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Jean-Michel Arrang

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Florence Gbahou; Agnès Rouleau; Jean-Michel Arrang
The histamine autoreceptor is a short isoform of the H₃ receptor.
Marie Humbert-Claude; Ludwig Vincent; Elisabeth Davenas; Florence Gbahou; Jean-Michel Arrang
Involvement of histamine receptors in the atypical antipsychotic profile of clozapine: a reassessment in vitro and in vivo.
Mouhammad Motawaj; Jean-Michel Arrang
Ciproxifan, a histamine H₃-receptor antagonist / inverse agonist, modulates methamphetamine-induced sensitization in mice.

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All Publications

2012: Florence Gbahou; Agnès Rouleau; Jean-Michel Arrang
The histamine autoreceptor is a short isoform of the H₃ receptor.
British journal of pharmacology 2012;166(6):1860-71.
2012: Marie Humbert-Claude; Ludwig Vincent; Elisabeth Davenas; Florence Gbahou; Jean-Michel Arrang
Involvement of histamine receptors in the atypical antipsychotic profile of clozapine: a reassessment in vitro and in vivo.
Psychopharmacology 2012;220(1):225-41.
2011: Mouhammad Motawaj; Jean-Michel Arrang
Ciproxifan, a histamine H₃-receptor antagonist / inverse agonist, modulates methamphetamine-induced sensitization in mice.
The European journal of neuroscience 2011;33(7):1197-204.
2011: M Motawaj; A Burban; E Davenas; Jean-Michel Arrang
Activation of brain histaminergic neurotransmission: a mechanism for cognitive effects of memantine in Alzheimer's disease.
The Journal of pharmacology and experimental therapeutics 2011;336(2):479-87.
2010: Mouhammad Motawaj; Aude Burban; Elisabeth Davenas; Florence Gbahou; Raphaël Faucard; Séverine Morisset; Jean-Michel Arrang
[The histaminergic system: a target for innovative treatments of cognitive deficits].
Thérapie 2010;65(5):415-22.
2010: F Gbahou; E Davenas; Séverine Morisset; Jean-Michel Arrang
Effects of betahistine at histamine H3 receptors: mixed inverse agonism/agonism in vitro and partial inverse agonism in vivo.
The Journal of pharmacology and experimental therapeutics 2010;334(3):945-54.
2010: Aude Burban; Chit Sadakhom; Dominique Dumoulin; Christiane Rose; Gwenaëlle Le Pen; Henriette Frances; Jean-Michel Arrang
Modulation of prepulse inhibition and stereotypies in rodents: no evidence for antipsychotic-like properties of histamine H3-receptor inverse agonists.
Psychopharmacology 2010;210(4):591-604.
2010: A Burban; R Faucard; V Armand; C Bayard; V Vorobjev; Jean-Michel Arrang
Histamine potentiates N-methyl-D-aspartate receptors by interacting with an allosteric site distinct from the polyamine binding site.
The Journal of pharmacology and experimental therapeutics 2010;332(3):912-21.
2010: Mouhammad Motawaj; Katell Peoc'h; Jacques Callebert; Jean-Michel Arrang
CSF levels of the histamine metabolite tele-methylhistamine are only slightly decreased in Alzheimer's disease.
Journal of Alzheimer's disease : JAD 2010;22(3):861-71.
2009: Walid Beghdadi; Adeline Porcherie; Bradley Schneider; Séverine Morisset; David Dubayle; Roger Peronet; Michel Dy; Jacques Louis; Jean-Michel Arrang; Salaheddine Mécheri
Histamine H(3) receptor-mediated signaling protects mice from cerebral malaria.
PloS one 2009;4(6):e6004.
2008: Valérie Biran; Véronique Cochois; A Karroubi; Jean-Michel Arrang; Christiane Charriaut-Marlangue; Anne Héron
Stroke induces histamine accumulation and mast cell degranulation in the neonatal rat brain.
Brain pathology (Zurich, Switzerland) 2008;18(1):1-9.
2007: Jean-Michel Arrang; Séverine Morisset; Florence Gbahou
Constitutive activity of the histamine H3 receptor.
Trends in pharmacological sciences 2007;28(7):350-7.
2007: Xavier Ligneau; Laurent Landais; David Perrin; Johanne Piriou; Marilyne Uguen; Emmanuel Denis; Philippe Robert; Régis Parmentier; Christelle Anaclet; Jian-Sheng Lin; Aude Burban; Jean-Michel Arrang; Jean-Charles Schwartz
Brain histamine and schizophrenia: potential therapeutic applications of H3-receptor inverse agonists studied with BF2.649.
