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Duane Miller
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57
Feller, Dennis
43
Dalton, James
23
Shams, Gamal
22
Patil, Popat
12
Uretsky, NJ
11
Wallace, Lane
11
Li, Wei
11
Bohl, Casey
10
Gao, Wenqing
10
Tigyi, Gabor
9
De Los Angeles, Joseph
7
Gududuru, Veeresa
7
He, Yali
7
Hong, Seoung Soo
7
Hwang, Dong Jin
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All Publications
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2009: Zeng Kui; Thompson Karin Emmons; Yates Charles R; Miller Duane D
Synthesis and biological evaluation of quinic acid derivatives as anti-inflammatory agents.
Bioorganic & medicinal chemistry letters 2009;19(18):5458-60.
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2009: Danquah Michael; Li Feng; Duke Charles B; Miller Duane D; Mahato Ram I
Micellar delivery of bicalutamide and embelin for treating prostate cancer.
Pharmaceutical research 2009;26(9):2081-92.
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2009: Wang Zhao; Lu Yan; Seibel William; Miller Duane D; Li Wei
Identifying novel molecular structures for advanced melanoma by ligand-based virtual screening.
Journal of chemical information and modeling 2009;49(6):1420-7.
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2009: Mohler Michael L; Bohl Casey E; Jones Amanda; Coss Christopher C; Narayanan Ramesh; He Yali; Hwang Dong Jin; Dalton James T; Miller Duane D
Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit.
Journal of medicinal chemistry 2009;52(12):3597-617.
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2009: Li Wei; Hwang Dong Jin; Cremer Dieter; Joo Hyun; Kraka Elfi; Kim Juhyun; Ross Charles R; Nguyen Viet Q; Dalton James T; Miller Duane D
Structure determination of chiral sulfoxide in diastereomeric bicalutamide derivatives.
Chirality 2009;21(6):578-83.
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2009: Ramagiri Suma; Ma Fei; Kosanam Hari; Wang XiangDi; Patil Renukadevi; Miller Duane D; Geisert Eldon; Yates Charles R
Fast and sensitive liquid chromatography/electrospray mass spectrometry method to study ocular penetration of EDL-155, a novel antitumor agent for retinoblastoma in rats.
Journal of mass spectrometry : JMS 2009;44(5):786-93.
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2009: Lu Yan; Li Chien-Ming; Wang Zhao; Ross Charles R; Chen Jianjun; Dalton James T; Li Wei; Miller Duane D
Discovery of 4-substituted methoxybenzoyl-aryl-thiazole as novel anticancer agents: synthesis, biological evaluation, and structure-activity relationships.
Journal of medicinal chemistry 2009;52(6):1701-11.
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2009: Zmijewski Michal A; Li Wei; Zjawiony Jordan K; Sweatman Trevor W; Chen Jianjun; Miller Duane D; Slominski Andrzej T
Photo-conversion of two epimers (20R and 20S) of pregna-5,7-diene-3beta, 17alpha, 20-triol and their bioactivity in melanoma cells.
Steroids 2009;74(2):218-28.
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2009: Jones Amanda; Chen Jiyun; Hwang Dong Jin; Miller Duane D; Dalton James T
Preclinical characterization of a (S)-N-(4-cyano-3-trifluoromethyl-phenyl)-3-(3-fluoro, 4-chlorophenoxy)-2-hydroxy-2-methyl-propanamide: a selective androgen receptor modulator for hormonal male contraception.
Endocrinology 2009;150(1):385-95.
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2009: Patil Shivaputra A; Patil Renukadevi; Miller Duane D
Solid phase synthesis of biologically important indoles.
Current medicinal chemistry 2009;16(20):2531-65.
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2008: Zmijewski Michal A; Li Wei; Zjawiony Jordan K; Sweatman Trevor W; Chen Jianjun; Miller Duane D; Slominski Andrzej T
Synthesis and photo-conversion of androsta- and pregna-5,7-dienes to vitamin D3-like derivatives.
Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 2008;7(12):1570-6.
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2008: DeCuypere Michael; Lu Yan; Miller Duane D; LeDoux Mark S
Regional distribution of tetrahydroisoquinoline derivatives in rodent, human, and Parkinson's disease brain.
Journal of neurochemistry 2008;107(5):1398-413.
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2008: Narayanan Ramesh; Coss Christopher C; Yepuru Muralimohan; Kearbey Jeffrey D; Miller Duane D; Dalton James T
Steroidal androgens and nonsteroidal, tissue-selective androgen receptor modulator, S-22, regulate androgen receptor function through distinct genomic and nongenomic signaling pathways.
Molecular endocrinology (Baltimore, Md.) 2008;22(11):2448-65.
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2008: Bohl Casey E; Wu Zengru; Chen Jiyun; Mohler Michael L; Yang Jun; Hwang Dong Jin; Mustafa Suni; Miller Duane D; Bell Charles E; Dalton James T
Effect of B-ring substitution pattern on binding mode of propionamide selective androgen receptor modulators.
Bioorganic & medicinal chemistry letters 2008;18(20):5567-70.
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2008: Kang Gyong-Suk; Wang Xiang Di; Mohler Michael L; Kirichenko Oleg V; Patil Renukadevi; Orr William E; Miller Duane D; Geisert Eldon E
Effects, in an in-vivo model system, of 1,2,3,4-tetrahydroisoquinoline on glioma.
Anti-cancer drugs 2008;19(9):859-70.
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2008: Bavadekar Supriya A; Hong Seoung-Soo; Lee Sang-Ii; Miller Duane D; Feller Dennis R
Bioisosteric phentolamine analogs as selective human alpha(2)- versus alpha(1)-adrenoceptor ligands.
European journal of pharmacology 2008;590(1-3):53-60.
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2008: DeCuypere Michael; Kalabokis Vassilios N; Hao Ruyi; Schroeder Dorothy; Miller Duane D; LeDoux Mark S
Localization of N-methyl-norsalsolinol within rodent and human brain.
Journal of neuroscience research 2008;86(11):2543-52.
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2008: Chen Jianjun; Wang Zhao; Lu Yan; Dalton James T; Miller Duane D; Li Wei
Synthesis and antiproliferative activity of imidazole and imidazoline analogs for melanoma.
Bioorganic & medicinal chemistry letters 2008;18(11):3183-7.
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2008: Song Pengfei; Ma Fei; Wang Fan; Wang XiangDi; Patil Renukadevi; Ramagiri Suma; Orr William E; Miller Duane D; Geisert Eldon; Yates Charles R
Plasma and cerebrospinal fluid pharmacokinetics of the novel tetrahydroisoquinoline EDL-155 in rats.
