Preview
Sign-in for full Details 
Sign-in free and Explore the Exciting World of BiomedExperts:
- Over 1.500.000 Profiles
- More than 1.800 Organizations worldwide
- State of the Art Network Visualizations
- Manage your own Profile
- Locate Experts in your Country/Region
- Locate Experts in your 1. and 2. Level Network
- Connect to Experts Worldwide
NetworkView
Gabriella Marucci
This is a preview profile on BiomedExperts - the first literature-based scientific social network. It brings the right researchers
together and allows them to collaborate online. Collexis and Dell provide the BiomedExperts network of +1.5 Million pre-calculated profiles
free of charge to researchers worldwide.
Research Profile (preview)
Concepts & Ideas
Anatomy
Living Beings
Chemicals & Drugs
Phenomena
Procedures
Sign-in to see full Profile
Network (preview)
33
Angeli, Piero
23
Melchiorre, Carlo
21
Buccioni, Michela
13
Brasili, Livio
13
Quaglia, Wilma
12
Giardinà, Dario
11
Pigini, Maria
11
Tumiatti, Vincenzo
10
Rosini, Michela
9
Scapecchi, Serena
9
Romanelli, Maria Novella
9
Minarini, Anna
9
Leonardi, Amedeo
8
Matucci, Rosanna
8
Piergentili, Alessandro
Sign-in to see all Coauthors
Publications
Sign-in to see all Publications
Sign in free and see...
Visualized networks:
See your personal network in
sophisticated graphical views
GeoTargeted Searches:
Locate experts around the world
and connect with global collaborators
Research Profiles:
See the visualized research activity
of experts around the globe
Sign-in to see more
Geonetwork of Gabriella Marucci (preview)
Cities where this author has publications
Cities where co-authors of this author have publications
Sign-in to see more
All Publications
-
2009: Volpini Rosaria; Mishra Ram Chandra; Kachare Dhuldeo D; Dal Ben Diego; Lambertucci Catia; Antonini Ippolito; Vittori Sauro; Marucci Gabriella; Sokolova Elena; Nistri Andrea; Cristalli Gloria
Adenine-based acyclic nucleotides as novel P2X3 receptor ligands.
Journal of medicinal chemistry 2009;52(15):4596-603.
-
2009: Volpini Rosaria; Dal Ben Diego; Lambertucci Catia; Marucci Gabriella; Mishra Ram Chandra; Ramadori Anna Teresa; Klotz Karl-Norbert; Trincavelli Maria Letizia; Martini Claudia; Cristalli Gloria
Adenosine A2A receptor antagonists: new 8-substituted 9-ethyladenines as tools for in vivo rat models of Parkinson's disease.
ChemMedChem 2009;4(6):1010-9.
-
2009: Sorbi Claudia; Franchini Silvia; Tait Annalisa; Prandi Adolfo; Gallesi Rossella; Angeli Piero; Marucci Gabriella; Pirona Lorenza; Poggesi Elena; Brasili Livio
1,3-Dioxolane-based ligands as rigid analogues of naftopidil: structure-affinity/activity relationships at alpha1 and 5-HT1A receptors.
ChemMedChem 2009;4(3):393-9.
-
2009: Franchini Silvia; Tait Annalisa; Prandi Adolfo; Sorbi Claudia; Gallesi Rossella; Buccioni Michela; Marucci Gabriella; De Stefani Carla; Cilia Antonio; Brasili Livio
(2,2-Diphenyl-[1,3]oxathiolan-5-ylmethyl)-(3-phenyl-propyl)-amine: a potent and selective 5-HT(1A) receptor agonist.
ChemMedChem 2009;4(2):196-203.
-
2009: Buccioni Michela; Kandhavelu Meenakshisundaram; Angeli Piero; Cristalli Gloria; Dal Ben Diego; Giardinà Dario; Lambertucci Catia; Lammi Carmen; Volpini Rosaria; Marucci Gabriella
Identification of alpha1-adrenoceptor subtypes involved in contraction of young CD rat epididymal vas deferens.
European journal of pharmacology 2009;602(2-3):388-94.
-
2008: Marucci Gabriella; Finaurini Sara; Buccioni Michela; Lammi Carmen; Kandhavelu Meenakshisundaram; Volpini Rosaria; Ricciutelli Massimo; Angeli Piero; Commandeur Jan N M; Cristalli Gloria
In vitro metabolism studies of new adenosine A 2A receptor antagonists.
