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Paolo La Colla
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43
Loddo, Roberta
32
Pani, Alessandra
31
Artico, Marino
28
Loi, Anna Giulia
27
Massa, Silvio
26
Marongiu, Maria Elena
19
Musiu, Chiara
14
Tramontano, Enzo
13
Mai, Antonello
13
Silvestri, Romano
13
Collu, Gabriella
12
De Montis, A
12
Sanna, Giuseppina
10
Busonera, Bernardetta
10
Novellino, Ettore
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All Publications
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2009: El-Brollosy Nasser R; Al-Deeb Omar A; El-Emam Ali A; Pedersen Erik B; La Colla Paolo; Collu Gabriella; Sanna Giuseppina; Loddo Roberta
Synthesis of novel uracil non-nucleoside derivatives as potential reverse transcriptase inhibitors of HIV-1.
Archiv der Pharmazie 2009;342(11):663-70.
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2009: Loksha Yasser M; Pedersen Erik B; Loddo Roberta; La Colla Paolo
Synthesis and anti-HIV-1 activity of 1-substiuted 6-(3-cyanobenzoyl) and [(3-cyanophenyl)fluoromethyl]-5-ethyl-uracils.
Archiv der Pharmazie 2009;342(9):501-6.
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2009: Giampieri Michele; Balbi Alessandro; Mazzei Mauro; La Colla Paolo; Ibba Cristina; Loddo Roberta
Antiviral activity of indole derivatives.
Antiviral research 2009;83(2):179-85.
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2009: Tonelli Michele; Vazzana Iana; Tasso Bruno; Boido Vito; Sparatore Fabio; Fermeglia Maurizio; Paneni Maria Silvia; Posocco Paola; Pricl Sabrina; La Colla Paolo; Ibba Cristina; Secci Barbara; Collu Gabriella; Loddo Roberta
Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives.
Bioorganic & medicinal chemistry 2009;17(13):4425-40.
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2009: Romanowska Joanna; Szymanska-Michalak Agnieszka; Boryski Jerzy; Stawinski Jacek; Kraszewski Adam; Loddo Roberta; Sanna Giuseppina; Collu Gabriella; Secci Barbara; La Colla Paolo
Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters.
Bioorganic & medicinal chemistry 2009;17(9):3489-98.
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2009: Franzetti Andrea; Caredda Paolo; Ruggeri Claudio; La Colla Paolo; Tamburini Elena; Papacchini Maddalena; Bestetti Giuseppina
Potential applications of surface active compounds by Gordonia sp. strain BS29 in soil remediation technologies.
Chemosphere 2009;75(6):801-7.
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2009: Spallarossa Andrea; Cesarini Sara; Ranise Angelo; Schenone Silvia; Bruno Olga; Borassi Alberto; La Colla Paolo; Pezzullo Margherita; Sanna Giuseppina; Collu Gabriella; Secci Barbara; Loddo Roberta
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
European journal of medicinal chemistry 2009;44(5):2190-201.
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2009: Spallarossa Andrea; Cesarini Sara; Ranise Angelo; Bruno Olga; Schenone Silvia; La Colla Paolo; Collu Gabriella; Sanna Giuseppina; Secci Barbara; Loddo Roberta
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors.
European journal of medicinal chemistry 2009;44(4):1650-63.
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2009: Vicini Paola; Incerti Matteo; La Colla Paolo; Loddo Roberta
Anti-HIV evaluation of benzo[d]isothiazole hydrazones.
European journal of medicinal chemistry 2009;44(4):1801-7.
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2009: Cesarini Sara; Spallarossa Andrea; Ranise Angelo; Schenone Silvia; Rosano Camillo; La Colla Paolo; Sanna Giuseppina; Busonera Bernardetta; Loddo Roberta
N-acylated and N,N'-diacylated imidazolidine-2-thione derivatives and N,N'-diacylated tetrahydropyrimidine-2(1H)-thione analogues: synthesis and antiproliferative activity.
European journal of medicinal chemistry 2009;44(3):1106-18.
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2009: Pani Alessandra; Mandas Antonella; Diaz Giacomo; Abete Claudia; Cocco Pier Luigi; Angius Fabrizio; Brundu Annalisa; Muçaka Nico; Pais Maria Elena; Saba Antonio; Barberini Luigi; Zaru Cristina; Palmas Manuela; Putzu Paolo F; Mocali Alessandra; Paoletti Francesco; La Colla Paolo; Dessì Sandra
Accumulation of neutral lipids in peripheral blood mononuclear cells as a distinctive trait of Alzheimer patients and asymptomatic subjects at risk of disease.
BMC medicine 2009;7():66.
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2008: Tonelli Michele; Paglietti Giuseppe; Boido Vito; Sparatore Fabio; Marongiu Fabio; Marongiu Esther; La Colla Paolo; Loddo Roberta
Antiviral activity of benzimidazole derivatives. I. Antiviral activity of 1-substituted-2-[(benzotriazol-1/2-yl)methyl]benzimidazoles.
Chemistry & biodiversity 2008;5(11):2386-401.
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2008: Vitale G; Carta A; Loriga M; Paglietti G; La Colla P; Busonera B; Collu D; Loddo R
2-Arylbenzimidazoles as antiviral and antiproliferative agents. Part 1.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2008;4(6):605-15.
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2008: Tonelli Michele; Boido Vito; Canu Caterina; Sparatore Anna; Sparatore Fabio; Paneni Maria Silvia; Fermeglia Maurizio; Pricl Sabrina; La Colla Paolo; Casula Laura; Ibba Cristina; Collu David; Loddo Roberta
Antimicrobial and cytotoxic arylazoenamines. Part III: antiviral activity of selected classes of arylazoenamines.
Bioorganic & medicinal chemistry 2008;16(18):8447-65.
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2008: Akhtar Tashfeen; Hameed Shahid; Al-Masoudi Najim A; Loddo Roberta; La Colla Paolo
In vitro antitumor and antiviral activities of new benzothiazole and 1,3,4-oxadiazole-2-thione derivatives.