Cancer chemotherapy and pharmacology 2008;61(6):1037-44.
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2008: Zhu Lin; Ye Zhaoyang; Cheng Kun; Miller Duane D; Mahato Ram I
Site-specific delivery of oligonucleotides to hepatocytes after systemic administration.
Bioconjugate chemistry 2008;19(1):290-8.
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2008: Ramagiri Suma; Gupte Renuka; Rakov Igor; Yates Charles R; Miller Duane D
Quantitative chiral analysis of phthaloylglutamic acid and related analogs by a single ratio kinetic method using electrospray ionization and matrix-assisted laser desorption techniques.
Rapid communications in mass spectrometry : RCM 2008;22(5):639-46.
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2007: Li Wei; Lu Yan; Wang Zhao; Dalton James T; Miller Duane D
Synthesis and antiproliferative activity of thiazolidine analogs for melanoma.
Bioorganic & medicinal chemistry letters 2007;17(15):4113-7.
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2007: Deng Wenlin; Shuyu E; Tsukahara Ryoko; Valentine William J; Durgam Gangadhar; Gududuru Veeresa; Balazs Louisa; Manickam Venkatraman; Arsura Marcello; VanMiddlesworth Lester; Johnson Leonard R; Parrill Abby L; Miller Duane D; Tigyi Gabor
The lysophosphatidic acid type 2 receptor is required for protection against radiation-induced intestinal injury.
Gastroenterology 2007;132(5):1834-51.
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2007: Bohl Casey E; Wu Zengru; Miller Duane D; Bell Charles E; Dalton James T
Crystal structure of the T877A human androgen receptor ligand-binding domain complexed to cyproterone acetate provides insight for ligand-induced conformational changes and structure-based drug design.
The Journal of biological chemistry 2007;282(18):13648-55.
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2007: Li Wei; Wang Zhao; Gududuru Veeresa; Zbytek Blazej; Slominski Andrzej T; Dalton James T; Miller Duane D
Structure-activity relationship studies of arylthiazolidine amides as selective cytotoxic agents for melanoma.
Anticancer research 2007;27(2):883-8.
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2007: Kearbey Jeffrey D; Gao Wenqing; Narayanan Ramesh; Fisher Scott J; Wu Di; Miller Duane D; Dalton James T
Selective Androgen Receptor Modulator (SARM) treatment prevents bone loss and reduces body fat in ovariectomized rats.
Pharmaceutical research 2007;24(2):328-35.
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2006: Bavadekar Supriya A; Ma Guoyi; Mustafa Suni M; Moore Bob M; Miller Duane D; Feller Dennis R
Tethered yohimbine analogs as selective human alpha2C-adrenergic receptor ligands.
The Journal of pharmacology and experimental therapeutics 2006;319(2):739-48.
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2006: Hwang Dong Jin; Yang Jun; Xu Huiping; Rakov Igor M; Mohler Michael L; Dalton James T; Miller Duane D
Arylisothiocyanato selective androgen receptor modulators (SARMs) for prostate cancer.
Bioorganic & medicinal chemistry 2006;14(19):6525-38.
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2006: Perera Minoli A; Yin Donghua; Wu Di; Chan Kenneth K; Miller Duane D; Dalton James
In vivo metabolism and final disposition of a novel nonsteroidal androgen in rats and dogs.
Drug metabolism and disposition: the biological fate of chemicals 2006;34(10):1713-21.
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2006: Mohler Michael L; Kang Gyong-Suk; Hong Seoung-Soo; Patil Renukadevi; Kirichenko Oleg V; Li Wei; Rakov Igor M; Geisert Eldon E; Miller Duane D
Discovery of antiglioma activity of biaryl 1,2,3,4-tetrahydroisoquinoline derivatives and conformationally flexible analogues.
Journal of medicinal chemistry 2006;49(19):5845-8.
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2006: Gourley Dick R; Rowell Crescent; Wingate LaMarcus; Yates Charles R; Gourley Greta K; Miller Duane D; Vleet Van
Status of PharmD/PhD programs in colleges of pharmacy: the University of Tennessee dual PharmD/PhD program.
American journal of pharmaceutical education 2006;70(2):44.
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2006: Boucher Bradley A; Chyka Peter J; Fitzgerald Walter L; Hak Lawrence J; Miller Duane D; Parker Robert B; Phelps Stephanie J; Wood George C; Gourley Dick R
A comprehensive approach to faculty development.
American journal of pharmaceutical education 2006;70(2):27.
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2006: Yang Jun; Bohl Casey E; Nair Vipin A; Mustafa Suni M; Hong Seoung Soo; Miller Duane D; Dalton James T
Preclinical pharmacology of a nonsteroidal ligand for androgen receptor-mediated imaging of prostate cancer.
The Journal of pharmacology and experimental therapeutics 2006;317(1):402-8.
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2006: Nikulin Victor I; Rakov Igor M; De Los Angeles Joseph E; Mehta Ratna C; Boyd LeNe'Sheya Y; Feller Dennis R; Miller Duane D
1-Benzyl-1,2,3,4-tetrahydroisoquinoline-6,7-diols as novel affinity and photoaffinity probes for beta-adrenoceptor subtypes.
Bioorganic & medicinal chemistry 2006;14(6):1684-97.
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2006: Wu Di; Wu Zengru; Yang Jun; Nair Vipin A; Miller Duane D; Dalton James T
Pharmacokinetics and metabolism of a selective androgen receptor modulator in rats: implication of molecular properties and intensive metabolic profile to investigate ideal pharmacokinetic characteristics of a propanamide in preclinical study.
Drug metabolism and disposition: the biological fate of chemicals 2006;34(3):483-94.
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2006: Gao Wenqing; Wu Zengru; Bohl Casey E; Yang Jun; Miller Duane D; Dalton James T
Characterization of the in vitro metabolism of selective androgen receptor modulator using human, rat, and dog liver enzyme preparations.
Drug metabolism and disposition: the biological fate of chemicals 2006;34(2):243-53.
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2006: Gao Wenqing; Johnston Jeffrey S; Miller Duane D; Dalton James T
Interspecies differences in pharmacokinetics and metabolism of S-3-(4-acetylamino-phenoxy)-2-hydroxy-2-methyl-N-(4-nitro-3-trifluoromethylphenyl)-propionamide: the role of N-acetyltransferase.
Drug metabolism and disposition: the biological fate of chemicals 2006;34(2):254-60.
