; Bartolini Manuela; Andrisano Vincenza; Recanatini Maurizio; Rampa Angela
Extensive SAR and computational studies of 3-{4-[(benzylmethylamino)methyl]phenyl}-6,7-dimethoxy-2H-2-chromenone (AP2238) derivatives.
Journal of medicinal chemistry 2007;50(17):4250-4.
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2007: Mancini Francesca; Naldi Marina; Cavrini Vanni; Andrisano Vincenza
Multiwell fluorometric and colorimetric microassays for the evaluation of beta-secretase (BACE-1) inhibitors.
Analytical and bioanalytical chemistry 2007;388(5-6):1175-83.
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2007: Bartolini Manuela; Cavrini Vanni; Andrisano Vincenza
Characterization of reversible and pseudo-irreversible acetylcholinesterase inhibitors by means of an immobilized enzyme reactor.
Journal of chromatography. A 2007;1144(1):102-10.
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2007: Piazzi Lorna; Belluti Federica; Bisi Alessandra; Gobbi Silvia; Rizzo Stefano; Bartolini Manuela; Andrisano Vincenza; Recanatini Maurizio; Rampa Angela
Cholinesterase inhibitors: SAR and enzyme inhibitory activity of 3-[omega-(benzylmethylamino)alkoxy]xanthen-9-ones.
Bioorganic & medicinal chemistry 2007;15(1):575-85.
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2007: Cavalli Andrea; Bolognesi Maria Laura; Capsoni Simona; Andrisano Vincenza; Bartolini Manuela; Margotti Elisa; Cattaneo Antonino; Recanatini Maurizio; Melchiorre Carlo
A small molecule targeting the multifactorial nature of Alzheimer's disease.
Angewandte Chemie (International ed. in English) 2007;46(20):3689-92.
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2006: Rosini Michela; Mancini Francesca; Tarozzi Andrea; Colizzi Francesco; Andrisano Vincenza; Bolognesi Maria L; Hrelia Patrizia; Melchiorre Carlo
Design, synthesis, and biological evaluation of substituted 2,3-dihydro-1H-cyclopenta[b]quinolin-9-ylamine related compounds as fructose-1,6-bisphosphatase inhibitors.
Bioorganic & medicinal chemistry 2006;14(23):7846-53.
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2006: Mancini Francesca; Fiori Jessica; Cavrini Vanni; Andrisano Vincenza
Separation and quantitation of fructose-6-phosphate and fructose-1 ,6-diphosphate by LC-ESI-MS for the evaluation of fructose-1,6-biphosphatase activity.
Journal of separation science 2006;29(15):2395-400.
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2006: Naldi M; Andrisano V; Fiori J; Calonghi N; Pagnotta E; Parolin C; Pieraccini G; Masotti L
Histone proteins determined in a human colon cancer by high-performance liquid chromatography and mass spectrometry.
Journal of chromatography. A 2006;1129(1):73-81.
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2006: Temporini C; Perani E; Mancini F; Bartolini M; Calleri E; Lubda D; Felix G; Andrisano V; Massolini G
Optimization of a trypsin-bioreactor coupled with high-performance liquid chromatography-electrospray ionization tandem mass spectrometry for quality control of biotechnological drugs.
Journal of chromatography. A 2006;1120(1-2):121-31.
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2005: Fiori J; Bragieri M; Zanotti M C; Liverani A; Borzatta V; Mancini F; Cavrini V; Andrisano V
Liquid chromatography-tandem mass spectrometry for the identification of impurities in d-allethrin samples.
Journal of chromatography. A 2005;1099(1-2):149-56.
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2005: Muñoz-Ruiz Pilar; Rubio Laura; García-Palomero Esther; Dorronsoro Isabel; del Monte-Millán María; Valenzuela Rita; Usán Paola; de Austria Celia; Bartolini Manuela; Andrisano Vincenza; Bidon-Chanal Axel; Orozco Modesto; Luque F Javier; Medina Miguel; Martínez Ana
Design, synthesis, and biological evaluation of dual binding site acetylcholinesterase inhibitors: new disease-modifying agents for Alzheimer's disease.
