Pawel Kafarski

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Matczak-Jon Ewa; Slepokura Katarzyna; Kafarski Pawel; Skrzynska Izabela; Jon Marek
Conformational isomers of the [(5-methyl-2-pyridinio)aminomethylene]diphosphonate dianion and [(5-methyl-2-pyridyl)aminomethylene]diphosphonate trianion in salts with 4-aminopyridine and ammonia.
Doskocz Marek; Strupinska Agnieszka; Roszak Szczepan; Prokopowicz Monika; Koole Leo H; Kafarski Pawel
Theoretical study of spin-spin coupling across the hydrogen (O-H...N) bond in adenosine derivatives.
McGowan Sheena; Porter Corrine J; Lowther Jonathan; Stack Colin M; Golding Sarah J; Skinner-Adams Tina S; Trenholme Katharine R; Teuscher Franka; Donnelly Sheila M; Grembecka Jolanta; Mucha Artur; Kafarski Pawel; Degori Ross; Buckle Ashley M; Gardiner Donald L; Whisstock James C; Dalton John P
Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase.

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2009: Matczak-Jon Ewa; Slepokura Katarzyna; Kafarski Pawel; Skrzynska Izabela; Jon Marek
Conformational isomers of the [(5-methyl-2-pyridinio)aminomethylene]diphosphonate dianion and [(5-methyl-2-pyridyl)aminomethylene]diphosphonate trianion in salts with 4-aminopyridine and ammonia.
Acta crystallographica. Section C, Crystal structure communications 2009;65(Pt 6):o261-6.
2009: Doskocz Marek; Strupinska Agnieszka; Roszak Szczepan; Prokopowicz Monika; Koole Leo H; Kafarski Pawel
Theoretical study of spin-spin coupling across the hydrogen (O-H...N) bond in adenosine derivatives.
Journal of molecular modeling 2009;15(6):651-8.
2009: McGowan Sheena; Porter Corrine J; Lowther Jonathan; Stack Colin M; Golding Sarah J; Skinner-Adams Tina S; Trenholme Katharine R; Teuscher Franka; Donnelly Sheila M; Grembecka Jolanta; Mucha Artur; Kafarski Pawel; Degori Ross; Buckle Ashley M; Gardiner Donald L; Whisstock James C; Dalton John P
Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase.
Proceedings of the National Academy of Sciences of the United States of America 2009;106(8):2537-42.
2008: Podstawka Edyta; Kafarski Pawel; Proniewicz Leonard M
Structural properties of L-X-L-Met-L-Ala phosphonate tripeptides: a combined FT-IR, FT-RS, and SERS spectroscopy studies and DFT calculations.
The journal of physical chemistry. A 2008;112(46):11744-55.
2008: Latajka R; Jewginski M; Makowski M; Pawelczak M; Huber T; Sewald N; Kafarski P
Pentapeptides containing two dehydrophenylalanine residues--synthesis, structural studies and evaluation of their activity towards cathepsin C.
Journal of peptide science : an official publication of the European Peptide Society 2008;14(10):1084-95.
2008: Vassiliou Stamatia; Grabowiecka Agnieszka; Kosikowska Paulina; Yiotakis Athanasios; Kafarski Pawel; Berlicki Lukasz
Design, synthesis, and evaluation of novel organophosphorus inhibitors of bacterial ureases.
Journal of medicinal chemistry 2008;51(18):5736-44.
2008: Cunningham Eithne; Drag Marcin; Kafarski Pawel; Bell Angus
Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors.
Antimicrobial agents and chemotherapy 2008;52(9):3221-8.
2008: Jaskula Barbara; Kafarski Pawel; Aerts Guido; De Cooman Luc
A kinetic study on the isomerization of hop alpha-acids.
Journal of agricultural and food chemistry 2008;56(15):6408-15.
2008: Forlani Giuseppe; Occhipinti Andrea; Berlicki Lukasz; Dziedziola Gabriela; Wieczorek Anna; Kafarski Pawel
Tailoring the structure of aminobisphosphonates to target plant P5C reductase.
Journal of agricultural and food chemistry 2008;56(9):3193-9.
2008: Forlani Giuseppe; Pavan Mauro; Gramek Magdalena; Kafarski Pawel; Lipok Jacek
Biochemical bases for a widespread tolerance of cyanobacteria to the phosphonate herbicide glyphosate.
Plant & cell physiology 2008;49(3):443-56.
2008: Mucha Artur; Lämmerhofer Michael; Lindner Wolfgang; Pawelczak Malgorzata; Kafarski Pawel
Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase.