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2006: Durgam Gangadhar G; Tsukahara Ryoko; Makarova Natalia; Walker Michelle D; Fujiwara Yuko; Pigg Kathryn R; Baker Daniel L; Sardar Vineet M; Parrill Abby L; Tigyi Gabor; Miller Duane D
Synthesis and pharmacological evaluation of second-generation phosphatidic acid derivatives as lysophosphatidic acid receptor ligands.
Bioorganic & medicinal chemistry letters 2006;16(3):633-40.
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2006: Gududuru Veeresa; Zeng Kui; Tsukahara Ryoko; Makarova Natalia; Fujiwara Yuko; Pigg Kathryn R; Baker Daniel L; Tigyi Gabor; Miller Duane D
Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors.
Bioorganic & medicinal chemistry letters 2006;16(2):451-6.
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2005: Chen Jiyun; Hwang Dong Jin; Chung Kiwon; Bohl Casey E; Fisher Scott J; Miller Duane D; Dalton James T
In vitro and in vivo structure-activity relationships of novel androgen receptor ligands with multiple substituents in the B-ring.
Endocrinology 2005;146(12):5444-54.
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2005: Hong Seoung-Soo; Bavadekar Supriya A; Lee Sang-Il; Patil Popat N; Lalchandani S G; Feller Dennis R; Miller Duane D
Bioisosteric phentolamine analogs as potent alpha-adrenergic antagonists.
Bioorganic & medicinal chemistry letters 2005;15(21):4691-5.
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2005: Bohl Casey E; Miller Duane D; Chen Jiyun; Bell Charles E; Dalton James T
Structural basis for accommodation of nonsteroidal ligands in the androgen receptor.
The Journal of biological chemistry 2005;280(45):37747-54.
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2005: Gao Wenqing; Reiser Peter J; Coss Christopher C; Phelps Mitch A; Kearbey Jeffrey D; Miller Duane D; Dalton James T
Selective androgen receptor modulator treatment improves muscle strength and body composition and prevents bone loss in orchidectomized rats.
Endocrinology 2005;146(11):4887-97.
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2005: Kim Juhyun; Wu Di; Hwang Dong Jin; Miller Duane D; Dalton James T
The para substituent of S-3-(phenoxy)-2-hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-phenyl)-propionamides is a major structural determinant of in vivo disposition and activity of selective androgen receptor modulators.
The Journal of pharmacology and experimental therapeutics 2005;315(1):230-9.
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2005: Gududuru Veeresa; Hurh Eunju; Sullivan Joshua; Dalton James T; Miller Duane D
SAR studies of 2-arylthiazolidine-4-carboxylic acid amides: a novel class of cytotoxic agents for prostate cancer.
Bioorganic & medicinal chemistry letters 2005;15(18):4010-3.
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2005: Durgam Gangadhar G; Virag Tamas; Walker Michelle D; Tsukahara Ryoko; Yasuda Satoshi; Liliom Karoly; van Meeteren Laurens A; Moolenaar Wouter H; Wilke Nicole; Siess Wolfgang; Tigyi Gabor; Miller Duane D
Synthesis, structure-activity relationships, and biological evaluation of fatty alcohol phosphates as lysophosphatidic acid receptor ligands, activators of PPARgamma, and inhibitors of autotaxin.
Journal of medicinal chemistry 2005;48(15):4919-30.
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2005: Mustafa Suni M; Bavadekar Supriya A; Ma Guoyi; Moore Bob M; Feller Dennis R; Miller Duane D
Synthesis and biological studies of yohimbine derivatives on human alpha2C-adrenergic receptors.
Bioorganic & medicinal chemistry letters 2005;15(11):2758-60.
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2005: Bohl Casey E; Gao Wenqing; Miller Duane D; Bell Charles E; Dalton James T
Structural basis for antagonism and resistance of bicalutamide in prostate cancer.
Proceedings of the National Academy of Sciences of the United States of America 2005;102(17):6201-6.
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2005: Gududuru Veeresa; Hurh Eunju; Dalton James T; Miller Duane D
Discovery of 2-arylthiazolidine-4-carboxylic acid amides as a new class of cytotoxic agents for prostate cancer.
Journal of medicinal chemistry 2005;48(7):2584-8.
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2005: Chen Jiyun; Hwang Dong Jin; Bohl Casey E; Miller Duane D; Dalton James T
A selective androgen receptor modulator for hormonal male contraception.
The Journal of pharmacology and experimental therapeutics 2005;312(2):546-53.
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2005: Narang Ajit S; Thoma Laura; Miller Duane D; Mahato Ram I
Cationic lipids with increased DNA binding affinity for nonviral gene transfer in dividing and nondividing cells.
Bioconjugate chemistry 2005;16(1):156-68.
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2004: Gao Wenqing; Kearbey Jeffrey D; Nair Vipin A; Chung Kiwon; Parlow A F; Miller Duane D; Dalton James T
Comparison of the pharmacological effects of a novel selective androgen receptor modulator, the 5alpha-reductase inhibitor finasteride, and the antiandrogen hydroxyflutamide in intact rats: new approach for benign prostate hyperplasia.
Endocrinology 2004;145(12):5420-8.
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2004: Gududuru Veeresa; Hurh Eunju; Dalton James T; Miller Duane D
Synthesis and antiproliferative activity of 2-aryl-4-oxo-thiazolidin-3-yl-amides for prostate cancer.
Bioorganic & medicinal chemistry letters 2004;14(21):5289-93.
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2004: Gududuru Veeresa; Hurh Eunju; Durgam Gangadhar G; Hong Seoung Soo; Sardar Vineet M; Xu Huiping; Dalton James T; Miller Duane D
Synthesis and biological evaluation of novel cytotoxic phospholipids for prostate cancer.
Bioorganic & medicinal chemistry letters 2004;14(19):4919-23.
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2004: Bohl Casey E; Chang Cheng; Mohler Michael L; Chen Jiyun; Miller Duane D; Swaan Peter W; Dalton James T
A ligand-based approach to identify quantitative structure-activity relationships for the androgen receptor.
Journal of medicinal chemistry 2004;47(15):3765-76.
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2004: Kearbey J D; Wu D; Gao W; Miller D D; Dalton J T
Pharmacokinetics of S-3-(4-acetylamino-phenoxy)-2-hydroxy-2-methyl-N-(4-nitro- 3-trifluoromethyl-phenyl)-propionamide in rats, a non-steroidal selective androgen receptor modulator.
Xenobiotica; the fate of foreign compounds in biological systems 2004;34(3):273-80.