Biochemical pharmacology 2007;73(8):1215-24.
2007: Marie Humbert-Claude; Séverine Morisset; Florence Gbahou; Jean-Michel Arrang
Histamine H3 and dopamine D2 receptor-mediated [35S]GTPgamma[S] binding in rat striatum: evidence for additive effects but lack of interactions.
Biochemical pharmacology 2007;73(8):1172-81.
2007: Jean-Michel Arrang
Histamine and schizophrenia.
International review of neurobiology 2007;78():247-87.
2007: Xavier Ligneau; D Perrin; L Landais; Jean-Claude Camelin; T P G Calmels; Isabelle Berrebi-Bertrand; J-M Lecomte; Régis Parmentier; Christelle Anaclet; Jian-Sheng Lin; Valérie Bertaina-Anglade; Christophe Drieu La Rochelle; F d'Aniello; Agnès Rouleau; Florence Gbahou; Jean-Michel Arrang; C Robin Ganellin; Holger Stark; Walter Schunack; Jean-Charles Schwartz
BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology.
The Journal of pharmacology and experimental therapeutics 2007;320(1):365-75.
2006: Raphaël Faucard; Vincent Armand; Anne Héron; Véronique Cochois; Jean-Charles Schwartz; Jean-Michel Arrang
N-methyl-D-aspartate receptor antagonists enhance histamine neuron activity in rodent brain.
Journal of neurochemistry 2006;98(5):1487-96.
2006: Florence Gbahou; Ludwig Vincent; Marie Humbert-Claude; Joël Tardivel-Lacombe; Claude Chabret; Jean-Michel Arrang
Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.
British journal of pharmacology 2006;147(7):744-54.
2005: Joachim Apelt; Sven Grassmann; Xavier Ligneau; Heinz H Pertz; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Search for histamine H3 receptor antagonists with combined inhibitory potency at Ntau-methyltransferase: ether derivatives.
Die Pharmazie 2005;60(2):97-106.
2004: Sven Grassmann; Joachim Apelt; Xavier Ligneau; Heinz H Pertz; Jean-Michel Arrang; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Search for histamine H(3) receptor ligands with combined inhibitory potency at histamine N-methyltransferase: omega-piperidinoalkanamine derivatives.
Archiv der Pharmazie 2004;337(10):533-45.
2004: Agnès Rouleau; Anne Héron; Véronique Cochois; Catherine Pillot; Jean-Charles Schwartz; Jean-Michel Arrang
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
Journal of neurochemistry 2004;90(6):1331-8.
2004: Nadia Pelloux-Léon; Abdellatif Fkyerat; Antonia Piripitsi; Wasyl Tertiuk; Walter Schunack; Holger Stark; Monique Garbarg; Xavier Ligneau; Jean-Michel Arrang; Jean-Charles Schwartz; C Robin Ganellin
Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain.
Journal of medicinal chemistry 2004;47(12):3264-74.
2004: Tibor Mikó; Xavier Ligneau; Heinz H Pertz; Jean-Michel Arrang; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Structural variations of 1-(4-(phenoxymethyl)benzyl)piperidines as nonimidazole histamine H3 receptor antagonists.
Bioorganic & medicinal chemistry 2004;12(10):2727-36.
2004: Galina Meier; Michael Krause; Annette Hüls; Xavier Ligneau; Heinz H Pertz; Jean-Michel Arrang; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack; Holger Stark
4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists.
Journal of medicinal chemistry 2004;47(10):2678-87.
2003: Florence Gbahou; Agnès Rouleau; Séverine Morisset; Régis Parmentier; Sylvain Crochet; Jian-Sheng Lin; Xavier Ligneau; Joël Tardivel-Lacombe; Holger Stark; Walter Schunack; C Robin Ganellin; Jean-Charles Schwartz; Jean-Michel Arrang
Protean agonism at histamine H3 receptors in vitro and in vivo.
Proceedings of the National Academy of Sciences of the United States of America 2003;100(19):11086-91.
2003: Sven Grassmann; Joachim Apelt; Wolfgang Sippl; Xavier Ligneau; Heinz H Pertz; Yuan Hui Zhao; Jean-Michel Arrang; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Imidazole derivatives as a novel class of hybrid compounds with inhibitory histamine N-methyltransferase potencies and histamine hH3 receptor affinities.
