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Jean Martinez

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Guillaume Miralles; Karine Puget; Jean Martinez; Amélie Maurras; Pascal Verdié; Gilles Subra
Microwave-mediated reduction of disulfide bridges with supported (tris(2-carboxyethyl)phosphine) as resin-bound reducing agent.
Rosella Spina; Jean Martinez; Evelina Colacino; Frédéric Lamaty
Poly(ethylene glycol) as a reaction matrix in platinum- or gold-catalyzed cycloisomerization: a mechanistic investigation.
Ludovic T Maillard; Jean Martinez; Ophélie Quinonéro; Gülhan Turan-Zitouni; Gülşen Akalin; Sébastien Bertout; Fatih Demirci; Pierre Fulcrand; Nicolas Masurier
Synthesis and anti-Candida activity of novel 2-hydrazino-1,3-thiazole derivatives.

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All Publications

2013: Guillaume Miralles; Karine Puget; Jean Martinez; Amélie Maurras; Pascal Verdié; Gilles Subra
Microwave-mediated reduction of disulfide bridges with supported (tris(2-carboxyethyl)phosphine) as resin-bound reducing agent.
ACS combinatorial science 2013;15(4):169-73.
2013: Rosella Spina; Jean Martinez; Evelina Colacino; Frédéric Lamaty
Poly(ethylene glycol) as a reaction matrix in platinum- or gold-catalyzed cycloisomerization: a mechanistic investigation.
Chemistry (Weinheim an der Bergstrasse, Germany) 2013;19(12):3817-21.
2013: Ludovic T Maillard; Jean Martinez; Ophélie Quinonéro; Gülhan Turan-Zitouni; Gülşen Akalin; Sébastien Bertout; Fatih Demirci; Pierre Fulcrand; Nicolas Masurier
Synthesis and anti-Candida activity of novel 2-hydrazino-1,3-thiazole derivatives.
Bioorganic & medicinal chemistry letters 2013;23(6):1803-7.
2013: Rosella Spina; Evelina Colacino; Bartolo Gabriele; Jean Martinez; Giuseppe Salerno; Frédéric Lamaty
Synthesis of pyrrolin-4-ones by Pt-catalyzed cycloisomerization in PEG under microwaves.
The Journal of organic chemistry 2013;78(6):2698-702.
2013: Marine Peuchmaur; Fabien Rodier; Jean Sévalle; Youness Touati-Jallabe; Frédéric Checler; Marie-Agnès Lacour; vincent lisowski; Jean Martinez; Jean-François Hernandez
Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor protein.
Bioorganic & medicinal chemistry 2013;21(4):1018-29.
2013: Sophie Mary; Pascal Verdié; Marjorie Damian; jean-alain fehrentz; Jacky Marie; Jean Martinez; Jean-Louis Banères
How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape.
Biochemical Society transactions 2013;41(1):144-7.
2013: David PARAMELLE; Gilles Subra; Guillaume Miralles; Jean Martinez
Chemical cross-linkers for protein structure studies by mass spectrometry.
Proteomics 2013;13(3-4):438-56.
2013: V Cassina; jean-alain fehrentz; Vittorio Locatelli; Elena Bresciani; Doriano Brogioli; Jean Martinez; R J Omeljaniuk; R Possenti; L Rizzi; D Salerno; L Tamiazzo; A Tempestini; Antonio Torsello; P Verdié; F Mantegazza
Biophysical characterization of a binding site for TLQP-21, a naturally occurring peptide which induces resistance to obesity.
Biochimica et biophysica acta 2013;1828(2):455-60.
2013: Aline Moulin; Johanne Ryan; Jean Martinez; Céline M'Kadmi; Damien Boeglin; Luc Brunel; Luc Demange; Séverine Denoyelle; jean-alain fehrentz
The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist.
Amino acids 2013;44(2):301-14.
2013: Marie Schaeffer; Eric Trinquet; Pascal Verdié; Vincent Prévot; Thomas Roux; Jean-Louis Banères; Emmanuel Bourrier; Bénédicte Dehouck; jean-alain fehrentz; David J Hodson; Chrystel Lafont; Laurent Lamarque; Fanny Langlet; Jacky Marie; Jean Martinez; Pierre-François Méry; François Molino; Patrice Mollard
Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons.
Proceedings of the National Academy of Sciences of the United States of America 2013;110(4):1512-7.
2013: Hiroshi Enomoto; Soultan Al Halifa; Jean Martinez; Benjamin Nottelet; Gilles Subra; Julien Tailhades; Jean Coudane; Mathieu Dupré; Christine Enjalbal; Muriel Amblard
Synthesis of peptide-grafted comb polypeptides via polymerisation of NCA-peptides.
Chemical communications (Cambridge, England) 2013;49(4):409-11.
2012: Mathieu Dupré; Christine Enjalbal; Toufik Hadjersi; Jean Martinez; Nacéra Megouda; Rabah Boukherroub; Sonia Cantel; Yannick Coffinier
Investigation of silicon-based nanostructure morphology and chemical termination on laser desorption ionization mass spectrometry performance.
Analytical chemistry 2012;84(24):10637-44.
2012: Thomas-Xavier Métro; Thomas Reidon; Jordi Sarpoulet; Julien Bonnamour; Jean Martinez; Frédéric Lamaty
Mechanosynthesis of amides in the total absence of organic solvent from reaction to product recovery.
Chemical communications (Cambridge, England) 2012;48(96):11781-3.
2012: Valérie Declerck; Xavier Bantreil; Evelina Colacino; Jean Martinez; Frédéric Lamaty
Poly(ethylene glycol) as reaction medium for mild Mizoroki-Heck reaction in a ball-mill.
Chemical communications (Cambridge, England) 2012;48(96):11778-80.
2012: Rosella Spina; Evelina Colacino; Bartolo Gabriele; Jean Martinez; Giuseppe Salerno; Frédéric Lamaty
Preparation of enantioenriched iodinated pyrrolinones by iodocyclization of α-amino-ynones.
Organic & biomolecular chemistry 2012;10(45):9085-9.
2012: Maxime Louet; Jean Martinez; Landry Charlier; NICOLAS FLOQUET
Dissociation of membrane-anchored heterotrimeric G-protein induced by G(α) subunit binding to GTP.
Journal of chemical information and modeling 2012;52(11):3022-7.
2012: Baptiste Legrand; Jean Martinez; Emmanuel Wenger; Christophe André; Marie Christine Averlant-Petit; M Calmes; Claude Didierjean; Muriel Amblard
Robust helix formation in a new family of oligoureas based on a constrained bicyclic building block.
Angewandte Chemie (International ed. in English) 2012;51(45):11267-70.
2012: Nicolas Masurier; Maciej Pawłowski; Muriel Amblard; Jean Martinez; Pascal Verdié; Pawel Zajdel; Gilles Subra
A new highly versatile handle for chemistry on a solid support: the pipecolic linker.
Chemistry (Weinheim an der Bergstrasse, Germany) 2012;18(37):11536-40.
2012: Mathieu Dupré; Jean-Olivier Durand; Sonia Cantel; Jean Martinez; Christine Enjalbal
Silica nanoparticles pre-spotted onto target plate for laser desorption/ionization mass spectrometry analyses of peptides.
Analytica chimica acta 2012;741():47-57.
2012: Sonia Cantel; Christine Enjalbal; Jean Martinez; Keiichiro Ohara; Luc Brunel; Jean-Jacques Vasseur; Michael Smietana
An innovative strategy for sulfopeptides analysis using MALDI-TOF MS reflectron positive ion mode.
Proteomics 2012;12(14):2247-57.
2012: C Martin; Jean Martinez; H Miramon; N Vanthuyne; Florine Cavelier
Resolution of protected silaproline for a gram scale preparation.
Amino acids 2012;43(2):649-55.
2012: Christophe André; Monique Calmès; Françoise Escale; Jean Martinez; Muriel Amblard; Olivier Songis
New 1,3-amino alcohols derived from enantiopure bridgehead β-aminobicyclo[2.2.2]oct-5-ene-2-carboxylic acids.
Amino acids 2012;43(1):415-21.
2012: Xiaoli Shi; Pascale Zimmermann; Sandrine Opi; Isabelle Parrot; Audrey Restouin; Stefan T Arold; Stephane Betzi; Yves Collette; Mingdong Huang; Patrick Lecine; Adrien Lugari; Jean Martinez; XAVIER MORELLI
Structural recognition mechanisms between human Src homology domain 3 (SH3) and ALG-2-interacting protein X (Alix).
FEBS letters 2012;586(13):1759-64.
2012: Sophie Mary; Marjorie Damian; jean-alain fehrentz; Nicolas Floquet; Maxime Louet; Jacky Marie; Jean Martinez; Jean-Louis Banères
Ligands and signaling proteins govern the conformational landscape explored by a G protein-coupled receptor.
Proceedings of the National Academy of Sciences of the United States of America 2012;109(21):8304-9.
2012: Nicolas Masurier; Emmanuel Moreau; Jean Martinez; Roberta Aruta; Séverine Denoyelle; Vincent Gaumet; vincent lisowski; Ludovic T Maillard
Selective C-acylation of 2-aminoimidazo[1,2-a]pyridine: application to the synthesis of imidazopyridine-fused [1,3]diazepinones.
The Journal of organic chemistry 2012;77(7):3679-85.
2012: Mathieu Dupré; Rabah Boukherroub; Sonia Cantel; Yannick Coffinier; Jean Martinez; Christine Enjalbal
Laser desorption ionization mass spectrometry of protein tryptic digests on nanostructured silicon plates.
Journal of proteomics 2012;75(7):1973-90.
2012: Amer Moussa; Jean Martinez; Patrick Meffre; Valérie Rolland
Chemoenzymatic routes to enantiomerically pure 2-azatyrosine and 2-, 3- and 4-pyridylalanine derivatives.
Amino acids 2012;42(4):1339-48.
2012: Pierrick Nun; Violaine Pérez; Monique Calmès; Jean Martinez; Frédéric Lamaty
Preparation of chiral amino esters by asymmetric phase-transfer catalyzed alkylations of Schiff bases in a ball mill.