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2004: Marhefka Craig A; Gao Wenqing; Chung Kiwon; Kim Juhyun; He Yali; Yin Donghua; Bohl Casey; Dalton James T; Miller Duane D
Design, synthesis, and biological characterization of metabolically stable selective androgen receptor modulators.
Journal of medicinal chemistry 2004;47(4):993-8.
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2004: Wu Zengru; Gao Wenqing; Phelps Mitch A; Wu Di; Miller Duane D; Dalton James T
Favorable effects of weak acids on negative-ion electrospray ionization mass spectrometry.
Analytical chemistry 2004;76(3):839-47.
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2004: Lalchandani Shilpa G; Zhang Xiaoyang; Hong Seoung Soo; Liggett Stephen B; Li Wei; Moore Bob M; Miller Duane D; Feller Dennis R
Medetomidine analogs as selective agonists for the human alpha2-adrenoceptors.
Biochemical pharmacology 2004;67(1):87-96.
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2003: Yates Charles R; Chang Cheng; Kearbey Jeffrey D; Yasuda Kazuto; Schuetz Erin G; Miller Duane D; Dalton James T; Swaan Peter W
Structural determinants of P-glycoprotein-mediated transport of glucocorticoids.
Pharmaceutical research 2003;20(11):1794-803.
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2003: Wagner Carl E; Mohler Michael L; Kang Gyong Suk; Miller Duane D; Geisert Eldon E; Chang Yu-An; Fleischer Everly B; Shea Kenneth J
Synthesis of 1-boraadamantaneamine derivatives with selective astrocyte vs C6 glioma antiproliferative activity. A novel class of anti-hepatitis C agents with potential to bind CD81.
Journal of medicinal chemistry 2003;46(14):2823-33.
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2003: Virag Tamas; Elrod Don B; Liliom Karoly; Sardar Vineet M; Parrill Abby L; Yokoyama Kazuaki; Durgam Gangadhar; Deng Wenlin; Miller Duane D; Tigyi Gabor
Fatty alcohol phosphates are subtype-selective agonists and antagonists of lysophosphatidic acid receptors.
Molecular pharmacology 2003;63(5):1032-42.
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2003: Yin Donghua; Gao Wenqing; Kearbey Jeffrey D; Xu Huiping; Chung Kiwon; He Yali; Marhefka Craig A; Veverka Karen A; Miller Duane D; Dalton James T
Pharmacodynamics of selective androgen receptor modulators.
The Journal of pharmacology and experimental therapeutics 2003;304(3):1334-40.
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2003: Yin Donghua; Xu Huiping; He Yali; Kirkovsky Leonid I; Miller Duane D; Dalton James T
Pharmacology, pharmacokinetics, and metabolism of acetothiolutamide, a novel nonsteroidal agonist for the androgen receptor.
The Journal of pharmacology and experimental therapeutics 2003;304(3):1323-33.
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2003: Yin Donghua; He Yali; Perera Minoli A; Hong Seoung Soo; Marhefka Craig; Stourman Nina; Kirkovsky Leonid; Miller Duane D; Dalton James T
Key structural features of nonsteroidal ligands for binding and activation of the androgen receptor.
Molecular pharmacology 2003;63(1):211-23.
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2003: Mahato Ram I; Narang Ajit S; Thoma Laura; Miller Duane D
Emerging trends in oral delivery of peptide and protein drugs.
Critical reviews in therapeutic drug carrier systems 2003;20(2-3):153-214.
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2002: Lalchandani Shilpa G; Lei Longping; Zheng Weiping; Suni Mustafa M; Moore Bob M; Liggett Stephen B; Miller Duane D; Feller Dennis R
Yohimbine dimers exhibiting selectivity for the human alpha 2C-adrenoceptor subtype.
The Journal of pharmacology and experimental therapeutics 2002;303(3):979-84.
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2002: Wang Dong-an; Narang Ajit S; Kotb Malak; Gaber A Osama; Miller Duane D; Kim Sung Wan; Mahato Ram I
Novel branched poly(ethylenimine)-cholesterol water-soluble lipopolymers for gene delivery.
Biomacromolecules 2002;3(6):1197-207.
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2002: He Yali; Yin Donghua; Perera Minoli; Kirkovsky Leonid; Stourman Nina; Li Wei; Dalton James T; Miller Duane D
Novel nonsteroidal ligands with high binding affinity and potent functional activity for the androgen receptor.
European journal of medicinal chemistry 2002;37(8):619-34.
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2001: Donkor I O; Zheng X; Han J; Lacy C; Miller D D
Significance of hydrogen bonding at the S(1)' subsite of calpain I.
Bioorganic & medicinal chemistry letters 2001;11(13):1753-5.
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2001: Marhefka C A; Moore B M; Bishop T C; Kirkovsky L; Mukherjee A; Dalton J T; Miller D D
Homology modeling using multiple molecular dynamics simulations and docking studies of the human androgen receptor ligand binding domain bound to testosterone and nonsteroidal ligands.
Journal of medicinal chemistry 2001;44(11):1729-40.
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2001: Baker D L; Desiderio D M; Miller D D; Tolley B; Tigyi G J
Direct quantitative analysis of lysophosphatidic acid molecular species by stable isotope dilution electrospray ionization liquid chromatography-mass spectrometry.
Analytical biochemistry 2001;292(2):287-95.
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2001: Liliom K; Sun G; Bünemann M; Virág T; Nusser N; Baker D L; Wang D A; Fabian M J; Brandts B; Bender K; Eickel A; Malik K U; Miller D D; Desiderio D M; Tigyi G; Pott L
Sphingosylphosphocholine is a naturally occurring lipid mediator in blood plasma: a possible role in regulating cardiac function via sphingolipid receptors.
The Biochemical journal 2001;355(Pt 1):189-97.
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2001: Konkar A A; Nikulin V I; De Los Angeles J; Hong S S; Fertel R H; Miller D D; Feller D R
Biochemical activities of trimetoquinol analogs at human beta(1)- and beta(3)-adrenergic receptors.
Pharmacology 2001;62(1):45-55.
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2000: Donkor I O; Zheng X; Miller D D
Synthesis and calpain inhibitory activity of alpha-ketoamides with 2,3-methanoleucine stereoisomers at the P2 position.
Bioorganic & medicinal chemistry letters 2000;10(22):2497-500.
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2000: Donkor I O; Zheng X; Han J; Miller D D
Asymmetric synthesis of 2,3-methanoleucine stereoisomers from common intermediates.
Chirality 2000;12(7):551-7.
