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Andreas Link

Research Profile

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Publications

TOP 3
Felix Wilde; Andreas Link
Advances in the design of a multipurpose fragment screening library.
Riad Schulz; Kristin Sydow; Thomas Emmrich; Carsten Hirt; Thomas Kiefer; Ulrike Leffler; Heidi Lemmerhirt; Andreas Link; Patrick J Bednarski
Identification of a glutathione peroxidase inhibitor that reverses resistance to anticancer drugs in human B-cell lymphoma cell lines.
Christoph Kamper; Katharina Korpis; Lennart Anger; Patrick J Bednarski; Martin Neuenschwander; Edgar Specker; Andreas Link
Sustainable synthesis and automated deposition: an accessible discovery screening library of fragment-like purines.

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All Publications

2013: Felix Wilde; Andreas Link
Advances in the design of a multipurpose fragment screening library.
Expert opinion on drug discovery 2013;8(5):597-606.
2012: Riad Schulz; Kristin Sydow; Thomas Emmrich; Carsten Hirt; Thomas Kiefer; Ulrike Leffler; Heidi Lemmerhirt; Andreas Link; Patrick J Bednarski
Identification of a glutathione peroxidase inhibitor that reverses resistance to anticancer drugs in human B-cell lymphoma cell lines.
Bioorganic & medicinal chemistry letters 2012;22(21):6712-5.
2012: Christoph Kamper; Katharina Korpis; Lennart Anger; Patrick J Bednarski; Martin Neuenschwander; Edgar Specker; Andreas Link
Sustainable synthesis and automated deposition: an accessible discovery screening library of fragment-like purines.
Molecular diversity 2012;16(3):541-51.
2011: Ulrike Nagel; Gregor Radau; Andreas Link
Short synthesis of ethyl 3-(3-aminophenyl)propanoate.
Archiv der Pharmazie 2011;344(12):840-2.
2011: Marcus Freitag; Manfred Jung; Tim Larsen; Tobias Rumpf; Jörg Schemies; Felix Schulz; Khattab El Gaghlab; Andreas Link
Synthesis and biological activity of splitomicin analogs targeted at human NAD(+)-dependent histone deacetylases (sirtuins).
Bioorganic & medicinal chemistry 2011;19(12):3669-77.
2010: Vida Zohrabi-Kalantari; Philipp Heidler; Marcel Kaiser; Reto Brun; Christoph Kamper; Andreas Link
Inhibitors of adenosine consuming parasites through polymer-assisted N-acylation of N6-substituted 5'-amino-5'-deoxyadenosines.
Molecular diversity 2010;14(2):307-20.
2010: Andreas Link; Philipp Heidler; Marcel Kaiser; Reto Brun
Parallel synthesis of a series of non-functional ATP/NAD analogs with activity against trypanosomatid parasites.
Molecular diversity 2010;14(2):215-24.
2010: Thomas Emmrich; Ali El-Tayeb; Hesham Taha; Roland Seifert; Christa E Müller; Andreas Link
Synthesis of a hydrolytically stable, fluorescent-labeled ATP analog as a tool for probing adenylyl cyclases.
Bioorganic & medicinal chemistry letters 2010;20(1):232-5.
2009: Andreas Link; Philipp Heidler; Marcel Kaiser; Reto Brun
Synthesis of a series of N6-substituted adenosines with activity against trypanosomatid parasites.
European journal of medicinal chemistry 2009;44(9):3665-71.
2009: Philipp Heidler; Vida Zohrabi-Kalantari; Marcel Kaiser; Reto Brun; Thomas Emmrich; Andreas Link
Inhibitors of adenosine consuming parasites through polymer-assisted solution phase synthesis of lipophilic 5'-amido-5'-deoxyadenosine derivatives.
Bioorganic & medicinal chemistry 2009;17(4):1428-36.
2009: Andreas Link; Manfred Schubert-Zsilavecz
[Pharmazie in unserer Zeit 3/2009].
Pharmazie in unserer Zeit 2009;38(3):201.