Chemistry (Weinheim an der Bergstrasse, Germany) 2012;18(12):3773-9.
2012: Jean-Daniel Malcor; Jean Martinez; Nadine Payrot; Geneviève ROUGON; Patrick Vlieghe; Karima Abouzid; Marion David; Franck Debarbieux; Aude Faucon; Nicolas Floquet; Guillaume Jacquot; Michel Khrestchatisky; vincent lisowski
Chemical optimization of new ligands of the low-density lipoprotein receptor as potential vectors for central nervous system targeting.
Journal of medicinal chemistry 2012;55(5):2227-41.
2012: Christophe André; Marie Christine Averlant-Petit; Muriel Amblard; Cheng Deng; Claude Didierjean; Baptiste Legrand; Jean Martinez; Guillaume Pickaert; M Calmes
(S)-ABOC: a rigid bicyclic β-amino acid as turn inducer.
Organic letters 2012;14(4):960-3.
2012: Marjorie Damian; jean-alain fehrentz; Jean-Philippe Leyris; Jacky Marie; Jean Martinez; Jean-Louis Banères; Pascal Verdié; Sophie Mary
High constitutive activity is an intrinsic feature of ghrelin receptor protein: a study with a functional monomeric GHS-R1a receptor reconstituted in lipid discs.
The Journal of biological chemistry 2012;287(6):3630-41.
2012: Mathieu Dupré; Sonia Cantel; Jean Martinez; Christine Enjalbal
Occurrence of C-terminal residue exclusion in peptide fragmentation by ESI and MALDI tandem mass spectrometry.
Journal of the American Society for Mass Spectrometry 2012;23(2):330-46.
2012: Maxime Louet; Jean Martinez; NICOLAS FLOQUET
GDP release preferentially occurs on the phosphate side in heterotrimeric G-proteins.
PLoS computational biology 2012;8(7):e1002595.
2011: Adrien Lugari; Jean Martinez; Stefan T Arold; Sebastian Breuer; Yves Collette; Thibault Coursindel; Alexis Nazabal; Sandrine Opi; Isabelle Parrot; Audrey Restouin; Xiaoli Shi; Bruce E Torbett; XAVIER MORELLI
A specific protein disorder catalyzer of HIV-1 Nef.
Bioorganic & medicinal chemistry 2011;19(24):7401-6.
2011: Pascal Verdié; Muriel Amblard; Sonia Cantel; M Cristau; Christine Enjalbal; Jean Martinez; Karine Puget; Luisa Ronga; Gilles Subra
Oxyfold: a simple and efficient solid-supported reagent for disulfide bond formation.
Chemistry, an Asian journal 2011;6(9):2382-9.
2011: Nikola Pavlov; Emmanuel Wenger; Claude Didierjean; Pierre Gilles; Jean Martinez; Emilia Naydenova; Monique Calmès
Asymmetric synthesis of β2-tryptophan analogues via Friedel-Crafts alkylation of indoles with a chiral nitroacrylate.
The Journal of organic chemistry 2011;76(15):6116-24.
2011: Maxime Louet; Jean Martinez; david perahia; NICOLAS FLOQUET
A concerted mechanism for opening the GDP binding pocket and release of the nucleotide in hetero-trimeric G-proteins.
Journal of molecular biology 2011;411(1):298-312.
2011: Julien Tailhades; Pascal Verdié; Sébastien Blanquer; Jean Coudane; Jean Martinez; Benjamin Nottelet; Etienne Schacht; Gilles Subra; Muriel Amblard
From polyesters to polyamides via O-N acyl migration: an original multi-transfer reaction.
Macromolecular rapid communications 2011;32(12):876-80.
2011: David PARAMELLE; Christine Enjalbal; Muriel Amblard; Eric Forest; Michaël Heymann; Sonia Cantel; Christophe Geourjon; Jean Martinez; Gilles Subra
Solid-Phase Cross-Linking (SPCL): a new tool for protein structure studies.
Proteomics 2011;11(7):1277-86.
2011: Monique Calmes; Françoise Escale; Claude Didierjean; Jean Martinez
Synthesis of enantiopure trans-N-Boc-3-aminobicyclo[2.2.2]octane-2-carboxylic acids and their bicyclic 1,3-amino alcohol derivatives via the [4+2] cycloaddition of 1,3-cyclohexadiene to a chiral β-nitroacrylate.
Chirality 2011;23(3):245-9.
2011: Fatimazohra Lenda; Nadine Crouzin; Mélanie Cavalier; Janique Guiramand; Fabien Lanté; Gérard Barbanel; Catherine Cohen-Solal; Jean Martinez; Farhate Guenoun; Frédéric Lamaty; Michel Vignes
Synthesis of C5-tetrazole derivatives of 2-amino-adipic acid displaying NMDA glutamate receptor antagonism.
Amino acids 2011;40(3):913-22.
2011: Youness Touati-Jallabe; Laurent Chiche; Abdallah Hamzé; André Aumelas; Vincent Lisowski; Dorothée Berthomieu; Jean Martinez; Jean-François Hernandez
Cyclic peptides with a diversely substituted guanidine bridge: solid-phase synthesis and structural analysis.
Chemistry (Weinheim an der Bergstrasse, Germany) 2011;17(9):2566-70.
2011: Alice Baron; Pascal Verdié; Jean Martinez; Frédéric Lamaty
cis-Apa: a practical linker for the microwave-assisted preparation of cyclic pseudopeptides via RCM cyclative cleavage.
The Journal of organic chemistry 2011;76(3):766-72.
2011: Mathieu Dupré; Sonia Cantel; Pascal Verdié; Jean Martinez; Christine Enjalbal
Sequencing Lys-N proteolytic peptides by ESI and MALDI tandem mass spectrometry.
Journal of the American Society for Mass Spectrometry 2011;22(2):265-79.
2011: Jean-Philippe Leyris; Thomas Roux; Eric Trinquet; Pascal Verdié; Jean-Alain Fehrentz; Nadia Oueslati; Stéphanie Douzon; Emmanuel Bourrier; Laurent Lamarque; Didier Gagne; Jean-Claude Galleyrand; Céline M'kadmi; Jean Martinez; Sophie Mary; Jean-Louis Banères; Jacky Marie
Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a.
Analytical biochemistry 2011;408(2):253-62.
2011: Emilie Pringos; Jean Martinez; Michel Vignes; Valerie Rolland
Peptide neurotoxins that affect voltage-gated calcium channels: a close-up on ω-agatoxins.
Toxins 2011;3(1):17-42.
2010: Pauline Petiot; Clarence Charnay; Jean Martinez; Lucy Puttergill; Francisco Galindo; Frederic Lamaty; Evelina Colacino
Synthesis of a new hydrophilic poly(ethylene glycol)-ionic liquid and its application in peptide synthesis.
Chemical communications (Cambridge, England) 2010;46(46):8842-4.
2010: David PARAMELLE; Gilles Subra; Lubomir L Vezenkov; Marie Maynadier; Christophe André; Christine Enjalbal; Monique Calmès; Marcel Garcia; Jean Martinez; Muriel Amblard
A straightforward approach for cellular-uptake quantification.
Angewandte Chemie (International ed. in English) 2010;49(44):8240-3.
2010: Lubomir L Vezenkov; Marie Maynadier; Jean-François Hernandez; Marie-Christine Averlant-Petit; Olivier Fabre; Ettore Benedetti; Marcel Garcia; Jean Martinez; Muriel Amblard
Noncationic dipeptide mimic oligomers as cell penetrating nonpeptides (CPNP).
Bioconjugate chemistry 2010;21(10):1850-4.
2010: Thibault Coursindel; Audrey Restouin; Georges Dewynter; Jean Martinez; Yves Collette; Isabelle Parrot
Stereoselective ring contraction of 2,5-diketopiperazines: An innovative approach to the synthesis of promising bioactive 5-membered scaffolds.
Bioorganic chemistry 2010;38(5):210-7.
2010: Catherine Gozé; Gilbert Bergé; Céline M'Kadmi; Nicolas Floquet; Didier Gagne; Jean-Claude Galleyrand; Jean-Alain Fehrentz; Jean Martinez
Involvement of tryptophan W276 and of two surrounding amino acid residues in the high constitutive activity of the ghrelin receptor GHS-R1a.
European journal of pharmacology 2010;643(2-3):153-61.
2010: Pawel Zajdel; Nicolas Masurier; Pierre Sanchez; Maciej Pawlowski; Aude Kreiter; Gaël Nomezine; Christine Enjalbal; Muriel Amblard; Jean Martinez; Gilles Subra
Recycling the versatile Pipecolic linker.
Journal of combinatorial chemistry 2010;12(5):747-53.
2010: Paweł Zajdel; Gaël Nomezine; Nicolas Masurier; Muriel Amblard; Maciej Pawłowski; Jean Martinez; Gilles Subra
A new highly versatile handle for chemistry on a solid support: the pipecolic linker.
Chemistry (Weinheim an der Bergstrasse, Germany) 2010;16(25):7547-53.
2010: Julien Schmidt; Véronique Garambois; Luc Rocheblave; Jean Martinez; André Pèlegrin; Florine Cavelier; Eric Vivès
Cyclization of peptides through a urea bond: application to the Arg-Gly-Asp tripeptide.
Chembiochem : a European journal of chemical biology 2010;11(8):1083-92.
2010: Aline Moulin; Mathieu Bibian; Anne-Laure Blayo; Sarah El Habnouni; Jean Martinez; Jean-Alain Fehrentz
Synthesis of 3,4,5-trisubstituted-1,2,4-triazoles.
Chemical reviews 2010;110(4):1809-27.
2010: Hélène Miramon; Florine Cavelier; Jean Martinez; Hervé Cottet
Highly resolutive separations of hardly soluble synthetic polypeptides by capillary electrophoresis.
Analytical chemistry 2010;82(1):394-9.
2010: Julien Tailhades; Marie-Aude Gidel; Benjamin Grossi; Jennifer Lécaillon; Luc Brunel; Gilles Subra; Jean Martinez; Muriel Amblard
Synthesis of peptide alcohols on the basis of an O-N acyl-transfer reaction.