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2000: Zheng W; Lei L; Lalchandani S; Sun G; Feller D R; Miller D D
Yohimbine dimers exhibiting binding selectivities for human alpha2a- versus alpha2b-adrenergic receptors.
Bioorganic & medicinal chemistry letters 2000;10(7):627-30.
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2000: Mehta R C; Salazar-Bookaman M M; Fertel R H; De Los Angeles J; Nikulin V I; Fraundorfer P F; Miller D D; Feller D R
Biochemical and functional characterization of 1-benzyl substituted trimetoquinol affinity analogs on rat and human beta-adrenoceptors.
Biochemical pharmacology 2000;59(5):517-29.
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2000: He Y; Nikulin V I; Vansal S S; Feller D R; Miller D D
Synthesis and human beta-adrenoceptor activity of 1-(3,5-diiodo-4- methoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-6-ol derivatives in vitro.
Journal of medicinal chemistry 2000;43(4):591-8.
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2000: Kirkovsky L; Mukherjee A; Yin D; Dalton J T; Miller D D
Chiral nonsteroidal affinity ligands for the androgen receptor. 1. Bicalutamide analogues bearing electrophilic groups in the B aromatic ring.
Journal of medicinal chemistry 2000;43(4):581-90.
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2000: Zheng X; Donkor I O; Miller D D; Ross C R
Unprecedented crystallization and X-ray crystal structure of racemic N(alpha)-(t-butyloxycarbonyl)-L-L-phenylalanine N-methoxy-N-methylamide.
Chirality 2000;12(1):2-6.
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1999: Konkar A A; Vansal S S; Shams G; Fraundorfer P F; Zheng W P; Nikulin V I; De Los Angeles J; Fertel R H; Miller D D; Feller D R
Beta-adrenoceptor subtype activities of trimetoquinol derivatives: biochemical studies on human beta-adrenoceptors expressed in chinese hamster ovary cells.
The Journal of pharmacology and experimental therapeutics 1999;291(2):875-83.
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1999: Mukherjee A; Kirkovsky L I; Kimura Y; Marvel M M; Miller D D; Dalton J T
Affinity labeling of the androgen receptor with nonsteroidal chemoaffinity ligands.
Biochemical pharmacology 1999;58(8):1259-67.
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1999: Jing L; Jagadeesh J M; De Los Angeles J; Miller D D; Patil P N
Depolarization of membrane potential and the smooth muscle contraction by isothiocyanatobenzyl imidazoline in guinea-pig stomach circular muscle.
Naunyn-Schmiedeberg's archives of pharmacology 1999;360(3):337-43.
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1999: Wolfe M S; De Los Angeles J; Miller D D; Xia W; Selkoe D J
Are presenilins intramembrane-cleaving proteases? Implications for the molecular mechanism of Alzheimer's disease.
Biochemistry 1999;38(35):11223-30.
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1999: Zheng W; Nikulin V I; Konkar A A; Vansal S S; Shams G; Feller D R; Miller D D
2-Amino-4-benzyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridines: novel selective beta3-adrenoceptor agonists.
Journal of medicinal chemistry 1999;42(12):2287-94.
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1999: Tigyi G; Fisher D J; Lilion K; Guo Z; Virag T; Sun G; Miller D D; Murakami-Murofushi K; Kobayashi S; Erickson J R
Determinants of receptor subtype specificity in the LPA-like lipid mediator family.
Advances in experimental medicine and biology 1999;469():245-51.
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1998: Fischer D J; Liliom K; Guo Z; Nusser N; Virág T; Murakami-Murofushi K; Kobayashi S; Erickson J R; Sun G; Miller D D; Tigyi G
Naturally occurring analogs of lysophosphatidic acid elicit different cellular responses through selective activation of multiple receptor subtypes.
Molecular pharmacology 1998;54(6):979-88.
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1998: Liliom K; Fischer D J; Virág T; Sun G; Miller D D; Tseng J L; Desiderio D M; Seidel M C; Erickson J R; Tigyi G
Identification of a novel growth factor-like lipid, 1-O-cis-alk-1'-enyl-2-lyso-sn-glycero-3-phosphate (alkenyl-GP) that is present in commercial sphingolipid preparations.
The Journal of biological chemistry 1998;273(22):13461-8.
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1998: Lei L; Vaghy P L; Slavica M; De Los Angeles J; Smith B; Miller D D; Feller D R
Activation of L-type calcium channel by tolazoline derivatives: role of isothiocyanate moiety.
Journal of cardiovascular pharmacology 1998;31(5):721-33.
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1998: Sun G; Slavica M; Uretsky N J; Wallace L J; Shams G; Weinstein D M; Miller J C; Miller D D
Design and synthesis of enantiomers of 3,5-dinitro-o-tyrosine: alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropanoic acid (AMPA) receptor antagonists.
Journal of medicinal chemistry 1998;41(7):1034-41.
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1998: Dalton J T; Mukherjee A; Zhu Z; Kirkovsky L; Miller D D
Discovery of nonsteroidal androgens.
Biochemical and biophysical research communications 1998;244(1):1-4.
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1997: Hill R A; Wallace L J; Miller D D; Weinstein D M; Shams G; Tai H; Layer R T; Willins D; Uretsky N J; Danthi S N
Structure--activity studies for alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropanoic acid receptors: acidic hydroxyphenylalanines.
Journal of medicinal chemistry 1997;40(20):3182-91.
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1997: Zhang X; De Los Angeles J E; He M Y; Dalton J T; Shams G; Lei L; Patil P N; Feller D R; Miller D D; Hsu F L
Medetomidine analogs as alpha 2-adrenergic ligands. 3. Synthesis and biological evaluation of a new series of medetomidine analogs and their potential binding interactions with alpha 2-adrenoceptors involving a "methyl pocket".
Journal of medicinal chemistry 1997;40(19):3014-24.
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1997: Shams G; Romstedt K J; Lust L A; Clark M T; Miller D D; Feller D R
Beta-adrenergic receptor and platelet inhibitory activities of a new series of trimetoquinol and related benzazepine analogs.
General pharmacology 1997;28(2):323-30.
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1997: Christoff J J; Bradley L; Miller D D; Lei L; Rodriguez F; Fraundorfer P; Romstedt K; Shams G; Feller D R
Synthesis and evaluation of trimetoquinol derivatives: novel thromboxane A2/prostaglandin H2 antagonists with diminished beta-adrenergic agonist activity.
Journal of medicinal chemistry 1997;40(1):85-91.
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1996: Ishikawa H; Miller D D; Patil P N
Comparison of post-junctional alpha-adrenoceptors in iris dilator muscle of humans, and albino and pigmented rabbits.