Acta pharmaceutica (Zagreb, Croatia) 2008;58(2):135-49.
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2008: Cesarini Sara; Spallarossa Andrea; Ranise Angelo; Schenone Silvia; Bruno Olga; La Colla Paolo; Casula Laura; Collu Gabriella; Sanna Giuseppina; Loddo Roberta
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
Bioorganic & medicinal chemistry 2008;16(12):6353-63.
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2008: Carta Antonio; Piras Sandra; Paglietti Giuseppe; Pricl Sabrina; La Colla Paolo; Busonera Bernardetta; Loddo Roberta
2(3)-Aryl-thio(oxy)-methylquinoxaline derivatives: a new class of P-glycoprotein-mediated drug efflux inhibitors.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2008;4(3):194-205.
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2008: Angusti Angela; Manfredini Stefano; Durini Elisa; Ciliberti Nunzia; Vertuani Silvia; Solaroli Nicola; Pricl Sabrina; Ferrone Marco; Fermeglia Maurizio; Loddo Roberta; Secci Barbara; Visioli Anna; Sanna Tiziana; Collu Gabriella; Pezzullo Margherita; La Colla Paolo
Design, synthesis and anti flaviviridae activity of N(6)-, 5',3'-O- and 5',2'-O-substituted adenine nucleoside analogs.
Chemical & pharmaceutical bulletin 2008;56(4):423-32.
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2008: Cesarini Sara; Spallarossa Andrea; Ranise Angelo; Bruno Olga; La Colla Paolo; Secci Barbara; Collu Gabriella; Loddo Roberta
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: Parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate.
Bioorganic & medicinal chemistry 2008;16(7):4173-85.
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2008: Cesarini Sara; Spallarossa Andrea; Ranise Angelo; Fossa Paola; La Colla Paolo; Sanna Giuseppina; Collu Gabriella; Loddo Roberta
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates.
Bioorganic & medicinal chemistry 2008;16(7):4160-72.
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2008: Mazzei Mauro; Nieddu Erika; Miele Mariangela; Balbi Alessandro; Ferrone Marco; Fermeglia Maurizio; Mazzei Marco T; Pricl Sabrina; La Colla Paolo; Marongiu Fabio; Ibba Cristina; Loddo Roberta
Activity of Mannich bases of 7-hydroxycoumarin against Flaviviridae.
Bioorganic & medicinal chemistry 2008;16(5):2591-605.
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2008: Franzetti Andrea; Bestetti Giuseppina; Caredda Paolo; La Colla Paolo; Tamburini Elena
Surface-active compounds and their role in the access to hydrocarbons in Gordonia strains.
FEMS microbiology ecology 2008;63(2):238-48.
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2008: El-Brollosy Nasser R; Sørensen Esben R; Pedersen Erik B; Sanna Giuseppina; La Colla Paolo; Loddo Roberta
Synthesis and antiviral evaluation of 6-(trifluoromethylbenzyl) and 6-(fluorobenzyl) analogues of HIV drugs emivirine and GCA-186.
Archiv der Pharmazie 2008;341(1):9-19.
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2008: Danel Krzysztof; Larsen Louise M; Pedersen Erik B; Sanna Giuseppina; La Colla Paolo; Loddo Roberta
Synthesis and antiviral activity of new dimeric inhibitors against HIV-1.
Bioorganic & medicinal chemistry 2008;16(1):511-7.
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2007: Carta A; Loriga M; Piras S; Paglietti G; Ferrone M; Fermeglia M; Pricl S; La Colla P; Collu G; Sanna T; Loddo R
Synthesis and anti-picornaviridae in vitro activity of a new class of helicase inhibitors the N,N'-bis[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl] alkyldicarboxamides.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2007;3(6):520-32.
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2007: Pani Alessandra; Norfo Claudia; Abete Claudia; Mulas Claudia; Putzolu Marirosa; Laconi Sergio; Orrù Christina Doriana; Cannas M Dolores; Vascellari Sarah; La Colla Paolo; Dessì Sandra
Antiprion activity of cholesterol esterification modulators: a comparative study using ex vivo sheep fibroblasts and lymphocytes and mouse neuroblastoma cell lines.
Antimicrobial agents and chemotherapy 2007;51(11):4141-7.
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2007: Aly Youssef L; Pedersen Erik B; La Colla Paolo; Loddo Roberta
Synthesis and anti-HIV-1 activity of new MKC-442 analogues with an alkynyl-substituted 6-benzyl group.
Archiv der Pharmazie 2007;340(5):225-35.
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2007: Filosa Rosanna; Peduto Antonella; de Caprariis Paolo; Saturnino Carmela; Festa Michela; Petrella Antonello; Pau Amedeo; Pinna Gérard Aimé; La Colla Paolo; Busonera Bernardetta; Loddo Roberta
Synthesis and antiproliferative properties of N3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine.
European journal of medicinal chemistry 2007;42(3):293-306.
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2007: Carta Antonio; Loriga Mario; Paglietti Giuseppe; Ferrone Marco; Fermeglia Maurizio; Pricl Sabrina; Sanna Tiziana; Ibba Cristina; La Colla Paolo; Loddo Roberta
Design, synthesis, and preliminary in vitro and in silico antiviral activity of [4,7]phenantrolines and 1-oxo-1,4-dihydro-[4,7]phenantrolines against single-stranded positive-sense RNA genome viruses.
Bioorganic & medicinal chemistry 2007;15(5):1914-27.
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2007: Benzaria Samira; Bardiot Dorothée; Bouisset Tony; Counor Clément; Rabeson Céline; Pierra Claire; Storer Richard; Loi Anna Giulia; Cadeddu Alessandra; Mura Massimo; Musiu Chiara; Liuzzi Michel; Loddo Roberta; Bergelson Svetlana; Bichko Vadim; Bridges Edward; Cretton-Scott Erika; Mao John; Sommadossi Jean-Pierre; Seifer Maria; Standring David; Tausek Michele; Gosselin Gilles; La Colla Paolo
2'-C-Methyl branched pyrimidine ribonucleoside analogues: potent inhibitors of RNA virus replication.