Bioorganic & medicinal chemistry 2003;11(10):2163-74.
2003: Tibor Mikó; Xavier Ligneau; Heinz H Pertz; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds.
Journal of medicinal chemistry 2003;46(8):1523-30.
2003: Jean-Charles Schwartz; Séverine Morisset; Agnès Rouleau; Xavier Ligneau; Florence Gbahou; Joël Tardivel-Lacombe; Holger Stark; Walter Schunack; C Robin Ganellin; Jean-Michel Arrang
Therapeutic implications of constitutive activity of receptors: the example of the histamine H3 receptor.
Journal of neural transmission. Supplementum 2003;(64):1-16.
2003: Catherine Pillot; Anne Héron; Jean-Charles Schwartz; Jean-Michel Arrang
Ciproxifan, a histamine H3-receptor antagonist/inverse agonist, modulates the effects of methamphetamine on neuropeptide mRNA expression in rat striatum.
The European journal of neuroscience 2003;17(2):307-14.
2002: Astrid Sasse; Xavier Ligneau; Agnès Rouleau; Sigurd Elz; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Influence of bulky substituents on histamine h(3) receptor agonist/antagonist properties.
Journal of medicinal chemistry 2002;45(18):4000-10.
2002: Catherine Pillot; Jordi Ortiz; Anne Héron; Sophie Ridray; Jean-Charles Schwartz; Jean-Michel Arrang
Ciproxifan, a histamine H3-receptor antagonist/inverse agonist, potentiates neurochemical and behavioral effects of haloperidol in the rat.
The Journal of neuroscience : the official journal of the Society for Neuroscience 2002;22(16):7272-80.
2002: Sven Grassmann; Bassem Sadek; Xavier Ligneau; Sigurd Elz; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Holger Stark; Walter Schunack
Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H(3)-receptor antagonists.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 2002;15(4):367-78.
2002: Joachim Apelt; Xavier Ligneau; Heinz H Pertz; Jean-Michel Arrang; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Development of a new class of nonimidazole histamine H(3) receptor ligands with combined inhibitory histamine N-methyltransferase activity.
Journal of medicinal chemistry 2002;45(5):1128-41.
2002: Séverine Morisset; C Pilon; Joël Tardivel-Lacombe; D Weinstein; W Rostene; C Betancur; Pierre Sokoloff; Jean-Charles Schwartz; Jean-Michel Arrang
Acute and chronic effects of methamphetamine on tele-methylhistamine levels in mouse brain: selective involvement of the D(2) and not D(3) receptor.
The Journal of pharmacology and experimental therapeutics 2002;300(2):621-8.
2002: Catherine Pillot; A Heron; Véronique Cochois; Joël Tardivel-Lacombe; Xavier Ligneau; Jean-Charles Schwartz; Jean-Michel Arrang
A detailed mapping of the histamine H(3) receptor and its gene transcripts in rat brain.
Neuroscience 2002;114(1):173-93.
2002: Agnès Rouleau; Xavier Ligneau; Joël Tardivel-Lacombe; Séverine Morisset; Florence Gbahou; Jean-Charles Schwartz; Jean-Michel Arrang
Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.
British journal of pharmacology 2002;135(2):383-92.
2001: Jean-Charles Schwartz; Séverine Morisset; Agnès Rouleau; Joël Tardivel-Lacombe; Florence Gbahou; Xavier Ligneau; Anne Héron; Astrid Sasse; Holger Stark; Walter Schunack; R C Ganellin; Jean-Michel Arrang
Application of genomics to drug design: the example of the histamine H3 receptor.
European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 2001;11(6):441-8.
2001: Anne Héron; Agnès Rouleau; Véronique Cochois; Catherine Pillot; Jean-Charles Schwartz; Jean-Michel Arrang
Expression analysis of the histamine H(3) receptor in developing rat tissues.
Mechanisms of development 2001;105(1-2):167-73.
2001: Holger Stark; Wolfgang Sippl; Xavier Ligneau; Jean-Michel Arrang; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack
Different antagonist binding properties of human and rat histamine H3 receptors.
Bioorganic & medicinal chemistry letters 2001;11(7):951-4.
2001: Joël Tardivel-Lacombe; Séverine Morisset; Florence Gbahou; Jean-Charles Schwartz; Jean-Michel Arrang
Chromosomal mapping and organization of the human histamine H3 receptor gene.