Naunyn-Schmiedeberg's archives of pharmacology 1996;354(6):765-72.
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1996: Sun G; Uretsky N J; Wallace L J; Shams G; Weinstein D M; Miller D D
Synthesis of chiral 1-(2'-amino-2'-carboxyethyl)-1,4-dihydro-6,7-quinoxaline-2,3-diones: alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptor agonists and antagonists.
Journal of medicinal chemistry 1996;39(22):4430-8.
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1996: De Los Angeles J E; Nikulin V I; Shams G; Konkar A A; Mehta R; Feller D R; Miller D D
Iodinated analogs of trimetoquinol as highly potent and selective beta 2-adrenoceptor ligands.
Journal of medicinal chemistry 1996;39(19):3701-11.
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1996: Ishikawa H; Miller D D; Patil P N
Irreversible agonist and antagonist properties of isothiocyanatobenzyl imidazoline in albino rabbit iris muscles.
Naunyn-Schmiedeberg's archives of pharmacology 1996;354(3):362-8.
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1996: Lezama E J; Konkar A A; Salazar-Bookaman M M; Miller D D; Feller D R
Pharmacological study of atypical beta-adrenoceptors in rat esophageal smooth muscle.
European journal of pharmacology 1996;308(1):69-80.
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1996: Zhang X; Yao X T; Dalton J T; Shams G; Lei L; Patil P N; Feller D R; Hsu F L; George C; Miller D D
Medetomidine analogs as alpha 2-adrenergic ligands. 2. Design, synthesis, and biological activity of conformationally restricted naphthalene derivatives of medetomidine.
Journal of medicinal chemistry 1996;39(15):3001-13.
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1996: Konkar A A; Fraundorfer P F; Fertel R H; Burkman A M; Miller D D; Feller D R
Pharmacological activities of trimetoquinol and 1-benzyl halogen-substituted analogues on rat beta-adrenoceptor subtypes.
European journal of pharmacology 1996;305(1-3):63-71.
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1996: Mukherjee A; Kirkovsky L; Yao X T; Yates R C; Miller D D; Dalton J T
Enantioselective binding of Casodex to the androgen receptor.
Xenobiotica; the fate of foreign compounds in biological systems 1996;26(2):117-22.
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1996: Ishikawa H; Miller D D; Patil P N
Actions of imidazolines on bovine ciliary artery.
Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics 1996;12(3):313-22.
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1994: Farooqui T; Brooks K; Harrold M W; Miller D D; Wallace L J; Uretsky N J
Interaction of permanently charged metoclopramide analogs with D-2 dopamine receptors.
General pharmacology 1994;25(8):1577-84.
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1994: Fraundorfer P F; Fertel R H; Miller D D; Feller D R
Biochemical and pharmacological characterization of high-affinity trimetoquinol analogs on guinea pig and human beta adrenergic receptor subtypes: evidence for partial agonism.
The Journal of pharmacology and experimental therapeutics 1994;270(2):665-74.
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1994: Hong S S; Romstedt K J; Feller D R; Hsu F L; Cupps T L; Lyon R A; Miller D D
A structure-activity relationship study of benzylic modifications of 4-[1-(1-naphthyl)ethyl]-1H-imidazoles on alpha 1- and alpha 2-adrenergic receptors.
Journal of medicinal chemistry 1994;37(15):2328-33.
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1994: Slavica M; Lei L; Patil P N; Kerezy A; Feller D R; Miller D D
Synthesis and biological activities of a new set of irreversibly acting 2-(4'-isothiocyanatobenzyl)imidazoline analogs in rat thoracic aorta.
Journal of medicinal chemistry 1994;37(12):1874-81.
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1994: Fraundorfer P F; Lezama E J; Salazar-Bookaman M M; Fertel R H; Miller D D; Feller D R
Isomeric-activity ratios of trimetoquinol enantiomers on beta-adrenergic receptor subtypes: functional and biochemical studies.
Chirality 1994;6(2):76-85.
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1993: Romstedt K J; Shin Y; Shams G; Doyle K; Tantishaiyakul V; Clark M T; Adejare A; Hamada A; Miller D D; Feller D R
Halogen-substituted trimetoquinol analogs as thromboxane A2 receptor antagonists in platelets and aorta.
Biochemical pharmacology 1993;46(11):2051-9.
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1993: Shin Y; Romstedt K J; Miller D D; Feller D R
Interactions of nonprostanoid trimetoquinol analogs with thromboxane A2/prostaglandin H2 receptors in human platelets, rat vascular endothelial cells and rat vascular smooth muscle cells.
The Journal of pharmacology and experimental therapeutics 1993;267(3):1017-23.
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1993: Harrold M W; Sriburi A; Matsumoto K; Miller D D; Farooqui T; Uretsky N
The interaction of ammonium, sulfonium, and sulfide analogues of metoclopramide with the dopamine D2 receptor.
Journal of medicinal chemistry 1993;36(21):3166-70.
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1993: Abdel-Ghany Y S; Ihnat M A; Miller D D; Kunin C M; Tong H H
Structure-activity relationship of glycine betaine analogs on osmotolerance of enteric bacteria.
Journal of medicinal chemistry 1993;36(6):784-9.
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1993: Kunin C M; Tong H H; Miller D D; Abdel-Ghany Y; Poggi M C; LeRudulier D
Effect of novel compound, 1-methyl-1-piperidino methane sulfonate (MPMS), on the osmoprotectant activity of glycine betaine, choline and L-proline in Escherichia coli.
Archives of microbiology 1993;160(2):81-6.
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1992: Smar M W; Ares J J; Nakayama T; Itabe H; Kador P F; Miller D D
Selective irreversible inhibitors of aldose reductase.
Journal of medicinal chemistry 1992;35(6):1117-20.
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1992: Willins D L; Wallace L J; Miller D D; Uretsky N J
alpha-Amino-3-hydroxy-5-methylisoxazole-4-propionate/kainate receptor antagonists in the nucleus accumbens and ventral pallidum decrease the hypermotility response to psychostimulant drugs.
The Journal of pharmacology and experimental therapeutics 1992;260(3):1145-51.
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1992: Amemiya Y; Hong S S; Venkataraman B V; Patil P N; Shams G; Romstedt K; Feller D R; Hsu F L; Miller D D
Synthesis and alpha-adrenergic activities of 2- and 4-substituted imidazoline and imidazole analogues.
Journal of medicinal chemistry 1992;35(4):750-5.
