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Anita Lewin

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Charles J McElhinny; Scott Runyon; Lawrence Brieaddy; Anita H Lewin; Wayne Mascarella; F Ivy Carroll
Hydrolytic instability of the important orexin 1 receptor antagonist SB-334867: possible confounding effects on in vivo and in vitro studies.
F Ivy Carroll; Anita H Lewin; Wayne Mascarella; Herbert H Seltzman; P Anantha Reddy
Designer drugs: a medicinal chemistry perspective.
P Anantha Reddy; Sean T Jones; Anita H Lewin; F Ivy Carroll
Synthesis of hemopressin peptides by classical solution phase fragment condensation.

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2012: Charles J McElhinny; Scott Runyon; Lawrence Brieaddy; Anita H Lewin; Wayne Mascarella; F Ivy Carroll
Hydrolytic instability of the important orexin 1 receptor antagonist SB-334867: possible confounding effects on in vivo and in vitro studies.
Bioorganic & medicinal chemistry letters 2012;22(21):6661-4.
2012: F Ivy Carroll; Anita H Lewin; Wayne Mascarella; Herbert H Seltzman; P Anantha Reddy
Designer drugs: a medicinal chemistry perspective.
Annals of the New York Academy of Sciences 2012;1248():18-38.
2012: P Anantha Reddy; Sean T Jones; Anita H Lewin; F Ivy Carroll
Synthesis of hemopressin peptides by classical solution phase fragment condensation.
International journal of peptides 2012;2012():186034.
2011: Anita H Lewin; Gregory M Miller; Brian Gilmour
Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class.
Bioorganic & medicinal chemistry 2011;19(23):7044-8.
2010: Susan C J Sumner; Timothy R Fennell; Rodney W Snyder; George F Taylor; Anita H Lewin
Distribution of carbon-14 labeled C60 ([14C]C60) in the pregnant and in the lactating dam and the effect of C60 exposure on the biochemical profile of urine.
Journal of applied toxicology : JAT 2010;30(4):354-60.
2009: Anita H Lewin; Hernán A Navarro; Brian P Gilmour
Amiodarone and its putative metabolites fail to activate wild type hTAAR1.
Bioorganic & medicinal chemistry letters 2009;19(20):5913-4.
2009: P Anantha Reddy; Anita H Lewin; Peter W Schiller
Synthesis and pharmacological evaluation of highly potent [Dmt1]DALDA analogs.
Advances in experimental medicine and biology 2009;611():473-4.
2008: Anita H Lewin; Hernán A Navarro; Wayne Mascarella
Structure-activity correlations for beta-phenethylamines at human trace amine receptor 1.
Bioorganic & medicinal chemistry 2008;16(15):7415-23.
2006: Hernán A Navarro; Brian P Gilmour; Anita H Lewin
A rapid functional assay for the human trace amine-associated receptor 1 based on the mobilization of internal calcium.
Journal of biomolecular screening 2006;11(6):688-93.
2006: Anita H Lewin
Receptors of mammalian trace amines.
The AAPS journal 2006;8(1):E138-45.
2005: Scott P Runyon; Jason P Burgess; Philip Abraham; Kathryn I Keverline-Frantz; Judith L Flippen-Anderson; Jeffrey Deschamps; Anita H Lewin; Hernán A Navarro; John W Boja; Michael J Kuhar; Frank carroll
Synthesis, structural identification, and ligand binding of tropane ring analogs of paroxetine and an unexpected aza-bicyclo[3.2.2]nonane rearrangement product.
Bioorganic & medicinal chemistry 2005;13(7):2439-49.
1998: Anita H Lewin; G Sun; L Fudala; Hernán A Navarro; L M Zhou; Piotr Popik; A Faynsteyn; Phil Skolnick
Molecular features associated with polyamine modulation of NMDA receptors.
Journal of medicinal chemistry 1998;41(6):988-95.
1998: K I Keverline-Frantz; John W Boja; Michael J Kuhar; Philip Abraham; Jason P Burgess; Anita H Lewin; Frank carroll
Synthesis and ligand binding of tropane ring analogues of paroxetine.