Neuroreport 2001;12(2):321-4.
2001: Astrid Sasse; Xavier Ligneau; Bassem Sadek; Sigurd Elz; Heinz H Pertz; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack; Holger Stark
Benzophenone derivatives and related compounds as potent histamine H3-receptor antagonists and potential PET/SPECT ligands.
Archiv der Pharmazie 2001;334(2):45-52.
2001: Séverine Morisset; Astrid Sasse; Florence Gbahou; Anne Héron; Xavier Ligneau; Joël Tardivel-Lacombe; Jean-Charles Schwartz; Jean-Michel Arrang
The rat H3 receptor: gene organization and multiple isoforms.
Biochemical and biophysical research communications 2001;280(1):75-80.
2001: Holger Stark; Jean-Michel Arrang; Xavier Ligneau; Monique Garbarg; C Robin Ganellin; Jean-Charles Schwartz; Walter Schunack
The histamine H3 receptor and its ligands.
Progress in medicinal chemistry 2001;38():279-308.
2000: Séverine Morisset; Agnès Rouleau; Xavier Ligneau; Florence Gbahou; Joël Tardivel-Lacombe; Holger Stark; Walter Schunack; C Robin Ganellin; Jean-Charles Schwartz; Jean-Michel Arrang
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
Nature 2000;408(6814):860-4.
2000: Xavier Ligneau; Séverine Morisset; Joël Tardivel-Lacombe; Florence Gbahou; C Robin Ganellin; Holger Stark; Walter Schunack; Jean-Charles Schwartz; Jean-Michel Arrang
Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain.
British journal of pharmacology 2000;131(7):1247-50.
2000: Holger Stark; Bassem Sadek; Michael Krause; Annette Hüls; Xavier Ligneau; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
Novel histamine H(3)-receptor antagonists with carbonyl-substituted 4-(3-(phenoxy)propyl)-1H-imidazole structures like ciproxifan and related compounds.
Journal of medicinal chemistry 2000;43(21):3987-94.
2000: Holger Stark; Xavier Ligneau; Bassem Sadek; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
Analogues and derivatives of ciproxifan, a novel prototype for generating potent histamine H3-receptor antagonists.
Bioorganic & medicinal chemistry letters 2000;10(20):2379-82.
2000: G Drutel; Markus Kathmann; Anne Héron; Claude Gros; S Macé; Jean-Charles Schwartz; Jean-Michel Arrang
Two splice variants of the hypoxia-inducible factor HIF-1alpha as potential dimerization partners of ARNT2 in neurons.
The European journal of neuroscience 2000;12(10):3701-8.
2000: Astrid Sasse; Bassem Sadek; Xavier Ligneau; Sigurd Elz; Heinz H Pertz; Peter Luger; C Robin Ganellin; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack; Holger Stark
New histamine H(3)-receptor ligands of the proxifan series: imoproxifan and other selective antagonists with high oral in vivo potency.
Journal of medicinal chemistry 2000;43(17):3335-43.
2000: Joël Tardivel-Lacombe; Agnès Rouleau; Anne Héron; Séverine Morisset; Catherine Pillot; Véronique Cochois; Jean-Charles Schwartz; Jean-Michel Arrang
Cloning and cerebral expression of the guinea pig histamine H3 receptor: evidence for two isoforms.
Neuroreport 2000;11(4):755-9.
2000: C Ito; Séverine Morisset; Marie-Odile Krebs; Jean-Pierre Olié; Henri Lôo; Marie-France Poirier; Lars Lannfelt; Jean-Charles Schwartz; Jean-Michel Arrang
Histamine H2 receptor gene variants: lack of association with schizophrenia.
Molecular psychiatry 2000;5(2):159-64.
2000: Séverine Morisset; Elisabeth Traiffort; Jean-Michel Arrang; Jean-Charles Schwartz
Changes in histamine H3 receptor responsiveness in mouse brain.
Journal of neurochemistry 2000;74(1):339-46.
1999: G Drutel; Anne Héron; Markus Kathmann; Claude Gros; S Macé; M Plotkine; Jean-Charles Schwartz; Jean-Michel Arrang
ARNT2, a transcription factor for brain neuron survival?
The European journal of neuroscience 1999;11(5):1545-53.