Drug metabolism letters 2008;2(4):301-7.
-
2008: Minarini Anna; Marucci Gabriella; Bellucci Cristina; Giorgi Gianluca; Tumiatti Vincenzo; Bolognesi Maria Laura; Matera Riccardo; Rosini Michela; Melchiorre Carlo
Design, synthesis, and biological evaluation of pirenzepine analogs bearing a 1,2-cyclohexanediamine and perhydroquinoxaline units in exchange for the piperazine ring as antimuscarinics.
Bioorganic & medicinal chemistry 2008;16(15):7311-20.
-
2008: Scapecchi Serena; Nesi Marta; Matucci Rosanna; Bellucci Cristina; Buccioni Michela; Dei Silvia; Guandalini Luca; Manetti Dina; Martini Elisabetta; Marucci Gabriella; Romanelli Maria Novella; Teodori Elisabetta; Cirilli Roberto
Synthesis and pharmacological characterization of chiral pyrrolidinylfuran derivatives: the discovery of new functionally selective muscarinic agonists.
Journal of medicinal chemistry 2008;51(13):3905-12.
-
2008: Dei Silvia; Bellucci Cristina; Buccioni Michela; Ferraroni Marta; Guandalini Luca; Manetti Dina; Marucci Gabriella; Matucci Rosanna; Nesi Marta; Romanelli Maria Novella; Scapecchi Serena; Teodori Elisabetta
Muscarinic antagonists with multiple stereocenters: Synthesis, affinity profile and functional activity of isomeric 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine sulfoxide derivatives.
Bioorganic & medicinal chemistry 2008;16(10):5490-500.
-
2008: Varoli Lucilla; Angeli Piero; Buccioni Michela; Burnelli Silvia; Fazio Nicola; Marucci Gabriella; Recanatini Maurizio; Spampinato Santi
Synthesis and pharmacological profile of a series of 1-substituted-2-carbonyl derivatives of Diphenidol: novel M4 muscarinic receptor antagonists.
Medicinal chemistry (Shariqah (United Arab Emirates)) 2008;4(2):121-8.
-
2007: Dei Silvia; Bellucci Cristina; Buccioni Michela; Ferraroni Marta; Guandalini Luca; Manetti Dina; Martini Elisabetta; Marucci Gabriella; Matucci Rosanna; Nesi Marta; Romanelli Maria Novella; Scapecchi Serena; Teodori Elisabetta
Synthesis, affinity profile, and functional activity of muscarinic antagonists with a 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine structure.
Journal of medicinal chemistry 2007;50(6):1409-13.
-
2007: Tumiatti Vincenzo; Minarini Anna; Milelli Andrea; Rosini Michela; Buccioni Michela; Marucci Gabriella; Ghelardini Carla; Bellucci Cristina; Melchiorre Carlo
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: effect of replacing the inner polymethylene chain with cyclic moieties.
Bioorganic & medicinal chemistry 2007;15(6):2312-21.
-
2007: Sagratini Gianni; Angeli Piero; Buccioni Michela; Gulini Ugo; Marucci Gabriella; Melchiorre Carlo; Leonardi Amedeo; Poggesi Elena; Giardinà Dario
Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.
Bioorganic & medicinal chemistry 2007;15(6):2334-45.
-
2006: Romeo Giuseppe; Materia Luisa; Marucci Gabriella; Modica Maria; Pittalà Valeria; Salerno Loredana; Siracusa Maria Angela; Buccioni Michela; Angeli Piero; Minneman Kenneth P
New pyrimido[5,4-b]indoles and [1]benzothieno[3,2-d]pyrimidines: high affinity ligands for the alpha(1)-adrenoceptor subtypes.
Bioorganic & medicinal chemistry letters 2006;16(24):6200-3.
-
2006: Scapecchi Serena; Matucci Rosanna; Bellucci Cristina; Buccioni Michela; Dei Silvia; Guandalini Luca; Martelli Cecilia; Manetti Dina; Martini Elisabetta; Marucci Gabriella; Nesi Marta; Romanelli Maria Novella; Teodori Elisabetta; Gualtieri Fulvio
Highly chiral muscarinic ligands: the discovery of (2S,2'R,3'S,5'R)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-sulfoxide methyl iodide, a potent, functionally selective, M2 partial agonist.