Antiviral chemistry & chemotherapy 2007;18(4):225-42.
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2006: Carta Antonio; Loriga Giovanni; Piras Sandra; Paglietti Giuseppe; Ferrone Marco; Fermeglia Maurizio; Pricl Sabrina; La Colla Paolo; Secci Barbara; Collu Gabriella; Loddo Roberta
Synthesis and in vitro evaluation of the anti-viral activity of N-[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkylcarboxamides.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2006;2(6):577-89.
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2006: Filosa Rosanna; Buonerba Mariafrancesca; Loddo Roberta; Busonera Bernardetta; La Colla Paolo; Saturnino Carmela
N, N' (4,5-dihydro-1h-imidazol-2-yl)3-aza-1,10-decane-diamine and N, N'(4,5-dihydro-1H-imidazol-2-yl)3-aza-1, 10-dodecane-diamine antagonize cell proliferation as selective ligands towards topoisomerase II.
The Journal of pharmacy and pharmacology 2006;58(10):1415-20.
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2006: Corona Paola; Vitale Gabriella; Loriga Mario; Paglietti Giuseppe; La Colla Paolo; Collu Gabriella; Sanna Giuseppina; Loddo Roberta
4-Substituted anilino imidazo[1,2-a] and triazolo[4,3-a]quinoxalines. Synthesis and evaluation of in vitro biological activity.
European journal of medicinal chemistry 2006;41(9):1102-7.
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2006: Al-Masoudi Najim A; Al-Masoudi Iman A; Ali Ibrahim A I; Al-Soud Yaseen A; Saeed Bahjat; La Colla Paolo
Amino acid derivatives. Part I. Synthesis, antiviral and antitumor evaluation of new alpha-amino acid esters bearing coumarin side chain.
Acta pharmaceutica (Zagreb, Croatia) 2006;56(2):175-88.
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2006: Vicini Paola; Incerti Matteo; Doytchinova Irini A; La Colla Paolo; Busonera Bernadetta; Loddo Roberta
Synthesis and antiproliferative activity of benzo[d]isothiazole hydrazones.
European journal of medicinal chemistry 2006;41(5):624-32.
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2006: Carta Antonio; Loriga Mario; Piras Sandra; Paglietti Giuseppe; La Colla Paolo; Busonera Bernardetta; Collu Gabriella; Loddo Roberta
Synthesis of variously substituted 3-phenoxymethyl quinoxalin-2-ones and quinoxalines capable to potentiate in vitro the antiproliferative activity of anticancer drugs in multi-drug resistant cell lines.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2006;2(2):113-22.
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2006: Szymanska Agnieszka; Szymczak Marzena; Boryski Jerzy; Stawinski Jacek; Kraszewski Adam; Collu Gabriella; Sanna Giseppina; Giliberti Gabriele; Loddo Roberta; La Colla Paolo
Aryl nucleoside H-phosphonates. Part 15: Synthesis, properties and, anti-HIV activity of aryl nucleoside 5'-alpha-hydroxyphosphonates.
Bioorganic & medicinal chemistry 2006;14(6):1924-34.
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2005: Ranise Angelo; Spallarossa Andrea; Cesarini Sara; Bondavalli Francesco; Schenone Silvia; Bruno Olga; Menozzi Giulia; Fossa Paola; Mosti Luisa; La Colla Massimiliano; Sanna Giuseppina; Murreddu Marta; Collu Gabriella; Busonera Bernardetta; Marongiu Maria Elena; Pani Alessandra; La Colla Paolo; Loddo Roberta
Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives.
Journal of medicinal chemistry 2005;48(11):3858-73.
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2005: Mai Antonello; Artico Marino; Ragno Rino; Sbardella Gianluca; Massa Silvio; Musiu Chiara; Mura Massimo; Marturana Flavia; Cadeddu Alessandra; Maga Giovanni; La Colla Paolo
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydropyrimidin-4(3H)-ones, a new series of potent, broad-spectrum non-nucleoside reverse transcriptase inhibitors belonging to the DABO family.
Bioorganic & medicinal chemistry 2005;13(6):2065-77.
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2005: Tramontano Enzo; Esposito Francesca; Badas Roberta; Di Santo Roberto; Costi Roberta; La Colla Paolo
6-[1-(4-Fluorophenyl)methyl-1H-pyrrol-2-yl)]-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro.
Antiviral research 2005;65(2):117-24.
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2005: Dukhan D; Leroy F; Peyronnet J; Bosc E; Chaves D; Durka M; Storer R; La Colla P; Seela F; Gosselin G
Synthesis of 5-aza-7-deazaguanine nucleoside derivatives as potential anti-flavivirus agents.
Nucleosides, nucleotides & nucleic acids 2005;24(5-7):671-4.
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2004: Menozzi Giulia; Merello Luisa; Fossa Paola; Schenone Silvia; Ranise Angelo; Mosti Luisa; Bondavalli Francesco; Loddo Roberta; Murgioni Chiara; Mascia Valeria; La Colla Paolo; Tamburini Elena
Synthesis, antimicrobial activity and molecular modeling studies of halogenated 4-[1H-imidazol-1-yl(phenyl)methyl]-1,5-diphenyl-1H-pyrazoles.
Bioorganic & medicinal chemistry 2004;12(20):5465-83.
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2004: Pierra Claire; Benzaria Samira; Dukhan David; Loi Anna Giulia; La Colla Paolo; Bridges Edward; Mao John; Standring David; Sommadossi Jean-Pierre; Gosselin Gilles
Synthesis, physicochemical and pharmacokinetic studies of potential prodrugs of beta-L-2'-deoxycytidine, a selective and specific anti-HBV agent.
Antiviral chemistry & chemotherapy 2004;15(5):269-79.