2008: Dirk Giessmann; Philipp Heidler; Timothy Haemers; Serge Van Calenbergh; Armin Reichenberg; Hassan Jomaa; Claus Weidemeyer; Silke Sanderbrand; Jochen Wiesner; Andreas Link
Towards new antimalarial drugs: synthesis of non-hydrolyzable phosphate mimics as feed for a predictive QSAR study on 1-deoxy-D-xylulose-5-phosphate reductoisomerase inhibitors.
Chemistry & biodiversity 2008;5(4):643-56.
2008: Timothy Haemers; Jochen Wiesner; Dirk Giessmann; Thomas Verbrugghen; Ulrik Hillaert; Regina Ortmann; Hassan Jomaa; Andreas Link; Martin Schlitzer; Serge Van Calenbergh
Synthesis of beta- and gamma-oxa isosteres of fosmidomycin and FR900098 as antimalarial candidates.
Bioorganic & medicinal chemistry 2008;16(6):3361-71.
2007: Marcus Freitag; Marcel Kaiser; Tim Larsen; Vida Zohrabi-Kalantari; Philipp Heidler; Andreas Link
Synthesis and antiplasmodial activity of new N-[3-(4-{3-[(7-chloroquinolin-4-yl)amino]propyl}piperazin-1-yl)propyl]carboxamides.
Bioorganic & medicinal chemistry 2007;15(7):2782-8.
2006: Conrad Kunick; Carola Bleeker; Christian Prühs; Frank Totzke; Christoph Schächtele; Michael H G Kubbutat; Andreas Link
Matrix compare analysis discriminates subtle structural differences in a family of novel antiproliferative agents, diaryl-3-hydroxy-2,3,3a,10a-tetrahydrobenzo[b]cycylopenta[e]azepine-4,10(1H,5H)-diones.
Bioorganic & medicinal chemistry letters 2006;16(8):2148-53.
2005: Vida Zohrabi-Kalantari; Philipp Heidler; Tim Larsen; Andreas Link
O,N,N'-trialkylisoureas as mild activating reagents for N-acylsulfonamide anchors.
Organic letters 2005;7(25):5665-7.
2005: Tim Larsen; Andreas Link
A timely reassessment of early prediction in the bioavailability of orally administered drugs.
Angewandte Chemie (International ed. in English) 2005;44(29):4432-4.
2005: Philipp Heidler; Vida Zohrabi-Kalantari; Thierry Calmels; Marc Capet; Isabelle Berrebi-Bertrand; Jean-Charles Schwartz; Holger Stark; Andreas Link
Parallel synthesis and dopamine D3/D2 receptor screening of novel {4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}carboxamides.
Bioorganic & medicinal chemistry 2005;13(6):2009-14.
2005: Philipp Heidler; Andreas Link
N-acyl-N-alkyl-sulfonamide anchors derived from Kenner's safety-catch linker: powerful tools in bioorganic and medicinal chemistry.
Bioorganic & medicinal chemistry 2005;13(3):585-99.
2004: Vida Zohrabi-Kalantari; Andreas Link
Practical synthesis of fenbufen ethanolamide.
Archiv der Pharmazie 2004;337(10):546-8.
2004: Claudia Herforth; Philipp Heidler; Stephan Franke; Andreas Link
Polymer-bound reagents for the introduction of spacer-modified biotin labels.
Bioorganic & medicinal chemistry 2004;12(11):2895-902.
2004: Claudia Herforth; Jochen Wiesner; Philipp Heidler; Silke Sanderbrand; Serge Van Calenbergh; Hassan Jomaa; Andreas Link
Antimalarial activity of N(6)-substituted adenosine derivatives. Part 3.
Bioorganic & medicinal chemistry 2004;12(4):755-62.
2003: Andreas Link
Combinatorial chemistry as a new approach in antiparasitic drug discovery.
Parasitology research 2003;90 Suppl 2():S86-90.
2003: Philipp Heidler; Claudia Herforth; Andreas Link
Synthesis and antimalarial activity of novel N6-substituted adenosine derivatives.
Nucleosides, nucleotides & nucleic acids 2003;22(5-8):977-9.
2003: Tommie L Lincecum; Michael Tukalo; Anna Yaremchuk; Richard S Mursinna; Amy M Williams; Brian S Sproat; Wendy Van Den Eynde; Andreas Link; Serge Van Calenbergh; Morten Grøtli; Susan A Martinis; Stephen Cusack