Journal of medicinal chemistry 2006;49(6):1925-31.
-
2006: Pittalà Valeria; Romeo Giuseppe; Salerno Loredana; Siracusa Maria Angela; Modica Maria; Materia Luisa; Mereghetti Ilario; Cagnotto Alfredo; Mennini Tiziana; Marucci Gabriella; Angeli Piero; Russo Filippo
3-Arylpiperazinylethyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione derivatives as novel, high-affinity and selective alpha(1)-adrenoceptor ligands.
Bioorganic & medicinal chemistry letters 2006;16(1):150-3.
-
2005: Marucci Gabriella; Angeli Piero; Buccioni Michela; Gulini Ugo; Melchiorre Carlo; Sagratini Gianni; Testa Rodolfo; Giardinà Dario
(+)-Cyclazosin, a selective alpha1B-adrenoceptor antagonist: functional evaluation in rat and rabbit tissues.
European journal of pharmacology 2005;522(1-3):100-7.
-
2005: Dei Silvia; Angeli Piero; Bellucci Cristina; Buccioni Michela; Gualtieri Fulvio; Marucci Gabriella; Manetti Dina; Matucci Rosanna; Romanelli Maria Novella; Scapecchi Serena; Teodori Elisabetta
Muscarinic subtype affinity and functional activity profile of 1-methyl-2-(2-methyl-1,3-dioxolan-4-yl)pyrrolidine and 1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine derivatives.
Biochemical pharmacology 2005;69(11):1637-45.
-
2005: Tait Annalisa; Luppi Amedeo; Franchini Silvia; Preziosi Elisa; Parenti Carlo; Buccioni Michela; Marucci Gabriella; Leonardi Amedeo; Poggesi Elena; Brasili Livio
1,2,4-Benzothiadiazine derivatives as alpha1 and 5-HT1A receptor ligands.
Bioorganic & medicinal chemistry letters 2005;15(4):1185-8.
-
2005: Antonello Alessandra; Hrelia Patrizia; Leonardi Amedeo; Marucci Gabriella; Rosini Michela; Tarozzi Andrea; Tumiatti Vincenzo; Melchiorre Carlo
Design, synthesis, and biological evaluation of prazosin-related derivatives as multipotent compounds.
Journal of medicinal chemistry 2005;48(1):28-31.
-
2004: Scapecchi Serena; Martini Elisabetta; Bellucci Cristina; Buccioni Michela; Dei Silvia; Guandalini Luca; Manetti Dina; Martelli Cecilia; Marucci Gabriella; Matucci Rosanna
Molecular modulation of muscarinic antagonists. Synthesis and affinity profile of 2,2-diphenyl-2-ethylthio-acetic acid esters designed to probe the binding site cavity.
Farmaco (Società chimica italiana : 1989) 2004;59(12):971-80.
-
2003: Rosini Michela; Antonello Alessandra; Cavalli Andrea; Bolognesi Maria L; Minarini Anna; Marucci Gabriella; Poggesi Elena; Leonardi Amedeo; Melchiorre Carlo
Prazosin-related compounds. Effect of transforming the piperazinylquinazoline moiety into an aminomethyltetrahydroacridine system on the affinity for alpha1-adrenoreceptors.
Journal of medicinal chemistry 2003;46(23):4895-903.
-
2003: Varoli Lucilla; Angeli Piero; Buccioni Michela; Burnelli Silvia; Cavalli Andrea; Marucci Gabriella; Recanatini Maurizio
Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol.
Farmaco (Società chimica italiana : 1989) 2003;58(9):651-7.
-
2003: Piergentili Alessandro; Gentili Francesco; Ghelfi Francesca; Marucci Gabriella; Pigini Maria; Quaglia Wilma; Giannella Mario
Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine.
Bioorganic & medicinal chemistry 2003;11(18):3901-11.
-
2003: Giardinà Dario; Polimanti O; Sagratini G; Angeli P; Gulini U; Marucci G; Melchiorre C; Poggesi E; Leonardi A
Searching for cyclazosin analogues as alpha(1B)-adrenoceptor antagonists.
Farmaco (Società chimica italiana : 1989) 2003;58(7):477-87.