Journal of medicinal chemistry 1998;41(2):247-57.
1997: B E Blough; Philip Abraham; A C Mills; Anita H Lewin; John W Boja; U Scheffel; Michael J Kuhar; Frank carroll
3 Beta-(4-ethyl-3-iodophenyl)nortropane-2 beta-carboxylic acid methyl ester as a high-affinity selective ligand for the serotonin transporter.
Journal of medicinal chemistry 1997;40(24):3861-4.
1996: B E Blough; Philip Abraham; Anita H Lewin; Michael J Kuhar; J W Boja; Frank carroll
Synthesis and transporter binding properties of 3 beta-(4'-alkyl-, 4'-alkenyl-, and 4'-alkynylphenyl)nortropane-2 beta-carboxylic acid methyl esters: serotonin transporter selective analogs.
Journal of medicinal chemistry 1996;39(20):4027-35.
1996: C W Sachs; L M Ballas; Wayne Mascarella; A R Safa; Anita H Lewin; C Loomis; Frank carroll; R M Bell; R L Fine
Effects of sphingosine stereoisomers on P-glycoprotein phosphorylation and vinblastine accumulation in multidrug-resistant MCF-7 cells.
Biochemical pharmacology 1996;52(4):603-12.
1996: P Kotian; Wayne Mascarella; Philip Abraham; Anita H Lewin; J W Boja; Michael J Kuhar; Frank carroll
Synthesis, ligand binding, and quantitative structure-activity relationship study of 3 beta-(4'-substituted phenyl)-2 beta-heterocyclic tropanes: evidence for an electrostatic interaction at the 2 beta-position.
Journal of medicinal chemistry 1996;39(14):2753-63.
1995: J K Staley; J W Boja; Frank carroll; Herbert H Seltzman; C D Wyrick; Anita H Lewin; Philip Abraham; Deborah C Mash
Mapping dopamine transporters in the human brain with novel selective cocaine analog [125I]RTI-121.
Synapse (New York, N.Y.) 1995;21(4):364-72.
1995: P Kotian; Philip Abraham; Anita H Lewin; Wayne Mascarella; J W Boja; Michael J Kuhar; Frank carroll
Synthesis and ligand binding study of 3 beta-(4'-substituted phenyl)-2 beta-(heterocyclic)tropanes.
Journal of medicinal chemistry 1995;38(18):3451-3.
1995: Anita H Lewin; S L Black; M E Bos; R R Goehring; X Nair; G Whiting; P Bouquin; G Tetrault; Frank carroll
Evaluation of retinoid lactones as topical therapeutic agents in dermatology.
Pharmaceutical research 1995;12(7):983-92.
1995: J W Boja; Jean Lud Cadet; Theresa A Kopajtic; John R Lever; Herbert H Seltzman; C D Wyrick; Anita H Lewin; Philip Abraham; Frank carroll
Selective labeling of the dopamine transporter by the high affinity ligand 3 beta-(4-[125I]iodophenyl)tropane-2 beta-carboxylic acid isopropyl ester.
Molecular pharmacology 1995;47(4):779-86.
1995: Frank carroll; P Kotian; A Dehghani; J L Gray; M A Kuzemko; K A Parham; Philip Abraham; Anita H Lewin; J W Boja; Michael J Kuhar
Cocaine and 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter.
Journal of medicinal chemistry 1995;38(2):379-88.
1994: Frank carroll; Wayne Mascarella; M A Kuzemko; Y Gao; Philip Abraham; Anita H Lewin; J W Boja; Michael J Kuhar
Synthesis, ligand binding, and QSAR (CoMFA and classical) study of 3 beta-(3'-substituted phenyl)-, 3 beta-(4'-substituted phenyl)-, and 3 beta-(3',4'-disubstituted phenyl)tropane-2 beta-carboxylic acid methyl esters.
Journal of medicinal chemistry 1994;37(18):2865-73.
