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Giovanni Greco

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Sabrina Taliani; Maria Letizia Trincavelli; Elisabetta Barresi; Sandro Cosconati; Barbara Cosimelli; Simona Daniele; Salvatore Di Maro; Giovanni Greco; Concettina La Motta; Luciana Marinelli; Anna Maria Marini; Claudia Martini; Ettore Novellino; Isabella Pugliesi; Silvia Salerno; Francesca Simorini; Federico Da Settimo
3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A₂B adenosine receptor antagonists.
Barbara Cosimelli; Luciana Marinelli; Ettore Novellino; Sandro Cosconati; Giovanni Greco
From the pharmacophore to the homology model of the benzodiazepine receptor: the indolyglyoxylamides affair.
Barbara Cosimelli; Federico Da Settimo; Simona Daniele; Matteo Fornai; Giovanni Greco; Concettina La Motta; Ettore Novellino; Isabella Pugliesi; Annalisa Sala; Elda Severi; Sabrina Taliani; Maria Letizia Trincavelli; luca Antonioli; Corrado Blandizzi; Rocchina Colucci; Claudia Martini
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility.

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All Publications

2012: Sabrina Taliani; Maria Letizia Trincavelli; Elisabetta Barresi; Sandro Cosconati; Barbara Cosimelli; Simona Daniele; Salvatore Di Maro; Giovanni Greco; Concettina La Motta; Luciana Marinelli; Anna Maria Marini; Claudia Martini; Ettore Novellino; Isabella Pugliesi; Silvia Salerno; Francesca Simorini; Federico Da Settimo
3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A₂B adenosine receptor antagonists.
Journal of medicinal chemistry 2012;55(4):1490-9.
2012: Barbara Cosimelli; Luciana Marinelli; Ettore Novellino; Sandro Cosconati; Giovanni Greco
From the pharmacophore to the homology model of the benzodiazepine receptor: the indolyglyoxylamides affair.
Current topics in medicinal chemistry 2012;12(4):321-32.
2011: Barbara Cosimelli; Federico Da Settimo; Simona Daniele; Matteo Fornai; Giovanni Greco; Concettina La Motta; Ettore Novellino; Isabella Pugliesi; Annalisa Sala; Elda Severi; Sabrina Taliani; Maria Letizia Trincavelli; luca Antonioli; Corrado Blandizzi; Rocchina Colucci; Claudia Martini
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility.
ChemMedChem 2011;6(10):1909-18.
2011: Barbara Cosimelli; Barbara Costa; Eleonora Da Pozzo; Federico Da Settimo; Giovanni Greco; Concettina La Motta; Ettore Novellino; Elda Severi; Francesca Simorini; Sabrina Taliani; Sara Bendinelli; Claudia Martini
Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein.
European journal of medicinal chemistry 2011;46(9):4506-20.
2010: Sabrina Taliani; Eleonora Da Pozzo; Marusca Bellandi; Sara Bendinelli; Isabella Pugliesi; Francesca Simorini; Concettina La Motta; Silvia Salerno; Anna Maria Marini; Federico Da Settimo; Barbara Cosimelli; Giovanni Greco; Ettore Novellino; Claudia Martini
Novel irreversible fluorescent probes targeting the 18 kDa translocator protein: synthesis and biological characterization.
Journal of medicinal chemistry 2010;53(10):4085-93.
2010: Sabrina Taliani; Concettina La Motta; Laura Mugnaini; Francesca Simorini; Silvia Salerno; Anna Maria Marini; Federico Da Settimo; Sandro Cosconati; Barbara Cosimelli; Giovanni Greco; Vittorio Limongelli; Luciana Marinelli; Ettore Novellino; Osele Ciampi; Simona Daniele; Maria Letizia Trincavelli; Claudia Martini
Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation.
Journal of medicinal chemistry 2010;53(10):3954-63.
2009: Sabrina Taliani; Barbara Cosimelli; Federico Da Settimo; Anna Maria Marini; Concettina La Motta; Francesca Simorini; Silvia Salerno; Ettore Novellino; Giovanni Greco; Sandro Cosconati; Luciana Marinelli; F Salvetti; Gianluca L'Abbate; Silvia Trasciatti; Marina Montali; Barbara Costa; Claudia Martini
Identification of anxiolytic/nonsedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the gamma-aminobutyric acid-A (GABAA) alpha2 benzodiazepine receptor.
Journal of medicinal chemistry 2009;52(12):3723-34.
2008: Federico Da Settimo; Francesca Simorini; Sabrina Taliani; Concettina La Motta; Anna Maria Marini; Silvia Salerno; Marusca Bellandi; Ettore Novellino; Giovanni Greco; Barbara Cosimelli; Eleonora Da Pozzo; Barbara Costa; Nicola Simola; Micaela Morelli; Claudia Martini
Anxiolytic-like effects of N,N-dialkyl-2-phenylindol-3-ylglyoxylamides by modulation of translocator protein promoting neurosteroid biosynthesis.