Journal of medicinal chemistry 2005;48(23):7223-33.
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2005: Bartolini M; Cavrini V; Andrisano V
Batchwise covalent immobilization of human acetylcholinesterase: kinetic and inhibition spectrophotometric studies.
Analytical biochemistry 2005;342(1):163-6.
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2005: Belluti Federica; Rampa Angela; Piazzi Lorna; Bisi Alessandra; Gobbi Silvia; Bartolini Manuela; Andrisano Vincenza; Cavalli Andrea; Recanatini Maurizio; Valenti Piero
Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation.
Journal of medicinal chemistry 2005;48(13):4444-56.
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2005: Bolognesi Maria Laura; Andrisano Vincenza; Bartolini Manuela; Cavalli Andrea; Minarini Anna; Recanatini Maurizio; Rosini Michela; Tumiatti Vincenzo; Melchiorre Carlo
Heterocyclic inhibitors of AChE acylation and peripheral sites.
Farmaco (Società chimica italiana : 1989) 2005;60(6-7):465-73.
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2005: Tarozzi Andrea; Marchesi Alessandra; Hrelia Silvana; Angeloni Cristina; Andrisano Vincenza; Fiori Jessica; Cantelli-Forti Giorgio; Hrelia Patrizia
Protective effects of cyanidin-3-O-beta-glucopyranoside against UVA-induced oxidative stress in human keratinocytes.
Photochemistry and photobiology 2005;81(3):623-9.
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2005: Abd El-Hady Deia; Gotti Roberto; Abo El-Maali Nagwa; Andrisano Vincenza
Simultaneous separation and determination of Tarabine PFS and Adriblastine using micellar electrokinetic chromatography and high performance liquid chromatography. Application to some biological fluids.
Journal of separation science 2005;28(6):534-42.
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2005: el-Hady D Abd; el-Maali N Abo; Gotti R; Bertucci C; Mancini F; Andrisano V
Methotrexate determination in pharmaceuticals by enantioselective HPLC.
Journal of pharmaceutical and biomedical analysis 2005;37(5):919-25.
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2005: El-Hady Deia Abd; El-Maali Nagwa Abo; Gotti Roberto; Andrisano Vincenza
Simultaneous micellar electrokinetic chromatography and liquid chromatography of adriblastina and tarabine PFS Their application to some biological fluids.
Talanta 2005;66(1):253-60.
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2005: Luppi B; Bigucci F; Cerchiara T; Andrisano V; Pucci V; Mandrioli R; Zecchi V
Micelles based on polyvinyl alcohol substituted with oleic acid for targeting of lipophilic drugs.
Drug delivery 2005;12(1):21-6.
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2005: Rosini Michela; Andrisano Vincenza; Bartolini Manuela; Bolognesi Maria L; Hrelia Patrizia; Minarini Anna; Tarozzi Andrea; Melchiorre Carlo
Rational approach to discover multipotent anti-Alzheimer drugs.
Journal of medicinal chemistry 2005;48(2):360-3.
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2005: Bolognesi Maria Laura; Andrisano Vincenza; Bartolini Manuela; Banzi Rita; Melchiorre Carlo
Propidium-based polyamine ligands as potent inhibitors of acetylcholinesterase and acetylcholinesterase-induced amyloid-beta aggregation.
Journal of medicinal chemistry 2005;48(1):24-7.
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2004: Tumiatti Vincenzo; Andrisano Vincenza; Banzi Rita; Bartolini Manuela; Minarini Anna; Rosini Michela; Melchiorre Carlo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties.
Journal of medicinal chemistry 2004;47(26):6490-8.
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2004: Bolognesi Maria Laura; Bartolini Manuela; Cavalli Andrea; Andrisano Vincenza; Rosini Michela; Minarini Anna; Melchiorre Carlo
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues.
Journal of medicinal chemistry 2004;47(24):5945-52.
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2004: Mancini F; Fiori J; Bertucci C; Cavrini V; Bragieri M; Zanotti M C; Liverani A; Borzatta V; Andrisano V
Stereoselective determination of allethrin by two-dimensional achiral/chiral liquid chromatography with ultraviolet/circular dichroism detection.