1994: Anita H Lewin; R R Goehring; F C Zusi; G J Gendimenico; X Nair; G Whitting; P Bouquin; G Tetrault; Frank carroll
The requirement for a retinoic acid lactone of 11-cis, 13-cis-stereochemistry for topical dermatologic activity.
Pharmaceutical research 1994;11(7):1065-7.
1994: J W Boja; Michael J Kuhar; Theresa A Kopajtic; Emily Boja; Philip Abraham; Anita H Lewin; Frank carroll
Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters.
Journal of medicinal chemistry 1994;37(8):1220-3.
1994: Anita H Lewin; M E Bos; F C Zusi; X Nair; G Whiting; P Bouquin; G Tetrault; Frank carroll
Evaluation of retinoids as therapeutic agents in dermatology.
Pharmaceutical research 1994;11(2):192-200.
1993: Frank carroll; J L Gray; Philip Abraham; M A Kuzemko; Anita H Lewin; J W Boja; Michael J Kuhar
3-Aryl-2-(3'-substituted-1',2',4'-oxadiazol-5'-yl)tropane analogues of cocaine: affinities at the cocaine binding site at the dopamine, serotonin, and norepinephrine transporters.
Journal of medicinal chemistry 1993;36(20):2886-90.
1993: Anita H Lewin; P Skolnick; J C Marvizon; I A Paul; J P Bowen
Requirements for high affinity binding of glycine analogs to the glycine site of the NMDA receptor complex.
European journal of pharmacology 1993;247(1):1-10.
1993: Frank carroll; Anita H Lewin; Michael J Kuhar; J W Boja
Cocaine receptor: a structure-activity relationship study.
NIDA research monograph 1993;134():229-37.
1992: KM Tramposch; S A Steiner; P L Stanley; D O Nettleton; R C Franson; Anita H Lewin; F I Carroll
Novel inhibitor of phospholipase A2 with topical anti-inflammatory activity.
Biochemical and biophysical research communications 1992;189(1):272-9.
1992: J W Boja; R M McNeill; Anita H Lewin; Philip Abraham; Frank carroll; Michael J Kuhar
Selective dopamine transporter inhibition by cocaine analogs.
Neuroreport 1992;3(11):984-6.
1992: E J Cline; Ursula Scheffel; J W Boja; W M Mitchell; Frank carroll; Philip Abraham; Anita H Lewin; Michael J Kuhar
In vivo binding of [125I]RTI-55 to dopamine transporters: pharmacology and regional distribution with autoradiography.
Synapse (New York, N.Y.) 1992;12(1):37-46.
1992: J W Boja; W M Mitchell; A Patel; Theresa A Kopajtic; Frank carroll; Anita H Lewin; Philip Abraham; Michael J Kuhar
High-affinity binding of [125I]RTI-55 to dopamine and serotonin transporters in rat brain.
Synapse (New York, N.Y.) 1992;12(1):27-36.
1992: J W Boja; E J Cline; Frank carroll; Anita H Lewin; A Philip; Robert F Dannals; Dean F Wong; Ursula Scheffel; Michael J Kuhar
High potency cocaine analogs: neurochemical, imaging, and behavioral studies.
Annals of the New York Academy of Sciences 1992;654():282-91.
1992: Frank carroll; Philip Abraham; Anita H Lewin; K A Parham; J W Boja; Michael J Kuhar
Isopropyl and phenyl esters of 3 beta-(4-substituted phenyl)tropan-2 beta-carboxylic acids. Potent and selective compounds for the dopamine transporter.
Journal of medicinal chemistry 1992;35(13):2497-500.
1992: Ursula Scheffel; Robert F Dannals; E J Cline; George A Ricaurte; Frank carroll; Philip Abraham; Anita H Lewin; Michael J Kuhar
[123/125I]RTI-55, an in vivo label for the serotonin transporter.
Synapse (New York, N.Y.) 1992;11(2):134-9.
1992: Frank carroll; Y Gao; Philip Abraham; Anita H Lewin; R Lew; A Patel; J W Boja; Michael J Kuhar
Probes for the cocaine receptor. Potentially irreversible ligands for the dopamine transporter.
