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Antonio Garofalo

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Bikash Debnath; Antonio Garofalo; Fedora Grande; Shili Xu; Nouri Neamati
Small molecule inhibitors of CXCR4.
Francesca Aiello; Adrian Esqueda; Antonio Garofalo; Fedora Grande; Tino W Sanchez; Yumna Shabaik; Nouri Neamati
Design and synthesis of 3-carbamoylbenzoic acid derivatives as inhibitors of human apurinic/apyrimidinic endonuclease 1 (APE1).
Takashi Oshima; Xuefei Cao; Fedora Grande; Roppei Yamada; Antonio Garofalo; Stan Louie; Nouri Neamati
Combination effects of SC144 and cytotoxic anticancer agents.

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All Publications

2013: Bikash Debnath; Antonio Garofalo; Fedora Grande; Shili Xu; Nouri Neamati
Small molecule inhibitors of CXCR4.
Theranostics 2013;3(1):47-75.
2012: Francesca Aiello; Adrian Esqueda; Antonio Garofalo; Fedora Grande; Tino W Sanchez; Yumna Shabaik; Nouri Neamati
Design and synthesis of 3-carbamoylbenzoic acid derivatives as inhibitors of human apurinic/apyrimidinic endonuclease 1 (APE1).
ChemMedChem 2012;7(10):1825-39.
2009: Takashi Oshima; Xuefei Cao; Fedora Grande; Roppei Yamada; Antonio Garofalo; Stan Louie; Nouri Neamati
Combination effects of SC144 and cytotoxic anticancer agents.
Anti-cancer drugs 2009;20(5):312-20.
2009: Fedora Grande; Roppei Yamada; Xuefei Cao; Francesca Aiello; Antonio Garofalo; Nouri Neamati
Synthesis and biological evaluation of novel hydrazide based cytotoxic agents.
Expert opinion on investigational drugs 2009;18(5):555-68.
2009: Carmen Plasencia; Fedora Grande; Takashi Oshima; Xuefei Cao; Roppei Yamada; Tino Sanchez; Francesca Aiello; Antonio Garofalo; Nouri Neamati
Discovery of a novel quinoxalinhydrazide with a broad-spectrum anticancer activity.
Cancer biology & therapy 2009;8(5):458-65.
2008: Jinxia Deng; Laleh Taheri; Fedora Grande; Francesca Aiello; Antonio Garofalo; Nouri Neamati
Discovery of novel anticancer compounds based on a quinoxalinehydrazine pharmacophore.
ChemMedChem 2008;3(11):1677-86.
2008: Antonio Garofalo; Fedora Grande; Antonella Brizzi; Francesca Aiello; Raveendra Dayam; Nouri Neamati
Naphthoxazepine inhibitors of HIV-1 integrase: synthesis and biological evaluation.
ChemMedChem 2008;3(6):986-90.
2008: Fedora Grande; Antonio Garofalo; Nouri Neamati
Small molecules anti-HIV therapeutics targeting CXCR4.
Current pharmaceutical design 2008;14(4):385-404.
2007: Jinxia Deng; Tino Sanchez; Laith Q Al-Mawsawi; Raveendra Dayam; Rosendo A Yunes; Antonio Garofalo; Michael B Bolger; Nouri Neamati
Discovery of structurally diverse HIV-1 integrase inhibitors based on a chalcone pharmacophore.
Bioorganic & medicinal chemistry 2007;15(14):4985-5002.
2007: Fedora Grande; Francesca Aiello; Osvaldo De Grazia; Antonella Brizzi; Antonio Garofalo; Nouri Neamati
Synthesis and antitumor activities of a series of novel quinoxalinhydrazides.
Bioorganic & medicinal chemistry 2007;15(1):288-94.
2006: Gaetano Ragno; Giuseppina Ioele; Michele De Luca; Antonio Garofalo; Fedora Grande; Antonella Risoli
A critical study on the application of the zero-crossing derivative spectrophotometry to the photodegradation monitoring of lacidipine.
Journal of pharmaceutical and biomedical analysis 2006;42(1):39-45.
2006: Francesca Aiello; Antonella Brizzi; O De Grazia; Antonio Garofalo; Fedora Grande; M S Sinicropi; Raveendra Dayam; Nouri Neamati
An approach to the stereo-controlled synthesis of polycyclic derivatives of l-4-thiazolidinecarboxylic acid active against HIV-1 integrase.
European journal of medicinal chemistry 2006;41(8):914-7.
2006: Raveendra Dayam; Francesca Aiello; Jinxia Deng; Yun Wu; Antonio Garofalo; Xiaoyuan Chen; Nouri Neamati
Discovery of small molecule integrin alphavbeta3 antagonists as novel anticancer agents.
Journal of medicinal chemistry 2006;49(15):4526-34.
2004: Francesca Aiello; Antonella Brizzi; Antonio Garofalo; Fedora Grande; Gaetano Ragno; Raveendra Dayam; Nouri Neamati
Synthesis of novel thiazolothiazepine based HIV-1 integrase inhibitors.
Bioorganic & medicinal chemistry 2004;12(16):4459-66.
2003: Gaetano Ragno; Francesca Aiello; Antonio Garofalo; Giuseppina Ioele; Maria Stefania Sinicropi
Multivariate least squares regression applied to the spectrophotometric analysis of manidipine and its main photoproduct.