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2004: Silvestri Romano; Artico Marino; De Martino Gabriella; La Regina Giuseppe; Loddo Roberta; La Colla Massimiliano; Mura Massimo; La Colla Paolo
Simple, short peptide derivatives of a sulfonylindolecarboxamide (L-737,126) active in vitro against HIV-1 wild type and variants carrying non-nucleoside reverse transcriptase inhibitor resistance mutations.
Journal of medicinal chemistry 2004;47(15):3892-6.
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2004: Sbardella Gianluca; Mai Antonello; Artico Marino; Setzu Maria Giovanna; Poni Graziella; La Colla Paolo
New 6-nitroquinolones: synthesis and antimicrobial activities.
Farmaco (Società chimica italiana : 1989) 2004;59(6):463-71.
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2004: Tramontano Enzo; Onidi Loredana; Esposito Francesca; Badas Roberta; La Colla Paolo
The use of a new in vitro reaction substrate reproducing both U3 and U5 regions of the HIV-1 3'-ends increases the correlation between the in vitro and in vivo effects of the HIV-1 integrase inhibitors.
Biochemical pharmacology 2004;67(9):1751-61.
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2004: Costi Roberta; Di Santo Roberto; Artico Marino; Roux Alessandra; Ragno Rino; Massa Silvio; Tramontano Enzo; La Colla Massimiliano; Loddo Roberta; Marongiu M Elena; Pani Alessandra; La Colla Paolo
6-aryl-2,4-dioxo-5-hexenoic acids, novel integrase inhibitors active against HIV-1 multiplication in cell-based assays.
Bioorganic & medicinal chemistry letters 2004;14(7):1745-9.
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2004: Sbardella Gianluca; Mai Antonello; Artico Marino; Loddo Roberta; Setzu Maria Grazia; La Colla Paolo
Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480.
Bioorganic & medicinal chemistry letters 2004;14(6):1537-41.
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2004: Silvestri Romano; Artico Marino; La Regina Giuseppe; De Martino Gabriella; La Colla Massimiliano; Loddo Roberta; La Colla Paolo
Anti-HIV-1 activity of pyrryl aryl sulfone (PAS) derivatives: synthesis and SAR studies of novel esters and amides at the position 2 of the pyrrole nucleus.
Farmaco (Società chimica italiana : 1989) 2004;59(3):201-10.
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2004: Ragno Rino; Mai Antonello; Sbardella Gianluca; Artico Marino; Massa Silvio; Musiu Chiara; Mura Massimo; Marturana Flavia; Cadeddu Alessandra; La Colla Paolo
Computer-aided design, synthesis, and anti-HIV-1 activity in vitro of 2-alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as novel potent non-nucleoside reverse transcriptase inhibitors, also active against the Y181C variant.
Journal of medicinal chemistry 2004;47(4):928-34.
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2004: Bolognese Adele; Correale Gaetano; Manfra Michele; Lavecchia Antonio; Mazzoni Orazio; Novellino Ettore; La Colla Paolo; Sanna Giuseppina; Loddo Roberta
Antitumor agents. 3. Design, synthesis, and biological evaluation of new pyridoisoquinolindione and dihydrothienoquinolindione derivatives with potent cytotoxic activity.
Journal of medicinal chemistry 2004;47(4):849-58.
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2004: Costi Roberta; Santo Roberto Di; Artico Marino; Massa Silvio; Ragno Rino; Loddo Roberta; La Colla Massimiliano; Tramontano Enzo; La Colla Paolo; Pani Alessandra
2,6-Bis(3,4,5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays.
Bioorganic & medicinal chemistry 2004;12(1):199-215.
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2003: Vicini Paola; Geronikaki Athina; Incerti Matteo; Busonera Bernadetta; Poni Graziella; Cabras Carla Alba; La Colla Paolo
Synthesis and biological evaluation of benzo[d]isothiazole, benzothiazole and thiazole Schiff bases.
Bioorganic & medicinal chemistry 2003;11(22):4785-9.
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2003: Alleca Sergio; Corona Paola; Loriga Mario; Paglietti Giuseppe; Loddo Roberta; Mascia Valeria; Busonera Bernardetta; La Colla Paolo
Quinoxaline chemistry. Part 16. 4-substituted anilino and 4-substituted phenoxymethyl pyrrolo[1,2-a]quinoxalines and N-[4-(pyrrolo[1,2-a]quinoxalin-4-yl)amino and hydroxymethyl]benzoyl glutamates. Synthesis and evaluation of in vitro biological activity.
Farmaco (Società chimica italiana : 1989) 2003;58(9):639-50.
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2003: Gomez-Monterrey Isabel; Campiglia Pietro; Grieco Paolo; Diurno Maria Vittoria; Bolognese Adele; La Colla Paolo; Novellino Ettore
New benzo[g]isoquinoline-5,10-diones and dihydrothieno [2,3-b]naphtho-4,9-dione derivatives: synthesis and biological evaluation as potential antitumoral agents.
Bioorganic & medicinal chemistry 2003;11(17):3769-75.
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2003: Silvestri Romano; De Martino Gabriella; La Regina Giuseppe; Artico Marino; Massa Silvio; Vargiu Laura; Mura Massimo; Loi Anna Giulia; Marceddu Tiziana; La Colla Paolo
Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: synthesis and SAR studies.
Journal of medicinal chemistry 2003;46(12):2482-93.
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2003: Ranise Angelo; Spallarossa Andrea; Schenone Silvia; Bruno Olga; Bondavalli Francesco; Pani Alessandra; Marongiu Maria Elena; Mascia Valeria; La Colla Paolo; Loddo Roberta
Synthesis and antiproliferative activity of basic thioanalogues of merbarone.
Bioorganic & medicinal chemistry 2003;11(12):2575-89.
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2003: Griffon J F; Dukhan D; Pierra C; Benzaria S; Loi A G; La Colla P; Sommadossi J P; Gosselin G
4'-C-methyl-beta-D-ribofuranosyl purine and pyrimidine nucleosides revisited.
Nucleosides, nucleotides & nucleic acids 2003;22(5-8):707-9.