-
2003: Brasili Livio; Sorbi Claudia; Franchini Silvia; Manicardi Massimo; Angeli Piero; Marucci Gabriella; Leonardi Amedeo; Poggesi Elena
1,3-dioxolane-based ligands as a novel class of alpha1-adrenoceptor antagonists.
Journal of medicinal chemistry 2003;46(8):1504-11.
-
2003: Tumiatti Vincenzo; Rosini Michela; Bartolini Manuela; Cavalli Andrea; Marucci Gabriella; Andrisano Vincenza; Angeli Piero; Banzi Rita; Minarini Anna; Recanatini Maurizio; Melchiorre Carlo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine.
Journal of medicinal chemistry 2003;46(6):954-66.
-
2002: Bolognesi Maria L; Bixel M Gabriele; Marucci Gabriella; Bartolini Manuela; Krauss Michael; Angeli Piero; Antonello Alessandra; Rosini Michela; Tumiatti Vincenzo; Hucho Ferdinand; Melchiorre Carlo
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure.
Journal of medicinal chemistry 2002;45(15):3286-95.
-
2002: Giardinà Dario; Crucianelli Mauro; Angeli Piero; Buccioni Michela; Gulini Ugo; Marucci Gabriella; Sagratini Gianni; Melchiorre Carlo
Structure--activity relationships among novel phenoxybenzamine-related beta-chloroethylamines.
Bioorganic & medicinal chemistry 2002;10(5):1291-303.
-
2002: Rosini Michela; Bixel M Gabriele; Marucci Gabriella; Budriesi Roberta; Krauss Michael; Bolognesi Maria L; Minarini Anna; Tumiatti Vincenzo; Hucho Ferdinand; Melchiorre Carlo
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms.
Journal of medicinal chemistry 2002;45(9):1860-78.
-
2002: Quaglia Wilma; Pigini Maria; Piergentili Alessandro; Giannella Mario; Gentili Francesco; Marucci Gabriella; Carrieri Antonio; Carotti Angelo; Poggesi Elena; Leonardi Amedeo; Melchiorre Carlo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes.
Journal of medicinal chemistry 2002;45(8):1633-43.
-
2002: Angeli Piero; Marucci Gabriella; Buccioni Michela; Piergentili Alessandro; Giannella Mario; Quaglia Wilma; Pigini Maria; Cantalamessa Franco; Nasuti Cinzia; Novi Francesca; Maggio Roberto; Qasem Ahmed R; Spampinato Santi
Deoxamuscaroneoxime derivatives as useful muscarinic agonists to explore the muscarinic subsite: demox, a modulator of orthosteric and allosteric sites at cardiac muscarinic M2 receptors.
Life sciences 2002;70(12):1427-46.
-
2002: Gentili Francesco; Bousquet Pascal; Brasili Livio; Caretto Mariangela; Carrieri Antonio; Dontenwill Monique; Giannella Mario; Marucci Gabriella; Perfumi Marina; Piergentili Alessandro; Quaglia Wilma; Rascente Carla; Pigini Maria
Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole.
Journal of medicinal chemistry 2002;45(1):32-40.
-
2001: Scapecchi S; Marucci G; Matucci R; Angeli P; Bellucci C; Buccioni M; Dei S; Gualtieri F; Manetti D; Romanelli M N; Teodori E
Structure-activity relationships in 2,2-diphenyl-2-ethylthioacetic acid esters: unexpected agonistic activity in a series of muscarinic antagonists.
Bioorganic & medicinal chemistry 2001;9(5):1165-74.
-
2001: Bolognesi M L; Marucci G; Angeli P; Buccioni M; Minarini A; Rosini M; Tumiatti V; Melchiorre C
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward alpha1-adrenoreceptor subtypes.
Journal of medicinal chemistry 2001;44(3):362-71.
-
2001: Gulini U; Angeli P; Marucci G; Buccioni M; Giardinà D; Antolini L; Franchini S; Sorbi C; Brasili L
Synthesis, absolute configuration and antimuscarinic activity of the enantiomers of [1-(2,2-diphenyl-[1,3]dioxolan-4-yl)-ethyl]-dimethyl-amine.
Bioorganic & medicinal chemistry letters 2001;11(2):247-50.