Bioorganic & medicinal chemistry letters 2008;18(5):1550-4.
2008: Lisowski M; Latajka R; Picur B; Lis T; Bryndal I; Rospenk M; Makowski M; Kafarski P
Combined effect of the DeltaPhe or DeltaAla residue and the p-nitroanilide group on a didehydropeptides conformation.
Biopolymers 2008;89(3):220-34.
2008: Minta Ewelina; Kafarski Pawel; Martinez Jean; Rolland Valérie
Synthesis of cyclooctapeptides: constraints analogues of the peptidic neurotoxin, omega-agatoxine IVB-an experimental point of view.
Journal of peptide science : an official publication of the European Peptide Society 2008;14(3):267-77.
2007: Skinner-Adams Tina S; Lowther Jonathan; Teuscher Franka; Stack Colin M; Grembecka Jolanta; Mucha Artur; Kafarski Pawel; Trenholme Katharine R; Dalton John P; Gardiner Donald L
Identification of phosphinate dipeptide analog inhibitors directed against the Plasmodium falciparum M17 leucine aminopeptidase as lead antimalarial compounds.
Journal of medicinal chemistry 2007;50(24):6024-31.
2007: Rudzinska Ewa; Berlicki Lukasz; Mucha Artur; Kafarski Pawel
Analysis of pD-dependent complexation of N-benzyloxycarbonylaminophosphonic acids by alpha-cyclodextrin. Enantiodifferentiation of phosphonic acid pKa values.
Chirality 2007;19(10):764-8.
2007: Teuscher Franka; Lowther Jonathan; Skinner-Adams Tina S; Spielmann Tobias; Dixon Matthew W A; Stack Colin M; Donnelly Sheila; Mucha Artur; Kafarski Pawel; Vassiliou Stamatia; Gardiner Donald L; Dalton John P; Trenholme Katharine R
The M18 aspartyl aminopeptidase of the human malaria parasite Plasmodium falciparum.
The Journal of biological chemistry 2007;282(42):30817-26.
2007: Forlani Giuseppe; Giberti Samuele; Berlicki Lukasz; Petrollino Davide; Kafarski Pawel
Plant P5C reductase as a new target for aminomethylenebisphosphonates.
Journal of agricultural and food chemistry 2007;55(11):4340-7.
2007: Vassiliou Stamatia; Xeilari Metaxia; Yiotakis Athanasios; Grembecka Jolanta; Pawelczak Malgorzata; Kafarski Pawel; Mucha Artur
A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.
Bioorganic & medicinal chemistry 2007;15(9):3187-200.
2007: Stack Colin M; Lowther Jonathan; Cunningham Eithne; Donnelly Sheila; Gardiner Donald L; Trenholme Katharine R; Skinner-Adams Tina S; Teuscher Franka; Grembecka Jolanta; Mucha Artur; Kafarski Pawel; Lua Linda; Bell Angus; Dalton John P
Characterization of the Plasmodium falciparum M17 leucyl aminopeptidase. A protease involved in amino acid regulation with potential for antimalarial drug development.
The Journal of biological chemistry 2007;282(3):2069-80.
2007: Rudzinska Ewa; Poliwoda Anna; Berlicki Lukasz; Mucha Artur; Dzygiel Pawel; Wieczorek Piotr P; Kafarski Pawel
Enantiodifferentiation of N-benzyloxycarbonylaminophosphonic and phosphinic acids and their esters using cyclodextrins by means of capillary electrophoresis.
Journal of chromatography. A 2007;1138(1-2):284-90.
2006: Preinerstorfer Beatrix; Lubda Dieter; Mucha Artur; Kafarski Pawel; Lindner Wolfgang; Lämmerhofer Michael
Stereoselective separations of chiral phosphinic acid pseudodipeptides by CEC using silica monoliths modified with an anion-exchange-type chiral selector.
Electrophoresis 2006;27(21):4312-20.
2006: Jagiello Monika; Minta Ewelina; Chojnacka Katarzyna; Kafarski Pawel
Mode of biosorption of chromium(III) by Spirulina species cells from aqueous solutions.
Water environment research : a research publication of the Water Environment Federation 2006;78(7):740-3.
2006: Berlicki Lukasz; Kafarski Pawel
Computer-aided analysis of the interactions of glutamine synthetase with its inhibitors.
Bioorganic & medicinal chemistry 2006;14(13):4578-85.
2006: Matczak-Jon Ewa; Kurzak Barbara; Kafarski Pawel; Wozna Agnieszka
Coordination abilities of piperyd-1-yl-methane-1,1-diphosphonic acids towards zinc(II), magnesium(II) and calcium(II): potentiometric and NMR studies.