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2003: Ranise Angelo; Spallarossa Andrea; Schenone Silvia; Bruno Olga; Bondavalli Francesco; Vargiu Laura; Marceddu Tiziana; Mura Massimo; La Colla Paolo; Pani Alessandra
Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: a novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives.
Journal of medicinal chemistry 2003;46(5):768-81.
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2003: Baraldi Pier Giovanni; Tabrizi Mojgan Aghazadeh; Pavani Maria Giovanna; Nuñez Maria del Carmen; Makaeva Rimma; Gambari Roberto; La Colla Paolo; Romagnoli Romeo
Design, synthesis and in vitro cytotoxicity of a cis-dichloroplatinum (II) complex linked to the minor groove binder stallimycin.
Arzneimittel-Forschung 2003;53(2):107-13.
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2002: Setzu Maria Giovanna; Stefancich Giorgio; La Colla Paolo; Castellano Sabrina
Synthesis and antifungal properties of N-[(1,1'-biphenyl)-4-ylmethyl]-1H-imidazol-1-amine derivatives.
Farmaco (Società chimica italiana : 1989) 2002;57(12):1015-8.
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2002: Bolognese Adele; Correale Gaetano; Manfra Michele; Lavecchia Antonio; Mazzoni Orazio; Novellino Ettore; Barone Vincenzo; La Colla Paolo; Loddo Roberta
Antitumor agents. 2. Synthesis, structure-activity relationships, and biological evaluation of substituted 5H-pyridophenoxazin-5-ones with potent antiproliferative activity.
Journal of medicinal chemistry 2002;45(24):5217-23.
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2002: Bolognese Adele; Correale Gaetano; Manfra Michele; Lavecchia Antonio; Mazzoni Orazio; Novellino Ettore; Barone Vincenzo; Pani Alessandra; Tramontano Enzo; La Colla Paolo; Murgioni Chiara; Serra Ilaria; Setzu Giovanna; Loddo Roberta
Antitumor agents. 1. Synthesis, biological evaluation, and molecular modeling of 5H-pyrido[3,2-a]phenoxazin-5-one, a compound with potent antiproliferative activity.
Journal of medicinal chemistry 2002;45(24):5205-16.
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2002: Abu Sheikha Ghassan; La Colla Paolo; Loi Anna Giulia
A new class of acyclic nucleoside phosphonates: synthesis and biological activity of 9-[[(phosphonomethyl)aziridin-1-yl]methyl]guanine (PMAMG) and analogues.
Nucleosides, nucleotides & nucleic acids 2002;21(10):619-35.
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2002: Jeannot Frédéric; Gosselin Gilles; Standring David; Bryant Martin; Sommadossi Jean Pierre; Giulia Loi Anna; La Colla Paolo; Mathé Christophe
Synthesis and studies of 3'-C-trifluoromethyl nucleoside analogues bearing adenine or cytosine as the base.
Bioorganic & medicinal chemistry 2002;10(10):3153-61.
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2002: Di Santo Roberto; Costi Roberta; Artico Marino; Massa Silvio; Ragno Rino; Marshall Garland R; La Colla Paolo
Design, synthesis and QSAR studies on N-aryl heteroarylisopropanolamines, a new class of non-peptidic HIV-1 protease inhibitors.
Bioorganic & medicinal chemistry 2002;10(8):2511-26.
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2002: Silvestri Romano; Artico Marino; De Martino Gabriella; Ragno Rino; Massa Silvio; Loddo Roberta; Murgioni Chiara; Loi Anna Giulia; La Colla Paolo; Pani Alessandra
Synthesis, biological evaluation, and binding mode of novel 1-[2-(diarylmethoxy)ethyl]-2-methyl-5-nitroimidazoles targeted at the HIV-1 reverse transcriptase.
Journal of medicinal chemistry 2002;45(8):1567-76.
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2002: Pani A; Loi A G; Mura M; Marceddu T; La Colla P; Marongiu M E
Targeting HIV: old and new players.
Current drug targets. Infectious disorders 2002;2(1):17-32.
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2001: Pinna G A; Loriga G; Murineddu G; Grella G; Mura M; Vargiu L; Murgioni C; La Colla P
Synthesis and anti-HIV-1 activity of new delavirdine analogues carrying arylpyrrole moieties.
Chemical & pharmaceutical bulletin 2001;49(11):1406-11.
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2001: Menozzi G; Mosti L; Fossa P; Musiu C; Murgioni C; La Colla P
Synthesis and biological evaluation of azole derivatives, analogues of bifonazole, with a phenylisoxazolyl or phenylpyrimidinyl moiety.
Farmaco (Società chimica italiana : 1989) 2001;56(9):633-40.
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2001: Mai A; Sbardella G; Artico M; Ragno R; Massa S; Novellino E; Greco G; Lavecchia A; Musiu C; La Colla M; Murgioni C; La Colla P; Loddo R
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase.
Journal of medicinal chemistry 2001;44(16):2544-54.
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2001: Pani A; Musiu C; Loi A G; Mai A; Loddo R; La Colla P; Marongiu M E
DABOs as candidates to prevent mucosal HIV transmission.
Antiviral chemistry & chemotherapy 2001;12 Suppl 1():51-9.
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2000: Aiello E; Aiello S; Mingoia F; Bacchi A; Pelizzi G; Musiu C; Setzu M G; Pani A; La Colla P; Marongiu M E
Synthesis and antimicrobial activity of new 3-(1-R-3(5)-methyl-4-nitroso-1H-5(3)-pyrazolyl)-5-methylisoxazoles.
Bioorganic & medicinal chemistry 2000;8(12):2719-28.
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2000: Castellano S; Stefancich G; Musiu C; La Colla P
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines.
Archiv der Pharmazie 2000;333(9):299-304.
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2000: Silvestri R; Artico M; De Martino G; Novellino E; Greco G; Lavecchia A; Massa S; Loi A G; Doratiotto S; La Colla P
Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors.
Bioorganic & medicinal chemistry 2000;8(9):2305-9.