Journal of chromatography. A 2004;1046(1-2):67-73.
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2004: Gotti Roberto; El-Hady Deia Abd; Andrisano Vincenza; Bertucci Carlo; El-Maali Nagwa Abo; Cavrini Vanni
Determination of the chiral and achiral related substances of methotrexate by cyclodextrin-modified micellar electrokinetic chromatography.
Electrophoresis 2004;25(16):2830-7.
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2004: Bartolini M; Cavrini V; Andrisano V
Monolithic micro-immobilized-enzyme reactor with human recombinant acetylcholinesterase for on-line inhibition studies.
Journal of chromatography. A 2004;1031(1-2):27-34.
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2004: Abd El-Hady D; Abdel-Hamid M I; Seliem M M; Andrisano V; Abo El-Maali N
Osteryoung square wave stripping voltammetry at mercury film electrode for monitoring ultra trace levels of Tarabine PFS and its interaction with ssDNA.
Journal of pharmaceutical and biomedical analysis 2004;34(5):879-90.
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2004: Bragieri Matteo; Liverani Alessandra; Zanotti Maria Cristina; Borzatta Valerio; Fiori Jessica; Cavrini Vanni; Andrisano Vincenza
GC-FID/MS method for the impurity profiling of synthetic d-allethrin.
Journal of separation science 2004;27(1-2):89-95.
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2003: Bertucci C; Bartolini M; Gotti R; Andrisano V
Drug affinity to immobilized target bio-polymers by high-performance liquid chromatography and capillary electrophoresis.
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 2003;797(1-2):111-29.
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2003: Gotti Roberto; Bertucci Carlo; Andrisano Vincenza; Pomponio Romeo; Cavrini Vanni
Study of donepezil binding to serum albumin by capillary electrophoresis and circular dichroism.
Analytical and bioanalytical chemistry 2003;377(5):875-9.
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2003: Fiori Jessica; Ballardini Roberto; Hrelia Patrizia; Andrisano Vincenza; Tarozzi Andrea; Cavrini Vanni
Investigation of the photochemical properties and in vitro phototoxic potential of bumetanide.
Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 2003;2(10):1011-7.
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2003: Bolognesi Maria Laura; Cavalli Andrea; Andrisano Vincenza; Bartolini Manuela; Banzi Rita; Antonello Alessandra; Rosini Michela; Melchiorre Carlo
Design, synthesis and biological evaluation of ambenonium derivatives as AChE inhibitors.
Farmaco (Società chimica italiana : 1989) 2003;58(9):917-28.
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2003: Fiori J; Ballardini R; Andrisano V; Cavrini V
Photostability studies on the furosemide-triamterene drug association.
Farmaco (Società chimica italiana : 1989) 2003;58(9):867-73.
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2003: Andrisano V; Bartolini M; Bertucci C; Cavrini V; Luppi B; Cerchiara T
Analytical methods for the determination of folic acid in a polymeric micellar carrier.
Journal of pharmaceutical and biomedical analysis 2003;32(4-5):983-9.
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2003: Piazzi Lorna; Rampa Angela; Bisi Alessandra; Gobbi Silvia; Belluti Federica; Cavalli Andrea; Bartolini Manuela; Andrisano Vincenza; Valenti Piero; Recanatini Maurizio
3-(4-[[Benzyl(methyl)amino]methyl]phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced beta-amyloid aggregation: a dual function lead for Alzheimer's disease therapy.
Journal of medicinal chemistry 2003;46(12):2279-82.
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2003: Tarozzi A; Andrisano V; Fiori J; Cavrini V; Forti G Cantelli; Hrelia P
Photomutagenic properties of terfenadine as revealed by a stepwise photostability, phototoxicity and photomutagenicity testing approach.
Photochemistry and photobiology 2003;77(4):356-61.
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2003: Tumiatti Vincenzo; Rosini Michela; Bartolini Manuela; Cavalli Andrea; Marucci Gabriella; Andrisano Vincenza; Angeli Piero; Banzi Rita; Minarini Anna; Recanatini Maurizio; Melchiorre Carlo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine.
Journal of medicinal chemistry 2003;46(6):954-66.