Angewandte Chemie (International ed. in English) 2010;49(1):117-20.
2009: David PARAMELLE; Sonia Cantel; Christine Enjalbal; Muriel Amblard; Eric Forest; Michaël Heymann; Christophe Geourjon; Jean Martinez; Gilles Subra
A new generation of cross-linkers for selective detection by MALDI MS.
Proteomics 2009;9(23):5384-8.
2009: Reine Nehmé; Catherine Perrin; Vincent Guerlavais; Jean-Alain Fehrentz; Hervé Cottet; Jean Martinez; Huguette Fabre
Use of coated capillaries for the electrophoretic separation of stereoisomers of a growth hormone secretagogue.
Electrophoresis 2009;30(21):3772-9.
2009: N Salomé; C Hansson; Maria Taube; L Gustafsson-Ericson; Emil Egecioglu; L Karlsson-Lindahl; Jean-Alain Fehrentz; Jean Martinez; Daniel Perrissoud; Suzanne Dickson
On the central mechanism underlying ghrelin's chronic pro-obesity effects in rats: new insights from studies exploiting a potent ghrelin receptor antagonist.
Journal of neuroendocrinology 2009;21(9):777-85.
2009: Pawel Zajdel; Gilles Subra; Pascal Verdie; Ewa Gabzdyl; Andrzej Jacek Bojarski; Beata Duszyńska; Jean Martinez; Maciej Pawłowski
Sulfonamides with the N-alkyl-N'-dialkylguanidine moiety as 5-HT7 receptor ligands.
Bioorganic & medicinal chemistry letters 2009;19(16):4827-31.
2009: Nawar Shenar; Sonia Cantel; Jean Martinez; Christine Enjalbal
Comparison of inert supports in laser desorption/ionization mass spectrometry of peptides: pencil lead, porous silica gel, DIOS-chip and NALDI target.
Rapid communications in mass spectrometry : RCM 2009;23(15):2371-9.
2009: Pawel Zajdel; Maciej Pawłowski; Jean Martinez; Gilles Subra
Combinatorial chemistry on solid support in the search for central nervous system agents.
Combinatorial chemistry & high throughput screening 2009;12(7):723-39.
2009: Jean Sevalle; Erwan Ayral; Jean-François Hernandez; Jean Martinez; Frédéric Checler
Pharmacological evidences for DFK167-sensitive presenilin-independent gamma-secretase-like activity.
Journal of neurochemistry 2009;110(1):275-83.
2009: Daniel Farran; Delphine Echalier; Jean Martinez; Georges Dewynter
Regioselective and sequential reactivity of activated 2,5-diketopiperazines.
Journal of peptide science : an official publication of the European Peptide Society 2009;15(7):474-8.
2009: Nicolas Salomé; David Haage; Daniel Perrissoud; Aline Moulin; Luc Demange; Emil Egecioglu; Jean-Alain Fehrentz; Jean Martinez; Suzanne Dickson
Anorexigenic and electrophysiological actions of novel ghrelin receptor (GHS-R1A) antagonists in rats.
European journal of pharmacology 2009;612(1-3):167-73.
2009: Anne-Claude Couffin-Hoarau; Anne-Marie Aubertin; Mahfoud Boustta; Sylvie Schmidt; Jean-Alain Fehrentz; Jean Martinez; Michel Vert
Peptide-poly(L-lysine citramide) conjugates and their in vitro anti-HIV behavior.
Biomacromolecules 2009;10(4):865-76.
2009: Valérie Declerck; loic toupet; Jean Martinez; Frédéric Lamaty
Selective [3 + 2] Huisgen cycloaddition. Synthesis of trans-disubstituted triazolodiazepines from aza-Baylis-Hillman adducts.
The Journal of organic chemistry 2009;74(5):2004-7.
2009: Erwan Ayral; Philippe Gloanec; Gilbert Bergé; Guillaume De Nanteuil; Philippe Mennecier; Alain Rupin; Tony J Verbeuren; Pierre Fulcrand; Jean Martinez; Jean-François Hernandez
Design, synthesis, and biological evaluation of 1,5-benzothiazepine-4-one derivatives targeting factor VIIa/tissue factor.
Bioorganic & medicinal chemistry letters 2009;19(5):1386-91.
2009: Pawel Zajdel; Gilles Subra; Pascal Verdie; Andrzej Jacek Bojarski; Beata Duszyńska; Katarzyna Basista; Jolanta Obniska; Jean Martinez; Maciej Pawłowski
The influence of an ethylene spacer on the 5-HT(1A) and 5-HT(2A) receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones.
European journal of medicinal chemistry 2009;44(2):800-8.
2009: Valérie Declerck; Pierrick Nun; Jean Martinez; Frédéric Lamaty
Solvent-free synthesis of peptides.
Angewandte Chemie (International ed. in English) 2009;48(49):9318-21.
2009: M'Barek Bouazaoui; Stéphane Mari; Pierre Czernic; Catherine Curie; Jean Martinez; Florine Cavelier
Synthesis and biological activity of nicotianamine and analogues.
Advances in experimental medicine and biology 2009;611():555-7.
2009: Youness Touati-Jallabe; Abdallah Hamzé; Gilbert Bergé; Claudia Verna; Anne-Dominique Lajoix; Pierre Fulcrand; Jean Martinez; Jean-François Hernandez
Solid-phase synthesis of dipeptidic and pseudo-dipeptidic potential NOS inhibitors through a side-chain anchoring approach.
Advances in experimental medicine and biology 2009;611():133-4.
2009: Valérie Declerck; Jean Martinez; Frédéric Lamaty
aza-Baylis-Hillman reaction.
Chemical reviews 2009;109(1):1-48.
2008: Daniel Farran; Isabelle Parrot; Loïc Toupet; Jean Martinez; Georges Dewynter
Transannular rearrangement of activated 2,5-diketopiperazines: a key route to original scaffolds.
Organic & biomolecular chemistry 2008;6(21):3989-96.
2008: Pierre-Emmanuel Stoebner; Lionel Le Gallic; Marie L Berthe; Nathalie Boulle; Benjamin Lallemant; Myriam Marque; Catherine Gaspard; Christophe Delfour; Thierry Lavabre-Bertrand; Jean Martinez; Laurent Meunier
Decreased expression of thymidine phosphorylase/platelet-derived endothelial cell growth factor in basal cell carcinomas.
Experimental dermatology 2008;17(11):908-15.
2008: Nawar Shenar; Jean Martinez; Christine Enjalbal
Laser desorption/ionization mass spectrometry on porous silica and alumina for peptide mass fingerprinting.
Journal of the American Society for Mass Spectrometry 2008;19(5):632-44.
2008: Aline Moulin; Luc Demange; Joanne Ryan; Delphine Mousseaux; Pierre Sanchez; Gilbert Bergé; Didier Gagne; Daniel Perrissoud; Vittorio Locatelli; Antonio Torsello; Jean-Claude Galleyrand; Jean-Alain Fehrentz; Jean Martinez
New trisubstituted 1,2,4-triazole derivatives as potent ghrelin receptor antagonists. 3. Synthesis and pharmacological in vitro and in vivo evaluations.
Journal of medicinal chemistry 2008;51(3):689-93.
2008: Aline Moulin; Luc Demange; Joanne Ryan; Céline M'Kadmi; Jean-Claude Galleyrand; Jean Martinez; Jean-Alain Fehrentz
Trisubstituted 1,2,4-triazoles as ligands for the ghrelin receptor: on the significance of the orientation and substitution at position 3.
Bioorganic & medicinal chemistry letters 2008;18(1):164-8.
2007: Aline Moulin; Luc Demange; Gilbert Bergé; Didier Gagne; Joanne Ryan; Delphine Mousseaux; Annie Heitz; Daniel Perrissoud; Vittorio Locatelli; Antonio Torsello; Jean-Claude Galleyrand; Jean-Alain Fehrentz; Jean Martinez
Toward potent ghrelin receptor ligands based on trisubstituted 1,2,4-triazole structure. 2. Synthesis and pharmacological in vitro and in vivo evaluations.
Journal of medicinal chemistry 2007;50(23):5790-806.
2007: Daniel Farran; Loïc Toupet; Jean Martinez; Georges Dewynter
Stereocontrolled synthesis of 2,4-diamino-3-hydroxyacids starting from diketopiperazines: a new route for the preparation of statine analogues.
Organic letters 2007;9(23):4833-6.
2007: Gülhan Turan-Zitouni; Jean-Alain Fehrentz; Pierre Chevallet; Jean Martinez; Zafer Asim Kaplancikli; Ahmet Ozdemir; Muhittin Arslanyolu; Mehmet Taha Yildiz
Synthesis and antibacterial activity of tert-butyl [1-benzyl-2[(4-aryl-2-thiazolyl)hydrazono]ethyl]carbamate derivatives.
Archiv der Pharmazie 2007;340(6):310-4.
2007: Luc Demange; Damien Boeglin; Aline Moulin; Delphine Mousseaux; Joanne Ryan; Gilbert Bergé; Didier Gagne; Annie Heitz; Daniel Perrissoud; Vittorio Locatelli; Antonio Torsello; Jean-Claude Galleyrand; Jean-Alain Fehrentz; Jean Martinez
Synthesis and pharmacological in vitro and in vivo evaluations of novel triazole derivatives as ligands of the ghrelin receptor. 1.
Journal of medicinal chemistry 2007;50(8):1939-57.
2007: Pawel Zajdel; Gilles Subra; Andrzej Jacek Bojarski; Beata Duszyńska; Ewa Tatarczyńska; Agnieszka Nikiforuk; Ewa Chojnacka-Wójcik; Maciej Pawłowski; Jean Martinez
Novel class of arylpiperazines containing N-acylated amino acids: their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation.
Bioorganic & medicinal chemistry 2007;15(8):2907-19.
2007: Laetitia Mouls; Jean-Louis Aubagnac; Jean Martinez; Christine Enjalbal
Low energy peptide fragmentations in an ESI-Q-Tof type mass spectrometer.
Journal of proteome research 2007;6(4):1378-91.