1999: Séverine Morisset; U G Sahm; Elisabeth Traiffort; Joël Tardivel-Lacombe; Jean-Michel Arrang; Jean-Charles Schwartz
Atypical neuroleptics enhance histamine turnover in brain via 5-Hydroxytryptamine2A receptor blockade.
The Journal of pharmacology and experimental therapeutics 1999;288(2):590-6.
1998: C Robin Ganellin; F Leurquin; A Piripitsi; Jean-Michel Arrang; Monique Garbarg; Xavier Ligneau; Walter Schunack; Jean-Charles Schwartz
Synthesis of potent non-imidazole histamine H3-receptor antagonists.
Archiv der Pharmazie 1998;331(12):395-404.
1998: Holger Stark; Xavier Ligneau; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
General construction pattern of histamine H3-receptor antagonists: change of a paradigm.
Bioorganic & medicinal chemistry letters 1998;8(15):2011-6.
1998: Holger Stark; Annette Hüls; Xavier Ligneau; K Purand; Heinz H Pertz; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
Development of FUB 181, a selective histamine H3-receptor antagonist of high oral in vivo potency with 4-(omega-(arylalkyloxy)alkyl)-1H-imidazole structure.
Archiv der Pharmazie 1998;331(6):211-8.
1997: Holger Stark; Annette Hüls; Xavier Ligneau; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
Search for novel leads for histamine H3-receptor antagonists: oxygen-containing derivatives.
Die Pharmazie 1997;52(7):495-500.
1997: Holger Stark; Xavier Ligneau; R Lipp; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
Search for novel leads for histamine H3-receptor antagonists: amine derivatives.
Die Pharmazie 1997;52(6):419-23.
1996: G Drutel; M Kathmann; A Heron; Jean-Charles Schwartz; Jean-Michel Arrang
Cloning and selective expression in brain and kidney of ARNT2 homologous to the Ah receptor nuclear translocator (ARNT).
Biochemical and biophysical research communications 1996;225(2):333-9.
1996: Annette Hüls; K Purand; Holger Stark; S Reidemeister; Xavier Ligneau; Jean-Michel Arrang; Jean-Charles Schwartz; Walter Schunack
Novel histamine H3-receptor antagonists with benzyl ether structure or related moieties: synthesis and structure-activity relationships.
Archiv der Pharmazie 1996;329(8-9):379-85.
1996: Holger Stark; K Purand; Xavier Ligneau; Agnès Rouleau; Jean-Michel Arrang; Monique Garbarg; Jean-Charles Schwartz; Walter Schunack
Novel carbamates as potent histamine H3 receptor antagonists with high in vitro and oral in vivo activity.
Journal of medicinal chemistry 1996;39(5):1157-63.
1996: Claas-Hinrich Lammers; Paul Schweitzer; P Facchinetti; Jean-Michel Arrang; Samuel G Madamba; George R Siggins; Daniele Piomelli
Arachidonate 5-lipoxygenase and its activating protein: prominent hippocampal expression and role in somatostatin signaling.
Journal of neurochemistry 1996;66(1):147-52.
1995: C Robin Ganellin; S K Hosseini; Y S Khalaf; W Tertiuk; Jean-Michel Arrang; Monique Garbarg; Xavier Ligneau; Jean-Charles Schwartz
Design of potent non-thiourea H3-receptor histamine antagonists.
Journal of medicinal chemistry 1995;38(17):3342-50.
1995: Jean-Michel Arrang; G Drutel; Monique Garbarg; Martial Ruat; Elisabeth Traiffort; Jean-Charles Schwartz
Molecular and functional diversity of histamine receptor subtypes.
Annals of the New York Academy of Sciences 1995;757():314-23.
1995: Jean-Michel Arrang; G Drutel; Jean-Charles Schwartz
Characterization of histamine H3 receptors regulating acetylcholine release in rat entorhinal cortex.
British journal of pharmacology 1995;114(7):1518-22.
1995: C Robin Ganellin; A Fkyerat; S K Hosseini; Y S Khalaf; A Piripitsi; W Tertiuk; Jean-Michel Arrang; Monique Garbarg; Xavier Ligneau; Jean-Charles Schwartz
Structure-activity studies with histamine H3-receptor ligands.
Journal de pharmacie de Belgique 1995;50(2-3):179-87.
1995: G Drutel; Jean-Michel Arrang; J Diaz; C Wisnewsky; K Schwartz; Jean-Charles Schwartz
Cloning of OL1, a putative olfactory receptor and its expression in the developing rat heart.