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2003: Bartolini Manuela; Andrisano Vincenza; Wainer Irving W
Development and characterization of an immobilized enzyme reactor based on glyceraldehyde-3-phosphate dehydrogenase for on-line enzymatic studies.
Journal of chromatography. A 2003;987(1-2):331-40.
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2003: Bartolini Manuela; Bertucci Carlo; Cavrini Vanni; Andrisano Vincenza
beta-Amyloid aggregation induced by human acetylcholinesterase: inhibition studies.
Biochemical pharmacology 2003;65(3):407-16.
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2002: Bartolini M; Bertucci C; Gotti R; Tumiatti V; Cavalli A; Recanatini M; Andrisano V
Determination of the dissociation constants (pKa) of basic acetylcholinesterase inhibitors by reversed-phase liquid chromatography.
Journal of chromatography. A 2002;958(1-2):59-67.
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2002: Piccoli A; Fiori J; Andrisano V; Orioli M
Determination of triclosan in personal health care products by liquid chromatography (HPLC).
Farmaco (Società chimica italiana : 1989) 2002;57(5):369-72.
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2002: Bertucci C; Andrisano V; Gotti R; Cavrini V
Use of an immobilised human serum albumin HPLC column as a probe of drug-protein interactions: the reversible binding of valproate.
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 2002;768(1):147-55.
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2002: Andrisano V; Gotti R; Recanatini M; Cavalli A; Varoli L; Bertucci C
Stereoselective binding of 2-(4-biphenylyl)-3-substituted-3-hydroxypropionic acids on an immobilised human serum albumin chiral stationary phase.
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 2002;768(1):137-45.
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2001: Rampa A; Piazzi L; Belluti F; Gobbi S; Bisi A; Bartolini M; Andrisano V; Cavrini V; Cavalli A; Recanatini M; Valenti P
Acetylcholinesterase inhibitors: SAR and kinetic studies on omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)methyl]aminoalkoxyaryl derivatives.
Journal of medicinal chemistry 2001;44(23):3810-20.
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2001: Andrisano V; Hrelia P; Gotti R; Leoni A; Cavrini V
Photostability and phototoxicity studies on diltiazem.
Journal of pharmaceutical and biomedical analysis 2001;25(3-4):589-97.
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2001: Andrisano V; Bartolini M; Gotti R; Cavrini V; Felix G
Determination of inhibitors' potency (IC50) by a direct high-performance liquid chromatographic method on an immobilised acetylcholinesterase column.
Journal of chromatography. B, Biomedical sciences and applications 2001;753(2):375-83.
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2001: Gotti R; Cavrini V; Pomponio R; Andrisano V
Analysis and enantioresolution of donepezil by capillary electrophoresis.
Journal of pharmaceutical and biomedical analysis 2001;24(5-6):863-70.
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2001: Andrisano V; Ballardini R; Hrelia P; Cameli N; Tosti A; Gotti R; Cavrini V
Studies on the photostability and in vitro phototoxicity of Labetalol.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 2001;12(4):495-504.
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2001: Bolognesi M L; Andrisano V; Bartolini M; Minarini A; Rosini M; Tumiatti V; Melchiorre C
Hexahydrochromeno[4,3-b]pyrrole derivatives as acetylcholinesterase inhibitors.
Journal of medicinal chemistry 2001;44(1):105-9.
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2000: Andrisano V; Bertucci C; Battaglia A; Cavrini V
Photostability of drugs: photodegradation of melatonin and its determination in commercial formulations.
Journal of pharmaceutical and biomedical analysis 2000;23(1):15-23.
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2000: Recanatini M; Cavalli A; Belluti F; Piazzi L; Rampa A; Bisi A; Gobbi S; Valenti P; Andrisano V; Bartolini M; Cavrini V
SAR of 9-amino-1,2,3,4-tetrahydroacridine-based acetylcholinesterase inhibitors: synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues.
Journal of medicinal chemistry 2000;43(10):2007-18.
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2000: Gotti R; Furlanetto S; Andrisano V; Cavrini V; Pinzauti S
Design of experiments for capillary electrophoretic enantioresolution of salbutamol using dermatan sulfate.