Journal of medicinal chemistry 2008;51(18):5798-806.
2008: Barbara Cosimelli; Giovanni Greco; Marina Ehlardo; Ettore Novellino; Federico Da Settimo; Sabrina Taliani; Concettina La Motta; Marusca Bellandi; Tiziano Tuccinardi; Adriano Martinelli; Osele Ciampi; Maria Letizia Trincavelli; Claudia Martini
Derivatives of 4-amino-6-hydroxy-2-mercaptopyrimidine as novel, potent, and selective A3 adenosine receptor antagonists.
Journal of medicinal chemistry 2008;51(6):1764-70.
2007: Federico Da Settimo; Giampaolo Primofiore; Sabrina Taliani; Anna Maria Marini; Concettina La Motta; Francesca Simorini; Silvia Salerno; Valentina Sergianni; Tiziano Tuccinardi; Adriano Martinelli; Barbara Cosimelli; Giovanni Greco; Ettore Novellino; Osele Ciampi; Maria Letizia Trincavelli; Claudia Martini
5-amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a versatile scaffold to obtain potent and selective A3 adenosine receptor antagonists.
Journal of medicinal chemistry 2007;50(23):5676-84.
2007: Giampaolo Primofiore; Sabrina Taliani; Federico Da Settimo; Anna Maria Marini; Concettina La Motta; Francesca Simorini; Maria Paola Patrizi; Valentina Sergianni; Ettore Novellino; Giovanni Greco; Barbara Cosimelli; Vincenzo Calderone; Marina Montali; Francois Besnard; Claudia Martini
Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands.
Journal of medicinal chemistry 2007;50(7):1627-34.
2007: Sabrina Taliani; Francesca Simorini; Valentina Sergianni; Concettina La Motta; Federico Da Settimo; Barbara Cosimelli; Enrico Abignente; Giovanni Greco; Ettore Novellino; Leonardo Rossi; Vittorio Gremigni; Francesca Spinetti; Beatrice Chelli; Claudia Martini
New fluorescent 2-phenylindolglyoxylamide derivatives as probes targeting the peripheral-type benzodiazepine receptor: design, synthesis, and biological evaluation.
Journal of medicinal chemistry 2007;50(2):404-7.
2006: Giampaolo Primofiore; Federico Da Settimo; Anna Maria Marini; Sabrina Taliani; Concettina La Motta; Francesca Simorini; Ettore Novellino; Giovanni Greco; Barbara Cosimelli; Marina Ehlardo; Annalisa Sala; Francois Besnard; Marina Montali; Claudia Martini
Refinement of the benzodiazepine receptor site topology by structure-activity relationships of new N-(heteroarylmethyl)indol-3-ylglyoxylamides.
Journal of medicinal chemistry 2006;49(8):2489-95.
2005: Ettore Novellino; Barbara Cosimelli; Marina Ehlardo; Giovanni Greco; Manuela Iadanza; Antonio Lavecchia; Maria Grazia Rimoli; Annalisa Sala; Antonio Da Settimo; Giampaolo Primofiore; Federico Da Settimo; Sabrina Taliani; Concettina La Motta; Karl-Norbert Klotz; Daniela Tuscano; Maria Letizia Trincavelli; Claudia Martini
2-(Benzimidazol-2-yl)quinoxalines: a novel class of selective antagonists at human A(1) and A(3) adenosine receptors designed by 3D database searching.
Journal of medicinal chemistry 2005;48(26):8253-60.
2005: Giampaolo Primofiore; Federico Da Settimo; Sabrina Taliani; Silvia Salerno; Ettore Novellino; Giovanni Greco; Barbara Cosimelli; Francois Besnard; Barbara Costa; Marina Montali; Claudia Martini
High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives.
Journal of medicinal chemistry 2005;48(8):2936-43.
2005: Luca Guandalini; Elisabetta Martini; Silvia Dei; Dina Manetti; Serena Scapecchi; Elisabetta Teodori; Maria Novella Romanelli; Katia Varani; Giovanni Greco; Loredana Spadola; Ettore Novellino
Design of novel nicotinic ligands through 3D database searching.
Bioorganic & medicinal chemistry 2005;13(3):799-807.
2005: Federico Da Settimo; Giampaolo Primofiore; Concettina La Motta; Silvia Salerno; Ettore Novellino; Giovanni Greco; Antonio Lavecchia; Sonia Laneri; Enrico Boldrini
Spirohydantoin derivatives of thiopyrano[2,3-b]pyridin-4(4H)-one as potent in vitro and in vivo aldose reductase inhibitors.
Bioorganic & medicinal chemistry 2005;13(2):491-9.