Receptors & channels 1995;3(1):33-40.
1994: M Le Coniat; Elisabeth Traiffort; Martial Ruat; Jean-Michel Arrang; R Berger
Chromosomal localization of the human histamine H1-receptor gene.
Human genetics 1994;94(2):186-8.
1994: Jorge Diaz; Marisa Vizuete; Elisabeth Traiffort; Jean-Michel Arrang; Martial Ruat; Jean-Charles Schwartz
Localization of the histamine H2 receptor and gene transcripts in rat stomach: back to parietal cells.
Biochemical and biophysical research communications 1994;198(3):1195-202.
1994: R Leurs; Elisabeth Traiffort; Jean-Michel Arrang; Joël Tardivel-Lacombe; Martial Ruat; Jean-Charles Schwartz
Guinea pig histamine H1 receptor. II. Stable expression in Chinese hamster ovary cells reveals the interaction with three major signal transduction pathways.
Journal of neurochemistry 1994;62(2):519-27.
1994: Elisabeth Traiffort; R Leurs; Jean-Michel Arrang; Joël Tardivel-Lacombe; Jorge Diaz; Jean-Charles Schwartz; Martial Ruat
Guinea pig histamine H1 receptor. I. Gene cloning, characterization, and tissue expression revealed by in situ hybridization.
Journal of neurochemistry 1994;62(2):507-18.
1993: Martial Ruat; Elisabeth Traiffort; R Leurs; Joël Tardivel-Lacombe; Jorge Diaz; Jean-Michel Arrang; Jean-Charles Schwartz
Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.
Proceedings of the National Academy of Sciences of the United States of America 1993;90(18):8547-51.
1993: Martial Ruat; Elisabeth Traiffort; Jean-Michel Arrang; Joël Tardivel-Lacombe; Jorge Diaz; R Leurs; Jean-Charles Schwartz
A novel rat serotonin (5-HT6) receptor: molecular cloning, localization and stimulation of cAMP accumulation.
Biochemical and biophysical research communications 1993;193(1):268-76.
1992: R Lipp; Jean-Michel Arrang; Monique Garbarg; P Luger; Jean-Charles Schwartz; Walter Schunack
Synthesis, absolute configuration, stereoselectivity, and receptor selectivity of (alpha R, beta S)-alpha,beta-dimethylhistamine, a novel high potent histamine H3 receptor agonist.
Journal of medicinal chemistry 1992;35(23):4434-41.
1992: Monique Garbarg; Jean-Michel Arrang; Agnès Rouleau; Xavier Ligneau; M D Tuong; Jean-Charles Schwartz; C Robin Ganellin
S-[2-(4-imidazolyl)ethyl]isothiourea, a highly specific and potent histamine H3 receptor agonist.
The Journal of pharmacology and experimental therapeutics 1992;263(1):304-10.
1992: Elisabeth Traiffort; Martial Ruat; Jean-Michel Arrang; R Leurs; Daniele Piomelli; Jean-Charles Schwartz
Expression of a cloned rat histamine H2 receptor mediating inhibition of arachidonate release and activation of cAMP accumulation.
Proceedings of the National Academy of Sciences of the United States of America 1992;89(7):2649-53.
1992: Martial Ruat; Elisabeth Traiffort; R Leurs; Jean-Michel Arrang; G Kouyoumdjian; Joël Tardivel-Lacombe; Daniele Piomelli; G Diaz; Jean-Charles Schwartz
Molecular biology and pharmacology of histamine receptor subtypes.
Clinical neuropharmacology 1992;15 Suppl 1 Pt A():149A-150A.
1991: Martial Ruat; Elisabeth Traiffort; Jean-Michel Arrang; R Leurs; Jean-Charles Schwartz
Cloning and tissue expression of a rat histamine H2-receptor gene.
Biochemical and biophysical research communications 1991;179(3):1470-8.
1991: Jean-Michel Arrang; C Gulat-Marnay; N Defontaine; Jean-Charles Schwartz
Regulation of histamine release in rat hypothalamus and hippocampus by presynaptic galanin receptors.
Peptides 1991;12(5):1113-7.
1991: J C Schwartz; Jean-Michel Arrang; Monique Garbarg; H Pollard; Martial Ruat
Histaminergic transmission in the mammalian brain.
Physiological reviews 1991;71(1):1-51.
1991: R Lipp; Jean-Michel Arrang; J Buschmann; Monique Garbarg; P Luger; Walter Schunack; Jean-Charles Schwartz
Novel chiral H3-receptor agonists.