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2000: Pani A; Batetta B; Putzolu M; Sanna F; Spano O; Piras S; Mulas M F; Bonatesta R R; Amat di S Filippo C; Vargiu L; Marceddu T; Sanna L; La Colla P; Dessì S
MDR1, cholesterol certification and cell growth: a comparative study in normal and multidrug-resistant KB cell lines.
Cellular and molecular life sciences : CMLS 2000;57(7):1094-102.
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2000: Castellano S; La Colla P; Musiu C; Stefancich G
Azole antifungal agents related to naftifine and butenafine.
Archiv der Pharmazie 2000;333(6):162-6.
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2000: Artico M; Silvestri R; Pagnozzi E; Bruno B; Novellino E; Greco G; Massa S; Ettorre A; Loi A G; Scintu F; La Colla P
Structure-based design, synthesis, and biological evaluation of novel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations.
Journal of medicinal chemistry 2000;43(9):1886-91.
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2000: Manfredini S; Baraldi P G; Bazzanini R; Durini E; Vertuani S; Pani A; Marceddu T; Demontis F; Vargiu L; La Colla P
Pyrazole related nucleosides 5. Synthesis and biological activity of 2'-deoxy-2',3'-dideoxy- and acyclo-analogues of 4-iodo-1-beta-D-ribofuranosyl-3-carboxymethyl pyrazole (IPCAR).
Nucleosides, nucleotides & nucleic acids 2000;19(4):705-22.
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2000: Costi R; Di Santo R; Artico M; Massa S; Lavecchia A; Marceddu T; Sanna L; La Colla P; Marongiu M E
Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase.
Antiviral chemistry & chemotherapy 2000;11(2):117-33.
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2000: Manfredini S; Marastoni-M; Tomatis R; Durini E; Spisani S; Pani A; Marceddu T; Musiu C; Marongiu M E; La Colla P
Peptide T-araC conjugates: solid-phase synthesis and biological activity of N4-(acylpeptidyl)-araC.
Bioorganic & medicinal chemistry 2000;8(3):539-47.
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2000: Silvestri R; Artico M; Massa S; Marceddu T; De Montis F; La Colla P
1-[2-(Diphenylmethoxy)ethyl]-2-methyl-5-nitroimidazole: a potent lead for the design of novel NNRTIs.
Bioorganic & medicinal chemistry letters 2000;10(3):253-6.
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1999: Barraja P; Diana P; Lauria A; Passannanti A; Almerico A M; Minnei C; Longu S; Congiu D; Musiu C; La Colla P
Indolo[3,2-c]cinnolines with antiproliferative, antifungal, and antibacterial activity.
Bioorganic & medicinal chemistry 1999;7(8):1591-6.
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1999: Cirrincione G; Almerico A M; Barraja P; Diana P; Lauria A; Passannanti A; Musiu C; Pani A; Murtas P; Minnei C; Marongiu M E; La Colla P
Derivatives of the new ring system indolo[1,2-c]benzo[1,2,3]triazine with potent antitumor and antimicrobial activity.
Journal of medicinal chemistry 1999;42(14):2561-8.
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1999: Menozzi G; Mosti L; Bruno O; Lo Presti E; Musiu C; Longu S; La Colla P; Filippelli W; Falcone G; Piucci B
Synthesis and biological evaluation of [alpha-(1,5-disubstituted 1H-pyrazol-4-yl)benzyl]azoles, analogues of bifonazole.
Farmaco (Società chimica italiana : 1989) 1999;54(6):416-22.
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1999: Artico M; Mai A; Sbardella G; Massa S; Musiu C; Lostia S; Demontis F; La Colla P
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro.
Bioorganic & medicinal chemistry letters 1999;9(12):1651-6.
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1999: Costi P M; Rinaldi M; Tondi D; Pecorari P; Barlocco D; Ghelli S; Stroud R M; Santi D V; Stout T J; Musiu C; Marangiu E M; Pani A; Congiu D; Loi G A; La Colla P
Phthalein derivatives as a new tool for selectivity in thymidylate synthase inhibition.
Journal of medicinal chemistry 1999;42(12):2112-24.
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1999: Diana P; Barraja P; Lauria A; Almerico A M; Cirrincione G; Minnei C; Longu S; Congiu D; Musiu C; La Colla P
Synthesis and antiproliferative activity of 2-triazenothiophenes.
Anticancer research 1999;19(3A):2127-31.
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1999: Abu Sheika G; Tramontano E; Loi A G; Franchetti P; Grifantini M; La Colla P
Effect of acyclic nucleoside phosphonates on the HIV-1 integrase in vitro.
Nucleosides & nucleotides 1999;18(4-5):849-51.
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1999: Mai A; Artico M; Sbardella G; Massa S; Novellino E; Greco G; Loi A G; Tramontano E; Marongiu M E; La Colla P
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3, 4-dihydropyrimidin-4(3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives.
Journal of medicinal chemistry 1999;42(4):619-27.
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1998: Tramontano E; Piras G; Mellors J W; Putzolu M; Bazmi H Z; La Colla P
Biochemical characterization of HIV-1 reverse transcriptases encoding mutations at amino acid residues 161 and 208 involved in resistance to phosphonoformate.
Biochemical pharmacology 1998;56(12):1583-9.
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1998: Desideri N; Sestili I; Stein M L; Tramontano E; Corrias S; La Colla P
Synthesis and anti-human immunodeficiency virus type 1 integrase activity of hydroxybenzoic and hydroxycinnamic acid flavon-3-yl esters.
Antiviral chemistry & chemotherapy 1998;9(6):497-509.
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1998: Artico M; Di Santo R; Costi R; Novellino E; Greco G; Massa S; Tramontano E; Marongiu M E; De Montis A; La Colla P
Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase: synthesis, biological evaluation, and molecular modeling.
Journal of medicinal chemistry 1998;41(21):3948-60.
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1998: Franchetti P; Perlini P; Abu Sheikha G; Cappellacci L; Grifantini M; Loi A G; De Montis A; Pani A; Marongiu M E; La Colla P
Potent and selective inhibitors of human immunodeficiency virus protease structurally related to L-694,746.