Journal of inorganic biochemistry 2006;100(7):1155-66.
2006: Mucha A; Kunert A; Grembecka J; Pawelczak M; Kafarski P
A phosphonamidate containing aromatic N-terminal amino group as inhibitor of leucine aminopeptidase-design, synthesis and stability.
European journal of medicinal chemistry 2006;41(6):768-72.
2006: Brzezinska-Rodak Malgorzata; Zymanczyk-Duda Ewa; Klimek-Ochab Magdalena; Kafarski Pawel; Lejczak Barbara
A simple and green procedure for the microbial effective synthesis of 1-phenylethyl alcohol in both enantiomeric forms.
Biotechnology letters 2006;28(7):511-3.
2006: Matczak-Jon Ewa; Slepokura Katarzyna; Kafarski Pawel
[(5-Bromopyridinium-2-ylamino)(phosphono)methyl]phosphonate.
Acta crystallographica. Section C, Crystal structure communications 2006;62(Pt 3):o132-5.
2006: Forlani Giuseppe; Obojska Agnieszka; Berlicki Lukasz; Kafarski Pawel
Phosphinothricin analogues as inhibitors of plant glutamine synthetases.
Journal of agricultural and food chemistry 2006;54(3):796-802.
2005: Berlicki Lukasz; Obojska Agnieszka; Forlani Giuseppe; Kafarski Pawel
Design, synthesis, and activity of analogues of phosphinothricin as inhibitors of glutamine synthetase.
Journal of medicinal chemistry 2005;48(20):6340-9.
2005: Drag Marcin; Grembecka Jolanta; Pawelczak Malgorzata; Kafarski Pawel
alpha-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases.
European journal of medicinal chemistry 2005;40(8):764-71.
2005: Jasicka-Misiak Izabela; Wieczorek Piotr P; Kafarski Pawel
Crotonic acid as a bioactive factor in carrot seeds (Daucus carota L.).
Phytochemistry 2005;66(12):1485-91.
2005: Matczak-Jon Ewa; Videnova-Adrabinska Veneta; Burzynska Agnieszka; Kafarski Pawel; Lis Tadeusz
Solid-state molecular organization and solution behavior of methane-1,1-diphosphonic acid derivatives of heterocyclic amines: the role of the topochemical ring modification and the intramolecular hydrogen bonds in monosubstituted piperid-1-ylmethane-1,1-diphosphonic acids.
Chemistry (Weinheim an der Bergstrasse, Germany) 2005;11(8):2357-72.
2004: Jasicka-Misiak Izabela; Lipok Jacek; Nowakowska Ewa M; Wieczorek Piotr P; Mlynarz Piotr; Kafarski Pawel
Antifungal activity of the carrot seed oil and its major sesquiterpene compounds.
Zeitschrift für Naturforschung. C, Journal of biosciences 2004;59(11-12):791-6.
2004: Gasowska Beata; Kafarski Pawel; Wojtasek Hubert
Interaction of mushroom tyrosinase with aromatic amines, o-diamines and o-aminophenols.
Biochimica et biophysica acta 2004;1673(3):170-7.
2004: Obojska Agnieszka; Berlicki Lukasz; Kafarski Pawel; Lejczak Barbara; Chicca Milvia; Forlani Giuseppe
Herbicidal pyridyl derivatives of aminomethylene-bisphosphonic acid inhibit plant glutamine synthetase.
Journal of agricultural and food chemistry 2004;52(11):3337-44.
2004: Mucha Artur; Pawel Malgorzata; Hurek Józef; Kafarski Pawel
Synthesis and activity of phosphinic tripeptide inhibitors of cathepsin C.
Bioorganic & medicinal chemistry letters 2004;14(12):3113-6.
2004: Drag Marcin; Jezierski Adam; Kafarski Pawel
First example of the chemical, oxidative cleavage of the C-P bond in aminophosphonate chemistry. The oxidation of 1-amino-1-(3,4-dihydroxyphenyl)methylphosphonic acid by NaIO4.
Chemical communications (Cambridge, England) 2004;(9):1132-3.
2004: Sanders John M; Ghosh Subhash; Chan Julian M W; Meints Gary; Wang Hong; Raker Amy M; Song Yongcheng; Colantino Alison; Burzynska Agnieszka; Kafarski Pawel; Morita Craig T; Oldfield Eric
Quantitative structure-activity relationships for gammadelta T cell activation by bisphosphonates.
Journal of medicinal chemistry 2004;47(2):375-84.