-
2000: De Amici M; Dallanoce C; Angeli P; Marucci G; Cantalamessa F; De Micheli C
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine.
Farmaco (Società chimica italiana : 1989) 2000;55(8):535-43.
-
2000: De Amici M; Dallanoce C; De Micheli C; Angeli P; Marucci G; Cantalamessa F; Sparapassi L
Pharmacological profile of enantiomerically pure chiral muscarinic agonists: desoxymuscarines.
Life sciences 2000;67(3):317-26.
-
2000: Pigini M; Quaglia W; Gentili F; Marucci G; Cantalamessa F; Franchini S; Sorbi C; Brasili L
Structure-activity relationship at alpha-adrenergic receptors within a series of imidazoline analogues of cirazoline.
Bioorganic & medicinal chemistry 2000;8(5):883-8.
-
2000: Tumiatti V; Angeli P; Andrisano V; Bolognesi M L; Cavalli A; Marucci G; Minarini A; Recanatini M; Rosini M; Melchiorre C
[4-[[N-(3-chlorophenyl)carbamoyl]oxy]-2-butynyl]-trimethylammonium (McN-A-343)-related compounds. Effect of the butynyl chain inclusion into an aromatic unit on the potency for muscarinic receptors.
Bioorganic & medicinal chemistry 2000;8(4):681-9.
-
2000: Melchiorre C; Angeli P; Bolognesi M L; Chiarini A; Giardinà D; Gulini U; Leonardi A; Marucci G; Minarini A; Pigini M; Quaglia W; Rosini M; Tumiatti V
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety.
Pharmaceutica acta Helvetiae 2000;74(2-3):181-90.
-
1999: Varoli L; Angeli P; Burnelli S; Marucci G; Recanatini M
Synthesis and antagonistic activity at muscarinic receptor subtypes of some 2-carbonyl derivatives of diphenidol.
Bioorganic & medicinal chemistry 1999;7(9):1837-44.
-
1999: Quaglia W; Pigini M; Piergentili A; Giannella M; Marucci G; Poggesi E; Leonardi A; Melchiorre C
Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes.
Journal of medicinal chemistry 1999;42(15):2961-8.
-
1998: Malmusi L; Franchini S; Mucci A; Schenetti L; Gulini U; Marucci G; Brasili L
Synthesis and antimuscarinic activity of some ether- and thioether-bearing 1,3-dioxolanes and related sulfoxides and sulfones.
Bioorganic & medicinal chemistry 1998;6(6):825-32.
-
1997: Giardinà D; Crucianelli M; Marucci G; Angeli P; Melchiorre C; Antolini L
Synthesis and alpha-adrenoceptor blocking activity of the enantiomers of benzyl-(2-chloroethyl)-[2-(2-methoxyphenoxy)-1-methylethyl]amine hydrochloride.
Bioorganic & medicinal chemistry 1997;5(9):1775-82.
-
1997: Scapecchi S; Angeli P; Dei S; Ghelardini C; Gualtieri F; Marucci G; Paparelli F; Romanelli M N; Teodori E
SAR studies on the potent and selective muscarinic antagonist 2-ethylthio-2,2-diphenylacetic acid N,N-diethylaminoethyl ester.
Archiv der Pharmazie 1997;330(5):122-8.
-
1997: Angeli P; Brasili L; Cingolani M L; Marucci G; Piergentili A; Pigini M; Quaglia W
Synthesis and structure-activity relationship studies in a series of 2-substituted 1,3-dioxolanes modified at the cationic head.
Bioorganic & medicinal chemistry 1997;5(4):731-7.
-
1997: Angeli P; Cantalamessa F; Cavagna R; Conti P; De Amici M; De Micheli C; Gamba A; Marucci G
Synthesis and pharmacological characterization of enantiomerically pure muscarinic agonists: difluoromuscarines.
Journal of medicinal chemistry 1997;40(7):1099-103.
-
1996: Malmusi L; Mucci A; Schenetti L; Gulini U; Marucci G; Brasili L
Synthesis, NMR spectroscopy study, and antimuscarinic activity of a series of 2-(acyloxymethyl)-1,3-dioxolanes.
Bioorganic & medicinal chemistry 1996;4(12):2071-80.