2007: Yann Brouillette; vincent lisowski; Pierre Fulcrand; Jean Martinez
Reactivity study of 1H-thieno[3,2-d][1,3]oxazine-2,4-dione toward the synthesis of bicyclic 3,4-dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione analogues.
The Journal of organic chemistry 2007;72(7):2662-5.
2007: Pascal Verdié; Gilles Subra; Lidia Feliu; Pierre Sanchez; Gilbert Bergé; Geneviève Garcin; Jean Martinez
On-line synthesis of pseudopeptide library incorporating a benzodiazepinone turn mimic: biological evaluation on MC1 receptors.
Journal of combinatorial chemistry 2007;9(2):254-62.
2007: Valérie Declerck; Hassan Allouchi; Jean Martinez; Frédéric Lamaty
2-Trimethylsilylethanesulfonyl (SES) versus tosyl (Ts) protecting group in the preparation of nitrogen-containing five-membered rings. A novel route for the synthesis of substituted pyrrolines and pyrrolidines.
The Journal of organic chemistry 2007;72(4):1518-21.
2007: Daniel Farran; Isabelle Parrot; Jean Martinez; Georges Dewynter
Transannular rearrangement of activated lactams: stereoselective synthesis of substituted pyrrolidine-2,4-diones from diketopiperazines.
Angewandte Chemie (International ed. in English) 2007;46(39):7488-90.
2007: Aline Moulin; Jean Martinez; Jean-Alain Fehrentz
Synthesis of peptide aldehydes.
Journal of peptide science : an official publication of the European Peptide Society 2007;13(1):1-15.
2006: Laetitia Mouls; Gilles Subra; Jean-Louis Aubagnac; Jean Martinez; Christine Enjalbal
Tandem mass spectrometry of amidated peptides.
Journal of mass spectrometry : JMS 2006;41(11):1470-83.
2006: Florine Cavelier; Damien Marchand; Patrick Mbassi; Jean Martinez; Michel Marraud
Conformational studies of proline-, thiaproline- and dimethylsilaproline-containing diketopiperazines.
Journal of peptide science : an official publication of the European Peptide Society 2006;12(10):621-5.
2006: Moustapha Alfa Cissé; Céline Gandreuil; Jean-François Hernandez; Jean Martinez; Frédéric Checler; Bruno Vincent
Design and characterization of a novel cellular prion-derived quenched fluorimetric substrate of alpha-secretase.
Biochemical and biophysical research communications 2006;347(1):254-60.
2006: Sílvia Pujals; Jimena Fernandez-Carneado; Marcelo J Kogan; Jean Martinez; Florine Cavelier; Ernest Giralt
Replacement of a proline with silaproline causes a 20-fold increase in the cellular uptake of a Pro-rich peptide.
Journal of the American Chemical Society 2006;128(26):8479-83.
2006: Muriel Amblard; Jean-Alain Fehrentz; Jean Martinez; Gilles Subra
Methods and protocols of modern solid phase Peptide synthesis.
Molecular biotechnology 2006;33(3):239-54.
2006: Pawel Zajdel; Gilles Subra; Andrzej Jacek Bojarski; Beata Duszyńska; Maciej Pawłowski; Jean Martinez
Arylpiperazines with N-acylated amino acids as 5-HT1A receptor ligands.
Bioorganic & medicinal chemistry letters 2006;16(13):3406-10.
2006: Cécile Ganneau; Aline Moulin; Luc Demange; Jean Martinez; Jean-Alain Fehrentz
The epimerization of peptide aldehydes--a systematic study.
Journal of peptide science : an official publication of the European Peptide Society 2006;12(7):497-501.
2006: Patrice Ribière; Valérie Declerck; Jean Martinez; Frédéric Lamaty
2-(Trimethylsilyl)ethanesulfonyl (or SES) group in amine protection and activation.
Chemical reviews 2006;106(6):2249-69.
2006: Delphine Mousseaux; Lionel Le Gallic; Joanne Ryan; Catherine Oiry; Didier Gagne; Jean-Alain Fehrentz; Jean-Claude Galleyrand; Jean Martinez
Regulation of ERK1/2 activity by ghrelin-activated growth hormone secretagogue receptor 1A involves a PLC/PKCvarepsilon pathway.
British journal of pharmacology 2006;148(3):350-65.
2006: Géraldine Ibarz; Catherine Oiry; Eric Carnazzi; Philippe Crespy; Chantal Escrieut; Daniel Fourmy; Jean-Claude Galleyrand; Didier Gagne; Jean Martinez
Cholecystokinin 1 receptor modulates the MEKK1-induced c-Jun trans-activation: structural requirements of the receptor.
British journal of pharmacology 2006;147(8):951-8.
2005: Caroline Morel; Géraldine Ibarz; Catherine Oiry; Eric Carnazzi; Gilbert Bergé; Didier Gagne; Jean-Claude Galleyrand; Jean Martinez
Cross-interactions of two p38 mitogen-activated protein (MAP) kinase inhibitors and two cholecystokinin (CCK) receptor antagonists with the CCK1 receptor and p38 MAP kinase.
The Journal of biological chemistry 2005;280(22):21384-93.
2005: Christine Enjalbal; Patrice Ribière; Frédéric Lamaty; Neerja Yadav-Bhatnagar; Jean Martinez; Jean-Louis Aubagnac
MALDI-TOF MS analysis of soluble PEG based multi-step synthetic reaction mixtures with automated detection of reaction failure.
Journal of the American Society for Mass Spectrometry 2005;16(5):670-8.
2005: Solveig Lefranc-Jullien; vincent lisowski; Jean-François Hernandez; Jean Martinez; Frédéric Checler
Design and characterization of a new cell-permeant inhibitor of the beta-secretase BACE1.
British journal of pharmacology 2005;145(2):228-35.
2005: Pawel Zajdel; Gilles Subra; Andrzej Jacek Bojarski; Beata Duszyńska; Maciej Pawłowski; Jean Martinez
Parallel solid-phase synthesis and characterization of new sulfonamide and carboxamide proline derivatives as potential CNS agents.
Bioorganic & medicinal chemistry 2005;13(8):3029-35.
2005: Muriel Amblard; Jean-Alain Fehrentz; Jean Martinez; Gilles Subra
Fundamentals of modern peptide synthesis.
Methods in molecular biology (Clifton, N.J.) 2005;298():3-24.
2004: Abdallah Hamzé; Jean Martinez; abdallah hamze
Solid-phase synthesis of arginine-containing peptides and fluorogenic substrates using a side-chain anchoring approach.
The Journal of organic chemistry 2004;69(24):8394-402.
2004: Valérie Declerck; Patrice Ribière; Jean Martinez; Frédéric Lamaty
Sequential aza-Baylis-Hillman/ring closing metathesis/aromatization as a novel route for the synthesis of substituted pyrroles.
The Journal of organic chemistry 2004;69(24):8372-81.
2004: Pawel Zajdel; Andrzej Jacek Bojarski; Ryszard Bugno; Slawomir Jurczyk; Marcin Kołaczkowski; Mateusz Nowak; Gilles Subra; Jean Martinez; Maciej Pawłowski
A study on application of impregnated synthetic peptide TLC stationary phases for the screening of 5-HT1A ligands. Part 2.
Biomedical chromatography : BMC 2004;18(8):542-9.
2004: Jérôme Giovannoni; Claude Didierjean; Philippe Durand; Michel Marraud; André Aubry; Patrice Renaut; Jean Martinez; Muriel Amblard
Synthesis and structure of symmetrical bicyclic hexapeptides bridged by metathesis reaction.
Organic letters 2004;6(20):3449-52.
2004: Sonia Cantel; Annie Heitz; Jean Martinez; Jean-Alain Fehrentz
Synthesis of chiral alpha-amino aldehydes linked by their amine function to solid support.
Journal of peptide science : an official publication of the European Peptide Society 2004;10(9):531-4.
2004: Pawel Zajdel; Gilles Subra; Andrzej Jacek Bojarski; Beata Duszyńska; Maciej Pawłowski; Jean Martinez
A new class of arylpiperazine derivatives: the library synthesis on SynPhase lanterns and biological evaluation on serotonin 5-HT(1A) and 5-HT(2A) receptors.
Journal of combinatorial chemistry 2004;6(5):761-7.
2004: Patrice Ribière; Christine Enjalbal; Jean-Louis Aubagnac; Neerja Yadav-Bhatnagar; Jean Martinez; Frédéric Lamaty
Preparation of poly(ethylene glycol) sulfonamide: synthesis of N-supported beta-aminoesters via the aza-Baylis-Hillman reaction.
Journal of combinatorial chemistry 2004;6(4):464-7.
2004: Sonia Cantel; Stéphane Desgranges; Jean Martinez; Jean-Alain Fehrentz
Saponification of esters of chiral alpha-amino acids anchored through their amine function on solid support.
Journal of peptide science : an official publication of the European Peptide Society 2004;10(6):326-8.
2004: Florine Cavelier; D Marchand; Jean Martinez; S Sagan
Biological activity of silylated amino acid containing substance P analogues.
The journal of peptide research : official journal of the American Peptide Society 2004;63(3):290-6.
2004: Jean-Louis Aubagnac; Christine Enjalbal; Jean Martinez; Pierre Sanchez; Gilles Subra
Automated vs manual profiling of peptide libraries by mass spectrometry.
Methods in molecular biology (Clifton, N.J.) 2004;251():377-86.
2003: J Huck; Marie-Louise Roumestant; Jean Martinez
From beta-N-tert-butyloxycarbonyl N-carboxyanhydrides to beta-aminoacid derivatives.
The journal of peptide research : official journal of the American Peptide Society 2003;62(6):233-7.
2003: Damien Boeglin; Sonia Cantel; Annie Heitz; Jean Martinez; Jean-Alain Fehrentz
Solution and solid-supported synthesis of 3,4,5-trisubstituted 1,2,4-triazole-based peptidomimetics.
Organic letters 2003;5(23):4465-8.