Agents and actions. Supplements 1991;33():277-82.
1991: Jean-Michel Arrang; Monique Garbarg; Jean-Charles Schwartz; R Lipp; Holger Stark; Walter Schunack; JM Lecomte
The histamine H3-receptor: pharmacology, roles and clinical implications studied with agonists.
Agents and actions. Supplements 1991;33():55-67.
1990: M I Martinez-Mir; H Pollard; J Moreau; Jean-Michel Arrang; Martial Ruat; Elisabeth Traiffort; Jean-Charles Schwartz; J M Palacios
Three histamine receptors (H1, H2 and H3) visualized in the brain of human and non-human primates.
Brain research 1990;526(2):322-7.
1990: C Gulat-Marnay; A Lafitte; Jean-Michel Arrang; Jean-Charles Schwartz
Modulation of histamine release in the rat brain by kappa-opioid receptors.
Journal of neurochemistry 1990;55(1):47-53.
1990: Jean-Michel Arrang; J Roy; J L Morgat; Walter Schunack; Jean-Charles Schwartz
Histamine H3 receptor binding sites in rat brain membranes: modulations by guanine nucleotides and divalent cations.
European journal of pharmacology 1990;188(4-5):219-27.
1990: Jean-Charles Schwartz; Jean-Michel Arrang; Monique Garbarg; H Pollard
Plenary lecture. A third histamine receptor subtype: characterisation, localisation and functions of the H3-receptor.
Agents and actions 1990;30(1-2):13-23.
1990: Jean-Charles Schwartz; Jean-Michel Arrang; M Garbarg; C Gulat-Marnay; H Pollard
Modulation of histamine synthesis and release in brain via presynaptic autoreceptors and heteroreceptors.
Annals of the New York Academy of Sciences 1990;604():40-54.
1989: C Gulat-Marnay; A Lafitte; Jean-Michel Arrang; Jean-Charles Schwartz
Modulation of histamine release and synthesis in the brain mediated by alpha 2-adrenoceptors.
Journal of neurochemistry 1989;53(2):513-8.
1989: Jean-Michel Arrang; Monique Garbarg; Jean-Charles Lancelot; JM Lecomte; H Pollard; M Robba; W Schunack; Jean-Charles Schwartz
The third histamine receptor. Highly potent and selective ligands.
International archives of allergy and applied immunology 1989;88(1-2):79-81.
1989: Jean-Charles Schwartz; Jean-Michel Arrang; Monique Garbarg; H Pollard
Histamine H3 receptors in the brain: potent and selective ligands.
Psychopharmacology series 1989;7():10-9.
1989: C Gulat-Marnay; A Lafitte; Jean-Michel Arrang; Jean-Charles Schwartz
Regulation of histamine release and synthesis in the brain by muscarinic receptors.
Journal of neurochemistry 1989;52(1):248-54.
1988: Jean-Michel Arrang; N Defontaine; Jean-Charles Schwartz
Phencyclidine blocks histamine H3-receptors in rat brain.
European journal of pharmacology 1988;157(1):31-5.
1988: Jean-Michel Arrang; Monique Garbarg; Jean-Charles Lancelot; JM Lecomte; H Pollard; M Robba; W Schunack; Jean-Charles Schwartz
[Potential interest in powerful and specific ligands for the histamine H3 receptor].
Allergie et immunologie 1988;20(9):327-9, 331.
1988: Jean-Michel Arrang; Monique Garbarg; Jean-Charles Lancelot; JM Lecomte; H Pollard; M Robba; W Schunack; Jean-Charles Schwartz
Highly potent and selective ligands for a new class H3 of histamine receptor.
Investigative radiology 1988;23 Suppl 1():S130-2.
1988: Jean-Michel Arrang; B Devaux; J P Chodkiewicz; Jean-Charles Schwartz
H3-receptors control histamine release in human brain.
Journal of neurochemistry 1988;51(1):105-8.
1987: Jean-Michel Arrang; Monique Garbarg; Jean-Charles Schwartz
Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors.
Neuroscience 1987;23(1):149-57.
1987: Jean-Michel Arrang; Monique Garbarg; Jean-Charles Lancelot; JM Lecomte; H Pollard; M Robba; W Schunack; J C Schwartz
Highly potent and selective ligands for histamine H3-receptors.
Nature 1987;327(6118):117-23.