-
1996: Giardinà D; Crucianelli M; Marucci G; Melchiorre C; Polidori C; Pompei P; Massi M
Pharmacological evaluation of prazosin- and doxazosin-related compounds with modified piperazine ring.
Arzneimittel-Forschung 1996;46(11):1054-9.
-
1996: Quaglia W; Giannella M; Marucci G; Piergentili A; Pigini M; Tayebati S K; Melchiorre C
Structure-activity relationships in 1,4-benzodioxan-related compounds. 5. Effects of modification of the side chain on alpha-adrenoreceptor blocking activity.
Farmaco (Società chimica italiana : 1989) 1996;51(1):27-32.
-
1995: Brasili L; Pigini M; Marucci G; Quaglia W; Malmusi L; Lanier S M; Lanier B
Separation of alpha-adrenergic and imidazoline/guanidinium receptive sites (IGRS) activity in a series of imidazoline analogues of cirazoline.
Bioorganic & medicinal chemistry 1995;3(11):1503-9.
-
1995: Giardinà D; Crucianelli M; Marucci G; Paparelli F; Melchiorre C
Synthesis and alpha-adrenoreceptor blocking properties of phenoxybenzamine-related (2-chloroethyl)-(2,3-dihydrobenzo[1,4]dioxin- 2-ylmethyl)-(2-phenoxyethyl) amines.
Bioorganic & medicinal chemistry 1995;3(1):85-94.
-
1994: Scapecchi S; Angeli P; Dei S; Gualtieri F; Marucci G; Moriconi R; Paparelli F; Romanelli M N; Teodori E
Dialkylaminoalkyl esters of 2,2-diphenyl-2-alkylthioacetic acids: a new class of potent and functionally selective muscarinic antagonists.
Bioorganic & medicinal chemistry 1994;2(10):1061-74.
-
1994: Teodori E; Dei S; Romanelli M N; Scappecchi S; Gualtieri F; Angeli P; Marucci G; Matucci R
1,3-oxathiolane muscarinic ligands modified at the cationic head.
Farmaco (Società chimica italiana : 1989) 1994;49(5):305-12.
-
1993: Quaglia W; Pigini M; Tayebati S K; Piergentili A; Giannella M; Marucci G; Melchiorre C
Structure-activity relationships in 1,4-benzodioxan-related compounds. 4. Effect of aryl and alkyl substituents at position 3 on alpha-adrenoreceptor blocking activity.
Journal of medicinal chemistry 1993;36(11):1520-8.
-
1992: Bravo P; Resnati G; Angeli P; Frigerio M; Viani F; Arnone A; Marucci G; Cantalamessa F
Synthesis and pharmacological evaluation of enantiomerically pure 4-deoxy-4-fluoromuscarines.
Journal of medicinal chemistry 1992;35(17):3102-10.
-
1992: Andrisano V; Marucci G; Melchiorre C; Tumiatti V
Stereoselectivity at alpha-adrenoreceptor subtypes: observations with the enantiomers of WB 4101 separated through their amides of N-tosyl-(S)-proline.
Chirality 1992;4(1):16-20.
-
1991: Angeli P; Brasili L; Cingolani M L; Marucci G; Pigini P; Tonnini M C
Pharmacological characterization of muscarinic receptor subtypes in rabbit isolated tissue preparations.
Journal of autonomic pharmacology 1991;11(5):315-21.
-
1991: Giardinà D; Marrazzo A; Marucci G; Piloni M G; Quaglia W
Methoctramine-related polymethylene tetraamines. 4. Chirality effect on M2 muscarinic receptor blocking activity.
Farmaco (Società chimica italiana : 1989) 1991;46(7-8):861-72.
-
1991: Quaglia W; Giardinà D; Marucci G; Melchiorre C; Minarini A; Tumiatti V
Structure-activity relationships among methoctramine-related polymethylene tetraamines. 3. Effect of the four nitrogens on M2 muscarinic blocking activity as revealed by symmetrical and unsymmetrical polyamines.
Farmaco (Società chimica italiana : 1989) 1991;46(3):417-34.
-
1990: Angeli P; Brasili L; Cantalamessa F; Marucci G; Wess J
Determination of muscarinic agonist potencies at M1 and M2 muscarinic receptors in a modified pithed rat preparation.
Naunyn-Schmiedeberg's archives of pharmacology 1990;342(6):625-9.
Sign-in to see more