2003: Agnès Petit; A Pasini; Cristine Alves da Costa; Erwan Ayral; Jean-François Hernandez; Cecile Dumanchin-Njock; C J Phiel; Philippe Marambaud; Sherwin Wilk; M Farzan; Pierre Fulcrand; Jean Martinez; D Andrau; Cristine Alves da Costa
JLK isocoumarin inhibitors: selective gamma-secretase inhibitors that do not interfere with notch pathway in vitro or in vivo.
Journal of neuroscience research 2003;74(3):370-7.
2003: Abdallah Hamzé; abdallah hamze; Pierre Fulcrand; Jean Martinez
Synthesis of various 3-substituted 1,2,4-oxadiazole-containing chiral beta 3- and alpha-amino acids from Fmoc-protected aspartic acid.
The Journal of organic chemistry 2003;68(19):7316-21.
2003: Johny Wehbe; Valérie Rolland; Jean Martinez; Marc Rolland
An intermediate in a new synthesis approach to beta-substituted beta-hydroxyaspartame.
Acta crystallographica. Section C, Crystal structure communications 2003;59(Pt 8):o473-5.
2003: David Andrau; Cecile Dumanchin-Njock; Erwan Ayral; Jean Vizzavona; Mike Farzan; Michel Boisbrun; Pierre Fulcrand; Jean-François Hernandez; Jean Martinez; Solveig Lefranc-Jullien; Frédéric Checler
BACE1- and BACE2-expressing human cells: characterization of beta-amyloid precursor protein-derived catabolites, design of a novel fluorimetric assay, and identification of new in vitro inhibitors.
The Journal of biological chemistry 2003;278(28):25859-66.
2003: Pawel Zajdel; Andrzej Jacek Bojarski; Hanna Byrtus; Grazyna Chłoń-Rzepa; Jolanta Obniska; Pierre Chevallet; Jean Martinez; Maciej Pawłowski
Preliminary study on application of impregnated synthetic peptide TLC stationary phases for the pre-screening of 5-HT1A ligands.
Biomedical chromatography : BMC 2003;17(5):312-7.
2003: Lidia Feliu; Gilles Subra; Jean Martinez; Muriel Amblard
Spiroimidazolidinone library derivatives on SynPhase lanterns.
Journal of combinatorial chemistry 2003;5(4):356-61.
2003: Johny Wehbe; Tarek Kassem; Valérie Rolland; Marc Rolland; Mohamad Tabcheh; Marie-Louise Roumestant; Jean Martinez
Optically pure beta-substituted beta-hydroxy aspartates as glutamate transporter blockers.
Organic & biomolecular chemistry 2003;1(11):1938-42.
2003: Celine Gales; Marc Poirot; Julien Taillefer; Bernard Maigret; Jean Martinez; Luis Moroder; Chantal Escrieut; Lucien Pradayrol; Daniel Fourmy; Sandrine Silvente-Poirot
Identification of tyrosine 189 and asparagine 358 of the cholecystokinin 2 receptor in direct interaction with the crucial C-terminal amide of cholecystokinin by molecular modeling, site-directed mutagenesis, and structure/affinity studies.
Molecular pharmacology 2003;63(5):973-82.
2003: Vincent Guerlavais; Damien Boeglin; Delphine Mousseaux; Catherine Oiry; Annie Heitz; Romano Deghenghi; Vittorio Locatelli; Antonio Torsello; Corrado Ghé; Filomena Catapano; Giampiero Muccioli; Jean-Claude Galleyrand; Jean-Alain Fehrentz; Jean Martinez
New active series of growth hormone secretagogues.
Journal of medicinal chemistry 2003;46(7):1191-203.
2003: Christine Enjalbal; Delphine Maux; Robert Combarieu; Jean Martinez; Jean-Louis Aubagnac
Imaging combinatorial libraries by mass spectrometry: from peptide to organic-supported syntheses.
Journal of combinatorial chemistry 2003;5(2):102-9.
2003: Christine Enjalbal; Frédéric Lamaty; Pierre Sanchez; E Suberchicot; Patrice Ribière; S Varray; R Lazaro; Neerja Yadav-Bhatnagar; Jean Martinez; J L Aubagna
Characterization of soluble polymer supported organic compounds by LC/electrospray ionization MS toward a complete automation of the liquid-phase process in combinatorial chemistry.
Analytical chemistry 2003;75(2):175-84.
2003: Rosa M Claramunt; Dionisia Sanz; Marta Pérez Torralba; José Elguero; Pierre Sanchez; Christine Enjalbal; Jean Martinez; Jean-Louis Aubagnac
Electrospray mass spectrometry of 2-aminotroponimines and 2-aminotropones.
European journal of mass spectrometry (Chichester, England) 2003;9(4):403-7.
2002: Daniel Fourmy; Chantal Escrieut; Elodie Archer; Céline Galès; Véronique Gigoux; Bernard Maigret; Luis Moroder; Sandrine Silvente-Poirot; Jean Martinez; Jean-Alain Fehrentz; Lucien Pradayrol
Structure of cholecystokinin receptor binding sites and mechanism of activation/inactivation by agonists/antagonists.
Pharmacology & toxicology 2002;91(6):313-20.
2002: Céline Douat; Annie Heitz; Marielle Paris; Jean Martinez; Jean-Alain Fehrentz
Post-synthesis incorporation of a lipidic side chain into a peptide on solid support.
Journal of peptide science : an official publication of the European Peptide Society 2002;8(11):601-14.
2002: V Lejeune; Florine Cavelier; Christine Enjalbal; Jean Martinez; Jean-Louis Aubagnac
ESI mass spectrometry of amino acid trimethylsilylethyl esters.
Journal of mass spectrometry : JMS 2002;37(11):1168-70.
2002: Fabio Broglio; François Boutignon; Andrea Benso; Cristina Gottero; Flavia Prodam; Emanuela Arvat; Corrado Ghè; Filomena Catapano; Antonio Torsello; Vittorio Locatelli; Giampiero Muccioli; Damien Boeglin; Vincent Guerlavais; Jean-Alain Fehrentz; Jean Martinez; Ezio Ghigo; Romano Deghenghi
EP1572: a novel peptido-mimetic GH secretagogue with potent and selective GH-releasing activity in man.
Journal of endocrinological investigation 2002;25(8):RC26-8.
2002: Jean-Alain Fehrentz; Jean Martinez; Damien Boeglin; Vincent Guerlavais; Romano Deghenghi
Growth hormone secretagogues: past, present and future.
IDrugs : the investigational drugs journal 2002;5(8):804-14.
2002: Julie Pannequin; Catherine Oiry; Caroline Morel; Jérôme Kucharczak; Isabelle Camby; Robert Kiss; Didier Gagne; Jean-Claude Galleyrand; Jean Martinez
C-terminal heptapeptide of gastrin inhibits astrocytomas motility by interacting with a new gastrin binding site.
The Journal of pharmacology and experimental therapeutics 2002;302(1):274-82.
2002: Florine Cavelier; Bertrand Vivet; Jean Martinez; André Aubry; Claude Didierjean; André Vicherat; Michel Marraud
Influence of silaproline on peptide conformation and bioactivity.
Journal of the American Chemical Society 2002;124(12):2917-23.
2002: Jean-Louis Aubagnac; Robert Combarieu; Christine Enjalbal; Jean Martinez
Quality control of solid-phase synthesis by mass spectrometry.
Methods in molecular biology (Clifton, N.J.) 2002;201():15-22.
2002: Delphine Maux; Christine Enjalbal; Jean Martinez; Jean-Louis Aubagnac
New example of proline-induced fragmentation in electrospray ionization mass spectrometry of peptides.
Rapid communications in mass spectrometry : RCM 2002;16(15):1470-5.
2001: Marc Rolland; Tarek Kassem; Valérie Rolland; Jean Martinez
Full stereochemical understanding in a new (2R,3R,4R)-4-hydroxyisoleucine synthesis.
Acta crystallographica. Section C, Crystal structure communications 2001;57(Pt 12):1415-7.
2001: Françoise Richard; Séverine Barroso; Jean Martinez; CATHERINE LABBE-JULLIE; Patrick Kitabgi
Agonism, inverse agonism, and neutral antagonism at the constitutively active human neurotensin receptor 2.
Molecular pharmacology 2001;60(6):1392-8.
2001: Jérôme Kucharczak; Julie Pannequin; Isabelle Camby; C Decaestecker; R Kiss; Jean Martinez
Gastrin induces over-expression of genes involved in human U373 glioblastoma cell migration.
Oncogene 2001;20(48):7021-8.
2001: M McKiernan; J Huck; Jean-Alain Fehrentz; Marie-Louise Roumestant; Ph Viallefont; Jean Martinez
Urethane N-carboxyanhydrides from beta-amino acids.
The Journal of organic chemistry 2001;66(20):6541-4.
2001: Delphine Maux; Christine Enjalbal; Jean Martinez; Jean-Louis Aubagnac; Robert Combarieu
Static secondary ion mass spectrometry to monitor solid-phase peptide synthesis.
Journal of the American Society for Mass Spectrometry 2001;12(10):1099-105.
2001: R Akkari; M Calmes; N Mai; M Rolland; Jean Martinez
Synthesis of a new insoluble polymer-supported chiral alcohol auxiliary and its first application to nucleophilic addition to ketenes.
The Journal of organic chemistry 2001;66(17):5859-65.
2001: Christine Enjalbal; Delphine Maux; Jean Martinez; Robert Combarieu; Jean-Louis Aubagnac
Mass spectrometry and combinatorial chemistry: new approaches for direct support-bound compound identification.
Combinatorial chemistry & high throughput screening 2001;4(4):363-73.
2001: Christine Farenc; Christine Enjalbal; Pierre Sanchez; Françoise Bressolle; Michel Audran; Jean Martinez; Jean-Louis Aubagnac
Quantitative determination of rocuronium in human plasma by liquid chromatography-electrospray ionization mass spectrometry.
Journal of chromatography. A 2001;910(1):61-7.
2001: S Bellahouel; Valérie Rolland; Marie-Louise Roumestant; Ph Viallefont; Jean Martinez
Chemoenzymatic synthesis of surfactants from carbohydrates, amino acids, and fatty acids.
Preparative biochemistry & biotechnology 2001;31(1):71-80.