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1992: Markovich K M; Tantishaiyakul V; Hamada A; Miller D D; Romstedt K J; Shams G; Shin Y; Fraundorfer P F; Doyle K; Feller D R
Synthesis of halogenated trimetoquinol derivatives and evaluation of their beta-agonist and thromboxane A2 (TXA2) antagonist activities.
Journal of medicinal chemistry 1992;35(3):466-79.
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1992: Hong S S; Romstedt K J; Feller D R; Hsu F L; George C; Cupps T L; Lyon R A; Miller D D
Resolution and adrenergic activities of the optical isomers of 4-[1-(1-naphthyl)ethyl]-1H-imidazole.
Chirality 1992;4(7):432-8.
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1992: Esbenshade T A; Hamada A; Miller D D; Feller D R
Effects of the stereochemical orientation of phenethylamines and imidazolines on alpha-adrenergic receptor-mediated DNA synthesis in primary cultured rat hepatocytes.
Chirality 1992;4(5):279-85.
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1991: Venkataraman B V; Shams G; Hamada A; Amemiya Y; Tantishaiyakul V; Hsu F; Fashempour J; Romstedt K J; Miller D D; Feller D R
Structure-activity studies of new imidazolines on adrenoceptors of rat aorta and human platelets.
Naunyn-Schmiedeberg's archives of pharmacology 1991;344(4):454-63.
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1991: Shams G; Venkataraman B V; Hamada A; Miller D D; Patil P N; Feller D R
Diversity of the pharmacological actions of some tolazoline analogues in human platelets and rat aorta.
European journal of pharmacology 1991;199(3):315-23.
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1991: Shin Y; Romstedt K J; Doyle K; Harrold M W; Gerhardt M A; Miller D D; Patil P N; Feller D R
Pharmacologic antagonism of thromboxane A2 receptors by trimetoquinol analogs in vitro and in vivo.
Chirality 1991;3(2):112-7.
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1991: Shams G; Fedyna J; Romstedt K J; Adejare A; Miller D D; Roche V F; Feller D R
Pharmacological properties of novel bicyclic isoquinoline analogs in isolated guinea pig atria, trachea and in human platelets: relationship to trimetoquinol.
General pharmacology 1991;22(6):1155-63.
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1990: Shams G; Harrold M W; Grazyl B; Miller D D; Feller D R
Pharmacological evaluation of the beta-adrenoceptor agonist properties of N-benzyl substituted trimetoquinol analogues.
European journal of pharmacology 1990;184(2-3):251-6.
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1990: Shams G; Romstedt K J; Gerhardt M A; Harrold M W; Miller D D; Feller D R
Pharmacological evaluation of the beta-adrenoceptor agonist and thromboxane receptor blocking properties of 1-benzyl substituted trimetoquinol analogues.
European journal of pharmacology 1990;184(1):21-31.
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1990: Ahn C H; Shams G; Schotzinger R L; Miller D D; Feller D R
Stereostructure activity relationships of catecholamines on human platelet function.
Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.) 1990;194(2):149-56.
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1990: Miller D D; Hamada A; Clark M T; Adejare A; Patil P N; Shams G; Romstedt K J; Kim S U; Intrasuksri U; McKenzie J L
Synthesis and alpha 2-adrenoceptor effects of substituted catecholimidazoline and catecholimidazole analogues in human platelets.
Journal of medicinal chemistry 1990;33(4):1138-44.
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1990: Shams G; Wallace L J; Miller D D; Feller D R
Effects of thromboxane A2 on thoracic aorta of young and old rats: use of selective thromboxane receptor antagonists.
Pharmacology 1990;40(1):27-32.
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1989: Rice P J; Miller D D; Patil P N
Epinephrine enantiomers: affinity, efficacy and potency relationships in rat smooth muscle tissues.
The Journal of pharmacology and experimental therapeutics 1989;249(1):242-8.
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1989: Harrold M W; Wallace R A; Farooqui T; Wallace L J; Uretsky N; Miller D D
Synthesis and D2 dopaminergic activity of pyrrolidinium, tetrahydrothiophenium, and tetrahydrothiophene analogues of sulpiride.
Journal of medicinal chemistry 1989;32(4):874-80.
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1989: Nichols A J; Hamada A; Adejare A; Miller D D; Patil P N; Ruffolo R R
Effect of aromatic fluorine substitution on the alpha and beta adrenoceptor-mediated effects of 3,4-dihydroxytolazoline in the pithed rat.
The Journal of pharmacology and experimental therapeutics 1989;248(2):671-6.
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1989: Farooqui T; Wallace R A; Miller D D; Uretsky N J
Effect of the inhibition of dopamine uptake on the dopamine- and dimethyldopamine-induced-inhibition of the potassium-evoked release of [3H]acetylcholine from striatal slices.
General pharmacology 1989;20(6):731-6.
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1989: Venkataraman B V; Hamada A; Shams G; Miller D D; Feller D R; Patil P N
Paradoxical effects of isothiocyanate analog of tolazoline on rat aorta and human platelets.
Blood vessels 1989;26(6):335-46.
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1989: Rice P J; Miller D D; Sokoloski T D; Patil P N
Pharmacologic implications of alpha-adrenoreceptor interactive parameters for epinephrine enantiomers in the rat vas deferens.
Chirality 1989;1(1):14-9.
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1988: Ruffolo R R; Nichols A J; Patil P N; Hamada A; Clark M; Miller D D
Effects of benzylic hydroxyl substitution on the alpha-adrenoceptor blocking activity of tolazoline.
European journal of pharmacology 1988;157(2-3):235-9.
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1988: Harrold M W; Grajzl B; Shin Y M; Romstedt K J; Feller D R; Miller D D
Synthesis and thromboxane A2 antagonist activity of N-benzyltrimetoquinol analogues.
Journal of medicinal chemistry 1988;31(8):1506-12.
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1988: Ahn C H; Romstedt K J; Wallace L J; Miller D D; Feller D R
Characterization of the inhibition of U46619-mediated human platelet activation by the trimetoquinol isomers. Evidence for endoperoxide/thromboxane A2 receptor blockade.
Biochemical pharmacology 1988;37(15):3023-33.
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1988: Miller D D; Harrold M; Wallace R A; Wallace L J; Uretsky N J
Dopaminergic drugs in the cationic form interact with D2 dopamine receptors.
Trends in pharmacological sciences 1988;9(8):282-4.
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1988: Lamba-Kanwal V K; Hamada A; Adejare A; Clark M T; Miller D D; Patil P N
Activation of alpha-1 adrenoreceptors of rat aorta by analogs of imidazoline.