Journal of chromatography. A 2000;875(1-2):411-22.
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2000: Andrisano V; Bertucci C; Cavrini V; Recanatini M; Cavalli A; Varoli L; Felix G; Wainer I W
Stereoselective binding of 2,3-substituted 3-hydroxypropionic acids on an immobilised human serum albumin chiral stationary phase: stereochemical characterisation and quantitative structure-retention relationship study.
Journal of chromatography. A 2000;876(1-2):75-86.
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2000: Tumiatti V; Angeli P; Andrisano V; Bolognesi M L; Cavalli A; Marucci G; Minarini A; Recanatini M; Rosini M; Melchiorre C
[4-[[N-(3-chlorophenyl)carbamoyl]oxy]-2-butynyl]-trimethylammonium (McN-A-343)-related compounds. Effect of the butynyl chain inclusion into an aromatic unit on the potency for muscarinic receptors.
Bioorganic & medicinal chemistry 2000;8(4):681-9.
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2000: Gotti R; Andrisano V; Cavrini V; Bertucci C; Furlanetto S
Analysis of ACE-inhibitors by CE using alkylsulfonic additives.
Journal of pharmaceutical and biomedical analysis 2000;22(3):423-31.
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2000: Rampa A; Bisi A; Belluti F; Gobbi S; Valenti P; Andrisano V; Cavrini V; Cavalli A; Recanatini M
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives.
Bioorganic & medicinal chemistry 2000;8(3):497-506.
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1999: Andrisano V; Gotti R; Leoni A; Cavrini V
Photodegradation studies on Atenolol by liquid chromatography.
Journal of pharmaceutical and biomedical analysis 1999;21(4):851-7.
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1999: Gotti R; Pomponio R; Andrisano V; Cavrini V
Analytical study of penicillamine in pharmaceuticals by capillary zone electrophoresis.
Journal of chromatography. A 1999;844(1-2):361-9.
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1999: Gotti R; Cavrini V; Andrisano V; Mascellani G
Semisynthetic chondroitins as chiral buffer additives in capillary electrophoresis.
Journal of chromatography. A 1999;845(1-2):247-56.
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1999: Simoni D; Roberti M; Andrisano V; Manferdini M; Rondanin R; Invidiata F P
Two-carbon bridge substituted cocaines: enantioselective synthesis, attribution of the absolute configuration and biological activity of novel 6- and 7-methoxylated cocaines.
Farmaco (Società chimica italiana : 1989) 1999;54(5):275-87.
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1998: Melchiorre C; Andrisano V; Bolognesi M L; Budriesi R; Cavalli A; Cavrini V; Rosini M; Tumiatti V; Recanatini M
Acetylcholinesterase noncovalent inhibitors based on a polyamine backbone for potential use against Alzheimer's disease.
Journal of medicinal chemistry 1998;41(22):4186-9.
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1998: Rampa A; Bisi A; Valenti P; Recanatini M; Cavalli A; Andrisano V; Cavrini V; Fin L; Buriani A; Giusti P
Acetylcholinesterase inhibitors: synthesis and structure-activity relationships of omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)- methyl]aminoalkoxyheteroaryl derivatives.
Journal of medicinal chemistry 1998;41(21):3976-86.
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1998: Gotti R; Cavrini V; Andrisano V; Mascellani G
Dermatan sulfate as useful chiral selector in capillary electrophoresis.
Journal of chromatography. A 1998;814(1-2):205-11.
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1998: Roveri P; Andrisano V; Di Pietra A M; Cavrini V
GC-MS analysis of incenses for possible presence of allergenic nitromusks.
Journal of pharmaceutical and biomedical analysis 1998;17(3):393-8.
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1998: Andrisano V; Gotti R; Cavrini V; Tumiatti V; Felix G; Wainer I W
Capillary electrophoretic and high-performance liquid chromatographic studies of the enantioselective separation of alpha1-adrenoreceptor antagonists.
Journal of chromatography. A 1998;803(1-2):189-95.