2001: Marc Rolland; A Jenhi ; J P Lavergne ; Jean Martinez; A Hasnaoui
[Dimethyl 3-benzyl-2-(4-methyl-2,5-dioxoimidazolidin-1-yl)butanedioate].
Acta crystallographica. Section C, Crystal structure communications 2001;57(Pt 1):62-3.
2000: Amor Belmeguenai; Hubert Vaudry; Jérôme Leprince; Bertrand Vivet; Florine Cavelier; Jean Martinez; Estelle Louiset
Neurotensin modulates the electrical activity of frog pituitary melanotropes via activation of a G-protein-coupled receptor pharmacologically related to both the NTS1 and nts2 receptors of mammals.
Neuroendocrinology 2000;72(6):379-91.
2000: Bertrand Vivet; Florine Cavelier; Jean Martinez; Claude Didierjean; Michel Marraud; André Aubry
A silaproline-containing dipeptide.
Acta crystallographica. Section C, Crystal structure communications 2000;56(Pt 12):1452-4.
2000: R Poosti; L di Malta; Didier Gagne; N Bernad; Jean-Claude Galleyrand; Chantal Escrieut; Sandrine Silvente-Poirot; Daniel Fourmy; Jean Martinez
The third intracellular loop of the rat and mouse cholecystokinin-A receptors is responsible for different patterns of gene activation.
Molecular pharmacology 2000;58(6):1381-8.
2000: M E Haddadi; Florine Cavelier; E Vives; A Azmani; J Verducci; Jean Martinez
All-L-Leu-Pro-Leu-Pro: a challenging cyclization.
Journal of peptide science : an official publication of the European Peptide Society 2000;6(11):560-70.
2000: R El Khalabi; A el Hallaoui; F Ouazzani; A Elachqar; A Atmani; Marie-Louise Roumestant; Ph Viallefont; Jean Martinez
Synthesis of phosphonic analogues of 4-hydroxyproline and 5-hydroxypipecolic acid.
Preparative biochemistry & biotechnology 2000;30(4):295-304.
2000: C Boyat; V Rolland-Fulcrand; Ph Viallefont; Jean Martinez
Chemo-enzymatic synthesis of new non ionic surfactants from unprotected carbohydrates.
Preparative biochemistry & biotechnology 2000;30(4):281-94.
2000: Catherine Oiry; Julie Pannequin; N Bernad; A M Artis; Jean-Claude Galleyrand; C Devin; M Cristau; Jean-Alain Fehrentz; Jean Martinez
A synthetic glycine-extended bombesin analogue interacts with the GRP/bombesin receptor.
European journal of pharmacology 2000;403(1-2):17-25.
2000: Pascal Nicole; laurence lins; Christiane Rouyer-Fessard; C Drouot; Pierre Fulcrand; Annick Thomas; Alain Couvineau; Jean Martinez; R Brasseur; Marc Laburthe
Identification of key residues for interaction of vasoactive intestinal peptide with human VPAC1 and VPAC2 receptors and development of a highly selective VPAC1 receptor agonist. Alanine scanning and molecular modeling of the peptide.
The Journal of biological chemistry 2000;275(31):24003-12.
2000: Tarek Kassem; Valérie Rolland; Jean Martinez; Marc Rolland
Two key chiral intermediates in a new 4-hydroxyisoleucine synthesis.
Acta crystallographica. Section C, Crystal structure communications 2000;56 ( Pt 8)():1037-9.
2000: P Bedos; Muriel Amblard; Gilles Subra; PR Dodey; Jean-Michel Luccarini; Jean-Luc Paquet; Didier Pruneau; A Aumelas; Jean Martinez
A rational approach to the design and synthesis of a new bradykinin B(1) receptor antagonist.
Journal of medicinal chemistry 2000;43(12):2387-94.
2000: Muriel Amblard; P Bedos; C Olivier; I Daffix; Jean-Michel Luccarini; PR Dodey; Didier Pruneau; Jean-Luc Paquet; Jean Martinez
Synthesis and biological evaluation of bradykinin B(1)/B(2) and selective B(1) receptor antagonists.
Journal of medicinal chemistry 2000;43(12):2382-6.
2000: M Cristau; C Devin; Catherine Oiry; O Chaloin; Muriel Amblard; N Bernad; Annie Heitz; Jean-Alain Fehrentz; Jean Martinez
Synthesis and biological evaluation of bombesin constrained analogues.
Journal of medicinal chemistry 2000;43(12):2356-61.
2000: Christine Enjalbal; Jean Martinez; Jean-Louis Aubagnac
Mass spectrometry in combinatorial chemistry.
Mass spectrometry reviews 2000;19(3):139-61.
2000: Marc Rolland; M Calmès; F Escale; Jean Martinez
[New derivatives of pantolactonyl N-phthalimido-2-arylpropanoate].
Acta crystallographica. Section C, Crystal structure communications 2000;56 ( Pt 4)():445-7.
2000: L Lecointe; Valérie Rolland; L Pappalardo; Marie-Louise Roumestant; Ph Viallefont; Jean Martinez
Diastereoselective synthesis of non-proteinogenic alpha-amino acids.
The journal of peptide research : official journal of the American Peptide Society 2000;55(4):300-7.
2000: B Sauvagnat; K Kulig; Frédéric Lamaty; R Lazaro; Jean Martinez
Soluble polymer supported synthesis of alpha-amino acid derivatives.
Journal of combinatorial chemistry 2000;2(2):134-42.
2000: Pascal Nicole; Christiane Rouyer-Fessard; Alain Couvineau; C Drouot; Pierre Fulcrand; Jean Martinez; Marc Laburthe
Alanine scanning of VIP. Structure-function relationship for binding to human recombinant VPAC1 receptor.
Annals of the New York Academy of Sciences 2000;921():352-6.
1999: Véronique Gigoux; Bernard Maigret; Chantal Escrieut; Sandrine Silvente-Poirot; Michèle Bouisson; Jean-Alain Fehrentz; Luis Moroder; D Gully; Jean Martinez; Nicole Vaysse; A D Fourmy
Arginine 197 of the cholecystokinin-A receptor binding site interacts with the sulfate of the peptide agonist cholecystokinin.
Protein science : a publication of the Protein Society 1999;8(11):2347-54.
1999: Muriel Amblard; I Daffix; Gilbert Bergé; M Calmès; PR Dodey; Didier Pruneau; Jean-Luc Paquet; Jean-Michel Luccarini; P Bélichard; Jean Martinez
Synthesis and characterization of bradykinin B(2) receptor agonists containing constrained dipeptide mimics.
Journal of medicinal chemistry 1999;42(20):4193-201.
1999: Muriel Amblard; I Daffix; P Bedos; Gilbert Bergé; Didier Pruneau; Jean-Luc Paquet; Jean-Michel Luccarini; P Bélichard; PR Dodey; Jean Martinez
Design and synthesis of potent bradykinin agonists containing a benzothiazepine moiety.
Journal of medicinal chemistry 1999;42(20):4185-92.
1999: M Giraud; Florine Cavelier; Jean Martinez
A side-reaction in the SPPS of Trp-containing peptides.
Journal of peptide science : an official publication of the European Peptide Society 1999;5(10):457-61.
1999: Jean-Louis Aubagnac; Muriel Amblard; Christine Enjalbal; Gilles Subra; Jean Martinez; P Durand; P Renaut
Identification of synthetic by-products in combinatorial libraries using high performance liquid chromatography-electrospray ionization mass spectrometry.
Combinatorial chemistry & high throughput screening 1999;2(5):289-96.
1999: Sandrine Silvente-Poirot; Chantal Escrieut; C Galès; Jean-Alain Fehrentz; Achim Escherich; Stephen A Wank; Jean Martinez; Luis Moroder; Bernard Maigret; Michèle Bouisson; Nicole Vaysse; Daniel Fourmy
Evidence for a direct interaction between the penultimate aspartic acid of cholecystokinin and histidine 207, located in the second extracellular loop of the cholecystokinin B receptor.
The Journal of biological chemistry 1999;274(33):23191-7.
1999: Véronique Gigoux; Chantal Escrieut; Jean-Alain Fehrentz; S Poirot; Bernard Maigret; Luis Moroder; D Gully; Jean Martinez; Nicole Vaysse; Daniel Fourmy
Arginine 336 and asparagine 333 of the human cholecystokinin-A receptor binding site interact with the penultimate aspartic acid and the C-terminal amide of cholecystokinin.
The Journal of biological chemistry 1999;274(29):20457-64.
1999: Jean-Louis Aubagnac; Christine Enjalbal; C Drouot; Robert Combarieu; Jean Martinez
Imaging time-of-flight secondary ion mass spectrometry of solid-phase peptide syntheses.
Journal of mass spectrometry : JMS 1999;34(7):749-54.
1999: Catherine Oiry; Julie Pannequin; A Cormier; Jean-Claude Galleyrand; Jean Martinez
L-365,260 inhibits in vitro acid secretion by interacting with a PKA pathway.
British journal of pharmacology 1999;127(1):259-67.
1999: C Devin; N Bernad; M Cristau; A M Artis-Noel; Annie Heitz; Jean-Alain Fehrentz; Jean Martinez
Synthesis and biological evaluation of C-terminal hydroxamide analogues of bombesin.
Journal of peptide science : an official publication of the European Peptide Society 1999;5(4):176-84.
1999: M Llinares; C Devin; O Chaloin; J Azay; A M Noel-Artis; N Bernad; Jean-Alain Fehrentz; Jean Martinez
Syntheses and biological activities of potent bombesin receptor antagonists.
The journal of peptide research : official journal of the American Peptide Society 1999;53(3):275-83.
1999: S Bouifraden; C Drouot; M el Hadrami; F Guenoun; L Lecointe; N Mai; M Paris; C Pothion; M Sadoune; B Sauvagnat; Muriel Amblard; Jean-Louis Aubagnac; M Calmes; Pierre Chevallet; J Daunis; Christine Enjalbal; Jean-Alain Fehrentz; Frédéric Lamaty; J P Lavergne; R Lazaro; Valérie Rolland; Marie-Louise Roumestant; Ph Viallefont; Y Vidal; Jean Martinez
Some of the amino acid chemistry going on in the Laboratory of Amino Acids, Peptides and Proteins.