Journal of medicinal chemistry 1992;35(10):1813-7.
1992: A Patel; J W Boja; John R Lever; R Lew; R Simantov; Frank carroll; Anita H Lewin; A Philip; Y Gao; Michael J Kuhar
A cocaine analog and a GBR analog label the same protein in rat striatal membranes.
Brain research 1992;576(1):173-4.
1992: Frank carroll; Anita H Lewin; J W Boja; Michael J Kuhar
Cocaine receptor: biochemical characterization and structure-activity relationships of cocaine analogues at the dopamine transporter.
Journal of medicinal chemistry 1992;35(6):969-81.
1992: Philip Abraham; J B Pitner; Anita H Lewin; J W Boja; Michael J Kuhar; Frank carroll
N-modified analogues of cocaine: synthesis and inhibition of binding to the cocaine receptor.
Journal of medicinal chemistry 1992;35(1):141-4.
1992: Anita H Lewin; Y G Gao; Philip Abraham; J W Boja; Michael J Kuhar; Frank carroll
2 beta-substituted analogues of cocaine. Synthesis and inhibition of binding to the cocaine receptor.
Journal of medicinal chemistry 1992;35(1):135-40.
1991: Robert L Balster; Frank carroll; J H Graham; R S Mansbach; M A Rahman; A Philip; Anita H Lewin; V M Showalter
Potent substituted-3 beta-phenyltropane analogs of cocaine have cocaine-like discriminative stimulus effects.
Drug and alcohol dependence 1991;29(2):145-51.
1991: W A Khan; Wayne Mascarella; Anita H Lewin; C D Wyrick; Frank carroll; Yusuf A Hannun
Use of D-erythro-sphingosine as a pharmacological inhibitor of protein kinase C in human platelets.
The Biochemical journal 1991;278 ( Pt 2)():387-92.
1991: Frank carroll; Y G Gao; M A Rahman; Philip Abraham; K Parham; Anita H Lewin; J W Boja; Michael J Kuhar
Synthesis, ligand binding, QSAR, and CoMFA study of 3 beta-(p-substituted phenyl)tropane-2 beta-carboxylic acid methyl esters.
Journal of medicinal chemistry 1991;34(9):2719-25.
1991: Frank carroll; Anita H Lewin; Philip Abraham; K Parham; J W Boja; Michael J Kuhar
Synthesis and ligand binding of cocaine isomers at the cocaine receptor.
Journal of medicinal chemistry 1991;34(3):883-6.
1991: J W Boja; M A Rahman; A Philip; Anita H Lewin; Frank carroll; Michael J Kuhar
Isothiocyanate derivatives of cocaine: irreversible inhibition of ligand binding at the dopamine transporter.
Molecular pharmacology 1991;39(3):339-45.
1991: J W Boja; A Patel; Frank carroll; M A Rahman; A Philip; Anita H Lewin; Theresa A Kopajtic; Michael J Kuhar
[125I]RTI-55: a potent ligand for dopamine transporters.
European journal of pharmacology 1991;194(1):133-4.
1991: X Nair; J Quigley; KM Tramposch; Frank carroll; Anita H Lewin; I Kiss
BMY 30047: a novel topically active retinoid with low local and systemic toxicity.
The Journal of pharmacology and experimental therapeutics 1991;256(1):365-70.
1991: Frank carroll; Anita H Lewin
Important compounds in the cocaine class: a synthesis overview.
NIDA research monograph 1991;112():284-99.
1990: J W Boja; Frank carroll; M A Rahman; A Philip; Anita H Lewin; Michael J Kuhar
New, potent cocaine analogs: ligand binding and transport studies in rat striatum.
European journal of pharmacology 1990;184(2-3):329-32.
1990: Frank carroll; A Philip; Anita H Lewin
Cocaine receptor--design of ligands.
NIDA research monograph 1990;96():112-21.
1990: Frank carroll; M A Rahman; A Philip; Anita H Lewin; J W Boja; Michael J Kuhar
Synthesis and receptor binding of cocaine analogs.
NIDA research monograph 1990;105():147-53.