2004: Giampaolo Primofiore; Federico Da Settimo; Sabrina Taliani; Francesca Simorini; Maria Paola Patrizi; Ettore Novellino; Giovanni Greco; Enrico Abignente; Barbara Costa; Beatrice Chelli; Claudia Martini
N,N-dialkyl-2-phenylindol-3-ylglyoxylamides. A new class of potent and selective ligands at the peripheral benzodiazepine receptor.
Journal of medicinal chemistry 2004;47(7):1852-5.
2003: Giampaolo Primofiore; Federico Da Settimo; Sabrina Taliani; Anna Maria Marini; Francesca Simorini; Ettore Novellino; Giovanni Greco; Letizia Trincavelli; Claudia Martini
Geometrically constrained analogues of N-benzylindolylglyoxylylamides: [1, 2, 4]triazino[4, 3-a]benzimidazol-4(10H)-one derivatives as potential new ligands at the benzodiazepine receptor.
Archiv der Pharmazie 2003;336(9):413-21.
2003: Federico Da Settimo; Giampaolo Primofiore; Antonio Da Settimo; Concettina La Motta; Francesca Simorini; Ettore Novellino; Giovanni Greco; Antonio Lavecchia; Enrico Boldrini
Novel, highly potent aldose reductase inhibitors: cyano(2-oxo-2,3-dihydroindol-3-yl)acetic acid derivatives.
Journal of medicinal chemistry 2003;46(8):1419-28.
2002: Ettore Novellino; Enrico Abignente; Barbara Cosimelli; Giovanni Greco; Manuela Iadanza; Sonia Laneri; Antonio Lavecchia; Maria Grazia Rimoli; Federico Da Settimo; Giampaolo Primofiore; Daniela Tuscano; Letizia Trincavelli; Claudia Martini
Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A(1) adenosine receptor antagonists.
Journal of medicinal chemistry 2002;45(23):5030-6.
2002: Anna Maria Dursi; Stefania Albrizio; Giovanni Greco; Sonia Mazzeo; Maria R Mazzoni; Ettore Novellino; Paolo Rovero
Conformational analysis of the Galpha(s) protein C-terminal region.
Journal of peptide science : an official publication of the European Peptide Society 2002;8(8):476-88.
2001: Federico Da Settimo; Giampaolo Primofiore; Antonio Da Settimo; Concettina La Motta; Sabrina Taliani; Francesca Simorini; Ettore Novellino; Giovanni Greco; Antonio Lavecchia; Enrico Boldrini
[1,2,4]Triazino[4,3-a]benzimidazole acetic acid derivatives: a new class of selective aldose reductase inhibitors.
Journal of medicinal chemistry 2001;44(25):4359-69.
2001: Giampaolo Primofiore; F D Settimo; Sabrina Taliani; Anna Maria Marini; Ettore Novellino; Giovanni Greco; Antonio Lavecchia; Francois Besnard; Letizia Trincavelli; Barbara Costa; Claudia Martini
Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships.
Journal of medicinal chemistry 2001;44(14):2286-97.
2001: Federico Da Settimo; Giampaolo Primofiore; Sabrina Taliani; Anna Maria Marini; Concettina La Motta; Ettore Novellino; Giovanni Greco; Antonio Lavecchia; Letizia Trincavelli; Claudia Martini
3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: a new class of selective A1 adenosine receptor antagonists.
Journal of medicinal chemistry 2001;44(3):316-27.
2000: Stefania Albrizio; Anna Maria D'Ursi; Caterina Fattorusso; C Galoppini; Giovanni Greco; Maria R Mazzoni; Ettore Novellino; Paolo Rovero
Conformational studies on a synthetic C-terminal fragment of the alpha subunit of G(S) proteins.
Biopolymers 2000;54(3):186-94.
2000: Maria R Mazzoni; Simone Taddei; Laura Giusti; Paolo Rovero; C Galoppini; Anna Maria D'Ursi; Stefania Albrizio; Antonio Triolo; Ettore Novellino; Giovanni Greco; Antonio Lucacchini; Heidi E Hamm
A galpha(s) carboxyl-terminal peptide prevents G(s) activation by the A(2A) adenosine receptor.
Molecular pharmacology 2000;58(1):226-36.
2000: Antonio Lavecchia; Giovanni Greco; Ettore Novellino; Franco Vittorio; Giuseppe Ronsisvalle
Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations.
Journal of medicinal chemistry 2000;43(11):2124-34.
2000: Giampaolo Primofiore; Federico Da Settimo; Sabrina Taliani; Anna Maria Marini; Concettina La Motta; Ettore Novellino; Giovanni Greco; Marco Gesi; Letizia Trincavelli; Claudia Martini
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands.
Journal of medicinal chemistry 2000;43(1):96-102.
1998: Antonio Da Settimo; Giampaolo Primofiore; Federico Da Settimo; Anna Maria Marini; Ettore Novellino; Giovanni Greco; Marco Gesi; Claudia Martini; Gino Giannaccini; Antonio Lucacchini
N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors.
Journal of medicinal chemistry 1998;41(20):3821-30.