Amino acids 1999;16(3-4):345-79.
1999: Isabelle Dubuc; Philippe Sarret; CATHERINE LABBE-JULLIE; Jean-Marie Botto; E Honoré; E Bourdel; Jean Martinez; Jean Costentin; Jean-Pierre Vincent; Patrick Kitabgi; Jean Mazella
Identification of the receptor subtype involved in the analgesic effect of neurotensin.
The Journal of neuroscience : the official journal of the Society for Neuroscience 1999;19(1):503-10.
1998: I Daffix; Muriel Amblard; Gilbert Bergé; PR Dodey; Didier Pruneau; Jean-Luc Paquet; C Fouchet; Rose-Marie Franck; E Defrêne; Jean-Michel Luccarini; P Bélichard; Jean Martinez
Synthesis and pharmacological evaluation of dimer derivatives of the bradykinin receptor antagonist HOE-140.
The journal of peptide research : official journal of the American Peptide Society 1998;52(1):1-14.
1998: Philippe Marambaud; N Chevallier; E Lopez-Perez; C Drouot; J Vizzanova; Pierre Fulcrand; Jean Martinez; Sherwin Wilk; Frédéric Checler
[Strategies for identification of secretases implicated in Alzheimer's disease].
Annales de biologie clinique 1998;56(3):277-84.
1998: J M Receveur; Janique Guiramand; Max Récasens; Marie-Louise Roumestant; Ph Viallefont; Jean Martinez
Synthesis and biological activity of glutamic acid derivatives.
Bioorganic & medicinal chemistry letters 1998;8(2):127-32.
1998: Eric Condamine; G Chapdeleine; L Demarcy; J F Duclos; Daniel Davoust; M Llinares; J Azay; Jean Martinez; S Chapelle
Biological activity and three-dimensional structure of an agonist analog of bombesin.
The journal of peptide research : official journal of the American Peptide Society 1998;51(1):55-64.
1998: J Azay; claire domaine; M Llinares; C Devin; Jean-Alain Fehrentz; N Bernad; C Roze; Jean Martinez
Comparative study of in vitro and in vivo activities of bombesin pseudopeptide analogs modified on the C-terminal dipeptide fragment.
Peptides 1998;19(1):57-63.
1997: J L Burgaud; R Poosti; jean-alain fehrentz; Jean Martinez; Jean-Louis Nahon
Melanin-concentrating hormone binding sites in human SVK14 keratinocytes.
Biochemical and biophysical research communications 1997;241(3):622-9.
1997: PASCAL FRAGNER; Olivier Presset; N Bernad; Jean Martinez; C Roze; S Aratan-Spire
A new biological contribution of cyclo(His-Pro) to the peripheral inhibition of pancreatic secretion.
The American journal of physiology 1997;273(6 Pt 1):E1127-32.
1997: H Barelli; A Lebeau; Jean Vizzavona; P Delaere; N Chevallier; C Drouot; Philippe Marambaud; Karine Ancolio; Joseph Buxbaum; OE Khorkova; J Heroux; Sudhir Sahasrabudhe; Jean Martinez; J M Warter; M Mohr; Frédéric Checler
Characterization of new polyclonal antibodies specific for 40 and 42 amino acid-long amyloid beta peptides: their use to examine the cell biology of presenilins and the immunohistochemistry of sporadic Alzheimer's disease and cerebral amyloid angiopathy cases.
Molecular medicine (Cambridge, Mass.) 1997;3(10):695-707.
1997: Catherine Oiry; Didier Gagne; E Cottin; N Bernad; Jean-Claude Galleyrand; Gilbert Bergé; M F Lignon; patrick eldin; Martine Le Cunff; J Léger; Pascal Clerc; Daniel Fourmy; Jean Martinez
CholecystokininB receptor from human Jurkat lymphoblastic T cells is involved in activator protein-1-responsive gene activation.
Molecular pharmacology 1997;52(2):292-9.
1997: N Chevallier; Jean Vizzavona; Philippe Marambaud; C P Baur; Maria Grazia Spillantini; Pierre Fulcrand; Jean Martinez; Michel Goedert; J P Vincent; Frédéric Checler
Cathepsin D displays in vitro beta-secretase-like specificity.
Brain research 1997;750(1-2):11-9.
1997: K Kennedy; Véronique Gigoux; Chantal Escrieut; Bernard Maigret; Jean Martinez; Luis Moroder; D Fréhel; D Gully; Nicole Vaysse; Daniel Fourmy
Identification of two amino acids of the human cholecystokinin-A receptor that interact with the N-terminal moiety of cholecystokinin.
The Journal of biological chemistry 1997;272(5):2920-6.
1997: Philippe Marambaud; F Rieunier; Sherwin Wilk; Jean Martinez; Frédéric Checler
Contribution of the proteasome to the alpha-secretase pathway in Alzheimer's disease.
Advances in experimental medicine and biology 1997;421():267-72.
1996: A C Lima-Leite; P Fulcrand; Jean-Claude Galleyrand; G Berge; A Aumelas; Jean-Pierre Bali; J Castel; Jean Martinez
Synthesis and biological activities of some human gastrin analogs.
Brazilian journal of medical and biological research = Revista brasileira de pesquisas médicas e biológicas / Sociedade Brasileira de Biofísica ... [et al.] 1996;29(10):1253-63.
1996: Isabelle Camby; Isabelle Salmon; Catherine Oiry; Jean-Claude Galleyrand; Nathalie Nagy; André Danguy; Jacques Brotchi; Jean-Lambert Pasteels; Jean Martinez; Robert Kiss
The influence of gastrin and/or cholecystokinin antagonists on the proliferation of three human astrocytic tumor cell lines.
Neuropeptides 1996;30(5):433-7.
1996: J Azay; D Gagne; C Devin; M Llinares; Jean-Alain Fehrentz; Jean Martinez
JMV641: a potent bombesin receptor antagonist that inhibits Swiss 3T3 cell proliferation.
Regulatory peptides 1996;65(1):91-7.
1996: Isabelle Camby; Isabelle Salmon; E Bourdel; Nathalie Nagy; André Danguy; Jacques Brotchi; Jean-Lambert Pasteels; Jean Martinez; Robert Kiss
Neurotensin-mediated effects on astrocytic tumor cell proliferation.
Neuropeptides 1996;30(2):133-9.
1996: C Carles-Bonnet; Jean Martinez; Claire Jarrousse; A Aumelas; H Niel; Dominique Bataille
H-Lys-Arg-Asn-Lys-Asn-Asn-OH is the minimal active structure of oxyntomodulin.
Peptides 1996;17(3):557-61.
1995: Catherine Oiry; Jean-Claude Galleyrand; A C Lima-Leite; P Fulcrand; Jean Martinez
Are C-terminal octapeptide of cholecystokinin and [Leu11]gastrin-(5-17) different in stimulating acid secretion in isolated rabbit gastric glands?
European journal of pharmacology 1995;294(2-3):511-9.
1995: J C Lallement; Catherine Oiry; A C Lima-Leite; M F Lignon; P Fulcrand; Jean-Claude Galleyrand; Jean Martinez
Cholecystokinin and gastrin are not equally sensitive to GTP gamma S at CCKB receptors: importance of the sulphated tyrosine.
European journal of pharmacology 1995;290(2):61-7.
1995: jean-alain fehrentz; C Genu-Dellac; Muriel Amblard; F Winternitz; A Loffet; Jean Martinez
The use of N-urethane-protected N-carboxyanhydrides (UNCAs) in amino acid and peptide synthesis.
Journal of peptide science : an official publication of the European Peptide Society 1995;1(2):124-31.
1994: Jean-Claude Galleyrand; A C Lima-Leite; J C Lallement; M F Lignon; N Bernad; P Fulcrand; Jean Martinez
Synthesis and characterization of a new labeled gastrin ligand, 125-I-BH-[Leu15]-gastrin-(5-17), on binding to canine fundic mucosal cells and Jurkat cells.
International journal of peptide and protein research 1994;44(4):348-56.
1994: J C Lallement; Jean-Claude Galleyrand; A C Lima-Leite; P Fulcrand; Jean Martinez
Gastrin13 and the C-terminal octapeptide of cholecystokinin are differently coupled to G-proteins in guinea-pig brain membranes.
European journal of pharmacology 1994;267(3):297-305.
1994: S S Poirot; Chantal Escrieut; Marlène Dufresne; Jean Martinez; Michèle Bouisson; Nicole Vaysse; Daniel Fourmy
Photoaffinity labeling of rat pancreatic cholecystokinin type A receptor antagonist binding sites demonstrates the presence of a truncated cholecystokinin type A receptor.
Molecular pharmacology 1994;45(4):599-607.
1994: J C Lallement; Jean-Claude Galleyrand; A C Lima-Leite; P Fulcrand; Jean Martinez
Gastrin13 binds to CCKB brain membrane receptors coupled to G protein in guinea pig brain membranes.
Annals of the New York Academy of Sciences 1994;713():346-9.
1994: M F Lignon; N Bernad; Jean Martinez
Cholecystokinin receptors in cells of the immune system.
Annals of the New York Academy of Sciences 1994;713():334-7.
1994: M Amblard; M F Lignon; N Bernad; A M Noel-Artis; L Hauad; J Laur; M Rodriguez; M C Galas; Daniel Fourmy; Jean Martinez
Biological evaluation of JMV180 cholecystokinin analogs.
Annals of the New York Academy of Sciences 1994;713():79-87.
1993: M F Lignon; N Bernad; Jean Martinez
Cholecystokinin increases intracellular Ca2+ concentration in the Human JURKAT T Lymphocyte cell line.
European journal of pharmacology 1993;245(3):241-6.
1993: Claire Jarrousse; C Carles-Bonnet; H Niel; R Sabatier; M P Audousset-Puech; philippe blache; A Kervran; Jean Martinez; Dominique Bataille
Inhibition of gastric acid secretion by oxyntomodulin and its 19-37 fragment in the conscious rat.