Antiviral chemistry & chemotherapy 1998;9(4):303-9.
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1998: Pani A; Marongiu M E; Pinna E; Scintu F; Perra G; Montis A D; Manfredini S; La Colla P
In vitro and in vivo antiproliferative activity of IPCAR, a new pyrazole nucleoside analog.
Anticancer research 1998;18(4A):2623-30.
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1998: Silvestri R; Artico M; Bruno B; Massa S; Novellino E; Greco G; Marongiu M E; Pani A; De Montis A; La Colla P
Synthesis and biological evaluation of 5H-indolo [3,2-b][1,5]benzothiazepine derivatives, designed as conformationally constrained analogues of the human immunodeficiency virus type 1 reverse transcriptase inhibitor L-737,126.
Antiviral chemistry & chemotherapy 1998;9(2):139-48.
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1998: Di Santo R; Costi R; Artico M; Massa S; Marongiu M E; Loi A G; De Montis A; La Colla P
1,2,5-Benzothiadiazepine and pyrrolo[2,1-d]-[1,2,5]benzothiadiazepine derivatives with specific anti-human immunodeficiency virus type 1 activity.
Antiviral chemistry & chemotherapy 1998;9(2):127-37.
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1998: Almerico A M; Diana P; Barraja P; Dattolo G; Mingoia F; Loi A G; Scintu F; Milia C; Puddu I; La Colla P
Glycosidopyrroles. Part 1. Acyclic derivatives: 1-(2-hydroxyethoxy)methylpyrroles as potential anti-viral agents.
Farmaco (Società chimica italiana : 1989) 1998;53(1):33-40.
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1997: Silvestri R; Artico M; Massa S; Stefancich G; Congeddu E; Putzolu M; La Colla P
Sulfone derivatives with anti-HIV activity.
Farmaco (Società chimica italiana : 1989) 1997;52(5):323-9.
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1997: Diana P; Barraja P; Almerico A M; Dattolo G; Mingoia F; Loi A G; Congeddu E; Musiu C; Putzolu M; La Colla P
Acyclic glycosidopyrroles analogues of ganciclovir: synthesis and biological activity.
Farmaco (Società chimica italiana : 1989) 1997;52(5):281-2.
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1997: Franchetti P; Cappellacci L; Sheikha G A; Jayaram H N; Gurudutt V V; Sint T; Schneider B P; Jones W D; Goldstein B M; Perra G; De Montis A; Loi A G; La Colla P; Grifantini M
Synthesis, structure, and antiproliferative activity of selenophenfurin, an inosine 5'-monophosphate dehydrogenase inhibitor analogue of selenazofurin.
Journal of medicinal chemistry 1997;40(11):1731-7.
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1997: Mai A; Artico M; Sbardella G; Quartarone S; Massa S; Loi A G; De Montis A; Scintu F; Putzolu M; La Colla P
Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines: novel non-nucleoside reverse transcriptase inhibitors of the S-DABO series.
Journal of medicinal chemistry 1997;40(10):1447-54.
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1997: Invidiata F P; Furnò G; Simoni D; Lampronti I; Musiu C; Milia C; Scintu F; La Colla P
3,6-Disubstituted 1,2,4-triazolo[3,4-b][1,3,4]thiadiazoles: synthesis and evaluation for antimicrobial and antiviral activity. III.
Farmaco (Società chimica italiana : 1989) 1997;52(4):259-61.
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1996: Baraldi P G; Cacciari B; Romagnoli R; Spalluto G; Garuti L; Roberti M; Pani A; Perra G; Scintu F; Pinna N; Musiu C; La Colla P
Synthesis, antiviral and antiproliferative activity of a new class of 5-(alkyl or arylthio)-6-vinyl uracils.
Anti-cancer drug design 1996;11(8):597-609.
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1996: Tondelli L; Colonna F P; Garbesi A; Zanella S; Marongiu M E; Corrias S; Loi A G; La Colla P
Native oligodeoxynucleotides specifically active against human immunodeficiency virus type 1 in vitro: a G-quartet-driven effect?
Antimicrobial agents and chemotherapy 1996;40(9):2034-8.
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1996: Artico M; Silvestri R; Pagnozzi E; Stefancich G; Massa S; Loi A G; Putzolu M; Corrias S; Spiga M G; La Colla P
5H-pyrrolo[1,2-b] [1,2,5]benzothiadiazepines (PBTDs): a novel class of non-nucleoside reverse transcriptase inhibitors.
Bioorganic & medicinal chemistry 1996;4(6):837-50.
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1996: Silvestri R; Artico M; Pagnozzi E; Stefancich G; Massa S; La Colla P; Loi A G; Spiga M G; Corrias S; Lichino D
Synthesis and anti-HIV activity of 10,11-dihydropyrrolo [1,2-b][1,2,5]benzothiadiazepine-11-acetic acid 5,5-dioxide derivatives and related compounds.
Farmaco (Società chimica italiana : 1989) 1996;51(6):425-30.
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1996: Mazzei M; Garzoglio R; Balbi A; Grandi T; De Montis A; Corrias S; La Colla P
Synthesis and antirhinovirus activity of 3-(diethylamino)-5-phenylisoxazole derivatives.
Farmaco (Società chimica italiana : 1989) 1996;51(5):351-9.
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1996: Valette G; Pompon A; Girardet J L; Cappellacci L; Franchetti P; Grifantini M; La Colla P; Loi A G; Périgaud C; Gosselin G; Imbach J L
Decomposition pathways and in vitro HIV inhibitory effects of isoddA pronucleotides: toward a rational approach for intracellular delivery of nucleoside 5'-monophosphates.
Journal of medicinal chemistry 1996;39(10):1981-90.
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1996: Manfredini S; Bazzanini R; Baraldi P G; Bonora M; Marangoni M; Simoni D; Pani A; Scintu F; Pinna E; Pisano L; La Colla P
Pyrazole-related nucleosides. 4. Synthesis and antitumor activity of some 1-tetrahydropyranyl-4-substituted pyrazoles.