The Journal of pharmacology and experimental therapeutics 1988;245(3):793-7.
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1988: Ahn C H; Wallace L J; Miller D D; Feller D R
Use of [3H]trimetoquinol as a radioligand in human platelets: interaction with putative endoperoxide/thromboxane A2 receptor sites.
Thrombosis research 1988;50(3):387-99.
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1987: Harrold M W; Chang Y A; Wallace R A; Farooqui T; Wallace L J; Uretsky N; Miller D D
Charged analogues of chlorpromazine as dopamine antagonists.
Journal of medicinal chemistry 1987;30(9):1631-5.
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1987: Rice P J; Hamada A; Miller D D; Patil P N
Asymmetric catecholimidazolines and catecholamidines: affinity and efficacy relationships at the alpha adrenoreceptor in rat aorta.
The Journal of pharmacology and experimental therapeutics 1987;242(1):121-30.
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1987: Fedyna J S; Adejare A; Miller D D; Feller D R
Pharmacological evaluation of the beta-adrenoceptor agonist and thromboxane antagonist properties of N-substituted trimetoquinol analogues.
European journal of pharmacology 1987;135(2):161-71.
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1987: Harrold M W; Gerhardt M A; Romstedt K; Feller D R; Miller D D
Synthesis and platelet antiaggregatory activity of trimetoquinol analogs as endoperoxide/thromboxane A2 antagonists.
Drug design and delivery 1987;1(3):193-207.
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1987: Chang Y A; Ares J; Anderson K; Sabol B; Wallace R A; Farooqui T; Uretsky N; Miller D D
Dopamine agonists: effects of charged and uncharged analogues of dopamine.
Journal of medicinal chemistry 1987;30(1):214-8.
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1987: Clark M T; Adejare A; Shams G; Feller D R; Miller D D
5-fluoro- and 8-fluorotrimetoquinol: selective beta 2-adrenoceptor agonists.
Journal of medicinal chemistry 1987;30(1):86-90.
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1986: Ahn C H; Hamada A; Miller D D; Feller D R
Alpha-adrenoceptor-mediated actions of optical isomers and desoxy analogs of catecholimidazoline and norepinephrine in human platelets: in vitro.
Biochemical pharmacology 1986;35(22):4095-102.
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1986: Adejare A; Miller D D; Fedyna J S; Ahn C H; Feller D R
Syntheses and beta-adrenergic agonist and antiaggregatory properties of N-substituted trimetoquinol analogues.
Journal of medicinal chemistry 1986;29(9):1603-9.
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1986: Clark M T; Chang J; Navran S S; Huzoor-Akbar; Mukhopadhyay A; Amin H; Feller D R; Miller D D
Synthesis and investigation of the beta-adrenoceptor agonist and platelet antiaggregatory properties of 1,7,8-trisubstituted 2,3,4,5-tetrahydro-1H-2-benzazepine analogues of trimetoquinol.
Journal of medicinal chemistry 1986;29(2):181-5.
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1985: Huzoor-Akbar; Mukhopadhyay A; Anderson K S; Navran S S; Romstedt K; Miller D D; Feller D R
Antagonism of prostaglandin-mediated responses in platelets and vascular smooth muscle by 13-azaprostanoic acid analogs. Evidence for selective blockade of thromboxane A2 responses.
Biochemical pharmacology 1985;34(5):641-7.
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1985: Mukhopadhyay A; Navran S S; Amin H M; Abdel-Aziz S A; Chang J; Sober D J; Miller D D; Feller D R
Effect of trimetoquinol analogs for antagonism of endoperoxide/thromboxane A2-mediated responses in human platelets and rat aorta.
The Journal of pharmacology and experimental therapeutics 1985;232(1):1-9.
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1984: Hamada A; Chang Y A; Uretsky N; Miller D D
Dopaminergic agonists: comparative actions of amine and sulfonium analogues of dopamine.
Journal of medicinal chemistry 1984;27(5):675-80.
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1984: Navran S S; Romstedt K; Chang J; Miller D D; Feller D R; Huzoor-Akbar
Human platelet activation by bacterial phospholipase C is mediated by phosphatidylinositol hydrolysis but not generation of phosphatidic acid: inhibition by a selective inhibitor of phospholipase C.
Thrombosis research 1984;33(5):499-510.
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1983: Miller D D; Hamada A; Craig E C; Christoph G G; Gallucci J C; Rice P J; Banning J W; Patil P N
Optically active catecholimidazolines: a study of steric interactions at alpha-adrenoreceptors.
Journal of medicinal chemistry 1983;26(7):957-63.
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1983: Ruffolo R R; Rice P J; Patil P N; Hamada A; Miller D D
Differences in the applicability of the easson-stedman hypothesis to the alpha 1- and alpha 2-adrenergic effects of phenethylamines and imidazolines.
European journal of pharmacology 1983;86(3-4):471-5.
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1982: Akbar H; Navran S S; Chang J; Miller D D; Feller D R
Investigation of the effects of phospholipase C on human platelets: evidence that aggregation induced by phospholipase C is independent of prostaglandin generation, released ADP and is modulated by cyclic AMP.
Thrombosis research 1982;27(4):405-17.
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1982: Akbar H; Navran S S; Miller D D; Feller D R
Antiplatelet actions of trimetoquinol isomers: evidence for inhibition of a prostaglandin-independent pathway of platelet aggregation.
Biochemical pharmacology 1982;31(5):886-9.
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1982: Mukhopadhyay A; Sober D J; Chang J; Slenn R T; Amin H M; Miller D D; Feller D R
Bronchoselective actions of a new series of trimetoquinol analogues.
European journal of pharmacology 1982;77(4):209-19.
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1981: Mayo J R; Navran S S; Huzoor-Akbar; Miller D D; Feller D R
Stereo-dependent inhibition of human platelet function by the optical isomers of trimetoquinol.
Biochemical pharmacology 1981;30(16):2237-41.
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1981: Sober D J; Chang J; Fowble J W; Mukhopadhyay A; Feller D R; Miller D D; Fairchild E H
Selective and potent beta 2-adrenoceptor agents within the tetrahydroisoquinoline class: effect of methyl substitution at the benzylic carbon of the 1-(3,4,5-trimethoxybenzyl) group of trimetoquinol.
Journal of medicinal chemistry 1981;24(8):970-4.
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1980: Hsu F L; Hamada A; Booher M E; Fuder H; Patil P N; Miller D D
Optically active derivatives of imidazolines. alpha-Adrenergic blocking properties.
Journal of medicinal chemistry 1980;23(11):1232-5.
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