Farmaco (Società chimica italiana : 1989) 2003;58(9):909-15.
2001: Giuseppe Campiani; Francesca Aiello; M Fabbrini; Elena Morelli; Anna Ramunno; S Armaroli; Vito Nacci; Antonio Garofalo; Giovanni Greco; Ettore Novellino; giovanni maga; Silvio Spadari; Alberto Bergamini; L Ventura; Barbara Bongiovanni; Marcella Capozzi; Francesca Bolacchi; Stefano Marini; Massimo Coletta; Giovanna Guiso; S Caccia
Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent.
Journal of medicinal chemistry 2001;44(3):305-15.
1999: Nouri Neamati; Jim A Turpin; Heather E Winslow; JL Christensen; K Williamson; Ann H Orr; William G Rice; Yves Pommier; Antonio Garofalo; Antonella Brizzi; Giuseppe Campiani; Isabella Fiorini; Vito Nacci
Thiazolothiazepine inhibitors of HIV-1 integrase.
Journal of medicinal chemistry 1999;42(17):3334-41.
1998: Giuseppe Campiani; Vito Nacci; S Bechelli; S M Ciani; Antonio Garofalo; Isabella Fiorini; H Wikström; P de Boer; Y Liao; P G Tepper; Alfredo Cagnotto; Tiziana Mennini
New antipsychotic agents with serotonin and dopamine antagonist properties based on a pyrrolo[2,1-b][1,3]benzothiazepine structure.
Journal of medicinal chemistry 1998;41(20):3763-72.
1996: Giuseppe Campiani; Vito Nacci; Isabella Fiorini; M P De Filippis; Antonio Garofalo; S M Ciani; Giovanni Greco; Ettore Novellino; D C Williams; Daniela M Zisterer; M J Woods; C Mihai; C Manzoni; Tiziana Mennini
Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific "peripheral-type" benzodiazepine receptor ligands.
Journal of medicinal chemistry 1996;39(18):3435-50.
1996: Giuseppe Campiani; Isabella Fiorini; M P De Filippis; S M Ciani; Antonio Garofalo; Vito Nacci; Gianluca Giorgi; A Sega; Maurizio Botta; Alberto Chiarini; Roberta Budriesi; Giancarlo Bruni; M R Romeo; C Manzoni; Tiziana Mennini
Cardiovascular characterization of pyrrolo[2,1-d][1,5]benzothiazepine derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): from dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blockers.
Journal of medicinal chemistry 1996;39(15):2922-38.
1996: Giuseppe Campiani; Vito Nacci; Isabella Fiorini; M P De Filippis; Antonio Garofalo; Giovanni Greco; Ettore Novellino; Sergio Altamura; L Di Renzo
Pyrrolobenzothiazepinones and pyrrolobenzoxazepinones: novel and specific non-nucleoside HIV-1 reverse transcriptase inhibitors with antiviral activity.
Journal of medicinal chemistry 1996;39(14):2672-80.
1995: Giuseppe Campiani; Antonio Garofalo; Isabella Fiorini; Maurizio Botta; Vito Nacci; Andrea Tafi; Alberto Chiarini; Roberta Budriesi; Giancarlo Bruni; M R Romeo
Pyrrolo[2,1-c][1,4]benzothiazines: synthesis, structure-activity relationships, molecular modeling studies, and cardiovascular activity.
Journal of medicinal chemistry 1995;38(22):4393-410.
1994: Giovanni Greco; Ettore Novellino; Isabella Fiorini; Vito Nacci; Giuseppe Campiani; S M Ciani; Antonio Garofalo; P Bernasconi; Tiziana Mennini
A comparative molecular field analysis model for 6-arylpyrrolo[2,1-d] [1,5]benzothiazepines binding selectively to the mitochondrial benzodiazepine receptor.
Journal of medicinal chemistry 1994;37(24):4100-8.
1994: Isabella Fiorini; Vito Nacci; S M Ciani; Antonio Garofalo; Giuseppe Campiani; Luisa Savini; Ettore Novellino; Giovanni Greco; P Bernasconi; Tiziana Mennini
Novel ligands specific for mitochondrial benzodiazepine receptors: 6-arylpyrrolo[2,1-d][1,5]benzothiazepine derivatives. Synthesis, structure-activity relationships, and molecular modeling studies.
Journal of medicinal chemistry 1994;37(10):1427-38.
1993: Antonio Garofalo; Giuseppe Campiani; Isabella Fiorini; Vito Nacci
Benzothiazine and benzothiazepine derivatives: synthesis and preliminary biological evaluation.
Farmaco (Società chimica italiana : 1989) 1993;48(2):275-83.
1990: Vito Nacci; Isabella Fiorini; Antonio Garofalo; Alfredo Cagnotto
Research on compounds with psychotropic activity. IX--Synthesis of 6-p-methoxyphenylpyrrolo[2,1-d][1,5]benzothiazepines and evaluation of their affinities for BDZ and GABA receptor subtypes.
Farmaco (Società chimica italiana : 1989) 1990;45(5):545-58.
1989: Maurizio Anzini; Salvatore Vomero; Antonio Garofalo; Andrea Cappelli; Alfredo Cagnotto
Synthesis and 5HT-receptors affinity of some 4-phenylquinoline derivatives.
Farmaco (Società chimica italiana : 1989) 1989;44(6):555-63.