Structural and mechanistic basis of pre- and posttransfer editing by leucyl-tRNA synthetase.
Molecular cell 2003;11(4):951-63.
2002: Claudia Herforth; Jochen Wiesner; Stephan Franke; Abolfasl Golisade; Hassan Jomaa; Andreas Link
Antimalarial activity of n(6)-substituted adenosine derivatives (part 2).
Journal of combinatorial chemistry 2002;4(4):302-14.
2002: Serge Van Calenbergh; Andreas Link; Shelly Fujikawa; Rianne A F de Ligt; Veerle Vanheusden; Abolfasl Golisade; Norbert Blaton; Jef Rozenski; Adriaan P IJzerman; Piet Herdewijn
5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists.
Journal of medicinal chemistry 2002;45(9):1845-52.
2002: Abolfasl Golisade; Jochen Wiesner; Claudia Herforth; Hassan Jomaa; Andreas Link
Anti-malarial activity of N(6)-substituted adenosine derivatives. Part I.
Bioorganic & medicinal chemistry 2002;10(3):769-77.
2002: Abolfasl Golisade; Claudia Herforth; Ludo Quirijnen; Louis Maes; Andreas Link
Improving an antitrypanosomal lead applying nucleophilic substitution on a safety catch linker.
Bioorganic & medicinal chemistry 2002;10(1):159-65.
2001: Kenneth Alan Jacobson; Zhan-Guo Gao; Aishe Chen; Dov Barak; Soon-Ai Kim; Kyeong Lee; Andreas Link; P V Rompaey; Serge Van Calenbergh; Bruce T Liang
Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides.
Journal of medicinal chemistry 2001;44(24):4125-36.
2001: Abolfasl Golisade; Claudia Herforth; Karen Wieking; Conrad Kunick; Andreas Link
Biotin labelling of amines by polymer-assisted solution-phase synthesis.
Bioorganic & medicinal chemistry letters 2001;11(13):1783-6.
2001: Christiane Schultz; Andreas Link; Conrad Kunick
Aryl rings are part of the darpone pharmacophore.
Archiv der Pharmazie 2001;334(5):163-6.
2000: Maryse Leost; Christiane Schultz; Andreas Link; Y Z Wu; J Biernat; Eva-Maria Mandelkow; James A Bibb; Gretchen L Snyder; Paul Greengard; Daniel W Zaharevitz; Rick Gussio; Adrian M Senderowicz; Edward A Sausville; Conrad Kunick; Laurent Meijer
Paullones are potent inhibitors of glycogen synthase kinase-3beta and cyclin-dependent kinase 5/p25.
European journal of biochemistry / FEBS 2000;267(19):5983-94.
2000: Abolfasl Golisade; J C Bressi; Serge Van Calenbergh; M H Gelb; Andreas Link
Polymer-assisted solution-phase synthesis of 2'-amido-2'-deoxyadenosine derivatives targeted at the NAD(+)-binding sites of parasite enzymes.
Journal of combinatorial chemistry 2000;2(5):537-44.
1999: Serge Van Calenbergh; Andreas Link; Conrad Kunick; Piet Herdewijn
Exploration of the effect of sterically demanding 3'-amido substitution of 3'-deoxyadenosines towards inhibition of cyclin-dependent kinase 1.
Die Pharmazie 1999;54(10):727-9.
1999: Christiane Schultz; Andreas Link; Maryse Leost; Daniel W Zaharevitz; Rick Gussio; Edward A Sausville; Laurent Meijer; Conrad Kunick
Paullones, a series of cyclin-dependent kinase inhibitors: synthesis, evaluation of CDK1/cyclin B inhibition, and in vitro antitumor activity.
Journal of medicinal chemistry 1999;42(15):2909-19.
1999: Andreas Link; Daniel W Zaharevitz; Conrad Kunick
Antitumor pyrido[3,2-d][1]benzazepines: synthesis and in vitro activity of thiophene analogs.
Die Pharmazie 1999;54(3):163-6.
1998: Andreas Link; Conrad Kunick
d-Fused [1]benzazepines with selective in vitro antitumor activity: synthesis and structure-activity relationships.
Journal of medicinal chemistry 1998;41(8):1299-305.
1996: Conrad Kunick; Andreas Link; M Hropot
Synthesis and in vivo testing of a potential aquaretic agent.
Die Pharmazie 1996;51(8):601-2.