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1997: Bonazzi D; Gotti R; Andrisano V; Cavrini V
Analysis of ACE inhibitors in pharmaceutical dosage forms by derivative UV spectroscopy and liquid chromatography (HPLC).
Journal of pharmaceutical and biomedical analysis 1997;16(3):431-8.
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1997: Andrisano V; Booth T D; Cavrini V; Wainer I W
Enantioselective separation of chiral arylcarboxylic acids on an immobilized human serum albumin chiral stationary phase.
Chirality 1997;9(2):178-83.
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1996: Di Pietra A M; Andrisano V; Gotti R; Cavrini V
On-line post-column photochemical derivatization in liquid chromatographic--diode-array detection analysis of binary drug mixtures.
Journal of pharmaceutical and biomedical analysis 1996;14(8-10):1191-9.
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1996: Di Pietra A M; Gatti R; Andrisano V; Cavrini V
Application of high-performance liquid chromatography with diode-array detection and on-line post-column photochemical derivatization to the determination of analgesics.
Journal of chromatography. A 1996;729(1-2):355-61.
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1995: Bonazzi D; Andrisano V; Gatti R; Cavrini V
Analysis of pharmaceutical creams: a useful approach based on solid-phase extraction (SPE) and UV spectrophotometry.
Journal of pharmaceutical and biomedical analysis 1995;13(11):1321-9.
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1995: Andrisano V; Bonazzi D; Cavrini V
HPLC analysis of liquorice triterpenoids--applications to the quality control of pharmaceuticals.
Journal of pharmaceutical and biomedical analysis 1995;13(4-5):597-605.
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1995: Gatti R; Andrisano V; Di Pietra A M; Cavrini V
Analysis of aliphatic dicarboxylic acids in pharmaceuticals and cosmetics by liquid chromatography (HPLC) with fluorescence detection.
Journal of pharmaceutical and biomedical analysis 1995;13(4-5):589-95.
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1994: Gotti R; Andrisano V; Gatti R; Cavrini V; Candeletti S
Determination of glutathione in biological samples by high performance liquid chromatography with fluorescence detection.
Biomedical chromatography : BMC 1994;8(6):306-8.
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1994: Bonazzi D; Andrisano V; Di Pietra A M; Cavrini V
Analysis of Trimethoprim--sulfonamide drug combinations in dosage forms by UV spectroscopy and liquid chromatography (HPLC).
Farmaco (Società chimica italiana : 1989) 1994;49(6):381-6.
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1994: Di Pietra A M; Gotti R; Bonazzi D; Andrisano V; Cavrini V
HPLC determination of glutathione and L-cysteine in pharmaceuticals after derivatization with ethacrynic acid.
Journal of pharmaceutical and biomedical analysis 1994;12(1):91-8.
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1992: Di Pietra A M; Cavrini V; Andrisano V; Gatti R
HPLC analysis of imidazole antimycotic drugs in pharmaceutical formulations.
Journal of pharmaceutical and biomedical analysis 1992;10(10-12):873-9.
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1992: Varoli L; Burnelli S; Guarnieri A; Scapini G; Andrisano V; Lumachi B
Nonsteroidal antiinflammatory agents. Part 21: optically active stereoisomers of p-trifluoromethylphenyl- and p-thioanisyl-biphenylyl- hydroxypropionic acids.
Die Pharmazie 1992;47(3):174-7.
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1992: Andrisano V; Marucci G; Melchiorre C; Tumiatti V
Stereoselectivity at alpha-adrenoreceptor subtypes: observations with the enantiomers of WB 4101 separated through their amides of N-tosyl-(S)-proline.
Chirality 1992;4(1):16-20.
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1990: Cavrini V; Andrisano V; Gatti R; Scapini G
HPLC determination of thioglycolic acid and other aliphatic thiols in cosmetic formulations using ethacrynic acid as precolumn derivatization reagent.
International journal of cosmetic science 1990;12(4):141-50.
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1990: Varoli L; Burnelli S; Guarnieri A; Scapini G; Andrisano V; Fantuz M
Nonsteroidal antiinflammatory agents. Part 20(3): Optically active thienyl-biphenylyl-hydroxypropionic acids.
Die Pharmazie 1990;45(7):488-90.
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