Anti-cancer drug design 1996;11(3):193-204.
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1996: Artico M; Silvestri R; Massa S; Loi A G; Corrias S; Piras G; La Colla P
2-Sulfonyl-4-chloroanilino moiety: a potent pharmacophore for the anti-human immunodeficiency virus type 1 activity of pyrrolyl aryl sulfones.
Journal of medicinal chemistry 1996;39(2):522-30.
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1995: Marongiu M E; Pani A; Tinti E; Grifantini M; Franchetti P; Cristalli G; La Colla P
Enhancement of the anti-HIV-1 activity of ddAdo by coformycin, EHNA and deaza-EHNA derivatives.
The new microbiologica : official journal of the Italian Society for Medical, Odontoiatric, and Clinical Microbiology (SIMMOC) 1995;18(4):359-70.
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1995: Franchetti P; Sheikha G A; Cappellacci L; Grifantini M; De Montis A; Piras G; Loi A G; La Colla P
Synthesis and antiviral activity of 8-aza analogs of chiral [2-(phosphonomethoxy) propyl]guanines.
Journal of medicinal chemistry 1995;38(20):4007-13.
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1995: Mai A; Artico M; Sbardella G; Massa S; Loi A G; Tramontano E; Scano P; La Colla P
Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines.
Journal of medicinal chemistry 1995;38(17):3258-63.
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1995: Massa S; Corelli F; Artico M; Mai A; Ragno R; De Montis A; Loi A G; Corrias S; Marongiu M E; La Colla P
[[[(Thienylcarbonyl)alkyl]oxy]phenyl]- and [[[(pyrrylcarbonyl)alkyl]oxy]phenyl]oxazoline derivatives with potent and selective antihuman rhinovirus activity.
Journal of medicinal chemistry 1995;38(5):803-9.
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1995: Artico M; Silvestri R; Stefancich G; Massa S; Pagnozzi E; Musu D; Scintu F; Pinna E; Tinti E; La Colla P
Synthesis of pyrryl aryl sulfones targeted at the HIV-1 reverse transcriptase.
Archiv der Pharmazie 1995;328(3):223-9.
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1994: Tramontano E; Marongiu M E; de Montis A; Loi A G; Artico M; Massa S; Mai A; la Colla P
Characterization of the anti-HIV-1 activity of 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), new non-nucleoside reverse transcriptase inhibitors.
The new microbiologica : official journal of the Italian Society for Medical, Odontoiatric, and Clinical Microbiology (SIMMOC) 1994;17(4):269-79.
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1994: Franchetti P; Cappellacci L; Grifantini M; Messini L; abu Sheikha G; Loi A G; Tramontano E; de Montis A; Spiga M G; La Colla P
Synthesis and evaluation of the anti-HIV activity of aza and deaza analogues of isoddA and their phosphates as prodrugs.
Journal of medicinal chemistry 1994;37(21):3534-41.
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1994: Pani A; Obino P; Guarracino P; La Colla P
The antimitotic drug 4,6-dimethyl-2-amino-3,4,5- trimethoxyphenyl-pyrimidine inhibits the nucleoside transport system of cells from various animal species.
Experientia 1994;50(1):29-33.
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1993: Pani A; Marongiu M E; La Colla P
Modulatory effect of N-acetyl-L-cysteine on the HIV-1 multiplication in chronically and acutely infected cell lines.
Antiviral research 1993;22(1):31-43.
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1993: Bravo P; Resnati G; Viani F; De Montis A; Corrias S; La Colla P
Synthesis and evaluation of the antiviral activity of acyclic nucleosides carrying fluorine and sulfur substituents.
Farmaco (Società chimica italiana : 1989) 1993;48(8):1113-20.
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1992: Manfredini S; Bazzanini R; Baraldi P G; Guarneri M; Simoni D; Marongiu M E; Pani A; Tramontano E; La Colla P
Pyrazole-related nucleosides. Synthesis and antiviral/antitumor activity of some substituted pyrazole and pyrazolo[4,3-d]-1,2,3-triazin-4-one nucleosides.
Journal of medicinal chemistry 1992;35(5):917-24.
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1991: Pani A; Marongiu M E; Obino P; Gavagnin M; La Colla P
Antimicrobial and antiviral activity of xylosyl-methylthio-adenosine, a naturally occurring analogue of methylthio-adenosine from Doris verrucosa.
Experientia 1991;47(11-12):1228-9.
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1991: Vicentini C B; Veronese A C; Giori P; Pani A; Piras G; Gabrielsen A; La Colla P
4-Diazo-5-alkylsulphonamidopyrazoles: synthesis and evaluation of biological activity.
Farmaco (Società chimica italiana : 1989) 1991;46(11):1351-63.
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1991: Botta M; De Angelis F; Corelli F; Menichincheri M; Nicoletti R; Marongiu M E; Pani A; La Colla P
Antiviral agents: synthesis of furylpyrimidinones and evaluation of their cytostatic and antiviral activity.
Archiv der Pharmazie 1991;324(4):203-7.
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1990: Massa S; Artico M; Corelli F; Mai A; Di Santo R; Cortes S; Marongiu M E; Pani A; La Colla P
Synthesis and antimicrobial and cytotoxic activities of pyrrole-containing analogues of trichostatin A.
Journal of medicinal chemistry 1990;33(10):2845-9.
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1989: La Colla P; Pani A; Marongiu M E; Corrias M V; Flore O; Marcello C; Lecca U
5-(2-bromoethyl)-2'-deoxyuridine: a selective inhibitor of herpes simplex viruses in vitro.
Clinical and experimental obstetrics & gynecology 1989;16(1):16-20.
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1985: La Colla P; Gelli G; Mura L; Landini M P; Corrias M V; Pani A; Marongiu M E
Antiherpes activity of 5-(2-bromoethyl)-2'-deoxyuridine.
Antiviral research 1985;Suppl 1():29-34.
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