2003: Sanders John M; Gómez Aurora Ortiz; Mao Junhong; Meints Gary A; Van Brussel Erin M; Burzynska Agnieszka; Kafarski Pawel; González-Pacanowska Dolores; Oldfield Eric
3-D QSAR investigations of the inhibition of Leishmania major farnesyl pyrophosphate synthase by bisphosphonates.
Journal of medicinal chemistry 2003;46(24):5171-83.
2003: Rudzinska Ewa; Wieczorek Piotr; Kafarski Pawel
Separation of aminoalkanephosphonic acid enantiomers by indirect UV detection capillary electrophoresis with application of cyclodextrins.
Electrophoresis 2003;24(15):2693-7.
2003: Grembecka Jolanta; Mucha Artur; Cierpicki Tomasz; Kafarski Pawel
The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.
Journal of medicinal chemistry 2003;46(13):2641-55.
2003: Drag Marcin; Pawelczak Malgorzata; Kafarski Pawel
Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase.
Chirality 2003;15 Suppl():S104-7.
2002: Rudzinska Ewa; Dzygiel Pawel; Wieczorek Piotr; Kafarski Pawel
Separation of aromatic aminophosphonic acid enantiomers by capillary electrophoresis with the application of cyclodextrins.
Journal of chromatography. A 2002;979(1-2):115-22.
2002: Brzezinska-Rodak Malorzata; Zymanczyk-Duda Ewa; Kafarski Paweal; Lejczak Barbara
Application of fungi as biocatalysts for the reduction of diethyl 1-oxoalkylphosphonates in anhydrous hexane.
Biotechnology progress 2002;18(6):1287-91.
2002: Gasowska Beata; Wojtasek Hubert; Hurek Józef; Drag Marcin; Nowak Kornel; Kafarski Pawel
Redox reaction between amino-(3,4-dihydroxyphenyl)methyl phosphonic acid and dopaquinone is responsible for the apparent inhibitory effect on tyrosinase.
European journal of biochemistry / FEBS 2002;269(16):4098-104.
2002: Martin Michael B; Sanders John M; Kendrick Howard; de Luca-Fradley Kate; Lewis Jared C; Grimley Joshua S; Van Brussel Erin M; Olsen Jeffrey R; Meints Gary A; Burzynska Agnieszka; Kafarski Pawel; Croft Simon L; Oldfield Eric
Activity of bisphosphonates against Trypanosoma brucei rhodesiense.
Journal of medicinal chemistry 2002;45(14):2904-14.
2002: Obojska Agnieszka; Ternan Nigel G; Lejczak Barbara; Kafarski Pawel; McMullan Geoff
Organophosphonate utilization by the thermophile Geobacillus caldoxylosilyticus T20.
Applied and environmental microbiology 2002;68(4):2081-4.
2001: Kafarski P; Lejczak B
Aminophosphonic acids of potential medical importance.
Current medicinal chemistry. Anti-cancer agents 2001;1(3):301-12.
2001: Ziora Z; Kafarski P; Holband J; Wójcik G
Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides.
Journal of peptide science : an official publication of the European Peptide Society 2001;7(9):466-73.
2001: Klimek M; Lejczak B; Kafarski P; Forlani G
Metabolism of the phosphonate herbicide glyphosate by a non-nitrate-utilizing strain of Penicillium chrysogenum.
Pest management science 2001;57(9):815-21.
2001: Grembecka J; Kafarski P
Leucine aminopeptidase as a target for inhibitor design.
Mini reviews in medicinal chemistry 2001;1(2):133-44.
2001: Makowski M; Pawelczak M; Latajka R; Nowak K; Kafarski P
Synthesis of tetrapeptide p-nitrophenylanilides containing dehydroalanine and dehydrophenylalanine and their influence on cathepsin C activity.
Journal of peptide science : an official publication of the European Peptide Society 2001;7(3):141-5.
2000: Dzygiel P; Rudzinska E; Wieczorek P; Kafarski P
Determination of optical purity of phosphonic acid analogues of aromatic amino acids by capillary electrophoresis with alpha-cyclodextrin.
Journal of chromatography. A 2000;895(1-2):301-7.
2000: Grembecka J; Sokalski W A; Kafarski P
Computer-aided design and activity prediction of leucine aminopeptidase inhibitors.
Journal of computer-aided molecular design 2000;14(6):531-44.
1997: Krzysko-Lupicka T; Strof W; Kubs K; Skorupa M; Wieczorek P; Lejczak B; Kafarski P
The ability of soil-borne fungi to degrade organophosphonate carbon-to-phosphorus bonds.
Applied microbiology and biotechnology 1997;48(4):549-52.

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Pawel Kafarski

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