The American journal of physiology 1993;264(5 Pt 1):G816-23.
1993: Sandrine Silvente-Poirot; C Hadjiivanova; Chantal Escrieut; Marlène Dufresne; Jean Martinez; Nicole Vaysse; Daniel Fourmy
Study of the states and populations of the rat pancreatic cholecystokinin receptor using the full peptide antagonist JMV 179.
European journal of biochemistry / FEBS 1993;212(2):529-38.
1992: Lenka Maletínská; M F Lignon; M C Galas; N Bernad; J Pírková; Jan Hlavácek; Jirina Slaninová; Jean Martinez
Pharmacological characterization of new cholecystokinin analogues.
European journal of pharmacology 1992;222(2-3):233-40.
1992: M C Galas; N Bernad; Jean Martinez
Pharmacological studies on CCKB receptors in guinea pig synaptoneurosomes.
European journal of pharmacology 1992;226(1):35-41.
1992: Jean-Claude Galleyrand; P Fulcrand; Jean-Pierre Bali; M Rodriguez; Richard Magous; J Laur; Jean Martinez
Biological effects of human gastrin I and II chemically modified at the C-terminal tetrapeptide amide.
Peptides 1992;13(3):519-25.
1992: M Rodriguez; A Heitz; Jean Martinez
"Carba" peptide bond surrogates. Different approaches to Gly-psi(CH2-CH2)-D,L-Xaa pseudo-dipeptide units.
International journal of peptide and protein research 1992;39(3):273-7.
1992: C Carles-Bonnet; Claire Jarrousse; H Niel; Jean Martinez; M Rolland; Dominique Bataille
N-acetyl oxyntomodulin30-37: pharmacokinetics and activity on gastric acid secretion.
Naunyn-Schmiedeberg's archives of pharmacology 1992;345(1):57-63.
1991: T Tani; A Le Quellec; Claire Jarrousse; F Sladeczek; Jean Martinez; Agnes Estival; Lucien Pradayrol; Dominique Bataille
Oxyntomodulin and related peptides control somatostatin secretion in RIN T3 cells.
Biochimica et biophysica acta 1991;1095(3):249-54.
1991: C Carles-Bonnet; Claire Jarrousse; H Niel; Jean Martinez; Dominique Bataille
Oxyntomodulin and its (19-37) and (30-37) fragments inhibit histamine-stimulated gastric acid secretion in the conscious rat.
European journal of pharmacology 1991;203(2):245-52.
1991: M Rolland; M Rodriguez; M F Lignon; M C Galas; J Laur; A Aumelas; Jean Martinez
Synthesis and biological activity of 2-phenylethyl ester analogues of C-terminal heptapeptide of cholecystokinin modified in Trp 30 region.
International journal of peptide and protein research 1991;38(2):181-92.
1991: M F Lignon; N Bernad; Jean Martinez
Pharmacological characterization of type B cholecystokinin binding sites on the human JURKAT T lymphocyte cell line.
Molecular pharmacology 1991;39(5):615-20.
1991: Jean Martinez; M Rodriguez; M F Lignon; M C Galas; M Amblard; M Rolland; C Mendre; P Fulcrand; J Laur; N Bernad
[Structure-activity relationship of cystokinins: analogs exhibiting selective activity].
Journal de pharmacie de Belgique 1991;46(1):9-16.
1990: A Kervran; M Dubrasquet; philippe blache; Jean Martinez; Dominique Bataille
Metabolic clearance rates of oxyntomodulin and glucagon in the rat: contribution of the kidney.
Regulatory peptides 1990;31(1):41-52.
1990: C Mendre; M Rodriguez; M F Lignon; M C Galas; C Gueudet; P Worms; Jean Martinez
Pharmacological activity of cholecystokinin analogues modified in the Met28-Gly29 region.
European journal of pharmacology 1990;186(2-3):213-22.
1990: M Rodriguez; M F Lignon; M C Galas; M Amblard; Jean Martinez
Cyclic cholecystokinin analogues that are highly selective for rat and guinea pig central cholecystokinin receptors.
Molecular pharmacology 1990;38(3):333-41.
1990: P Dubreuil; P Fulcrand; M Rodriguez; J Laur; Jean-Pierre Bali; Jean Martinez
ACE-like hydrolysis of gastrin analogs and CCK-8 by fundic mucosal cells of different species with release of the amidated C-terminal dipeptide.
Biochimica et biophysica acta 1990;1039(2):171-6.
1990: M Rodriguez; M Amblard; M C Galas; M F Lignon; A Aumelas; Jean Martinez
Synthesis of cyclic analogues of cholecystokinin highly selective for central receptors.
International journal of peptide and protein research 1990;35(5):441-51.
1990: M F Lignon; M C Galas; M Rodriguez; Jean Martinez
Correlation between phospholipid breakdown, intracellular calcium mobilization and enzyme secretion in rat pancreatic acini treated with Boc-[Nle28, Nle31]-CCK-7 and JMV180, two cholecystokinin analogues.
Cellular signalling 1990;2(4):339-46.
1989: M Rodriguez; M Rolland; M F Lignon; M C Galas; J Laur; A Aumelas; Jean Martinez
Synthesis and biological activities of some cholecystokinin analogues substituted in position 29 by a beta-alanine.
International journal of peptide and protein research 1989;34(5):394-404.
1989: A Aumelas; M P Audousset-Puech; Annie Heitz; Dominique Bataille; Jean Martinez
1H n.m.r. conformational studies on the C-terminal octapeptide of oxyntomodulin, a beta-turn locked by a salt bridge.
International journal of peptide and protein research 1989;34(4):268-76.
1989: M Rodriguez; M C Galas; M F Lignon; C Mendre; J Laur; A Aumelas; Jean Martinez
Synthesis and biological activity of some partially modified retro-inverso analogues of cholecystokinin.
Journal of medicinal chemistry 1989;32(10):2331-9.
1989: P Dubreuil; P Fulcrand; M Rodriguez; H Fulcrand; J Laur; Jean Martinez
Novel activity of angiotensin-converting enzyme. Hydrolysis of cholecystokinin and gastrin analogues with release of the amidated C-terminal dipeptide.
The Biochemical journal 1989;262(1):125-30.
1989: M Rodriguez; P Fulcrand; J Laur; A Aumelas; Jean-Pierre Bali; Jean Martinez
Synthesis of gastrin antagonists, analogues of the C-terminal tetrapeptide of gastrin, by introduction of a beta-homo residue.
Journal of medicinal chemistry 1989;32(3):522-8.
1988: P Fulcrand; M Rodriguez; M C Galas; M F Lignon; J Laur; A Aumelas; Jean Martinez
2-Phenylethyl ester and 2-phenylethyl amide derivative analogues of the C-terminal hepta- and octapeptide of cholecystokinin.
International journal of peptide and protein research 1988;32(5):384-95.
1988: philippe blache; A Kervran; Jean Martinez; Dominique Bataille
Development of an oxyntomodulin/glicentin C-terminal radioimmunoassay using a "thiol-maleoyl" coupling method for preparing the immunogen.
Analytical biochemistry 1988;173(1):151-9.
1988: C Mendre; M Rodriquez; C Gueudet; M F Lignon; M C Galas; J Laur; P Worms; Jean Martinez
A pseudopeptide that is a potent cholecystokinin agonist in the peripheral system is able to inhibit the dopamine-like effects of cholecystokinin in the striatum.
The Journal of biological chemistry 1988;263(22):10641-5.
1988: M C Galas; M F Lignon; M Rodriguez; C Mendre; P Fulcrand; J Laur; Jean Martinez
Structure-activity relationship studies on cholecystokinin: analogues with partial agonist activity.
The American journal of physiology 1988;254(2 Pt 1):G176-82.
1987: A Aumelas; M Rodriguez; Annie Heitz; B Castro; Jean Martinez
1H and 13C n.m.r. studies of pseudo-peptide analogues of the C-terminal tetrapeptide of gastrin.
International journal of peptide and protein research 1987;30(5):596-604.
1987: P Dubreuil; M F Lignon; Richard Magous; M Rodriguez; Jean-Pierre Bali; Jean Martinez
Degradation of a tetragastrin analogue by a membrane fraction from rat gastric mucosa.
Drug design and delivery 1987;2(1):49-54.
1987: M Rodriguez; M F Lignon; M C Galas; P Fulcrand; C Mendre; A Aumelas; J Laur; Jean Martinez
Synthesis and biological activities of pseudopeptide analogues of the C-terminal heptapeptide of cholecystokinin. On the importance of the peptide bonds.
Journal of medicinal chemistry 1987;30(8):1366-73.
1986: M P Audousset-Puech; M Dufour; A Kervran; Claire Jarrousse; B Castro; Dominique Bataille; Jean Martinez
Solid-phase peptide synthesis of human(Nle-27)-oxyntomodulin. Preliminary evaluation of its biological activities.
FEBS letters 1986;200(1):181-5.
1986: Claire Jarrousse; H Niel; M P Audousset-Puech; Jean Martinez; Dominique Bataille
Oxyntomodulin and its C-terminal octapeptide inhibit liquid meal-stimulated acid secretion.
Peptides 1986;7 Suppl 1():253-6.
1986: J M Dubrasquet; M P Audousset-Puech; Jean Martinez; Dominique Bataille
Somatostatin enhances the inhibitory effect of oxyntomodulin and its C-terminal octapeptide on acid secretion.
Peptides 1986;7 Suppl 1():257-9.
1985: M P Audousset-Puech; Claire Jarrousse; M Dubrasquet; A Aumelas; B Castro; Dominique Bataille; Jean Martinez
Synthesis of the C-terminal octapeptide of pig oxyntomodulin. Lys-Arg-Asn-Lys-Asn-Asn-Ile-Ala: a potent inhibitor of pentagastrin-induced acid secretion.
Journal of medicinal chemistry 1985;28(10):1529-33.
1985: Claire Jarrousse; M P Audousset-Puech; M Dubrasquet; H Niel; Jean Martinez; Dominique Bataille
Oxyntomodulin (glucagon-37) and its C-terminal octapeptide inhibit gastric acid secretion.
FEBS letters 1985;188(1):81-4.